BDBM50274260 2-(6,8-Dichloro-2-(4-methoxyphenyl)imidazo[1,2-a]pyridin-3-yl)-N-methyl-N-phenylacetamide::CHEMBL485606
SMILES: COc1ccc(cc1)-c1nc2c(Cl)cc(Cl)cn2c1CC(=O)N(C)c1ccccc1
InChI Key: InChIKey=QJCLUBBQLHBLOP-UHFFFAOYSA-N
Data: 1 KI
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
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Peripheral-Type Benzodiazepine Receptor (Rattus norvegicus (rat)) | BDBM50274260 (2-(6,8-Dichloro-2-(4-methoxyphenyl)imidazo[1,2-a]p...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.230 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universita degli Studi di Bari Curated by ChEMBL | Assay Description Displacement of [3H]PK11195 from peripheral benzodiazepine receptor in Sprague-Dawley rat cerebral cortex membrane by liquid scintillation counting | J Med Chem 51: 6876-88 (2008) Article DOI: 10.1021/jm8006728 BindingDB Entry DOI: 10.7270/Q23B612K | |||||||||||
More data for this Ligand-Target Pair |