The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
27940419 |
31 |
Novel CLK1 inhibitors based on N-aryloxazol-2-amine skeleton - A possible way to dual VEGFR2 TK/CLK ligands. |
Comenius University In Bratislava |
15080993 |
23 |
Novel GSK-3 inhibitors with improved cellular activity. |
Glaxosmithkline |
27474927 |
76 |
Synthesis, biological evaluation and molecular modeling studies of imidazo[1,2-a]pyridines derivatives as protein kinase inhibitors. |
Paris-Sud University |
26562543 |
14 |
Pivotal role of glycogen synthase kinase-3: A therapeutic target for Alzheimer's disease. |
Central University |
25827523 |
275 |
Isosteric replacements of the carboxylic acid of drug candidate VX-787: Effect of charge on antiviral potency and kinase activity of azaindole-based influenza PB2 inhibitors. |
Vertex Pharmaceuticals |
25198388 |
47 |
The design and synthesis of potent and selective inhibitors of Trypanosoma brucei glycogen synthase kinase 3 for the treatment of human african trypanosomiasis. |
University of Dundee |
20363627 |
56 |
Identification and structure-activity relationship of 8-hydroxy-quinoline-7-carboxylic acid derivatives as inhibitors of Pim-1 kinase. |
Universit£ |
17303421 |
56 |
Synthesis and activity of quinolinyl-methylene-thiazolinones as potent and selective cyclin-dependent kinase 1 inhibitors. |
Roche Research Center |
16789733 |
41 |
Discovery and evaluation of N-cyclopropyl- 2,4-difluoro-5-((2-(pyridin-2-ylamino)thiazol-5- ylmethyl)amino)benzamide (BMS-605541), a selective and orally efficacious inhibitor of vascular endothelial growth factor receptor-2. |
Bristol-Myers Squibb Pharmaceutical Research Institute |
16765046 |
63 |
Discovery of 2-pyrimidyl-5-amidothiophenes as potent inhibitors for AKT: synthesis and SAR studies. |
Chiron |
16366598 |
51 |
(6,7-Dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)phenylamines: platelet-derived growth factor receptor tyrosine kinase inhibitors with broad antiproliferative activity against tumor cells. |
Johnson & Johnson Pharmaceutical Research and Development |
30639897 |
48 |
Recent development of CDK inhibitors: An overview of CDK/inhibitor co-crystal structures. |
The First Affiliated Hospital of Zhengzhou University |
31404862 |
138 |
Imidazopyridine-based selective and multifunctional ligands of biological targets associated with psychiatric and neurodegenerative diseases. |
Palack£ |
30909021 |
21 |
Insights into the chemistry and therapeutic potential of furanones: A versatile pharmacophore. |
Jamia Hamdard |
31054862 |
14 |
1-Aryl-3-(4-methoxybenzyl)ureas as potentially irreversible glycogen synthase kinase 3 inhibitors: Synthesis and biological evaluation. |
Stellenbosch University |
23683591 |
23 |
Synthesis and evaluation of 8-amino-[1,2,4]triazolo[4,3-a]pyridin-3(2H)-one derivatives as glycogen synthase kinase-3 (GSK-3) inhibitors. |
Jeil Pharmaceutical |
15715498 |
7 |
CH...O and CH...N hydrogen bonds in ligand design: a novel quinazolin-4-ylthiazol-2-ylamine protein kinase inhibitor. |
Vertex Pharmaceuticals |
15686883 |
59 |
The development of potent and selective bisarylmaleimide GSK3 inhibitors. |
Lilly Research Laboratories |
15603961 |
35 |
3D QSAR studies on GSK-3 inhibition by aloisines. |
Zhejiang University |
29985601 |
64 |
Dual-Specificity Tyrosine Phosphorylation-Regulated Kinase 1A (DYRK1A) Inhibitors as Potential Therapeutics. |
Seoul National University |
27689729 |
17 |
Natural and synthetic bioactive inhibitors of glycogen synthase kinase. |
Jamia Hamdard (Hamdard University) |