Compile Data Set for Download or QSAR

Found 7 hits of Enzyme Inhibition Constant Data   

TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50390982(CHEMBL2075008)copy SMILEScopy InChI
Affinity DataKi:  1.01E+3nMAssay Description:TP_TRANSPORTER: inhibition of BQ-123 uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6KF8PubMed
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50390985(CHEMBL2074707)copy SMILEScopy InChI
Affinity DataKi:  8.32E+3nMAssay Description:TP_TRANSPORTER: inhibition of BQ-123 uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6KF8PubMed
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50390987(CHEMBL2074660)copy SMILEScopy InChI
Affinity DataKi:  4.00E+4nMAssay Description:TP_TRANSPORTER: inhibition of BQ-123 uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6KF8PubMed
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50390983(CHEMBL2074699)copy SMILEScopy InChI
Affinity DataKi:  5.41E+4nMAssay Description:TP_TRANSPORTER: inhibition of BQ-123 uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6KF8PubMed
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50390984(CHEMBL2074702)copy SMILEScopy InChI
Affinity DataKi:  6.55E+4nMAssay Description:TP_TRANSPORTER: inhibition of BQ-123 uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6KF8PubMed
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50329850((R)-3-Amino-4-[(S)-2-((R)-1-{(S)-1-[(R)-1-(1H-indo...)copy SMILEScopy InChI
Affinity DataKi:  8.41E+4nMAssay Description:TP_TRANSPORTER: inhibition of BQ-485 uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6KF8PubMed
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50390986(CHEMBL2074710)copy SMILEScopy InChI
Affinity DataKi:  8.54E+4nMAssay Description:TP_TRANSPORTER: inhibition of BQ-123 uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6KF8PubMed
* indicates data uncertainty>20%