Compile Data Set for Download or QSAR
Found 10 of ic50 data for polymerid = 50005714,50007118
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373848(CHEMBL255779)copy SMILEScopy InChI
Affinity DataIC50: 4.90E+4nMAssay Description:Antagonist activity at human Dvl1 assessed as inhibition of interaction between Dvl1 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8SPTPubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373845(CHEMBL402939)copy SMILEScopy InChI
Affinity DataIC50: 7.80E+4nMAssay Description:Antagonist activity at human Dvl1 assessed as inhibition of interaction between Dvl1 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8SPTPubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373844(CHEMBL272948)copy SMILEScopy InChI
Affinity DataIC50: 9.70E+4nMAssay Description:Antagonist activity at human Dvl1 assessed as inhibition of interaction between Dvl1 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8SPTPubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373847(CHEMBL256605)copy SMILEScopy InChI
Affinity DataIC50: 1.57E+5nMAssay Description:Antagonist activity at human Dvl1 assessed as inhibition of interaction between Dvl1 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8SPTPubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373851(CHEMBL256431)copy SMILEScopy InChI
Affinity DataIC50: 1.59E+5nMAssay Description:Antagonist activity at human Dvl1 assessed as inhibition of interaction between Dvl1 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8SPTPubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373846(CHEMBL401537)copy SMILEScopy InChI
Affinity DataIC50: 1.97E+5nMAssay Description:Antagonist activity at human Dvl1 assessed as inhibition of interaction between Dvl1 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8SPTPubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373843(CHEMBL410400)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+5nMAssay Description:Antagonist activity at human Dvl1 assessed as inhibition of interaction between Dvl1 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8SPTPubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373849(CHEMBL255988)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+5nMAssay Description:Antagonist activity at human Dvl1 assessed as inhibition of interaction between Dvl1 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8SPTPubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373850(CHEMBL404331)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+5nMAssay Description:Antagonist activity at human Dvl1 assessed as inhibition of interaction between Dvl1 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8SPTPubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50231890(2-((2-carboxyethyl)carbamoyl)-6-methyl-3-phenethyl...)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+5nMAssay Description:Antagonist activity at human Dvl1 assessed as inhibition of interaction between Dvl1 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8SPTPubMed