Compile Data Set for Download or QSAR

Found 56 hits of Enzyme Inhibition Constant Data   

TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366609(CHEMBL4177507)copy SMILEScopy InChI
Affinity DataIC50: 55nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366609(CHEMBL4177507)copy SMILEScopy InChI
Affinity DataIC50: 55nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366614(CHEMBL4176482)copy SMILEScopy InChI
Affinity DataIC50: 93nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366614(CHEMBL4176482)copy SMILEScopy InChI
Affinity DataIC50: 94nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366616(CHEMBL4176427)copy SMILEScopy InChI
Affinity DataIC50: 105nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366616(CHEMBL4176427)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50327884((2S,3S)-2-amino-3-(3-(4-(trifluoromethyl)benzamido...)copy SMILEScopy InChI
Affinity DataIC50: 117nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50327884((2S,3S)-2-amino-3-(3-(4-(trifluoromethyl)benzamido...)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366626(CHEMBL4165811)copy SMILEScopy InChI
Affinity DataIC50: 129nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366626(CHEMBL4165811)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366648(CHEMBL4173045)copy SMILEScopy InChI
Affinity DataIC50: 288nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366648(CHEMBL4173045)copy SMILEScopy InChI
Affinity DataIC50: 290nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366656(CHEMBL4162363)copy SMILEScopy InChI
Affinity DataIC50: 525nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366656(CHEMBL4162363)copy SMILEScopy InChI
Affinity DataIC50: 530nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366638(CHEMBL4166966)copy SMILEScopy InChI
Affinity DataIC50: 840nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366638(CHEMBL4166966)copy SMILEScopy InChI
Affinity DataIC50: 851nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366610(CHEMBL4169695)copy SMILEScopy InChI
Affinity DataIC50: 860nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366610(CHEMBL4169695)copy SMILEScopy InChI
Affinity DataIC50: 860nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366610(CHEMBL4169695)copy SMILEScopy InChI
Affinity DataIC50: 860nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366610(CHEMBL4169695)copy SMILEScopy InChI
Affinity DataIC50: 871nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366617(CHEMBL4163105)copy SMILEScopy InChI
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366655(CHEMBL4177165)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366617(CHEMBL4163105)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366655(CHEMBL4177165)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366650(CHEMBL4166282)copy SMILEScopy InChI
Affinity DataIC50: 1.55E+3nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366640(CHEMBL4166545)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366650(CHEMBL4166282)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366640(CHEMBL4166545)copy SMILEScopy InChI
Affinity DataIC50: 1.62E+3nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM86712(CAS_868359-05-1 | N-[4-(2-BROMO-4,5-DIFLUOROPHENOX...)copy SMILEScopy InChI
Affinity DataIC50: 1.86E+3nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM86712(CAS_868359-05-1 | N-[4-(2-BROMO-4,5-DIFLUOROPHENOX...)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366651(CHEMBL4173825)copy SMILEScopy InChI
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366651(CHEMBL4173825)copy SMILEScopy InChI
Affinity DataIC50: 2.14E+3nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366637(CHEMBL4164207)copy SMILEScopy InChI
Affinity DataIC50: 2.57E+3nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366637(CHEMBL4164207)copy SMILEScopy InChI
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366628(CHEMBL4165574)copy SMILEScopy InChI
Affinity DataIC50: 2.69E+3nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366628(CHEMBL4165574)copy SMILEScopy InChI
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366602(CHEMBL4159467)copy SMILEScopy InChI
Affinity DataIC50: 3.09E+3nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366602(CHEMBL4159467)copy SMILEScopy InChI
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366602(CHEMBL4159467)copy SMILEScopy InChI
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366602(CHEMBL4159467)copy SMILEScopy InChI
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50093753((2S,3S)-2-Amino-3-benzyloxy-succinic acid | (2S,3S...)copy SMILEScopy InChI
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50093753((2S,3S)-2-Amino-3-benzyloxy-succinic acid | (2S,3S...)copy SMILEScopy InChI
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM85209(DL-THA)copy SMILEScopy InChI
Affinity DataIC50: 9.55E+3nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM85209(DL-THA)copy SMILEScopy InChI
Affinity DataIC50: 9.60E+3nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366653(CHEMBL4163625)copy SMILEScopy InChI
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366653(CHEMBL4163625)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM18125((2S)-2-aminobutanedioic acid | Aspartate | CHEMBL2...)copy SMILEScopy InChI
Affinity DataIC50: 1.95E+4nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMedDrugBank
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM18125((2S)-2-aminobutanedioic acid | Aspartate | CHEMBL2...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMedDrugBank
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366654(CHEMBL4168620)copy SMILEScopy InChI
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50366654(CHEMBL4168620)copy SMILEScopy InChI
Affinity DataIC50: 2.82E+4nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
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