Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Retinoic acid receptor gamma (Homo sapiens (Human)) | BDBM50048291 (6-(3-Adamantan-1-yl-4-hydroxy-phenyl)-naphthalene-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | PDB PubMed | 77 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
CIRD GALDERMA Curated by ChEMBL | Assay Description Binding affinity to retinoic acid receptor (RAR) gamma using [3H]-CD 367 as radioligand | J Med Chem 38: 4993-5006 (1996) BindingDB Entry DOI: 10.7270/Q20G3J8S | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Retinoic acid receptor gamma (Homo sapiens (Human)) | BDBM50048291 (6-(3-Adamantan-1-yl-4-hydroxy-phenyl)-naphthalene-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | n/a | n/a | n/a | n/a | 49 | n/a | n/a | n/a | n/a |
Nestle Skin Health Curated by ChEMBL | Assay Description Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr... | Bioorg Med Chem Lett 28: 1736-1741 (2018) Article DOI: 10.1016/j.bmcl.2018.04.036 BindingDB Entry DOI: 10.7270/Q2N300JQ | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) |