Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Retinoic acid receptor gamma (Homo sapiens (Human)) | BDBM50457541 (CHEMBL4216161) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 7.40 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor alpha (Homo sapiens (Human)) | BDBM50457542 (CHEMBL4212472) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 11 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARalpha (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor alpha (Homo sapiens (Human)) | BDBM50457543 (CHEMBL3934863) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARalpha (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor beta (Homo sapiens (Human)) | BDBM50457544 (CHEMBL3936922) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 25 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARbeta (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hrs... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor gamma (Homo sapiens (Human)) | BDBM50457545 (CHEMBL4210286) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 353 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Inverse agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated f... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor alpha (Homo sapiens (Human)) | BDBM50457546 (CHEMBL4206237) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 212 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARalpha (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor alpha (Homo sapiens (Human)) | BDBM50457547 (CHEMBL3953756) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 103 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARalpha (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor alpha (Homo sapiens (Human)) | BDBM50457548 (CD-5789 | Trifarotene) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 500 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARalpha (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor beta (Homo sapiens (Human)) | BDBM50457549 (CHEMBL3960035) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 17 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARbeta (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hrs... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor beta (Homo sapiens (Human)) | BDBM50457550 (CHEMBL4207978) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARbeta (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hrs... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor gamma (Homo sapiens (Human)) | BDBM31888 (CD666) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 46 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor gamma (Homo sapiens (Human)) | BDBM393289 (US9963439, BMS961) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 51 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor gamma (Homo sapiens (Human)) | BDBM50048291 (6-(3-Adamantan-1-yl-4-hydroxy-phenyl)-naphthalene-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | n/a | n/a | n/a | n/a | 49 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Retinoic acid receptor gamma (Homo sapiens (Human)) | BDBM50457551 (CHEMBL4217953) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 6 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor gamma (Homo sapiens (Human)) | BDBM50457552 (CHEMBL4210595) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 0.220 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor gamma (Homo sapiens (Human)) | BDBM50457553 (CHEMBL4210099) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 4.40 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor gamma (Homo sapiens (Human)) | BDBM50457554 (CHEMBL4202830) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.40 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor gamma (Homo sapiens (Human)) | BDBM50457555 (CHEMBL4214493) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 60 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor gamma (Homo sapiens (Human)) | BDBM50457556 (CHEMBL4217018) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 47 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor gamma (Homo sapiens (Human)) | BDBM50457557 (CHEMBL4215630) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 120 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor gamma (Homo sapiens (Human)) | BDBM50457558 (CHEMBL4203950) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 422 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor gamma (Homo sapiens (Human)) | BDBM50457559 (CHEMBL4212684) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 85 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor gamma (Homo sapiens (Human)) | BDBM50457549 (CHEMBL3960035) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 4.70 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor gamma (Homo sapiens (Human)) | BDBM50457560 (CHEMBL3939687) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.90 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor gamma (Homo sapiens (Human)) | BDBM50457561 (CHEMBL3916016) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 2.10 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor gamma (Homo sapiens (Human)) | BDBM50457544 (CHEMBL3936922) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 3.60 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor gamma (Homo sapiens (Human)) | BDBM50457550 (CHEMBL4207978) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 67 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor alpha (Homo sapiens (Human)) | BDBM50048280 (6-(3-(1-Adamantyl)-4-methoxyphenyl)-2-naphthoic ac...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid UniChem Patents Similars | DrugBank Article PubMed | n/a | n/a | n/a | n/a | 22 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARalpha (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor alpha (Homo sapiens (Human)) | BDBM393289 (US9963439, BMS961) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARalpha (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor alpha (Homo sapiens (Human)) | BDBM50048291 (6-(3-Adamantan-1-yl-4-hydroxy-phenyl)-naphthalene-...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARalpha (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor alpha (Homo sapiens (Human)) | BDBM50457562 (CHEMBL4203742) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 59 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARalpha (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor alpha (Homo sapiens (Human)) | BDBM50457563 (CHEMBL4205733) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 40 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARalpha (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor alpha (Homo sapiens (Human)) | BDBM50457564 (CHEMBL4215021) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARalpha (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor alpha (Homo sapiens (Human)) | BDBM50457553 (CHEMBL4210099) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 336 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARalpha (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor alpha (Homo sapiens (Human)) | BDBM50457549 (CHEMBL3960035) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 180 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARalpha (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor alpha (Homo sapiens (Human)) | BDBM50457560 (CHEMBL3939687) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 180 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARalpha (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor alpha (Homo sapiens (Human)) | BDBM50457545 (CHEMBL4210286) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARalpha (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor alpha (Homo sapiens (Human)) | BDBM50457544 (CHEMBL3936922) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.01E+3 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARalpha (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor alpha (Homo sapiens (Human)) | BDBM50457565 (CHEMBL3910072) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARalpha (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor alpha (Homo sapiens (Human)) | BDBM50457566 (CHEMBL4211171) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARalpha (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor beta (Homo sapiens (Human)) | BDBM50048280 (6-(3-(1-Adamantyl)-4-methoxyphenyl)-2-naphthoic ac...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid UniChem Patents Similars | DrugBank Article PubMed | n/a | n/a | n/a | n/a | 2 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARbeta (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hrs... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor beta (Homo sapiens (Human)) | BDBM50457542 (CHEMBL4212472) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 2.5 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARbeta (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hrs... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor beta (Homo sapiens (Human)) | BDBM50457562 (CHEMBL4203742) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 8.60 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARbeta (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hrs... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor beta (Homo sapiens (Human)) | BDBM50457551 (CHEMBL4217953) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 40 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARbeta (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hrs... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor beta (Homo sapiens (Human)) | BDBM50457563 (CHEMBL4205733) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 6.80 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARbeta (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hrs... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor beta (Homo sapiens (Human)) | BDBM50457564 (CHEMBL4215021) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 13 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARbeta (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hrs... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor beta (Homo sapiens (Human)) | BDBM50457554 (CHEMBL4202830) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 40 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARbeta (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hrs... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor beta (Homo sapiens (Human)) | BDBM50457561 (CHEMBL3916016) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 60 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARbeta (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hrs... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor beta (Homo sapiens (Human)) | BDBM50457567 (CHEMBL3891815) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 35 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARbeta (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hrs... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor beta (Homo sapiens (Human)) | BDBM50457548 (CD-5789 | Trifarotene) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 125 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARbeta (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hrs... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair |
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