The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
15916423 |
28 |
Decoys for docking. |
University of California San Francisco |
14521410 |
36 |
Identification and prediction of promiscuous aggregating inhibitors among known drugs. |
Northwestern University |
13678405 |
23 |
A specific mechanism of nonspecific inhibition. |
Northwestern University |
11931626 |
124 |
A common mechanism underlying promiscuous inhibitors from virtual and high-throughput screening. |
Northwestern University |
8809160 |
132 |
Design, synthesis, and evaluation of 2 beta-alkenyl penam sulfone acids as inhibitors of beta-lactamases. |
F. Hoffmann-La Roche |
15109638 |
7 |
Design and synthesis of bridged gamma-lactams as analogues of beta-lactam antibiotics. |
Aventis Pharma |
20308379 |
3 |
In vitro properties of BAL30072, a novel siderophore sulfactam with activity against multiresistant gram-negative bacilli. |
Basilea Pharmaceutica International |
17072304 |
5 |
Deconstructing fragment-based inhibitor discovery. |
TBA |
17447748 |
20 |
A high-throughput screen for aggregation-based inhibition in a large compound library. |
University of California San Francisco |
15225711 |
16 |
Aza-boronic acids as non-beta-lactam inhibitors of AmpC-beta-lactamase. |
Università |
15214794 |
20 |
Mechanism of inactivation of beta-lactamases by novel 6-methylidene penems elucidated using electrospray ionization mass spectrometry. |
Wyeth Research |
14980686 |
50 |
Penicillin-derived inhibitors that simultaneously target both metallo- and serine-beta-lactamases. |
Southern Methodist University |
12109906 |
9 |
Structure-based approach for binding site identification on AmpC beta-lactamase. |
Northwestern University |
12039585 |
52 |
Cephalosporin-derived inhibitors of beta-lactamase. Part 4: The C3 substituent. |
Southern Methodist University |
11327608 |
45 |
Allyl and propargyl substituted penam sulfones as versatile intermediates toward the syntheses of new beta-lactamase inhibitors. |
Wyeth-Ayerst Research |
10498206 |
25 |
Synthesis and SAR of thioester and thiol inhibitors of IMP-1 metallo-beta-lactamase. |
Merck Research Laboratorie |
10230627 |
14 |
6-(1-Hydroxyalkyl))penam sulfone derivatives as inhibitors of class A and class C beta-lactamases II. |
Wyeth-Ayerst Research |
10230626 |
22 |
6-(1-Hydroxyalkyl)penam sulfone derivatives as inhibitors of class A and class C beta-lactamases I. |
Wyeth-Ayerst Research |
9804697 |
61 |
Structure-based enhancement of boronic acid-based inhibitors of AmpC beta-lactamase. |
Northwestern University Medical School |
9767633 |
76 |
Structure-based design of beta-lactamase inhibitors. 1. Synthesis and evaluation of bridged monobactams. |
F. Hoffmann-La Roche |
29784271 |
1 |
Boronic acid inhibitors of the class A?-lactamase KPC-2. |
Ucl School of Pharmacy |
16892341 |
8 |
Selective indole-based ECE inhibitors: synthesis and pharmacological evaluation. |
Bayer Healthcare |
12893846 |
3 |
A natural product ligand of the oxysterol receptor, liver X receptor. |
Eli Lilly |