The following articles (labelled with PubMed ID or TBD) are for your review
| PMID | Data | Article Title | Organization |
|---|
| 18537233 |
108 |
Selective influence on contextual memory: physiochemical properties associated with selectivity of benzodiazepine ligands at GABAA receptors containing the alpha5 subunit. |
Moltech |
| 20646926 |
13 |
The GABA(A) receptor as a target for photochromic molecules. |
University of Massachusetts |
| 20888240 |
254 |
Design, synthesis, and subtype selectivity of 3,6-disubstitutedß-carbolines at Bz/GABA(A)ergic receptors. SAR and studies directed toward agents for treatment of alcohol abuse. |
University of Wisconsin-Milwaukee |
| 15537339 |
18 |
An orally bioavailable, functionally selective inverse agonist at the benzodiazepine site of GABAA alpha5 receptors with cognition enhancing properties. |
Merck Sharp & Dohme Research Laboratories |
| 15214791 |
147 |
Synthesis and biological evaluation of 3-heterocyclyl-7,8,9,10-tetrahydro-(7,10-ethano)-1,2,4-triazolo[3,4-a]phthalazines and analogues as subtype-selective inverse agonists for the GABA(A)alpha5 benzodiazepine binding site. |
Merck Sharp and Dohme Research Laboratories |
| 15026049 |
42 |
Tricyclic pyridones as functionally selective human GABAA alpha 2/3 receptor-ion channel ligands. |
The Neuroscience Research Centre |
| 15006383 |
12 |
Determination of the stable conformation of GABA(A)-benzodiazepine receptor bivalent ligands by low temperature NMR and X-ray analysis. |
University of Wisconsin-Milwaukee |
| 14667209 |
32 |
Synthesis, in vitro affinity, and efficacy of a bis 8-ethynyl-4H-imidazo[1,5a]- [1,4]benzodiazepine analogue, the first bivalent alpha5 subtype selective BzR/GABA(A) antagonist. |
University of Wisconsin-Milwaukee |
| 11412984 |
66 |
Bioisosteric determinants for subtype selectivity of ligands for heteromeric GABA(A) receptors. |
The Royal Danish School of Pharmacy |
| 31117514 |
167 |
Five-Membered N-Heterocyclic Scaffolds as Novel Amino Bioisosteres at ?-Aminobutyric Acid (GABA) Type A Receptors and GABA Transporters. |
University of Copenhagen |
| 28606760 |
57 |
Progress in the discovery of small molecule modulators of the Cys-loop superfamily receptors. |
Amgen |
| 28753313 |
45 |
Neuroactive Steroids. 2. 3?-Hydroxy-3?-methyl-21-(4-cyano-1H-pyrazol-1'-yl)-19-nor-5?-pregnan-20-one (SAGE-217): A Clinical Next Generation Neuroactive Steroid Positive Allosteric Modulator of the (?-Aminobutyric Acid) |
Sage Therapeutics |
| 18973287 |
87 |
Structural Requirements for Eszopiclone and Zolpidem Binding to the gamma-Aminobutyric Acid Type-A (GABAA) Receptor Are Different. |
University of Wisconsin At Madison |
| 18790643 |
42 |
A study of the structure-activity relationship of GABA(A)-benzodiazepine receptor bivalent ligands by conformational analysis with low temperature NMR and X-ray analysis. |
University of Wisconsin-Milwaukee |
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