Compile Data Set for Download or QSAR

Found 9 hits of Enzyme Inhibition Constant Data   

TargetLysine-specific demethylase 4E(Homo sapiens (Human))
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50396018(CHEMBL1230640)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of recombinant JMJD2E (unknown origin) incubated for 15 mins prior to substrate addition by AlphaScreen methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028VHDPubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50495468(CHEMBL3108958)copy SMILEScopy InChI
Affinity DataIC50: 420nMAssay Description:Inhibition of recombinant JMJD2E (unknown origin) incubated for 15 mins prior to substrate addition by AlphaScreen methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028VHDPubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50495470(CHEMBL3108954)copy SMILEScopy InChI
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of recombinant JMJD2E (unknown origin) incubated for 15 mins prior to substrate addition by AlphaScreen methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028VHDPubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50495472(CHEMBL3108952)copy SMILEScopy InChI
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of recombinant JMJD2E (unknown origin) incubated for 15 mins prior to substrate addition by AlphaScreen methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028VHDPubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM26119(2-[4-(methoxycarbonyl)pyridin-2-yl]pyridine-4-carb...)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant JMJD2E (unknown origin) incubated for 15 mins prior to substrate addition by AlphaScreen methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028VHDPubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50495473(CHEMBL3108955)copy SMILEScopy InChI
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of recombinant JMJD2E (unknown origin) incubated for 15 mins prior to substrate addition by AlphaScreen methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028VHDPubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50495469(CHEMBL3108953)copy SMILEScopy InChI
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of recombinant JMJD2E (unknown origin) incubated for 15 mins prior to substrate addition by AlphaScreen methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028VHDPubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50495471(CHEMBL3108959)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of recombinant JMJD2E (unknown origin) incubated for 15 mins prior to substrate addition by AlphaScreen methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028VHDPubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50240772((1R,2S)-(-)-2-phenylcyclopropylamine | (1R,2S)-2-p...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant JMJD2E (unknown origin) incubated for 15 mins prior to substrate addition by AlphaScreen methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028VHDPubMed
Displayed 1 to 50 (of 74 total ) | Next | Last >>* indicates data uncertainty>20%