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16 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
26303893 93 A novel series of indazole-/indole-based glucagon receptor antagonists.EBI Merck Research Laboratories
24881566 140 Identification of diarylsulfonamides as agonists of the free fatty acid receptor 4 (FFA4/GPR120).EBI Glaxosmithkline
24527772 262 The discovery of N-((2H-tetrazol-5-yl)methyl)-4-((R)-1-((5r,8R)-8-(tert-butyl)-3-(3,5-dichlorophenyl)-2-oxo-1,4-diazaspiro[4.5]dec-3-en-1-yl)-4,4-dimethylpentyl)benzamide (SCH 900822): a potent and selective glucagon receptor antagonist.EBI Merck Research Laboratories
22708876 106 Discovery of a novel glucagon receptor antagonist N-[(4-{(1S)-1-[3-(3, 5-dichlorophenyl)-5-(6-methoxynaphthalen-2-yl)-1H-pyrazol-1-yl]ethyl}phenyl)carbonyl]-ß-alanine (MK-0893) for the treatment of type II diabetes.EBI Merck Research Laboratories
19702274 31 Eleven amino acid glucagon-like peptide-1 receptor agonists with antidiabetic activity.EBI Bristol-Myers Squibb
22119466 38 A novel series of glucagon receptor antagonists with reduced molecular weight and lipophilicity.EBI Pfizer
22030028 55 Discovery of N-aryl-2-acylindole human glucagon receptor antagonists.EBI Merck Research Laboratories
22001094 78 Discovery of cyclic guanidines as potent, orally active, human glucagon receptor antagonists.EBI Merck Research Laboratories
21147532 82 Discovery of novel, potent, selective, and orally active human glucagon receptor antagonists containing a pyrazole core.EBI Merck Research Laboratories
18707090 68 Novel glucagon receptor antagonists with improved selectivity over the glucose-dependent insulinotropic polypeptide receptor.EBI Novo Nordisk
17126016 69 Design and synthesis of conformationally constrained tri-substituted ureas as potent antagonists of the human glucagon receptor.EBI Merck Research Laboratories
16102966 55 Discovery of novel, potent, and orally active spiro-urea human glucagon receptor antagonists.EBI Merck Research Laboratories
29153547 50 Optimization of peptide-based polyagonists for treatment of diabetes and obesity.EBI Novo Nordisk Research Center Indianapolis
29879354 54 Dual Glucagon-like Peptide 1 (GLP-1)/Glucagon Receptor Agonists Specifically Optimized for Multidose Formulations.EBI Sanofi-Aventis Deutschland
21108268 67 Biological evaluation and structural determinants of p38α mitogen-activated-protein kinase and c-Jun-N-terminal kinase 3 inhibition by flavonoids.BDB Eberhard Karls University of Tuebingen