BindingDB logo
myBDB logout

33 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
23270988 4 Carbon-11 N-methyl alkylation of L-368,899 and in vivo PET imaging investigations for neural oxytocin receptors.EBI Yerkes National Primate Research Center
7629809 140 Amino acid side chain descriptors for quantitative structure-activity relationship studies of peptide analogues.EBI University of Illinois At Chicago
7752199 71 Effects of a D-Cys6/L-Cys6 interchange in nonselective and selective vasopressin and oxytocin antagonists.EBI Medical College of Ohio
17300166 88 Design and synthesis of the first selective agonists for the rat vasopressin V(1b) receptor: based on modifications of deamino-[Cys1]arginine vasopressin at positions 4 and 8.EBI University of Montpellier
16297621 17 Pyridobenzodiazepines: a novel class of orally active, vasopressin V2 receptor selective agonists.EBI Wyeth Research
16302826 129 Discovery and development of a new class of potent, selective, orally active oxytocin receptor antagonists.EBI Serono Pharmaceutical Research Institute
1331448 101 Development of a novel class of cyclic hexapeptide oxytocin antagonists based on a natural product.EBI Merck Research Laboratories
2167976 33 Receptor ligands which bind the oxytocin receptor with selectivity and high affinity. Chemical modification of a Streptomyces silvensis derived cyclic hexapeptide.EBI Merck
20550119 96 Oral oxytocin antagonists.EBI Drugmoldesign
 66 Non-peptide oxytocin antagonists: identification and synthesis of a potent camphor aminosuccinimideEBI TBA
 9 Potent, non-peptidic oxytocin receptor antagonists from a natural sourceEBI TBA
17316912 63 Synthesis and biological activity of oxytocin analogues containing conformationally-restricted residues in position 7.EBI University of Patras
11992787 37 Identification of potent and selective oxytocin antagonists. Part 2: further investigation of benzofuran derivatives.EBI Glaxosmithkline
10780900 5 A study of the relationship between biological activity and prolyl amide isomer geometry in oxytocin using 5-tert-butylproline to augment the Cys(6)-Pro(7) amide cis-isomer population.EBI Université
10340620 30 Nonpeptide oxytocin antagonists: analogs of L-371,257 with improved potency.EBI Merck Research Laboratories
9873680 21 Nonpeptide oxytocin antagonists: potent, orally bioavailable analogs of L-371,257 containing a 1-R-(pyridyl)ethyl ether terminus.EBI Merck Research Laboratories
9622556 63 Development of orally active oxytocin antagonists: studies on 1-(1-[4-[1-(2-methyl-1-oxidopyridin-3-ylmethyl)piperidin-4-yloxy]-2- methoxybenzoyl]piperidin-4-yl)-1,4-dihydrobenz[d][1,3]oxazin-2-one (L-372,662) and related pyridines.EBI Merck Research Laboratories
9083475 4 Synthesis and pharmacology of novel analogues of oxytocin and deaminooxytocin: directed methods for the construction of disulfide and trisulfide bridges in peptides.EBI University of Minnesota
8258821 491 Nanomolar-affinity, non-peptide oxytocin receptor antagonists.EBI Merck Research Laboratories
8126695 35 1-((7,7-Dimethyl-2(S)-(2(S)-amino-4-(methylsulfonyl)butyramido)bicyclo [2.2.1]-heptan-1(S)-yl)methyl)sulfonyl)-4-(2-methylphenyl)piperaz ine (L-368,899): an orally bioavailable, non-peptide oxytocin antagonist with potential utility for managing preterm labor.EBI Merck Research Laboratories
8021923 27 A new series of photoactivatable and iodinatable linear vasopressin antagonists.EBI Upr 9023 Cnrs
7473590 37 1-(1-[4-[(N-acetyl-4-piperidinyl)oxy]-2-methoxybenzoyl]piperidin-4- yl)-4H-3,1-benzoxazin-2(1H)-one (L-371,257): a new, orally bioavailable, non-peptide oxytocin antagonist.EBI Merck Research Laboratories
30199637 172 LIT-001, the First Nonpeptide Oxytocin Receptor Agonist that Improves Social Interaction in a Mouse Model of Autism.EBI Umr7200 Cnrs/Universit£
2163451 45 Cyclic hexapeptide oxytocin antagonists. Potency-, selectivity-, and solubility-enhancing modifications.EBI Merck Sharp & Dohme Research Laboratories
1331449 268 Orally active, nonpeptide oxytocin antagonists.EBI Merck Research Laboratories