The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
27894044 |
37 |
An insight on synthetic and medicinal aspects of pyrazolo[1,5-a]pyrimidine scaffold. |
University of Kwazulu-Natal |
18023192 |
2 |
Synthesis of fluorine substituted pyrazolopyrimidines as potential leads for the development of PET-imaging agents for the GABAA receptors. |
Abx Advanced Biochemical Compounds |
16610792 |
15 |
Refinement of the benzodiazepine receptor site topology by structure-activity relationships of new N-(heteroarylmethyl)indol-3-ylglyoxylamides. |
Universit£ |
16250647 |
71 |
2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine and analogues as A2A adenosine receptor antagonists. Design, synthesis, and pharmacological characterization. |
Universit£ |
7799410 |
46 |
Four amino acid exchanges convert a diazepam-insensitive, inverse agonist-preferring GABAA receptor into a diazepam-preferring GABAA receptor. |
Heidelberg |
18851913 |
11 |
Azaflavones compared to flavones as ligands to the benzodiazepine binding site of brain GABA(A) receptors. |
Lund University |
19469479 |
44 |
Identification of anxiolytic/nonsedative agents among indol-3-ylglyoxylamides acting as functionally selective agonists at the gamma-aminobutyric acid-A (GABAA) alpha2 benzodiazepine receptor. |
Universita Di Pisa |
18651727 |
15 |
Synthesis of GABAA receptor agonists and evaluation of their alpha-subunit selectivity and orientation in the GABA binding site. |
Johannes Gutenberg University |
17335185 |
21 |
Novel N-substituted indol-3-ylglyoxylamides probing the LDi and L1/L2 lipophilic regions of the benzodiazepine receptor site in search for subtype-selective ligands. |
Università |
17306981 |
8 |
Novel 3-iodo-8-ethoxypyrazolo[5,1-c][1,2,4]benzotriazine 5-oxide as promising lead for design of alpha5-inverse agonist useful tools for therapy of mnemonic damage. |
Università |
15828832 |
14 |
High affinity central benzodiazepine receptor ligands: synthesis and biological evaluation of a series of phenyltriazolobenzotriazindione derivatives. |
Università |
12519068 |
32 |
Synthesis and benzodiazepine receptor affinity of pyrazolo[1,5-a]pyrimidine derivatives. 3. New 6-(3-thienyl) series as alpha 1 selective ligands. |
University of Firenze |
12477354 |
8 |
Benzodiazepine receptor ligands. 7. Synthesis and pharmacological evaluation of new 3-esters of the 8-chloropyrazolo[5,1-c][1,2,4]benzotriazine 5-oxide. 3-(2-Thienylmethoxycarbonyl) derivative: an anxioselective agent in rodents. |
Università |
11428922 |
21 |
Novel N-(arylalkyl)indol-3-ylglyoxylylamides targeted as ligands of the benzodiazepine receptor: synthesis, biological evaluation, and molecular modeling analysis of the structure-activity relationships. |
Università |
20684859 |
12 |
Homology modeling and atomic level binding study of GABA(A) receptor with novel enaminone amides. |
Wuhan Institute of Technology |
29657102 |
19 |
Agonists of the ?-aminobutyric acid type B (GABA |
University of Mississippi |
29650463 |
17 |
A new class of pyrazolo[5,1-c][1,2,4]triazines as ?-aminobutyric type A (GABA |
Universit£ |
28606760 |
57 |
Progress in the discovery of small molecule modulators of the Cys-loop superfamily receptors. |
Amgen |
29451785 |
45 |
Structure-Function Evaluation of Imidazopyridine Derivatives Selective for ?-Subunit-Containing ?-Aminobutyric Acid Type A (GABA |
Johannes Gutenberg University Mainz |
29146472 |
71 |
Discovery of the first low-shift positive allosteric modulators for the muscarinic M1 receptor. |
Roche Pharma Research and Early Development |
26950400 |
37 |
Design, synthesis and biological evaluation of 1H-pyrrolo[2,3-b]pyridine and 1H-pyrazolo[3,4-b]pyridine derivatives as c-Met inhibitors. |
Tianjin University of Science and Technology |
26398141 |
14 |
Evaluation of 2-indolcarbohydrazones as potent a-glucosidase inhibitors, in silico studies and DFT based stereochemical predictions. |
Universiti Teknologi Mara (Uitm) |
25511999 |
3 |
Design, Synthesis, and Biological Evaluation of Novel Benzoyl Diarylamine/ether Derivatives as Potential Anti-HIV-1 Agents. |
Shandong University |
26364932 |
22 |
Structure and Inhibition of Microbiome ß-Glucuronidases Essential to the Alleviation of Cancer Drug Toxicity. |
University of North Carolina At Chapel Hill |
26158339 |
24 |
Type II Inhibitors Targeting CDK2. |
University of Oxford |