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39 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
26824643 69 Mimicking of Arginine by Functionalized N(¿)-Carbamoylated Arginine As a New Broadly Applicable Approach to Labeled Bioactive Peptides: High Affinity Angiotensin, Neuropeptide Y, Neuropeptide FF, and Neurotensin Receptor Ligands As Examples.EBI University of Regensburg
24900634 36 Design and Synthesis of Peptide YY Analogues with C-terminal Backbone Amide-to-Ester Modifications.EBI University of Copenhagen
24074877 135 Dimeric argininamide-type neuropeptide Y receptor antagonists: chiral discrimination between Y1 and Y4 receptors.EBI University of Regensburg
24090364 96 Replacement of Thr32 and Gln34 in the C-terminal neuropeptide Y fragment 25-36 by cis-cyclobutane and cis-cyclopentane β-amino acids shifts selectivity toward the Y(4) receptor.EBI University of Regensburg
18160282 40 Discovery of novel orally active ureido NPY Y5 receptor antagonists.EBI Schering-Plough Research Institute
21782428 61 Discovery of Lu AA33810: a highly selective and potent NPY5 antagonist with in vivo efficacy in a model of mood disorder.EBI Lundbeck Research Usa
19616955 34 Discovery of pyridone-containing imidazolines as potent and selective inhibitors of neuropeptide Y Y5 receptor.EBI Tsukuba Research Institute
21493077 39 Red-fluorescent argininamide-type NPY Y1 receptor antagonists as pharmacological tools.EBI Universit£T Regensburg
19864135 43 Discovery and SAR of cyclic isothioureas as novel NPY Y1 receptor antagonists.EBI Schering-Plough Research Institute
20042335 12 [Lys(DOTA)4]BVD15, a novel and potent neuropeptide Y analog designed for Y1 receptor-targeted breast tumor imaging.EBI Universit£
19679469 26 Identification of positron emission tomography ligands for NPY Y5 receptors in the brain.EBI Tsukuba Research Institute
19640706 25 Synthesis and evaluation of a series of 2,4-diaminopyridine derivatives as potential positron emission tomography tracers for neuropeptide Y Y1 receptors.EBI Tsukuba Research Institute
19596193 72 Design, synthesis and evaluation of a novel cyclohexanamine class of neuropeptide Y Y1 receptor antagonists.EBI Tsukuba Research Institute
19464889 43 Aryl urea derivatives of spiropiperidines as NPY Y5 receptor antagonists.EBI Tsukuba Research Institute
19459652 56 Discovery of tetrasubstituted imidazolines as potent and selective neuropeptide Y Y5 receptor antagonists: reduced human ether-a-go-go related gene potassium channel binding affinity and potent antiobesity effect.EBI Tsukuba Research Institute
19053784 19 Guanidine-acylguanidine bioisosteric approach in the design of radioligands: synthesis of a tritium-labeled N(G)-propionylargininamide ([3H]-UR-MK114) as a highly potent and selective neuropeptide Y Y1 receptor antagonist.EBI University of Regensburg
18752943 36 Syntheses and structure-activity relationships of novel, potent, and selective trans-2-[3-oxospiro[isobenzofuran-1(3H),1'-cyclohexan]-4'-yl]benzimidazole NPY Y5 receptor antagonists.EBI Banyu Tsukuba Research Institute
18723347 59 Design, syntheses, and structure-activity relationships of novel NPY Y5 receptor antagonists: 2-{3-Oxospiro[isobenzofuran-1(3H),4'-piperidin]-1'-yl}benzimidazole derivatives.EBI Banyu Tsukuba Research Institute
18637668 38 (9S)-9-(2-hydroxy-4,4-dimethyl-6-oxo-1-cyclohexen-1-yl)-3,3-dimethyl-2,3,4,9-tetrahydro-1H-xanthen-1-one, a selective and orally active neuropeptide Y Y5 receptor antagonist.EBI Tsukuba Research Institute
16610810 39 Neuropeptide Y (NPY) Y4 receptor selective agonists based on NPY(32-36): development of an anorectic Y4 receptor selective agonist with picomolar affinity.EBI University of Cincinnati
15109631 86 Discovery and SAR of potent, orally available and brain-penetrable 5,6-dihydro-4H-3-thia-1-aza-benzo[e]azulen- and 4,5-dihydro-6-oxa-3-thia-1-aza-benzo[e]azulen derivatives as neuropeptide Y Y5 receptor antagonists.EBI Novartis Pharma
32614182 299 Oligopeptides as Neuropeptide Y YEBI University of Regensburg
11334558 42 Highly selective and potent neuropeptide Y (NPY) Y1 receptor antagonists based on [Pro(30), Tyr(32), Leu(34)]NPY(28-36)-NH2 (BW1911U90).EBI University of Cincinnati and Va Medical Centers
27223253 89 High Affinity Agonists of the Neuropeptide Y (NPY) Y4 Receptor Derived from the C-Terminal Pentapeptide of Human Pancreatic Polypeptide (hPP): Synthesis, Stereochemical Discrimination, and Radiolabeling.EBI University of Regensburg
10866375 50 Design, synthesis and SAR of a series of 2-substituted 4-amino-quinazoline neuropeptide Y Y5 receptor antagonists.EBI Novartis Pharma
27295337 54 Optically Pure, Structural, and Fluorescent Analogues of a Dimeric Y4 Receptor Agonist Derived by an Olefin Metathesis Approach.EBI Monash University (Parkville Campus)
32364733 32 Heterodimeric Analogues of the Potent Y1R Antagonist 1229U91, Lacking One of the Pharmacophoric C-Terminal Structures, Retain Potent Y1R Affinity and Show Improved Selectivity over Y4R.EBI Monash University (Parkville Campus)
32184966 13 An Alkyne-functionalized Arginine for Solid-Phase Synthesis Enabling "Bioorthogonal" Peptide Conjugation.EBI University of Regensburg
9371234 49 Potent and selective 1,2,3-trisubstituted indole NPY Y-1 antagonists.EBI Eli Lilly
26466164 115 N(?)-Carbamoylation of the Argininamide Moiety: An Avenue to Insurmountable NPY Y1 Receptor Antagonists and a Radiolabeled Selective High-Affinity Molecular Tool ([(3)H]UR-MK299) with Extended Residence Time.EBI Cnrs/Ipbs (Institut De Pharmacologie Et Biologie Structurale)
30399314 532 Design of YEBI TBA
28795803 20 Identification and Characterization of the First Selective YEBI Leipzig University