Found 6 hits of Enzyme Inhibition Constant Data
TargetGeranylgeranyl pyrophosphate synthase(Homo sapiens (Human))
University of Iowa
Curated by ChEMBL
University of Iowa
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of recombinant GGDPS (unknown origin) assessed as decrease in radiolabeld GGPP level using FPP and [14C]IPP as substrate treated with enzy...More data for this Ligand-Target Pair
TargetGeranylgeranyl pyrophosphate synthase(Homo sapiens (Human))
University of Iowa
Curated by ChEMBL
University of Iowa
Curated by ChEMBL
Affinity DataIC50: 380nMAssay Description:Inhibition of recombinant GGDPS (unknown origin) assessed as decrease in radiolabeld GGPP level using FPP and [14C]IPP as substrate treated with enzy...More data for this Ligand-Target Pair
TargetGeranylgeranyl pyrophosphate synthase(Homo sapiens (Human))
University of Iowa
Curated by ChEMBL
University of Iowa
Curated by ChEMBL
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of recombinant GGDPS (unknown origin) assessed as decrease in radiolabeld GGPP level using FPP and [14C]IPP as substrate treated with enzy...More data for this Ligand-Target Pair
TargetGeranylgeranyl pyrophosphate synthase(Homo sapiens (Human))
University of Iowa
Curated by ChEMBL
University of Iowa
Curated by ChEMBL
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of recombinant GGDPS (unknown origin) assessed as decrease in radiolabeld GGPP level using FPP and [14C]IPP as substrate treated with enzy...More data for this Ligand-Target Pair
TargetGeranylgeranyl pyrophosphate synthase(Homo sapiens (Human))
University of Iowa
Curated by ChEMBL
University of Iowa
Curated by ChEMBL
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of recombinant GGDPS (unknown origin) assessed as decrease in radiolabeld GGPP level using FPP and [14C]IPP as substrate treated with enzy...More data for this Ligand-Target Pair
TargetGeranylgeranyl pyrophosphate synthase(Homo sapiens (Human))
University of Iowa
Curated by ChEMBL
University of Iowa
Curated by ChEMBL
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of recombinant GGDPS (unknown origin) assessed as decrease in radiolabeld GGPP level using FPP and [14C]IPP as substrate treated with enzy...More data for this Ligand-Target Pair