Reaction Details
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Target
Serine/threonine-protein kinase WNK2 [166-489]
Ligand
BDBM207990
Substrate
n/a
Meas. Tech.
WNK In Vitro Radiometric Assays
pH
7.3±n/a
IC50
50±n/a nM
Comments
extracted
Citation
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More Info.:
Target
Name:
Serine/threonine-protein kinase WNK2 [166-489]
Synonyms:
KIAA1760 | PRKWNK2 | SDCCAG43 | WNK2 | WNK2_HUMAN | With-No-Lysine kinase 2 (WNK2)
Type:
Protein
Mol. Mass.:
37413.16
Organism:
Homo sapiens (Human)
Description:
WNK2 truncation (166-489 aa)
Residue:
324
Sequence:
GRTRRDEPEEEEDDEDDLKAVATSLDGRFLKFDIELGRGSFKTVYKGLDTETWVEVAWCELQDRKLTKLERQRFKEEAEMLKGLQHPNIVRFYDFWESSAKGKRCIVLVTELMTSGTLKTYLKRFKVMKPKVLRSWCRQILKGLLFLHTRTPPIIHRDLKCDNIFITGPTGSVKIGDLGLATLKRASFAKSVIGTPEFMAPEMYEEHYDESVDVYAFGMCMLEMATSEYPYSECQNAAQIYRKVTCGIKPASFEKVHDPEIKEIIGECICKNKEERYEIKDLLSHAFFAEDTGVRVELAEEDHGRKSTIALRLWVEDPKKLKGK