The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
24035485 |
48 |
Bicyclic and tricyclic heterocycle derivatives as histamine H3 receptor antagonists for the treatment of obesity. |
Merck Research Laboratories |
23535326 |
10 |
Novel and highly potent histamine H3 receptor ligands. Part 3: an alcohol function to improve the pharmacokinetic profile. |
Bioprojet-Biotech |
24900450 |
44 |
Discovery of a potent thiadiazole class of histamine h3 receptor antagonist for the treatment of diabetes. |
TBA |
22464130 |
27 |
Fused bicycles as arylketone bioisosteres leading to potent, orally active thiadiazole H3 antagonists. |
Merck Research Laboratories |
22153663 |
59 |
Ligand based design of novel histamine H4 receptor antagonists; fragment optimization and analysis of binding kinetics. |
Griffin Discoveries |
21783360 |
52 |
Novel and highly potent histamine H3 receptor ligands. Part 2: exploring the cyclohexylamine-based series. |
Bioprojet-Biotech |
20833043 |
28 |
Investigation of 4-piperidinols as novel H3 antagonists. |
Athersys |
19773164 |
53 |
Synthesis and structure-activity relationships of 2-(1,4'-bipiperidin-1'-yl)thiazolopyridine as H3 receptor antagonists. |
Schering-Plough Research Institute |
19520574 |
49 |
Synthesis, structure-activity relationships, and biological profiles of a dihydrobenzoxathiin class of histamine H(3) receptor inverse agonists. |
Tsukuba Research Institute |
19553110 |
16 |
Development of a selective and potent radioactive ligand for histamine H(3) receptors: A compound potentially useful for receptor occupancy studies. |
Tsukuba Research Institute |
18841880 |
82 |
Synthesis and evaluation of structurally constrained quinazolinone derivatives as potent and selective histamine H3 receptor inverse agonists. |
Tsukuba Research Institute |
18752952 |
31 |
Benzimidazole-substituted (3-phenoxypropyl)amines as histamine H3 receptor ligands. |
The Schering Plough Research Institute |
31675226 |
63 |
4-(3-Aminoazetidin-1-yl)pyrimidin-2-amines as High-Affinity Non-imidazole Histamine H |
Vrije Universiteit Amsterdam |
29681486 |
33 |
Novel naphthyloxy derivatives - Potent histamine H |
Jagiellonian University Medical College |