The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
26862980 |
37 |
Tweaking Subtype Selectivity and Agonist Efficacy at (S)-2-Amino-3-(3-hydroxy-5-methyl-isoxazol-4-yl)propionic acid (AMPA) Receptors in a Small Series of BnTetAMPA Analogues. |
University of Copenhagen |
26653877 |
47 |
Studies on Aryl-Substituted Phenylalanines: Synthesis, Activity, and Different Binding Modes at AMPA Receptors. |
University of Copenhagen |
24824658 |
8 |
Structure-activity relationship studies of N-methylated and N-hydroxylated spider polyamine toxins as inhibitors of ionotropic glutamate receptors. |
University of Copenhagen |
23320429 |
48 |
Structure-activity relationship studies of argiotoxins: selective and potent inhibitors of ionotropic glutamate receptors. |
University of Copenhagen |
23092360 |
19 |
General synthesis ofß-alanine-containing spider polyamine toxins and discovery of nephila polyamine toxins 1 and 8 as highly potent inhibitors of ionotropic glutamate receptors. |
University of Copenhagen |
21188966 |
2 |
Solid-phase synthesis and biological evaluation of Joro spider toxin-4 from Nephila clavata. |
University of Copenhagen |
19588945 |
55 |
The glutamate receptor GluR5 agonist (S)-2-amino-3-(3-hydroxy-7,8-dihydro-6H-cyclohepta[d]isoxazol-4-yl)propionic acid and the 8-methyl analogue: synthesis, molecular pharmacology, and biostructural characterization. |
University of Copenhagen |
18811139 |
126 |
1H-cyclopentapyrimidine-2,4(1H,3H)-dione-related ionotropic glutamate receptors ligands. structure-activity relationships and identification of potent and Selective iGluR5 modulators. |
European Research Centre For Drug Discovery and Development (Natsyndrugs) |
18338843 |
57 |
Synthesis and pharmacological characterization at glutamate receptors of the four enantiopure isomers of tricholomic acid. |
Universit£ |
16250647 |
71 |
2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine and analogues as A2A adenosine receptor antagonists. Design, synthesis, and pharmacological characterization. |
Universit£ |
9357531 |
58 |
Synthesis of willardiine and 6-azawillardiine analogs: pharmacological characterization on cloned homomeric human AMPA and kainate receptor subtypes. |
University of Bristol |
1977908 |
10 |
(R)-4-oxo-5-phosphononorvaline: a new competitive glutamate antagonist at the NMDA receptor complex. |
Merrell Dow Research Institute |
21923187 |
5 |
A new phenylalanine derivative acts as an antagonist at the AMPA receptor GluA2 and introduces partial domain closure: synthesis, resolution, pharmacology, and crystal structure. |
University of Copenhagen |
21067182 |
37 |
Biostructural and Pharmacological Studies of Bicyclic Analogues of the 3-Isoxazolol Glutamate Receptor Agonist Ibotenic Acid |
TBA |
20684595 |
374 |
Quinazolin-4-one derivatives: A novel class of noncompetitive NR2C/D subunit-selective N-methyl-D-aspartate receptor antagonists. |
Emory University |
20096591 |
84 |
Developing a complete pharmacology for AMPA receptors: a perspective on subtype-selective ligands. |
University of California |
| 10 |
Synthesis and biology of the rigidified glutamate analogue, trans-2-carboxyazetidine-3-acetic acid (t-CAA) |
TBA |
17455929 |
36 |
A tetrazolyl-substituted subtype-selective AMPA receptor agonist. |
University of Copenhagen |
16942015 |
43 |
Uncompetitive antagonism of AMPA receptors: Mechanistic insights from studies of polyamine toxin derivatives. |
The Danish University of Pharmaceutical Sciences |
15615543 |
56 |
Bioisosteric modifications of 2-arylureidobenzoic acids: selective noncompetitive antagonists for the homomeric kainate receptor subtype GluR5. |
The Danish University of Pharmaceutical Sciences |
12747796 |
39 |
Design, synthesis, and pharmacology of a highly subtype-selective GluR1/2 agonist, (RS)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)propionic acid (Cl-HIBO). |
The Danish University of Pharmaceutical Sciences |
30943028 |
66 |
Use of the 4-Hydroxytriazole Moiety as a Bioisosteric Tool in the Development of Ionotropic Glutamate Receptor Ligands. |
University of Turin |
7629789 |
8 |
Synthesis, resolution, and biological evaluation of the four stereoisomers of 4-methylglutamic acid: selective probes of kainate receptors. |
Symphony Pharmaceuticals |
30125106 |
4 |
Controlling Ca |
University of Copenhagen |