BDBM108293 US8604046, 73
SMILES: C[C@H]1CCCN1[C@H]1CCN(C1)c1ccc(cc1)N1CCCC2(CCN(CC3CC3)CC2)C1=O
InChI Key: InChIKey=XJXJPAVAMSBCQC-NVQXNPDNSA-N
Data: 1 KI
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Histamine H3 receptor (Macaca mulatta (Rhesus macaque)) | BDBM108293 (US8604046, 73) | UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 0.200 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Patent | Assay Description The compounds of this invention have been demonstrated to displace [3H]- methylhistamine radioligand binding to mammalian cell membranes expressing r... | US Patent US8604046 (2013) BindingDB Entry DOI: 10.7270/Q2W957TB | |||||||||||
More data for this Ligand-Target Pair |