Compile Data Set for Download or QSAR
Found 51 of ic50 data for polymerid = 50000347
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 1.80nMAssay Description:Inhibition of human ZIPK using KKLNRTLSFAEPG as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5KB8PubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 3.5nMAssay Description:Inhibition of human ZIPK using KKLNRTLSFAEPG as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W380MTPubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50172243(CHEMBL3103192)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of Dapk3 (unknown origin) at by quantitative PCRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53NRMPubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of human recombinant DAPK3 by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67H7NPubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant human DAPK3 in presence of ATP at Km concentration by radiometric filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DN48PPPubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50166251(CHEMBL3799389)copy SMILEScopy InChI
Affinity DataIC50: 140nMAssay Description:Inhibition of DAPK3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N29ZTZPubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50314672(2-(3-bromophenyl)-4-(pyridin-3-ylmethylene)oxazol-...)copy SMILEScopy InChI
Affinity DataIC50: 148nMAssay Description:Inhibition of human recombinant DAPK3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB74R2PubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50314673(2-(2-bromo-4-methoxyphenyl)-4-(pyridin-3-ylmethyle...)copy SMILEScopy InChI
Affinity DataIC50: 157nMAssay Description:Inhibition of human recombinant DAPK3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB74R2PubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50314664(2-(2-chloro-5-iodophenyl)-4-(pyridin-4-ylmethylene...)copy SMILEScopy InChI
Affinity DataIC50: 227nMAssay Description:Inhibition of human recombinant DAPK3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB74R2PubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50554817(CHEMBL4764610)copy SMILES
Affinity DataIC50: 260nMAssay Description:Inhibition of human DAPK3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9GG7PubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50314665(2-(4-chloro-3-nitrophenyl)-4-(pyridin-3-ylmethylen...)copy SMILEScopy InChI
Affinity DataIC50: 279nMAssay Description:Inhibition of human recombinant DAPK3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB74R2PubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50314670(2-(4-bromo-3-methylphenyl)-4-(pyridin-3-ylmethylen...)copy SMILEScopy InChI
Affinity DataIC50: 279nMAssay Description:Inhibition of human recombinant DAPK3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB74R2PubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50314671(2-(4-nitrophenyl)-4-(pyridin-3-ylmethylene)oxazol-...)copy SMILEScopy InChI
Affinity DataIC50: 291nMAssay Description:Inhibition of human recombinant DAPK3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB74R2PubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50314668(2-(3,4-difluorophenyl)-4-(pyridin-3-ylmethylene)ox...)copy SMILEScopy InChI
Affinity DataIC50: 346nMAssay Description:Inhibition of human recombinant DAPK3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB74R2PubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50314669(2-(3-chlorophenyl)-4-(pyridin-3-ylmethylene)oxazol...)copy SMILEScopy InChI
Affinity DataIC50: 360nMAssay Description:Inhibition of human recombinant DAPK3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB74R2PubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50314674(2-(3-methoxyphenyl)-4-(pyridin-3-ylmethylene)oxazo...)copy SMILEScopy InChI
Affinity DataIC50: 395nMAssay Description:Inhibition of human recombinant DAPK3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB74R2PubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50166254(CHEMBL3797466)copy SMILEScopy InChI
Affinity DataIC50: 450nMAssay Description:Inhibition of DAPK3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N29ZTZPubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50166076(CHEMBL3799585)copy SMILEScopy InChI
Affinity DataIC50: 510nMAssay Description:Inhibition of DAPK3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N29ZTZPubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50314667(2-(4-chlorophenyl)-4-(pyridin-3-ylmethylene)oxazol...)copy SMILEScopy InChI
Affinity DataIC50: 530nMAssay Description:Inhibition of human recombinant DAPK3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB74R2PubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50314675(2-(4-methyl-3-nitrophenyl)-4-(pyridin-3-ylmethylen...)copy SMILEScopy InChI
Affinity DataIC50: 534nMAssay Description:Inhibition of human recombinant DAPK3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB74R2PubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50314663(2-phenyl-4-(pyridin-3-ylmethylene)oxazol-5(4H)-one...)copy SMILEScopy InChI
Affinity DataIC50: 583nMAssay Description:Inhibition of human recombinant DAPK3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB74R2PubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50166077(CHEMBL513703)copy SMILEScopy InChI
Affinity DataIC50: 700nMAssay Description:Inhibition of DAPK3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N29ZTZPubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50314666(4-(pyridin-3-ylmethylene)-2-m-tolyloxazol-5(4H)-on...)copy SMILEScopy InChI
Affinity DataIC50: 714nMAssay Description:Inhibition of human recombinant DAPK3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB74R2PubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50566949(CHEMBL4877302)copy SMILES
Affinity DataIC50: 720nMAssay Description:Inhibition of recombinant human ZIPK (1 to 290 residues) using KKLNRTLSFAEPG substrate incubated for 40 mins in presence of [gamma33P]ATP by scintill...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20K2D97PubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50315888(CHEMBL1090360 | N-(3-(5-(2-(3-morpholinophenylamin...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of ZipKMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M908VTPubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM311210((S)-methyl (5-((2-amino-2,4-dimethylpentyl)oxy)-6-...)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RSPPubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM311261((S)-methyl (5-((2-amino-2,4-dimethylpentyl)oxy)-6-...)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RSPPubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50235830(CHEMBL2006765)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of ZIPK (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WQ061VPubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50166121(CHEMBL3797480)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of DAPK3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N29ZTZPubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50580((2Z)-2-(3,4-dihydroxybenzylidene)-6-hydroxy-coumar...)copy SMILEScopy InChI
Affinity DataIC50: 2.33E+3nMAssay Description:Inhibition of human DAPK3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4N3PPubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50305006(5-(2-aminoethyl)-7-(7-(benzo[b]thiophen-2-yl)-1H-i...)copy SMILEScopy InChI
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of ZIPKMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD6ZJJPubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50235820(CHEMBL4066664)copy SMILEScopy InChI
Affinity DataIC50: 4.86E+3nMAssay Description:Inhibition of ZIPK (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WQ061VPubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50235833(CHEMBL4062803)copy SMILEScopy InChI
Affinity DataIC50: 4.98E+3nMAssay Description:Inhibition of ZIPK (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WQ061VPubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50519662(CHEMBL4438748)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human ZIPK (1 to 290 residues) using KKLNRTLSFAEPG substrate incubated for 40 mins in presence of [gamma33P]ATP by radiomet...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC93FGPubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50499634(CHEMBL3741589)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of ZIPK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5CV4PubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50235816(CHEMBL4069365)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of ZIPK (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WQ061VPubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50235817(CHEMBL4078893)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of ZIPK (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WQ061VPubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50429867(CHEMBL2333365)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of ZIPK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC847XPubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50166260(CHEMBL3799505)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of DAPK3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N29ZTZPubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50389320(CHEMBL2063926)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of DAPK3 by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9BV6PubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50135286(CHEMBL3745885)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human ZIPK using [KKLNRTLSFAEPG] as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24Q7WT8PubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50516171(CHEMBL4446892)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human ZIPK (1 to 290 residues) using KKLNRTLSFAEPG as substrate measured after 40 mins in presence of [gamma33P]ATP by radi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7SNDPubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50238989(CHEMBL4087337)copy SMILEScopy InChI
Affinity DataIC50: 1.22E+4nMAssay Description:Inhibition of human DAPK3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4N3PPubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50238990(CHEMBL4105195)copy SMILEScopy InChI
Affinity DataIC50: 1.89E+4nMAssay Description:Inhibition of human DAPK3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4N3PPubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM13533(1-[2-(4-methylphenyl)-5-tert-butyl-pyrazol-3-yl]-3...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of ZIPKMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC61NHPubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50359359(CHEMBL1929238)copy SMILEScopy InChI
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of ZIPKMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC61NHPubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50024284(CHEMBL3334979)copy SMILEScopy InChI
Affinity DataIC50: 3.98E+4nMAssay Description:Inhibition of human DAPK3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4N3PPubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50380246(CHEMBL2017214)copy SMILEScopy InChI
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of DAPK3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ88N1PubMed
TargetDeath-associated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50537742(CHEMBL4634634 | US11179389, Compound 1-14)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human full-length GST-tagged DAPK3 expressed in baculovirus expression system using FRET-labeled Ser/Thr 13 peptide as subs...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
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