The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
28074653 |
3 |
The Essential Medicinal Chemistry of Curcumin.![EBI](/images/logo_chembl.png) |
University of Minnesota |
18280153 |
9 |
Rational design of 4-amino-5,6-diaryl-furo[2,3-d]pyrimidines as potent glycogen synthase kinase-3 inhibitors.![EBI](/images/logo_chembl.png) |
Glaxosmithkline |
28803677 |
5 |
Indole-fused azepines and analogues as anticancer lead molecules: Privileged findings and future directions.![EBI](/images/logo_chembl.png) |
Babasaheb Bhimrao Ambedkar University |
30026041 |
139 |
Synthesis and anticancer activity of novel bisindolylhydroxymaleimide derivatives with potent GSK-3 kinase inhibition.![EBI](/images/logo_chembl.png) |
University College Cork |
19271755 |
78 |
Design, synthesis, and structure-activity relationship of substrate competitive, selective, and in vivo active triazole and thiadiazole inhibitors of the c-Jun N-terminal kinase.![BDB](/images/logo_bindingdb.png) |
Burnham Institute For Medical Research |
19072652 |
64 |
Synthesis and evaluation of novel inhibitors of Pim-1 and Pim-2 protein kinases.![BDB](/images/logo_bindingdb.png) |
Medical University of South Carolina |
17600705 |
43 |
N-4-Pyrimidinyl-1H-indazol-4-amine inhibitors of Lck: indazoles as phenol isosteres with improved pharmacokinetics.![BDB](/images/logo_bindingdb.png) |
Gsk |
17948975 |
12 |
Synthesis, Crystal Structure, and Activity of Pyrazole-Based Inhibitors of p38 Kinase.![BDB](/images/logo_bindingdb.png) |
Pfizer |
17927165 |
58 |
Toward Potent Ghrelin Receptor Ligands Based on Trisubstituted 1,2,4-Triazole Structure. 2. Synthesis and Pharmacological in Vitro and in Vivo Evaluations.![BDB](/images/logo_bindingdb.png) |
Cnrs |
17585753 |
26 |
Acridone-based inhibitors of inosine 5'-monophosphate dehydrogenase: discovery and SAR leading to the identification of N-(2-(6-(4-ethylpiperazin-1-yl)pyridin-3-yl)propan-2-yl)-2- fluoro-9-oxo-9,10-dihydroacridine-3-carboxamide (BMS-566419).![BDB](/images/logo_bindingdb.png) |
Bristol-Myers Squibb |
17914785 |
67 |
Discovery of 1-(4-Methoxyphenyl)-7-oxo-6-(4-(2-oxopiperidin-1-yl)phenyl)-4,5,6,7-tetrahydro- 1H-pyrazolo[3,4-c]pyridine-3-carboxamide (Apixaban, BMS-562247), a Highly Potent, Selective, Efficacious, and Orally Bioavailable Inhibitor of Blood Coagulation Factor Xa.![BDB](/images/logo_bindingdb.png) |
Bristol-Myers Squibb |
15177471 |
82 |
Thyroid receptor ligands. Part 2: Thyromimetics with improved selectivity for the thyroid hormone receptor beta.![BDB](/images/logo_bindingdb.png) |
Bristol-Myers Squibb |
16279780 |
36 |
Synthesis of N-{4-[(2,4-diamino-5-methyl-4,7-dihydro-3H-pyrrolo[2,3-d]pyrimidin-6-yl)thio]benzoyl}-L-glutamic acid and N-{4-[(2-amino-4-oxo-5-methyl-4,7-dihydro-3H-pyrrolo[2,3-d]pyrimidin-6-yl)thio]benzoyl}-L-glutamic acid as dual inhibitors of dihydrofolate reductase and thymidylate synthase and a![BDB](/images/logo_bindingdb.png) |
Duquesne University |