The following articles (labelled with PubMed ID or TBD) are for your review
| PMID | Data | Article Title | Organization |
|---|
| 28174065 |
7 |
Synthesis of new derivatives of 21-imidazolyl-16-dehydropregnenolone as inhibitors of 5a-reductase 2 and with cytotoxic activity in cancer cells. |
Universidad Nacional Aut£Noma De M£Xico |
| 27994731 |
3 |
Identification of Triptophenolide from |
Chinese Academy of Medical Science |
| 23403082 |
28 |
Cinnamides as selective small-molecule inhibitors of a cellular model of breast cancer stem cells. |
Broad Institute of Mit and Harvard |
| 23466225 |
2 |
Discovery of AZD3514, a small-molecule androgen receptor downregulator for treatment of advanced prostate cancer. |
Astrazeneca |
| 16134935 |
119 |
Impact of induced fit on ligand binding to the androgen receptor: a multidimensional QSAR study to predict endocrine-disrupting effects of environmental chemicals. |
University of Basel |
| 17606915 |
4 |
Discovery of antiandrogen activity of nonsteroidal scaffolds of marketed drugs. |
The Scripps Research Institute |
| 16942875 |
32 |
A bioisosteric approach to the discovery of indole carbinol androgen receptor ligands. |
Johnson and Johnson Pharmaceutical Research and Development |
| 16603353 |
26 |
Discovery of indole-containing tetracycles as a new scaffold for androgen receptor ligands. |
Johnson & Johnson Pharmaceutical Research and Development |
| 15454212 |
16 |
Synthesis and structure-activity investigation of iodinated arylhydantoins and arylthiohydantoins for development as androgen receptor radioligands. |
The University of Michigan Medical School |
| 11101354 |
18 |
Chiral derivatives of 2-cyclohexylideneperhydro-4,7-methanoindenes, a novel class of nonsteroidal androgen receptor ligand: synthesis, X-ray analysis, and biological activity. |
The University of Sydney |
| 10966753 |
5 |
Design, synthesis, and pharmacological characterization of 4-[4, 4-dimethyl-3-(4-hydroxybutyl)-5-oxo-2-thioxo-1-imidazolidinyl]- 2-iodobenzonitrile as a high-affinity nonsteroidal androgen receptor ligand. |
The University of Michigan Medical School |
| 1588549 |
9 |
Antiandrogenic steroidal sulfonyl heterocycles. Utility of electrostatic complementarity in defining bioisosteric sulfonyl heterocycles. |
Sterling Winthrop Pharmaceuticals Research Division |
| 3783591 |
225 |
Azasteroids: structure-activity relationships for inhibition of 5 alpha-reductase and of androgen receptor binding. |
TBA |
| 11327585 |
15 |
Synthesis and structure-activity studies of side-chain derivatized arylhydantoins for investigation as androgen receptor radioligands. |
The University of Michigan Medical School |
| 21944856 |
51 |
Tetrahydroquinolines as a novel series of nonsteroidal selective androgen receptor modulators: structural requirements for better physicochemical and biological properties. |
Kaken Pharmaceutical |
| 21349712 |
15 |
Design and synthesis of tricyclic tetrahydroquinolines as a new series of nonsteroidal selective androgen receptor modulators (SARMs). |
Kaken Pharmaceutical |
| 17328524 |
1 |
Synthesis and biological evaluation of [18F]bicalutamide, 4-[76Br]bromobicalutamide, and 4-[76Br]bromo-thiobicalutamide as non-steroidal androgens for prostate cancer imaging. |
University of Illinois |
| 17149866 |
4 |
Identification of the brominated flame retardant 1,2-dibromo-4-(1,2-dibromoethyl)cyclohexane as an androgen agonist. |
Orebro University |
| 27131065 |
26 |
Design and synthesis of novel bicalutamide and enzalutamide derivatives as antiproliferative agents for the treatment of prostate cancer. |
School of Pharmacy and Pharmaceutical Sciences |
| 31493989 |
14 |
Synthesis, biological evaluation and molecular docking of 4-Amino-2H-benzo[h]chromen-2-one (ABO) analogs containing the piperazine moiety. |
Luoyang Normal University |
| 31288149 |
8 |
A new series of bicalutamide, enzalutamide and enobosarm derivatives carrying pentafluorosulfanyl (SF |
Cardiff University |
| 30482547 |
6 |
Synthesis and biological evaluation of arylpiperazine derivatives as potential anti-prostate cancer agents. |
Southern Medical University |
| 15715462 |
70 |
Three-dimensional structure-activity relationships of nonsteroidal ligands in complex with androgen receptor ligand-binding domain. |
Csc-Scientific Computing |
| 30193215 |
20 |
Small molecule-induced degradation of the full length and V7 truncated variant forms of human androgen receptor. |
Vancouver Prostate Centre (Vpc) |
| 28757062 |
6 |
Design, synthesis and biological evaluation of novel 3-oxo-4-oxa-5?-androst-17?-amide derivatives as dual 5?-reductase inhibitors and androgen receptor antagonists. |
China Pharmaceutical University |
| 28937774 |
107 |
Selective Nonsteroidal Glucocorticoid Receptor Modulators for the Inhaled Treatment of Pulmonary Diseases. |
Astrazeneca |
| 28314097 |
8 |
Fragment-Sized EthR Inhibitors Exhibit Exceptionally Strong Ethionamide Boosting Effect in Whole-Cell Mycobacterium tuberculosis Assays. |
University of Cambridge |
| 27250740 |
15 |
Electrostatic Control of Isoform Selective Inhibitor Binding in Nitric Oxide Synthase. |
University of California Irvine |
| 6135157 |
11 |
Specific binding of 3H-tiotidine to histamine H2 receptors in guinea pig cerebral cortex. |
Hoechst Pharmaceutical Research Laboratories |
| 10908357 |
9 |
Recognition of a cognate RNA aptamer by neomycin B: quantitative evaluation of hydrogen bonding and electrostatic interactions. |
The Ohio State University |
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