Reaction Details
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Target
Serine/threonine-protein kinase WNK4 [1-444]
Ligand
BDBM207990
Substrate
n/a
Meas. Tech.
WNK In Vitro Radiometric Assays
pH
7.3±n/a
IC50
187±n/a nM
Comments
extracted
Citation
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More Info.:
Target
Name:
Serine/threonine-protein kinase WNK4 [1-444]
Synonyms:
PRKWNK4 | WNK4 | WNK4_HUMAN | With-No-Lysine kinase 4 (WNK4)
Type:
Protein
Mol. Mass.:
49727.70
Organism:
Homo sapiens (Human)
Description:
WNK4 truncation (1-444 aa)
Residue:
444
Sequence:
MLASPATETTVLMSQTEADLALRPPPPLGTAGQPRLGPPPRRARRFSGKAEPRPRSSRLSRRSSVDLGLLSSWSLPASPAPDPPDPPDSAGPGPARSPPPSSKEPPEGTWTEGAPVKAAEDSARPELPDSAVGPGSREPLRVPEAVALERRREQEEKEDMETQAVATSPDGRYLKFDIEIGRGSFKTVYRGLDTDTTVEVAWCELQTRKLSRAERQRFSEEVEMLKGLQHPNIVRFYDSWKSVLRGQVCIVLVTELMTSGTLKTYLRRFREMKPRVLQRWSRQILRGLHFLHSRVPPILHRDLKCDNVFITGPTGSVKIGDLGLATLKRASFAKSVIGTPEFMAPEMYEEKYDEAVDVYAFGMCMLEMATSEYPYSECQNAAQIYRKVTSGRKPNSFHKVKIPEVKEIIEGCIRTDKNERFTIQDLLAHAFFREERGVHVELAE