The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
25047579 |
130 |
Synthesis and binding profile of haloperidol-based bivalent ligands targeting dopamine D(2)-like receptors. |
Friedrich-Alexander University |
24100078 |
59 |
Click chemistry based synthesis of dopamine D4 selective receptor ligands for the selection of potential PET tracers. |
Friedrich-Alexander University |
23730937 |
55 |
Functionally selective dopamine D2/D3 receptor agonists comprising an enyne moiety. |
Friedrich-Alexander University |
23099096 |
88 |
Novel azulene derivatives for the treatment of erectile dysfunction. |
Friedrich-Alexander University |
18164618 |
36 |
Discovery of a dopamine D4 selective PET ligand candidate taking advantage of a click chemistry based REM linker. |
Clinic of Nuclear Medicine |
18307287 |
60 |
Synthesis, radiofluorination, and in vitro evaluation of pyrazolo[1,5-a]pyridine-based dopamine D4 receptor ligands: discovery of an inverse agonist radioligand for PET. |
Friedrich-Alexander University |
17154515 |
40 |
trans-2,3-dihydroxy-6a,7,8,12b-tetrahydro-6H-chromeno[3,4-c]isoquinoline: synthesis, resolution, and preliminary pharmacological characterization of a new dopamine D1 receptor full agonist. |
Purdue University |
16789750 |
155 |
2-[(4-phenylpiperazin-1-yl)methyl]imidazo(di)azines as selective D4-ligands. Induction of penile erection by 2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]imidazo[1,2-a]pyridine (PIP3EA), a potent and selective D4 partial agonist. |
Laboratoire De Chimie Th�Rapeutique |
16134944 |
85 |
Pharmacophore-guided drug discovery investigations leading to bioactive 5-aminotetrahydropyrazolopyridines. Implications for the binding mode of heterocyclic dopamine D3 receptor agonists. |
Friedrich-Alexander University |
15916420 |
68 |
Fancy bioisosteres: metallocene-derived G-protein-coupled receptor ligands with subnanomolar binding affinity and novel selectivity profiles. |
Friedrich-Alexander University |
22100258 |
124 |
Bivalent molecular probes for dopamine D2-like receptors. |
Friedrich-Alexander University |
22039961 |
21 |
Evaluation of 18F-labeled benzodioxine piperazine-based dopamine D4 receptor ligands: lipophilicity as a determinate of nonspecific binding. |
Forschungszentrum J£Lich |
21999579 |
40 |
Development of a bivalent dopamine D2 receptor agonist. |
Friedrich-Alexander University |
21599022 |
66 |
Bivalent dopamine D2 receptor ligands: synthesis and binding properties. |
Friedrich-Alexander University |
21273071 |
73 |
Aromatic ring functionalization of benzolactam derivatives: new potent dopamine D3 receptor ligands. |
University of Santiago De Compostela |
21388142 |
57 |
Highly potent 5-aminotetrahydropyrazolopyridines: enantioselective dopamine D3 receptor binding, functional selectivity, and analysis of receptor-ligand interactions. |
Friedrich-Alexander University |
21030255 |
18 |
Synthesis, biological evaluation and radiolabelling by 18F-fluoroarylation of a dopamine D3-selective ligand as prospective imaging probe for PET. |
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg |
20860381 |
61 |
Novel pyridylmethylamines as highly selective 5-HT(1A) superagonists. |
Friedrich-Alexander University |
20839776 |
105 |
Bioisosteric replacement leading to biologically active [2.2]paracyclophanes with altered binding profiles for aminergic G-protein-coupled receptors. |
Friedrich-Alexander University |
19807103 |
14 |
1,1'-Disubstituted ferrocenes as molecular hinges in mono- and bivalent dopamine receptor ligands. |
Friedrich-Alexander University |
19592258 |
20 |
Parallel synthesis of potent dopaminergic N-phenyltriazole carboxamides applying a novel click chemistry based phenol linker. |
Friedrich-Alexander University |
18834111 |
68 |
Novel D3 selective dopaminergics incorporating enyne units as nonaromatic catechol bioisosteres: synthesis, bioactivity, and mutagenesis studies. |
Friedrich-Alexander University |
17827018 |
64 |
Click chemistry based solid phase supported synthesis of dopaminergic phenylacetylenes. |
Friedrich-Alexander University |
17765546 |
36 |
In vitro affinities of various halogenated benzamide derivatives as potential radioligands for non-invasive quantification of D(2)-like dopamine receptors. |
Johannes Gutenberg University |
17266201 |
13 |
Structure-selectivity investigations of D2-like receptor ligands by CoMFA and CoMSIA guiding the discovery of D3 selective PET radioligands. |
Friedrich-Alexander University |
16563764 |
100 |
Synthesis and biological investigations of dopaminergic partial agonists preferentially recognizing the D4 receptor subtype. |
Friedrich-Alexander University |
16139501 |
54 |
Synthesis and evaluation of 18F-labeled dopamine D3 receptor ligands as potential PET imaging agents. |
University of Erlangen-Nuremberg |
15225707 |
42 |
Synthesis and radioiodination of selective ligands for the dopamine D3 receptor subtype. |
University of Erlangen-Nuremberg |