The following articles (labelled with PubMed ID or TBD) are for your review
| PMID | Data | Article Title | Organization |
|---|
| 27155470 |
4 |
Discovery of a sulfamate-based steroid sulfatase inhibitor with intrinsic selective estrogen receptor modulator properties. |
Chu De Qu£Bec - Research Center (Chul, T4) |
| 27155469 |
8 |
Recent developments of C-4 substituted coumarin derivatives as anticancer agents. |
Central University of Punjab |
| 26974384 |
94 |
Sulfatase inhibitors for recidivist breast cancer treatment: A chemical review. |
Punjabi University |
| 27143133 |
2 |
Design, synthesis, and biological evaluation of new arylamide derivatives possessing sulfonate or sulfamate moieties as steroid sulfatase enzyme inhibitors. |
University of Sharjah |
| 26301554 |
49 |
Recent developments in steroidal and nonsteroidal aromatase inhibitors for the chemoprevention of estrogen-dependent breast cancer. |
American University of Ras Al Khaimah |
| 25992880 |
90 |
Discovery and Development of the Aryl O-Sulfamate Pharmacophore for Oncology and Women's Health. |
University of Bath |
| 26163883 |
16 |
Synthesis of bicoumarin thiophosphate derivatives as steroid sulfatase inhibitors. |
Gdansk University of Technology |
| 26211459 |
16 |
A-ring substituted 17ß-arylsulfonamides of 17ß-aminoestra-1,3,5(10)-trien-3-ol as highly potent reversible inhibitors of steroid sulfatase. |
University of Waterloo |
| 24630694 |
11 |
Design and synthesis of silicon-containing steroid sulfatase inhibitors possessing pro-estrogen antagonistic character. |
The University of Tokyo |
| 24463645 |
1 |
Synthesis, structure-activity relationship of iodinated-4-aryloxymethyl-coumarins as potential anti-cancer and anti-mycobacterial agents. |
P.C. Jabin Science College |
| 21570853 |
5 |
Evaluation of sulfatase-directed quinone methide traps for proteomics. |
Bielefeld University |
| 22455789 |
32 |
Synthesis and evaluation of analogues of estrone-3-O-sulfamate as potent steroid sulfatase inhibitors. |
University of Bath |
| 20148564 |
60 |
Highly potent first examples of dual aromatase-steroid sulfatase inhibitors based on a biphenyl template. |
University of Bath |
| 18260615 |
8 |
Structure-activity relationships of C-17 cyano-substituted estratrienes as anticancer agents. |
University of Bath |
| 15293998 |
25 |
2-(1-adamantyl)-4-(thio)chromenone-6-carboxylic acids: potent reversible inhibitors of human steroid sulfatase. |
Novartis Institute For Biomedical Research Vienna |
| 15341968 |
13 |
Estrone formate: a novel type of irreversible inhibitor of human steroid sulfatase. |
Novartis Institutes For Biomedical Research Gdc |
| 14584960 |
11 |
Estrogenic potential of 2-alkyl-4-(thio)chromenone 6-O-sulfamates: potent inhibitors of human steroid sulfatase. |
Novartis Research Institute Vienna |
| 12213072 |
29 |
2-Substituted 4-(thio)chromenone 6-O-sulfamates: potent inhibitors of human steroid sulfatase. |
Novartis Research Institute Vienna |
| 11087571 |
35 |
Structure-activity relationships of 17alpha-derivatives of estradiol as inhibitors of steroid sulfatase. |
Laval University |
| 10447965 |
2 |
Synthesis and biological activity of the superestrogen (E)-17-oximino-3-O-sulfamoyl-1,3,5(10)-estratriene: x-ray crystal structure of (E)-17-oximino-3-hydroxy-1,3,5(10)-estratriene. |
University of Bath |
| 10377235 |
10 |
Potent inhibition of steroid sulfatase activity by 3-O-sulfamate 17alpha-benzyl(or 4'-tert-butylbenzyl)estra-1,3,5(10)-trienes: combination of two substituents at positions C3 and c17alpha of estradiol. |
Laval University |
| 8691463 |
3 |
Active site directed inhibition of estrone sulfatase by nonsteroidal coumarin sulfamates. |
University of Bath |
| 8295207 |
2 |
Estrone sulfamates: potent inhibitors of estrone sulfatase with therapeutic potential. |
University of Bath |
| 14741252 |
17 |
Inhibition of estrone sulfatase (ES) by alkyl and cycloalkyl ester derivatives of 4-[(aminosulfonyl)oxy] benzoic acid. |
Kingston University |
| 15149660 |
2 |
2-Alkylsulfanyl estrogen derivatives: synthesis of a novel class of multi-targeted anti-tumour agents. |
University of Bath |
| 14684318 |
8 |
The difluoromethylene group as a replacement for the labile oxygen in steroid sulfates: a new approach to steroid sulfatase inhibitors. |
University of Waterloo |
| 14643316 |
11 |
6-(2-adamantan-2-ylidene-hydroxybenzoxazole)-O-sulfamate: a potent non-steroidal irreversible inhibitor of human steroid sulfatase. |
Novartis Forschungsinstitut |
| 11965370 |
18 |
The mechanism of the irreversible inhibition of estrone sulfatase (ES) through the consideration of a range of methane- and amino-sulfonate-based compounds. |
Kingston University |
| 12161140 |
12 |
Inhibition of estrone sulfatase (ES) by derivatives of 4-[(aminosulfonyl)oxy] benzoic acid. |
Kingston University |
| 12127511 |
13 |
4,4'-Benzophenone-O,O'-disulfamate: a potent inhibitor of steroid sulfatase. |
Novartis Research Institute Vienna |
| 11992773 |
10 |
Design, synthesis and biochemical evaluation of AC ring mimics as novel inhibitors of the enzyme estrone sulfatase (ES). |
Kingston University |
| 11992772 |
34 |
A novel type of nonsteroidal estrone sulfatase inhibitors. |
Hans-Kn�Ll Institute of Natural Products Research |
| 11294387 |
15 |
Acid dissociation constant, a potential physicochemical factor in the inhibition of the enzyme estrone sulfatase (ES). |
Kingston University |
| 11277533 |
13 |
Novel inhibitors of the enzyme estrone sulfatase (ES). |
Kingston University |
| 11714597 |
5 |
Determination and use of a transition state for the enzyme estrone sulfatase (ES) from a proposed reaction mechanism. |
Kingston University |
| 11549461 |
13 |
Hydrophobicity, a physicochemical factor in the inhibition of the enzyme estrone sulfatase (ES). |
Kingston University |
| 10397493 |
4 |
Derivation of a possible transition-state for the reaction catalysed by the enzyme estrone Sulfatase (ES). |
Kingston University |
| 9873454 |
15 |
17 alpha-alkyl- or 17 alpha-substituted benzyl-17 beta-estradiols: a new family of estrone-sulfatase inhibitors. |
Laval University |
| | 4 |
Phosphonates and thiophosphonates as sulfate surrogates: synthesis of estrone 3-methylthiophosphonate, a potent inhibitor of estrone sulfatase |
TBA |
| 22264754 |
36 |
17ß-Arylsulfonamides of 17ß-aminoestra-1,3,5(10)-trien-3-ol as highly potent inhibitors of steroid sulfatase. |
University of Waterloo |
| 21925885 |
23 |
Inhibition of steroid sulfatase with 4-substituted estrone and estradiol derivatives. |
University of Waterloo |
| 24900302 |
27 |
Hybrid Dual Aromatase-Steroid Sulfatase Inhibitors with Exquisite Picomolar Inhibitory Activity |
TBA |
| 17696419 |
2 |
3,17-disubstituted 2-alkylestra-1,3,5(10)-trien-3-ol derivatives: synthesis, in vitro and in vivo anticancer activity. |
University of Bath |
| 17580843 |
38 |
Thiosemicarbazones of formyl benzoic acids as novel potent inhibitors of estrone sulfatase. |
Institute For Natural Products Research and Infection Biology |
| 17181151 |
10 |
2-substituted estradiol bis-sulfamates, multitargeted antitumor agents: synthesis, in vitro SAR, protein crystallography, and in vivo activity. |
University of Bath |
| 16078843 |
7 |
A-ring-substituted estrogen-3-O-sulfamates: potent multitargeted anticancer agents. |
University of Bath |
| 15686949 |
33 |
N-Acyl arylsulfonamides as novel, reversible inhibitors of human steroid sulfatase. |
Novartis Institutes For Biomedical Research |
| 14552755 |
28 |
Nortropinyl-arylsulfonylureas as novel, reversible inhibitors of human steroid sulfatase. |
Novartis Research Institute Vienna |
| 32122754 |
8 |
Design and synthesis of dansyl-labeled inhibitors of steroid sulfatase for optical imaging. |
Chu De Qu£Bec - Research Center |
| 32173116 |
8 |
A new series of aryl sulfamate derivatives: Design, synthesis, and biological evaluation. |
University of Sharjah |
| 31422224 |
11 |
Synthesis and in vitro evaluation of piperazinyl-ureido sulfamates as steroid sulfatase inhibitors. |
University of Cagliari |
| 31255926 |
46 |
Sulfamates in drug design and discovery: Pre-clinical and clinical investigations. |
University of Sharjah |
| 31129450 |
72 |
Estrogen signaling: An emanating therapeutic target for breast cancer treatment. |
Indian Institute of Technology (Bhu) |
| 29400967 |
136 |
Fluorine and Fluorinated Motifs in the Design and Application of Bioisosteres for Drug Design. |
Bristol-Myers Squibb |
| 28152429 |
17 |
Synthesis and biological evaluation of fluorinated N-benzoyl and N-phenylacetoyl derivatives of 3-(4-aminophenyl)-coumarin-7-O-sulfamate as steroid sulfatase inhibitors. |
Gdansk University of Technology |
| 28406629 |
51 |
First Dual Inhibitors of Steroid Sulfatase (STS) and 17?-Hydroxysteroid Dehydrogenase Type 1 (17?-HSD1): Designed Multiple Ligands as Novel Potential Therapeutics for Estrogen-Dependent Diseases. |
Saarland University |
| 18096504 |
19 |
URB602 inhibits monoacylglycerol lipase and selectively blocks 2-arachidonoylglycerol degradation in intact brain slices. |
University of California Irvine |
| 18022559 |
4 |
Inverse in silico screening for identification of kinase inhibitor targets. |
University of Munich |
| 14703393 |
52 |
Thermodynamics of the molecular and chiral recognition of cycloalkanols and camphor by modified beta-cyclodextrins possessing simple aromatic tethers. |
Nankai University |
| 18318466 |
41 |
Indoleamine 2,3-dioxygenase is the anticancer target for a novel series of potent naphthoquinone-based inhibitors. |
Bryn Mawr College |
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