Found 78 hits of Enzyme Inhibition Constant Data
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
The M. S. University of Baroda
Curated by ChEMBL
The M. S. University of Baroda
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Binding affinity to angiotensin AT1 receptorMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
The M. S. University of Baroda
Curated by ChEMBL
The M. S. University of Baroda
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Binding affinity to angiotensin AT1 receptorMore data for this Ligand-Target Pair
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
The M. S. University of Baroda
Curated by ChEMBL
The M. S. University of Baroda
Curated by ChEMBL
Affinity DataKi: 4.5nMAssay Description:Binding affinity to angiotensin AT2 receptorMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
The M. S. University of Baroda
Curated by ChEMBL
The M. S. University of Baroda
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Displacement of [3H]-angiotensin 2 from angiotensin AT1 receptor in human PLC-PRF5 cellsMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
The M. S. University of Baroda
Curated by ChEMBL
The M. S. University of Baroda
Curated by ChEMBL
Affinity DataKi: 24nMAssay Description:Binding affinity to angiotensin AT1 receptorMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
The M. S. University of Baroda
Curated by ChEMBL
The M. S. University of Baroda
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Displacement of [3H]-angiotensin 2 from angiotensin AT1 receptor in human PLC-PRF5 cellsMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
The M. S. University of Baroda
Curated by ChEMBL
The M. S. University of Baroda
Curated by ChEMBL
Affinity DataKi: 29nMAssay Description:Binding affinity to angiotensin AT1 receptorMore data for this Ligand-Target Pair
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
The M. S. University of Baroda
Curated by ChEMBL
The M. S. University of Baroda
Curated by ChEMBL
Affinity DataKi: 480nMAssay Description:Binding affinity to angiotensin AT2 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0550nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortic strip assessed as inhibition of angiotensin 2-induced contractile responseMore data for this Ligand-Target Pair
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
The M. S. University of Baroda
Curated by ChEMBL
The M. S. University of Baroda
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Binding affinity to angiotensin AT2 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Binding affinity to angiotensin AT1 receptor in rabbit aortic ringsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortaMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Binding affinity to angiotensin AT1 receptor in rabbit aortic ringsMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
The M. S. University of Baroda
Curated by ChEMBL
The M. S. University of Baroda
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Antagonist activity at angiotensin AT1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.420nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortaMore data for this Ligand-Target Pair
Affinity DataIC50: 0.550nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aorta assessed as reduction of angiotensin 2-induced contractile responseMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Binding affinity to angiotensin AT1 receptor in rabbit aortic ringsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.770nMAssay Description:Binding affinity to angiotensin AT1 receptor in rabbit aortic ringsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Binding affinity to angiotensin AT1 receptor in rabbit aortic ringsMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Binding affinity to angiotensin AT1 receptor in rabbit aortic ringsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Displacement of [125I]-Sar1Ile8-angiotensin 2 from angiotensin AT1 receptor in rabbit aortic membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Displacement of [125I]-Sar1Ile8-angiotensin 2 from angiotensin AT1 receptor in rabbit aortic membranesMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
The M. S. University of Baroda
Curated by ChEMBL
The M. S. University of Baroda
Curated by ChEMBL
Affinity DataIC50: 1.40nMAssay Description:Binding affinity to angiotensin AT1 receptorMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
The M. S. University of Baroda
Curated by ChEMBL
The M. S. University of Baroda
Curated by ChEMBL
Affinity DataIC50: 1.80nMAssay Description:Antagonist activity at angiotensin AT1 receptorMore data for this Ligand-Target Pair
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
The M. S. University of Baroda
Curated by ChEMBL
The M. S. University of Baroda
Curated by ChEMBL
Affinity DataIC50: 2.30nMAssay Description:Binding affinity to angiotensin AT2 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:Displacement of radiolabeled angiotensin 2 from angiotensin AT1 receptor in bovine adrenal cortex membranesMore data for this Ligand-Target Pair
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
The M. S. University of Baroda
Curated by ChEMBL
The M. S. University of Baroda
Curated by ChEMBL
Affinity DataIC50: 3.5nMAssay Description:Binding affinity to angiotensin AT2 receptorMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Cavia porcellus)
The M. S. University of Baroda
Curated by ChEMBL
The M. S. University of Baroda
Curated by ChEMBL
Affinity DataIC50: 3.80nMAssay Description:Binding affinity to angiotensin AT1 receptor in guinea pig adrenal cortex membranesMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
The M. S. University of Baroda
Curated by ChEMBL
The M. S. University of Baroda
Curated by ChEMBL
Affinity DataIC50: 4.70nMAssay Description:Binding affinity to angiotensin AT1 receptorMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
The M. S. University of Baroda
Curated by ChEMBL
The M. S. University of Baroda
Curated by ChEMBL
Affinity DataIC50: 4.90nMAssay Description:Binding affinity to angiotensin AT1 receptorMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Cavia porcellus)
The M. S. University of Baroda
Curated by ChEMBL
The M. S. University of Baroda
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Binding affinity to angiotensin AT1 receptor in guinea pig adrenal cortex membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Binding affinity to angiotensin AT1 receptor in rabbit aortic ringsMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
The M. S. University of Baroda
Curated by ChEMBL
The M. S. University of Baroda
Curated by ChEMBL
Affinity DataIC50: 5.60nMAssay Description:Binding affinity to angiotensin AT1 receptorMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
The M. S. University of Baroda
Curated by ChEMBL
The M. S. University of Baroda
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Binding affinity to angiotensin AT1 receptorMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
The M. S. University of Baroda
Curated by ChEMBL
The M. S. University of Baroda
Curated by ChEMBL
Affinity DataIC50: 6.5nMAssay Description:Binding affinity to angiotensin AT1 receptorMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
The M. S. University of Baroda
Curated by ChEMBL
The M. S. University of Baroda
Curated by ChEMBL
Affinity DataIC50: 6.90nMAssay Description:Binding affinity to angiotensin AT1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 7.70nMAssay Description:Displacement of radiolabeled angiotensin 2 from angiotensin AT1 receptor in bovine adrenal cortex membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 8.10nMAssay Description:Binding affinity to angiotensin AT1 receptor in bovine adrenal cortex membranesMore data for this Ligand-Target Pair
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
The M. S. University of Baroda
Curated by ChEMBL
The M. S. University of Baroda
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Binding affinity to angiotensin AT2 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Binding affinity to angiotensin AT1 receptor in bovine adrenal cortex membranesMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
The M. S. University of Baroda
Curated by ChEMBL
The M. S. University of Baroda
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Binding affinity to angiotensin AT1 receptorMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
The M. S. University of Baroda
Curated by ChEMBL
The M. S. University of Baroda
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Antagonist activity at angiotensin AT1 receptor in human PLC-PRF5 cellsMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
The M. S. University of Baroda
Curated by ChEMBL
The M. S. University of Baroda
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Binding affinity to angiotensin AT1 receptorMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
The M. S. University of Baroda
Curated by ChEMBL
The M. S. University of Baroda
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Binding affinity to angiotensin AT1 receptorMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
The M. S. University of Baroda
Curated by ChEMBL
The M. S. University of Baroda
Curated by ChEMBL
Affinity DataIC50: 20.8nMAssay Description:Binding affinity to angiotensin AT1 receptorMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
The M. S. University of Baroda
Curated by ChEMBL
The M. S. University of Baroda
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Antagonist activity at angiotensin AT1 receptor in human PLC-PRF5 cellsMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
The M. S. University of Baroda
Curated by ChEMBL
The M. S. University of Baroda
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Binding affinity to angiotensin AT1 receptorMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Cavia porcellus)
The M. S. University of Baroda
Curated by ChEMBL
The M. S. University of Baroda
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Binding affinity to angiotensin AT1 receptor in guinea pig adrenal cortex membranesMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Cavia porcellus)
The M. S. University of Baroda
Curated by ChEMBL
The M. S. University of Baroda
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Binding affinity to angiotensin AT1 receptor in guinea pig adrenal cortex membranesMore data for this Ligand-Target Pair
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
The M. S. University of Baroda
Curated by ChEMBL
The M. S. University of Baroda
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Binding affinity to angiotensin AT2 receptorMore data for this Ligand-Target Pair