The following articles (labelled with PubMed ID or TBD) are for your review
| PMID | Data | Article Title | Organization |
|---|
| 7381854 |
9 |
Structure--antitubulin activity relationship in steganacin congeners and analogues. Inhibition of tubulin polymerization in vitro by (+/-)-isodeoxypodophyllotoxin. |
TBA |
| 12372531 |
6 |
Synthesis and mechanism of action of novel pyrimidinyl pyrazole derivatives possessing antiproliferative activity. |
Daiichi Pharmaceutical |
| 11140732 |
10 |
Antimitotic and cell growth inhibitory properties of combretastatin A-4-like ethers. |
The University of Manchester |
| 9873473 |
4 |
Asymmetric synthesis of antimitotic combretadioxolane with potent antitumor activity against multi-drug resistant cells. |
University of Tokyo |
| 27149641 |
5 |
Synthesis, Evaluation, and Mechanism Study of Novel Indole-Chalcone Derivatives Exerting Effective Antitumor Activity Through Microtubule Destabilization in Vitro and in Vivo. |
Sun Yat-Sen University |
| 26970659 |
3 |
Design, synthesis of phenstatin/isocombretastatin-oxindole conjugates as antimitotic agents. |
Csir-Indian Institute of Chemical Technology |
| 26927488 |
4 |
Discovery of novel 2-phenyl-imidazo[1,2-a]pyridine analogues targeting tubulin polymerization as antiproliferative agents. |
Shanghai Institute of Materia Medica |
| 27066215 |
3 |
Synthesis and anti-cancer screening of novel heterocyclic-(2H)-1,2,3-triazoles as potential anti-cancer agents. |
University of Arkansas For Medical Sciences |
| 26204510 |
6 |
4-Fluoro-3',4',5'-trimethoxychalcone as a new anti-invasive agent. From discovery to initial validation in an in vivo metastasis model. |
Ghent University |
| 25108078 |
13 |
Synthesis and biological evaluations of new analogs of 2-methoxyestradiol: inhibitors of tubulin and angiogenesis. |
University of Oslo |
| 25313318 |
4 |
Development of a new benzophenone-diketopiperazine-type potent antimicrotubule agent possessing a 2-pyridine structure. |
Tokyo University of Pharmacy and Life Sciences |
| 14552774 |
13 |
The total synthesis of an aurone isolated from Uvaria hamiltonii: aurones and flavones as anticancer agents. |
Cardiff University |
| 27515320 |
3 |
Design and synthesis of cis-restricted benzimidazole and benzothiazole mimics of combretastatin A-4 as antimitotic agents with apoptosis inducing ability. |
Csir-Indian Institute of Chemical Technology |
| 27172319 |
5 |
Design, Synthesis, and Biological Evaluation of 1-Methyl-1,4-dihydroindeno[1,2-c]pyrazole Analogues as Potential Anticancer Agents Targeting Tubulin Colchicine Binding Site. |
Shandong University |
| 30580241 |
4 |
A class of novel tubulin polymerization inhibitors exert effective anti-tumor activity via mitotic catastrophe. |
Nanjing University |
| 30530194 |
6 |
Design, synthesis and biological evaluation of quinoline-indole derivatives as anti-tubulin agents targeting the colchicine binding site. |
China Pharmaceutical University |
| 30472600 |
2 |
Synthesis, biological evaluation, and molecular docking investigation of 3-amidoindoles as potent tubulin polymerization inhibitors. |
Southern Medical University |
| 31880942 |
1 |
Scaffold Hopping of Natural Product Evodiamine: Discovery of a Novel Antitumor Scaffold with Excellent Potency against Colon Cancer. |
Second Military Medical University |
| 31860298 |
3 |
Structure-Activity Relationship Study of Novel 6-Aryl-2-benzoyl-pyridines as Tubulin Polymerization Inhibitors with Potent Antiproliferative Properties. |
University of Tennessee Health Science Center |
| 31499359 |
1 |
Design, synthesis, and biological evaluation of novel benzodiazepine derivatives as anticancer agents through inhibition of tubulin polymerization in vitro and in vivo. |
The Second Affiliated Hospital of Guangzhou University of Chinese Medicine |
| 31185410 |
2 |
Design, synthesis, antitumor activities and biological studies of novel diaryl substituted fused heterocycles as dual ligands targeting tubulin and katanin. |
Fudan University |
| 30901597 |
1 |
Synthesis and bioevaluation of diarylpyrazoles as antiproliferative agents. |
Shenyang Pharmaceutical University |
| 30525584 |
2 |
Discovery of Novel Quinoline-Chalcone Derivatives as Potent Antitumor Agents with Microtubule Polymerization Inhibitory Activity. |
China Pharmaceutical University |
| 31610372 |
3 |
Design, synthesis, and biological evaluation of 1-substituted -2-aryl imidazoles targeting tubulin polymerization as potential anticancer agents. |
Southern Medical University |
| 31541870 |
2 |
Design and synthesis of (2-(phenylamino)thieno[3,2-d]pyrimidin-4-yl)(3,4,5-trimethoxyphenyl)methanone analogues as potent anti-tubulin polymerization agents. |
Peking University |
| 31536891 |
13 |
Potent combretastatin A-4 analogs containing 1,2,4-triazole: Synthesis, antiproliferative, anti-tubulin activity, and docking study. |
Minia University |
| 26985296 |
4 |
New Colchicine-Derived Triazoles and Their Influence on Cytotoxicity and Microtubule Morphology. |
University of Cologne |
| 26580420 |
13 |
An Orally Bioavailable, Indole-3-glyoxylamide Based Series of Tubulin Polymerization Inhibitors Showing Tumor Growth Inhibition in a Mouse Xenograft Model of Head and Neck Cancer. |
University of Sheffield |
| 24139940 |
5 |
Design and synthesis of silicon-containing tubulin polymerization inhibitors: replacement of the ethylene moiety of combretastatin A-4 with a silicon linker. |
The University of Tokyo |
| 23895532 |
11 |
Structure-activity relationship and in vitro and in vivo evaluation of the potent cytotoxic anti-microtubule agent N-(4-methoxyphenyl)-N,2,6-trimethyl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-aminium chloride and its analogues as antitumor agents. |
Duquesne University |
| 23790539 |
6 |
Design, synthesis and biological studies of novel tubulin inhibitors. |
The Ohio State University |
| 23750455 |
2 |
Design, synthesis, and biological evaluation of (E)-N-aryl-2-arylethenesulfonamide analogues as potent and orally bioavailable microtubule-targeted anticancer agents. |
Icahn School of Medicine At Mount Sinai |
| 23176628 |
21 |
Synthesis and biological evaluation of colchicine B-ring analogues tethered with halogenated benzyl moieties. |
University of Bradford |
| 23010271 |
7 |
Novel cyanocombretastatins as potent tubulin polymerisation inhibitors. |
University of Salford |
| 23259031 |
2 |
Synthesis and Biological Evaluation of a Biotinylated Paclitaxel With an Extra-Long Chain Spacer Arm. |
University of Minnesota |
| 22676247 |
8 |
Synthesis and biological evaluation of 1-benzylidene-3,4-dihydronaphthalen-2-one as a new class of microtubule-targeting agents. |
Second Military Medical University |
| 22329561 |
5 |
Synthesis and biological evaluation of 1,4-diaryl-2-azetidinones as specific anticancer agents: activation of adenosine monophosphate activated protein kinase and induction of apoptosis. |
University of Milan-Bicocca |
| 22185476 |
3 |
Synthesis and structure-activity relationship study of antimicrotubule agents phenylahistin derivatives with a didehydropiperazine-2,5-dione structure. |
Tokyo University of Pharmacy and Life Sciences |
| 22137934 |
9 |
Synthesis, biological evaluation and molecular modeling of 1,2,3-triazole analogs of combretastatin A-1. |
University of Oslo |
| 21920767 |
1 |
Synthesis and biological evaluation of phenstatin metabolites. |
University of Lille |
| 21705223 |
20 |
Phenylimino-10H-anthracen-9-ones as novel antimicrotubule agents-synthesis, antiproliferative activity and inhibition of tubulin polymerization. |
Westphalian Wilhelms-University |
| 21563750 |
45 |
N-benzoylated phenoxazines and phenothiazines: synthesis, antiproliferative activity, and inhibition of tubulin polymerization. |
Westphalian Wilhelms-University |
| 21480626 |
23 |
Synthesis and biological evaluation of 2,4,5-substituted pyrimidines as a new class of tubulin polymerization inhibitors. |
Chinese Academy of Sciences |
| 21106379 |
3 |
Tubulin photoaffinity labeling study with a plinabulin chemical probe possessing a biotin tag at the oxazole. |
Tokyo University of Pharmacy and Life Sciences |
| 21106374 |
5 |
Synthesis and biological evaluation of tubulysin D analogs related to stereoisomers of tubuvaline. |
Kyorin Pharmaceutical |
| 20708408 |
6 |
1,2,3-triazole analogs of combretastatin A-4 as potential microtubule-binding agents. |
University of Oslo |
| 20537765 |
34 |
Synthesis, antiproliferative activity and inhibition of tubulin polymerization by 1,5- and 1,8-disubstituted 10H-anthracen-9-ones bearing a 10-benzylidene or 10-(2-oxo-2-phenylethylidene) moiety. |
Westphalian Wilhelms-University |
| 20395148 |
3 |
Anti-microtubule 'plinabulin' chemical probe KPU-244-B3 labeled both alpha- and beta-tubulin. |
Tokyo University of Pharmacy and Life Sciences |
| 19220018 |
26 |
10-(2-oxo-2-phenylethylidene)-10H-anthracen-9-ones as highly active antimicrotubule agents: synthesis, antiproliferative activity, and inhibition of tubulin polymerization. |
Westphalian Wilhelms-University |
| 18678497 |
2 |
Structure-activity relationship studies on a novel class of antiproliferative agents derived from Lavendustin A. Part I: Ring A modifications. |
Novartis Institutes For Biomedical Research |
| 18396050 |
9 |
1,5-Disubstituted 1,2,3-triazoles as cis-restricted analogues of combretastatin A-4: Synthesis, molecular modeling and evaluation as cytotoxic agents and inhibitors of tubulin. |
University of Oslo |
| 17973361 |
19 |
Sulfonate derivatives of naphtho[2,3-b]thiophen-4(9H)-one and 9(10H)-anthracenone as highly active antimicrotubule agents. Synthesis, antiproliferative activity, and inhibition of tubulin polymerization. |
Cancercare Manitoba |
| 17618122 |
5 |
Synthesis, biological evaluation, and molecular modeling of 3,5-substituted-N1-phenyl-N4,N4-di-n-butylsulfanilamides as antikinetoplastid antimicrotubule agents. |
The Ohio State University |
| 17181164 |
21 |
9-Benzylidene-naphtho[2,3-b]thiophen-4-ones as novel antimicrotubule agents-synthesis, antiproliferative activity, and inhibition of tubulin polymerization. |
Westphalian Wilhelms-University |
| 16870433 |
4 |
Tubulin polymerization inhibitors with a fluorinated phthalimide skeleton derived from thalidomide. |
The University of Tokyo |
| 16213720 |
9 |
Conformationally restricted analogs of Combretastatin A-4 derived from SU5416. |
The Ohio State University |
| 12852768 |
32 |
Novel benzylidene-9(10H)-anthracenones as highly active antimicrotubule agents. Synthesis, antiproliferative activity, and inhibition of tubulin polymerization. |
Westphalian Wilhelms-University |
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