44 articles for thisTarget

---

The following articles (labelled with PubMed ID or TBD) are for your review

PMID	Data	Article Title	Organization
24915003	34	Probing of primed and unprimed sites of calpains: Design, synthesis and evaluation of epoxysuccinyl-peptide derivatives as selective inhibitors.	E£Tv£S Lor£Nd University (Elte)
19715320	87	Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation.	University of Florida
18396356	13	Design and synthesis of calpain inhibitory 6-pyridone 2-carboxamide derivatives.	Kyung Hee University
19419206	77	Identification of 3-acetyl-2-aminoquinolin-4-one as a novel, nonpeptidic scaffold for specific calpain inhibitory activity.	Ewha Womans University
19041242	25	Design and synthesis of 4-aryl-4-oxobutanoic acid amides as calpain inhibitors.	Shenyang Pharmaceutical University
10669559	180	Protease inhibitors: current status and future prospects.	University of Queensland
9667954	47	D-amino acid containing, high-affinity inhibitors of recombinant human calpain I.	Cephalon
14980679	30	Dipeptidyl aspartyl fluoromethylketones as potent caspase-3 inhibitors: SAR of the P2 amino acid.	Maxim Pharmaceuticals
15013018	48	1,2-Benzothiazine 1,1-dioxide alpha-ketoamide analogues as potent calpain I inhibitors.	Cephalon
10476870	9	Hydroxyoxazolidines as alpha-aminoacetaldehye equivalents: novel inhibitors of calpain.	Hoechst Marion Roussel
21504847	12	Synthesis of cinnamoyl ketoamides as hybrid structures of antioxidants and calpain inhibitors.	College of Pharmacy Kyung Hee University
	65	Subsite requirements for peptide aldehyde inhibitors of human calpain I	TBA
	10	Nonpeptidic inhibitors of recombinant human calpain I	TBA
	2	Oligopresentation of protease inhibitors with β-cyclodextrin as template	TBA
	6	Xanthene derived potent nonpeptidic inhibitors of recombinant human calpain I	TBA
	1	Synthesis of cystamidin a (pyrrole-3-propanamide), a reported calpain inhibitor	TBA
	17	Characterization of a continuous fluorogenic assay for calpain I. Kinetic evaluation of peptide aldehydes, halomethyl ketones and (acyloxy)methyl ketones as inhibitors of the enzyme	TBA
	22	Inhibition of human erythrocyte calpain I by novel quinolinecarboxamides	TBA
18789863	10	Molecular design to enhance the penetration into the retina via ocular instillation.	Senju Pharmaceutical
18024028	14	Design and synthesis of 4-quinolinone 2-carboxamides as calpain inhibitors.	Kyung Hee University
16789748	31	Exploration of orally available calpain inhibitors 2: peptidyl hemiacetal derivatives.	Senju Pharmaceutical
16380258	17	Novel dual inhibitors of calpain and lipid peroxidation with enhanced cellular activity.	Institut Henri Beaufour
15911268	13	Synthesis and biological evaluation of chromone carboxamides as calpain inhibitors.	Institute of Science & Technology
15713391	19	Dipeptidyl aspartyl fluoromethylketones as potent caspase inhibitors: peptidomimetic replacement of the P2 alpha-amino acid by a alpha-hydroxy acid.	Maxim Pharmaceuticals
15634028	5	Retro hydrazino-azapeptoids as peptidomimetics of proteasome inhibitors.	Université
15203170	7	Novel dual inhibitors of calpain and lipid peroxidation.	Institut Henri Beaufour
12773044	18	Benzoylalanine-derived ketoamides carrying vinylbenzyl amino residues: discovery of potent water-soluble calpain inhibitors with oral bioavailability.	Abbott
12593666	30	Structure-activity relationship study and drug profile of N-(4-fluorophenylsulfonyl)-L-valyl-L-leucinal (SJA6017) as a potent calpain inhibitor.	Senju Pharmaceutical
11992771	19	Discovery of phenyl alanine derived ketoamides carrying benzoyl residues as novel calpain inhibitors.	Abbott
11585453	52	1,2-Benzothiazine 1,1-dioxide P(2)-P(3) peptide mimetic aldehyde calpain I inhibitors.	Cephalon
11551769	2	Synthesis of a reported calpain inhibitor isolated from Streptomyces griseus.	The University of Tennessee Health Science Center
11551762	16	Potent peptide alpha-ketohydroxamate inhibitors of recombinant human calpain I.	Cephalon
11012026	18	Synthesis and biological evaluation of novel piperidine carboxamide derived calpain inhibitors.	Knoll
10476871	22	P2-achiral, P'-extended alpha-ketoamide inhibitors of calpain I.	Cephalon
9873596	18	P2-proline-derived inhibitors of calpain I.	Cephalon
9871656	1	Selective inhibition of the chymotrypsin-like activity of the 20S proteasome by 5-methoxy-1-indanone dipeptide benzamides.	Cv Therapeutics
9748367	11	Novel peptidyl phosphorus derivatives as inhibitors of human calpain I.	Cephalon
8831774	261	Novel peptidyl alpha-keto amide inhibitors of calpains and other cysteine proteases.	Georgia Institute of Technology
8230139	165	Peptide alpha-keto ester, alpha-keto amide, and alpha-keto acid inhibitors of calpains and other cysteine proteases.	Georgia Institute of Technology
8071940	32	Stereospecific synthesis of peptidyl alpha-keto amides as inhibitors of calpain.	Alkermes
27996267	22	Covalent Modifiers: A Chemical Perspective on the Reactivity of?,?-Unsaturated Carbonyls with Thiols via Hetero-Michael Addition Reactions.	University of Pittsburgh