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28 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
25047579 130 Synthesis and binding profile of haloperidol-based bivalent ligands targeting dopamine D(2)-like receptors.EBI Friedrich-Alexander University
24100078 59 Click chemistry based synthesis of dopamine D4 selective receptor ligands for the selection of potential PET tracers.EBI Friedrich-Alexander University
23730937 55 Functionally selective dopamine D2/D3 receptor agonists comprising an enyne moiety.EBI Friedrich-Alexander University
23099096 88 Novel azulene derivatives for the treatment of erectile dysfunction.EBI Friedrich-Alexander University
18164618 36 Discovery of a dopamine D4 selective PET ligand candidate taking advantage of a click chemistry based REM linker.EBI Clinic of Nuclear Medicine
18307287 60 Synthesis, radiofluorination, and in vitro evaluation of pyrazolo[1,5-a]pyridine-based dopamine D4 receptor ligands: discovery of an inverse agonist radioligand for PET.EBI Friedrich-Alexander University
17154515 40 trans-2,3-dihydroxy-6a,7,8,12b-tetrahydro-6H-chromeno[3,4-c]isoquinoline: synthesis, resolution, and preliminary pharmacological characterization of a new dopamine D1 receptor full agonist.EBI Purdue University
16789750 155 2-[(4-phenylpiperazin-1-yl)methyl]imidazo(di)azines as selective D4-ligands. Induction of penile erection by 2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]imidazo[1,2-a]pyridine (PIP3EA), a potent and selective D4 partial agonist.EBI Laboratoire De Chimie Th�Rapeutique
16134944 85 Pharmacophore-guided drug discovery investigations leading to bioactive 5-aminotetrahydropyrazolopyridines. Implications for the binding mode of heterocyclic dopamine D3 receptor agonists.EBI Friedrich-Alexander University
15916420 68 Fancy bioisosteres: metallocene-derived G-protein-coupled receptor ligands with subnanomolar binding affinity and novel selectivity profiles.EBI Friedrich-Alexander University
22100258 124 Bivalent molecular probes for dopamine D2-like receptors.EBI Friedrich-Alexander University
22039961 21 Evaluation of 18F-labeled benzodioxine piperazine-based dopamine D4 receptor ligands: lipophilicity as a determinate of nonspecific binding.EBI Forschungszentrum J£Lich
21999579 40 Development of a bivalent dopamine D2 receptor agonist.EBI Friedrich-Alexander University
21599022 66 Bivalent dopamine D2 receptor ligands: synthesis and binding properties.EBI Friedrich-Alexander University
21273071 73 Aromatic ring functionalization of benzolactam derivatives: new potent dopamine D3 receptor ligands.EBI University of Santiago De Compostela
21388142 57 Highly potent 5-aminotetrahydropyrazolopyridines: enantioselective dopamine D3 receptor binding, functional selectivity, and analysis of receptor-ligand interactions.EBI Friedrich-Alexander University
21030255 18 Synthesis, biological evaluation and radiolabelling by 18F-fluoroarylation of a dopamine D3-selective ligand as prospective imaging probe for PET.EBI Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
20860381 61 Novel pyridylmethylamines as highly selective 5-HT(1A) superagonists.EBI Friedrich-Alexander University
20839776 105 Bioisosteric replacement leading to biologically active [2.2]paracyclophanes with altered binding profiles for aminergic G-protein-coupled receptors.EBI Friedrich-Alexander University
19807103 14 1,1'-Disubstituted ferrocenes as molecular hinges in mono- and bivalent dopamine receptor ligands.EBI Friedrich-Alexander University
19592258 20 Parallel synthesis of potent dopaminergic N-phenyltriazole carboxamides applying a novel click chemistry based phenol linker.EBI Friedrich-Alexander University
18834111 68 Novel D3 selective dopaminergics incorporating enyne units as nonaromatic catechol bioisosteres: synthesis, bioactivity, and mutagenesis studies.EBI Friedrich-Alexander University
17827018 64 Click chemistry based solid phase supported synthesis of dopaminergic phenylacetylenes.EBI Friedrich-Alexander University
17765546 36 In vitro affinities of various halogenated benzamide derivatives as potential radioligands for non-invasive quantification of D(2)-like dopamine receptors.EBI Johannes Gutenberg University
17266201 13 Structure-selectivity investigations of D2-like receptor ligands by CoMFA and CoMSIA guiding the discovery of D3 selective PET radioligands.EBI Friedrich-Alexander University
16563764 100 Synthesis and biological investigations of dopaminergic partial agonists preferentially recognizing the D4 receptor subtype.EBI Friedrich-Alexander University
16139501 54 Synthesis and evaluation of 18F-labeled dopamine D3 receptor ligands as potential PET imaging agents.EBI University of Erlangen-Nuremberg
15225707 42 Synthesis and radioiodination of selective ligands for the dopamine D3 receptor subtype.EBI University of Erlangen-Nuremberg