Compile Data Set for Download or QSAR
Found 26 of ic50 data for polymerid = 8936
TargetSerine/threonine-protein kinase PAK 3(Homo sapiens (Human))TBA
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 0.235nMAssay Description:Inhibition of human PAK3 using RRRLSFAEPG as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5KB8PubMed
TargetSerine/threonine-protein kinase PAK 3(Homo sapiens (Human))TBA
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 0.343nMAssay Description:Inhibition of human PAK3 using RRRLSFAEPG as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W380MTPubMed
TargetSerine/threonine-protein kinase PAK 3(Homo sapiens (Human))TBA
LigandPNGBDBM50468260(CHEMBL4282837)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of GST-tagged PAK3 (unknown origin) expressed in Escherichia coli using peptide PC9 substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9DG3PubMed
TargetSerine/threonine-protein kinase PAK 3(Homo sapiens (Human))TBA
LigandPNGBDBM50112347(CHEMBL3609327 | FRAX597)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Inhibition of recombinant human PAK3 by Z'-LYTE assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 3(Homo sapiens (Human))TBA
LigandPNGBDBM50112347(CHEMBL3609327 | FRAX597)copy SMILEScopy InChI
Affinity DataIC50: 19.3nMAssay Description:IC50 values were determined using a 10 concentration point, non-radioactive, functional assay that employs a fluorescence-based, coupled enzyme forma...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 3(Homo sapiens (Human))TBA
LigandPNGBDBM50112347(CHEMBL3609327 | FRAX597)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Inhibition of PAK3 (unknown origin) using lipid substrate measured after 40 mins by ADP-glo kinase assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 3(Homo sapiens (Human))TBA
LigandPNGBDBM50112355(CHEMBL3609326)copy SMILEScopy InChI
Affinity DataIC50: 55nMAssay Description:Inhibition of full length PAK3 (unknown origin) by Z'-LYTE assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2BQSPubMed
TargetSerine/threonine-protein kinase PAK 3(Homo sapiens (Human))TBA
LigandPNGBDBM50434330(CHEMBL2386715)copy SMILEScopy InChI
Affinity DataIC50: 64nMAssay Description:Inhibition of PAK3-mediated MEK1 phosphorylation at Ser298 in human EBC1 cells after 2 hrs by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X068DZPubMed
TargetSerine/threonine-protein kinase PAK 3(Homo sapiens (Human))TBA
LigandPNGBDBM50434331(CHEMBL2386717)copy SMILEScopy InChI
Affinity DataIC50: 71nMAssay Description:Inhibition of PAK3-mediated MEK1 phosphorylation at Ser298 in human EBC1 cells after 2 hrs by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X068DZPubMed
TargetSerine/threonine-protein kinase PAK 3(Homo sapiens (Human))TBA
LigandPNGBDBM101618(US8530652, 114)copy SMILEScopy InChI
Affinity DataIC50: 99nMAssay Description:Inhibition of PAK3 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 3(Homo sapiens (Human))TBA
LigandPNGBDBM50434332(CHEMBL2386716)copy SMILEScopy InChI
Affinity DataIC50: 133nMAssay Description:Inhibition of PAK3-mediated MEK1 phosphorylation at Ser298 in human EBC1 cells after 2 hrs by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X068DZPubMed
TargetSerine/threonine-protein kinase PAK 3(Homo sapiens (Human))TBA
LigandPNGBDBM50601538(CHEMBL5090394)copy SMILES
Affinity DataIC50: 140nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66QTGPubMed
TargetSerine/threonine-protein kinase PAK 3(Homo sapiens (Human))TBA
LigandPNGBDBM50434333(CHEMBL2386718)copy SMILEScopy InChI
Affinity DataIC50: 244nMAssay Description:Inhibition of PAK3-mediated MEK1 phosphorylation at Ser298 in human EBC1 cells after 2 hrs by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X068DZPubMed
TargetSerine/threonine-protein kinase PAK 3(Homo sapiens (Human))TBA
LigandPNGBDBM50462709(CHEMBL4245507)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PAK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XP77MHPubMed
TargetSerine/threonine-protein kinase PAK 3(Homo sapiens (Human))TBA
LigandPNGBDBM50564348(CHEMBL4780410)copy SMILES
Affinity DataIC50: 1.37E+3nMAssay Description:Inhibition of PAK3 (unknown origin) using lipid substrate measured after 40 mins by ADP-glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20C50JGPubMed
TargetSerine/threonine-protein kinase PAK 3(Homo sapiens (Human))TBA
LigandPNGBDBM50579499(CHEMBL4847875)copy SMILES
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of wild-type human full length PAK3 (M1 to R544 residues) expressed in bacterial expression system by Kinomescan methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W3815DPubMed
TargetSerine/threonine-protein kinase PAK 3(Homo sapiens (Human))TBA
LigandPNGBDBM50429867(CHEMBL2333365)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PAK3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC847XPubMed
TargetSerine/threonine-protein kinase PAK 3(Homo sapiens (Human))TBA
LigandPNGBDBM50448771(CHEMBL3128042)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PAK3 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 3(Homo sapiens (Human))TBA
LigandPNGBDBM50519662(CHEMBL4438748)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant full-length human PAK3 using RRRLSFAEPG as substrate measured after 40 mins in presence of [gamma33P]ATP by radiometric sci...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC93FGPubMed
TargetSerine/threonine-protein kinase PAK 3(Homo sapiens (Human))TBA
LigandPNGBDBM50389320(CHEMBL2063926)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PAK3 by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9BV6PubMed
TargetSerine/threonine-protein kinase PAK 3(Homo sapiens (Human))TBA
LigandPNGBDBM50135286(CHEMBL3745885)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human PAK3 using [KKLNRTLSFAEPG] substrateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24Q7WT8PubMed
TargetSerine/threonine-protein kinase PAK 3(Homo sapiens (Human))TBA
LigandPNGBDBM50001733(CHEMBL3133821)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human PAK3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CN0PubMed
TargetSerine/threonine-protein kinase PAK 3(Homo sapiens (Human))TBA
LigandPNGBDBM13533(1-[2-(4-methylphenyl)-5-tert-butyl-pyrazol-3-yl]-3...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of PAK3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC61NHPubMed
TargetSerine/threonine-protein kinase PAK 3(Homo sapiens (Human))TBA
LigandPNGBDBM50359359(CHEMBL1929238)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of PAK3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC61NHPubMed
TargetSerine/threonine-protein kinase PAK 3(Homo sapiens (Human))TBA
LigandPNGBDBM50380246(CHEMBL2017214)copy SMILEScopy InChI
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of PAK3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ88N1PubMed
TargetSerine/threonine-protein kinase PAK 3(Homo sapiens (Human))TBA
LigandPNGBDBM50537742(CHEMBL4634634 | US11179389, Compound 1-14)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant full length human His-tagged PAK3 expressed in baculovirus expression system using serine/threonine-20 peptide as substrate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed