Compile Data Set for Download or QSAR
Found 731 of ki data for polymerid = 9852
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50565825(CHEMBL4777048)copy SMILES
Affinity DataKi:  0.0219nMAssay Description:Displacement of [125I]-[NIe,DPhe7]-alpha-MSH from human MC3R expressed in HEK293 cell membranes incubated for 120 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53QMNPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50565825(CHEMBL4777048)copy SMILES
Affinity DataKi:  0.0220nMAssay Description:Displacement of [125I]-[NIe,DPhe7]-alpha-MSH from human MC3R expressed in HEK293 cell membranes incubated for 120 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53QMNPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50565826(CHEMBL4794121)copy SMILES
Affinity DataKi:  0.0309nMAssay Description:Displacement of [125I]-[NIe,DPhe7]-alpha-MSH from human MC3R expressed in HEK293 cell membranes incubated for 120 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53QMNPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50565826(CHEMBL4794121)copy SMILES
Affinity DataKi:  0.0310nMAssay Description:Displacement of [125I]-[NIe,DPhe7]-alpha-MSH from human MC3R expressed in HEK293 cell membranes incubated for 120 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53QMNPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50565828(CHEMBL4798971)copy SMILES
Affinity DataKi:  0.0320nMAssay Description:Displacement of [125I]-[NIe,DPhe7]-alpha-MSH from human MC3R expressed in HEK293 cell membranes incubated for 120 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53QMNPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50565828(CHEMBL4798971)copy SMILES
Affinity DataKi:  0.0324nMAssay Description:Displacement of [125I]-[NIe,DPhe7]-alpha-MSH from human MC3R expressed in HEK293 cell membranes incubated for 120 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53QMNPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50165935(Ac-YRMEHdFRWGSPPKD-NH2 | CHEMBL414718)copy SMILEScopy InChI
Affinity DataKi:  0.110nMAssay Description:Inhibition of [125I]-NDP-alpha-MSH binding to melanocortin-3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2251HQZPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50080576(CHEMBL3422426)copy SMILES
Affinity DataKi:  0.129nMAssay Description:Displacement of [125I]-[NIe,DPhe7]-alpha-MSH from human MC3R expressed in HEK293 cell membranes incubated for 120 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53QMNPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50080576(CHEMBL3422426)copy SMILES
Affinity DataKi:  0.129nMAssay Description:Displacement of [125I]-[NIe,DPhe7]-alpha-MSH from human MC3R expressed in HEK293 cell membranes incubated for 120 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53QMNPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50565819(CHEMBL4794168)copy SMILES
Affinity DataKi:  0.135nMAssay Description:Displacement of [125I]-[NIe,DPhe7]-alpha-MSH from human MC3R expressed in HEK293 cell membranes incubated for 120 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53QMNPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50565819(CHEMBL4794168)copy SMILES
Affinity DataKi:  0.135nMAssay Description:Displacement of [125I]-[NIe,DPhe7]-alpha-MSH from human MC3R expressed in HEK293 cell membranes incubated for 120 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53QMNPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50134955(CHEMBL2370968 | H-Tyr-Val-Nle-Gly-Pro-D-Nal(2')-Ar...)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Binding affinity against human Melanocortin 3 receptor by gamma-MCH displacement.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SJ1K0PPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM82411(CAS_75921-69-6 | NDP-MSH)copy SMILEScopy InChI
Affinity DataKi:  0.224nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M32T8HPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM85021(alpha-MSH, [Nle4, D-Phe7])copy SMILEScopy InChI
Affinity DataKi:  0.224nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W98M7PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50105879(15-(2-Acetylamino-hexanoylamino)-6-(3-guanidino-pr...)copy SMILEScopy InChI
Affinity DataKi:  0.230nMAssay Description:Binding affinity against human melanocortin receptor 3 (hMC3R) (concentration of the peptide at 50% specific binding)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RF5T9SPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50165931(CHEMBL415165 | NDP-SYSMEHFRWGKPVG)copy SMILEScopy InChI
Affinity DataKi:  0.230nMAssay Description:Inhibition of [125I]-NDP-alpha-MSH binding to melanocortin-3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2251HQZPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50565829(CHEMBL4788071)copy SMILES
Affinity DataKi:  0.330nMAssay Description:Displacement of [125I]-[NIe,DPhe7]-alpha-MSH from human MC3R expressed in HEK293 cell membranes incubated for 120 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53QMNPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50565829(CHEMBL4788071)copy SMILES
Affinity DataKi:  0.331nMAssay Description:Displacement of [125I]-[NIe,DPhe7]-alpha-MSH from human MC3R expressed in HEK293 cell membranes incubated for 120 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53QMNPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50565827(CHEMBL4794990)copy SMILES
Affinity DataKi:  0.352nMAssay Description:Displacement of [125I]-[NIe,DPhe7]-alpha-MSH from human MC3R expressed in HEK293 cell membranes incubated for 120 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53QMNPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50565827(CHEMBL4794990)copy SMILES
Affinity DataKi:  0.355nMAssay Description:Displacement of [125I]-[NIe,DPhe7]-alpha-MSH from human MC3R expressed in HEK293 cell membranes incubated for 120 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53QMNPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50565831(CHEMBL4791788)copy SMILES
Affinity DataKi:  0.378nMAssay Description:Displacement of [125I]-[NIe,DPhe7]-alpha-MSH from human MC3R expressed in HEK293 cell membranes incubated for 120 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53QMNPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50565831(CHEMBL4791788)copy SMILES
Affinity DataKi:  0.380nMAssay Description:Displacement of [125I]-[NIe,DPhe7]-alpha-MSH from human MC3R expressed in HEK293 cell membranes incubated for 120 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53QMNPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50565830(CHEMBL4793821)copy SMILES
Affinity DataKi:  0.389nMAssay Description:Displacement of [125I]-[NIe,DPhe7]-alpha-MSH from human MC3R expressed in HEK293 cell membranes incubated for 120 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53QMNPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50565830(CHEMBL4793821)copy SMILES
Affinity DataKi:  0.391nMAssay Description:Displacement of [125I]-[NIe,DPhe7]-alpha-MSH from human MC3R expressed in HEK293 cell membranes incubated for 120 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53QMNPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50590042(CHEMBL5175981)copy SMILES
Affinity DataKi:  0.631nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20C50R5PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM82411(CAS_75921-69-6 | NDP-MSH)copy SMILEScopy InChI
Affinity DataKi:  0.680nMAssay Description:Binding affinity towards human Melanocortin 3 receptor (hMC3R)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2474BD9PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50565824(CHEMBL4800268)copy SMILES
Affinity DataKi:  0.690nMAssay Description:Displacement of [125I]-[NIe,DPhe7]-alpha-MSH from human MC3R expressed in HEK293 cell membranes incubated for 120 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53QMNPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50565824(CHEMBL4800268)copy SMILES
Affinity DataKi:  0.692nMAssay Description:Displacement of [125I]-[NIe,DPhe7]-alpha-MSH from human MC3R expressed in HEK293 cell membranes incubated for 120 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53QMNPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataKi:  0.780nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC3 receptor expressed in BHK570 cells after 1 hr in presence of ovalbuminMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DN464PPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50134946(CHEMBL2370964 | H-Tyr-Val-Nle-Gly-His-D-Nal(2')-Ar...)copy SMILEScopy InChI
Affinity DataKi:  0.810nMAssay Description:Binding affinity against human Melanocortin 3 receptor by gamma-MCH displacement.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SJ1K0PPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50105880(15-Acetylamino-6-(3-guanidino-propyl)-12-(3H-imida...)copy SMILEScopy InChI
Affinity DataKi:  0.960nMAssay Description:Binding affinity against human melanocortin receptor 3 (hMC3R) (concentration of the peptide at 50% specific binding)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RF5T9SPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50114077(6-(3-Guanidino-propyl)-12-(3H-imidazol-4-ylmethyl)...)copy SMILEScopy InChI
Affinity DataKi: <1nMAssay Description:Binding affinity for human Melanocortin-3 receptor (hMC3R) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RB75B3PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50189010((S)-2-[(S)-4-{(R)-2-[(S)-2-acetylamino-3-(4-hydrox...)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Binding affinity to human MC3RMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66KDFPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50189013((S)-2-[(S)-4-{(R)-2-[(S)-2-acetylamino-3-(3H-imida...)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Binding affinity to human MC3RMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66KDFPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50189024((S)-2-[(S)-4-[(R)-2-[(S)-2-acetylamino-3-(4-hydrox...)copy SMILEScopy InChI
Affinity DataKi:  1.10nMAssay Description:Binding affinity to human MC3RMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66KDFPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50114079(15-(2-Acetylamino-hexanoylamino)-9-benzyl-6-(3-gua...)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:Binding affinity for human Melanocortin-3 receptor (hMC3R) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RB75B3PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50165932(Ac-YRMEHdFRWG-NH2 | CHEMBL266879)copy SMILEScopy InChI
Affinity DataKi:  1.40nMAssay Description:Inhibition of [125I]-NDP-alpha-MSH binding to melanocortin-3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2251HQZPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50389783(CHEMBL2070245)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC3 receptor expressed in BHK570 cells after 1 hr in presence of ovalbuminMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DN464PPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50389771(CHEMBL2070243)copy SMILEScopy InChI
Affinity DataKi:  2.5nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC3 receptor expressed in BHK570 cells after 1 hr in presence of ovalbuminMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DN464PPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50105883(3-[25-Acetylamino-4-carbamoyl-13-(3-guanidino-prop...)copy SMILEScopy InChI
Affinity DataKi:  2.60nMAssay Description:Binding affinity against human melanocortin receptor 3 (hMC3R) (concentration of the peptide at 50% specific binding)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RF5T9SPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50165929(Ac-YR[CEH(pCl-dF)RWC]-NH2 | CHEMBL415661)copy SMILEScopy InChI
Affinity DataKi:  3.10nMAssay Description:Inhibition of [125I]-NDP-alpha-MSH binding to melanocortin-3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2251HQZPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50565833(CHEMBL4776340)copy SMILES
Affinity DataKi:  3.20nMAssay Description:Displacement of [125I]-[NIe,DPhe7]-alpha-MSH from human MC3R expressed in HEK293 cell membranes incubated for 120 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53QMNPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50565833(CHEMBL4776340)copy SMILES
Affinity DataKi:  3.25nMAssay Description:Displacement of [125I]-[NIe,DPhe7]-alpha-MSH from human MC3R expressed in HEK293 cell membranes incubated for 120 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53QMNPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50189025((S)-2-acetamido-N1-((R)-3-(4-fluorophenyl)-1-((S)-...)copy SMILEScopy InChI
Affinity DataKi:  3.30nMAssay Description:Binding affinity to human MC3RMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66KDFPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM82406(desacetyl-alpha-MSH)copy SMILEScopy InChI
Affinity DataKi:  3.68nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M32T8HPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM82406(desacetyl-alpha-MSH)copy SMILEScopy InChI
Affinity DataKi:  3.68nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W98M7PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50565818(CHEMBL4776915)copy SMILES
Affinity DataKi:  3.70nMAssay Description:Displacement of [125I]-[NIe,DPhe7]-alpha-MSH from human MC3R expressed in HEK293 cell membranes incubated for 120 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53QMNPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50565818(CHEMBL4776915)copy SMILES
Affinity DataKi:  3.75nMAssay Description:Displacement of [125I]-[NIe,DPhe7]-alpha-MSH from human MC3R expressed in HEK293 cell membranes incubated for 120 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53QMNPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50027084(Melatonan)copy SMILES
Affinity DataKi:  3.98nMAssay Description:Displacement of [125I]-[NIe,DPhe7]-alpha-MSH from human MC3R expressed in HEK293 cell membranes incubated for 120 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53QMNPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50027084(Melatonan)copy SMILES
Affinity DataKi:  4nMAssay Description:Displacement of [125I]-[NIe,DPhe7]-alpha-MSH from human MC3R expressed in HEK293 cell membranes incubated for 120 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53QMNPubMed
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