Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
72 kDa type IV collagenase (Homo sapiens (Human)) | BDBM50026872![]() (CHEMBL1233506 | SC-74020) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL DrugBank PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | <0.100 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of full length MMP2 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured after 3... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Matrix metalloproteinase-9 (Homo sapiens (Human)) | BDBM50366175![]() (CHEMBL1957606) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of MMP9 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured af... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
72 kDa type IV collagenase (Homo sapiens (Human)) | BDBM50366175![]() (CHEMBL1957606) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.800 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of full length MMP2 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured after 3... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 1/2 (Homo sapiens (Human)) | BDBM50475205![]() (CHEMBL190899) | PDB KEGG UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet ![]() | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.80 | n/a | n/a | n/a | n/a | n/a | n/a |
Domp£ S.p.A. Curated by ChEMBL | Assay Description Inhibition of CXCL8-induced chemotaxis in human polymorphonuclear cells | J Med Chem 48: 4312-31 (2005) Article DOI: 10.1021/jm049082i BindingDB Entry DOI: 10.7270/Q2Z89G5H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Matrix metalloproteinase-9 (Homo sapiens (Human)) | BDBM50366203![]() (CHEMBL1957601) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of MMP9 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured af... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutrophil collagenase (Homo sapiens (Human)) | BDBM50366175![]() (CHEMBL1957606) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of MMP8 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured af... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Matrix metalloproteinase-14 (Homo sapiens (Human)) | BDBM50366175![]() (CHEMBL1957606) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of MMP14 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured a... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Matrix metalloproteinase-9 (Homo sapiens (Human)) | BDBM50366205![]() (CHEMBL1957603) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of MMP9 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured af... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 1/2 (Homo sapiens (Human)) | BDBM50169045![]() ((R)-2-(4-isobutylphenyl)-N-(methylsulfonyl)propana...) | PDB KEGG UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 5.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Domp£ S.p.A. Curated by ChEMBL | Assay Description Inhibition of CXCL8-induced chemotaxis in human polymorphonuclear cells | J Med Chem 48: 4312-31 (2005) Article DOI: 10.1021/jm049082i BindingDB Entry DOI: 10.7270/Q2Z89G5H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
72 kDa type IV collagenase (Homo sapiens (Human)) | BDBM50366203![]() (CHEMBL1957601) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of full length MMP2 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured after 3... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
72 kDa type IV collagenase (Homo sapiens (Human)) | BDBM50366173![]() (CHEMBL1957604) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of full length MMP2 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured after 3... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
72 kDa type IV collagenase (Homo sapiens (Human)) | BDBM50366205![]() (CHEMBL1957603) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of full length MMP2 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured after 3... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
72 kDa type IV collagenase (Homo sapiens (Human)) | BDBM50366204![]() (CHEMBL1957602) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 13 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of full length MMP2 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured after 3... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Matrix metalloproteinase-9 (Homo sapiens (Human)) | BDBM50366204![]() (CHEMBL1957602) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 16 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of MMP9 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured af... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Macrophage metalloelastase (Homo sapiens (Human)) | BDBM50366175![]() (CHEMBL1957606) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 19 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of MMP12 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured a... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 1/2 (Homo sapiens (Human)) | BDBM50169048![]() ((R)-2-(3-Benzoyl-phenyl)-propionic acid | (R)-2-(3...) | PDB KEGG UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 34 | n/a | n/a | n/a | n/a | n/a | n/a |
Domp£ S.p.A. Curated by ChEMBL | Assay Description Inhibition of CXCL8-induced chemotaxis in human polymorphonuclear cells | J Med Chem 48: 4312-31 (2005) Article DOI: 10.1021/jm049082i BindingDB Entry DOI: 10.7270/Q2Z89G5H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 1/2 (Homo sapiens (Human)) | BDBM50088570![]() ((S)-2-(3-Benzoyl-phenyl)-propionic acid | (S)-2-(3...) | PDB KEGG UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 50 | n/a | n/a | n/a | n/a | n/a | n/a |
Domp£ S.p.A. Curated by ChEMBL | Assay Description Inhibition of CXCL8-induced chemotaxis in human polymorphonuclear cells | J Med Chem 48: 4312-31 (2005) Article DOI: 10.1021/jm049082i BindingDB Entry DOI: 10.7270/Q2Z89G5H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
72 kDa type IV collagenase (Homo sapiens (Human)) | BDBM50366174![]() (CHEMBL1957605) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 53 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of full length MMP2 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured after 3... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 1/2 (Homo sapiens (Human)) | BDBM50475204![]() (CHEMBL192943) | PDB KEGG UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet ![]() | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 80 | n/a | n/a | n/a | n/a | n/a | n/a |
Domp£ S.p.A. Curated by ChEMBL | Assay Description Inhibition of CXCL8-induced chemotaxis in human polymorphonuclear cells | J Med Chem 48: 4312-31 (2005) Article DOI: 10.1021/jm049082i BindingDB Entry DOI: 10.7270/Q2Z89G5H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutrophil collagenase (Homo sapiens (Human)) | BDBM50366174![]() (CHEMBL1957605) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of MMP8 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured af... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 1/2 (Homo sapiens (Human)) | BDBM50169047![]() ((S)-2-(4-Isobutyl-phenyl)-propionic acid | (S)-2-(...) | PDB KEGG UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
Domp£ S.p.A. Curated by ChEMBL | Assay Description Inhibition of CXCL8-induced chemotaxis in human polymorphonuclear cells | J Med Chem 48: 4312-31 (2005) Article DOI: 10.1021/jm049082i BindingDB Entry DOI: 10.7270/Q2Z89G5H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 1/2 (Homo sapiens (Human)) | BDBM50169044![]() ((-)-ibuprofen | (2R)-2-(4-isobutylphenyl)propanoic...) | PDB KEGG UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 110 | n/a | n/a | n/a | n/a | n/a | n/a |
Domp£ S.p.A. Curated by ChEMBL | Assay Description Inhibition of CXCL8-induced chemotaxis in human polymorphonuclear cells | J Med Chem 48: 4312-31 (2005) Article DOI: 10.1021/jm049082i BindingDB Entry DOI: 10.7270/Q2Z89G5H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Stromelysin-1 (Homo sapiens (Human)) | BDBM50366204![]() (CHEMBL1957602) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 160 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of MMP3 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured af... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Matrix metalloproteinase-14 (Homo sapiens (Human)) | BDBM50366173![]() (CHEMBL1957604) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 160 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of MMP14 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured a... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
72 kDa type IV collagenase (Homo sapiens (Human)) | BDBM50366200![]() (CHEMBL1957598) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of full length MMP2 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured after 3... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Matrix metalloproteinase-9 (Homo sapiens (Human)) | BDBM50366200![]() (CHEMBL1957598) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 230 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of MMP9 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured af... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutrophil collagenase (Homo sapiens (Human)) | BDBM50366173![]() (CHEMBL1957604) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 400 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of MMP8 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured af... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Matrix metalloproteinase-9 (Homo sapiens (Human)) | BDBM50366174![]() (CHEMBL1957605) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 480 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of MMP9 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured af... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Macrophage metalloelastase (Homo sapiens (Human)) | BDBM50366174![]() (CHEMBL1957605) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 500 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of MMP12 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured a... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Matrix metalloproteinase-9 (Homo sapiens (Human)) | BDBM50366202![]() (CHEMBL1957600) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 560 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of MMP9 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured af... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Matrix metalloproteinase-9 (Homo sapiens (Human)) | BDBM50366173![]() (CHEMBL1957604) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 600 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of MMP9 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured af... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Stromelysin-1 (Homo sapiens (Human)) | BDBM50366205![]() (CHEMBL1957603) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 700 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of MMP3 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured af... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
72 kDa type IV collagenase (Homo sapiens (Human)) | BDBM50366202![]() (CHEMBL1957600) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 710 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of full length MMP2 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured after 3... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Interstitial collagenase (Homo sapiens (Human)) | BDBM50366204![]() (CHEMBL1957602) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of MMP1 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured af... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
72 kDa type IV collagenase (Homo sapiens (Human)) | BDBM50366198![]() (CHEMBL1957596) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of full length MMP2 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured after 3... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Matrix metalloproteinase-9 (Homo sapiens (Human)) | BDBM50366198![]() (CHEMBL1957596) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of MMP9 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured af... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Stromelysin-1 (Homo sapiens (Human)) | BDBM50366173![]() (CHEMBL1957604) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of MMP3 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured af... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Macrophage metalloelastase (Homo sapiens (Human)) | BDBM50366173![]() (CHEMBL1957604) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of MMP12 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured a... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Interstitial collagenase (Homo sapiens (Human)) | BDBM50366174![]() (CHEMBL1957605) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of MMP1 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured af... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
72 kDa type IV collagenase (Homo sapiens (Human)) | BDBM50366176![]() (CHEMBL1957575) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of full length MMP2 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured after 3... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Matrix metalloproteinase-14 (Homo sapiens (Human)) | BDBM50366174![]() (CHEMBL1957605) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of MMP14 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured a... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Interstitial collagenase (Homo sapiens (Human)) | BDBM50366173![]() (CHEMBL1957604) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of MMP1 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured af... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
72 kDa type IV collagenase (Homo sapiens (Human)) | BDBM50366199![]() (CHEMBL1957597) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of full length MMP2 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured after 3... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Stromelysin-1 (Homo sapiens (Human)) | BDBM50366174![]() (CHEMBL1957605) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of MMP3 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured af... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
72 kDa type IV collagenase (Homo sapiens (Human)) | BDBM50366197![]() (CHEMBL1957595) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of full length MMP2 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured after 3... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
72 kDa type IV collagenase (Homo sapiens (Human)) | BDBM50366185![]() (CHEMBL1957584) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of full length MMP2 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured after 3... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Matrix metalloproteinase-9 (Homo sapiens (Human)) | BDBM50366176![]() (CHEMBL1957575) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of MMP9 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured af... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
72 kDa type IV collagenase (Homo sapiens (Human)) | BDBM50366201![]() (CHEMBL1957599) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of full length MMP2 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured after 3... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Matrix metalloproteinase-9 (Homo sapiens (Human)) | BDBM50366197![]() (CHEMBL1957595) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of MMP9 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured af... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Interstitial collagenase (Homo sapiens (Human)) | BDBM50366205![]() (CHEMBL1957603) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Colosseum Combinatorial Chemistry Centre for Technology (C4T SCarl) Curated by ChEMBL | Assay Description Inhibition of MMP1 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured af... | Bioorg Med Chem 20: 2323-37 (2012) Article DOI: 10.1016/j.bmc.2012.02.010 BindingDB Entry DOI: 10.7270/Q2N29XD5 | |||||||||||
More data for this Ligand-Target Pair |
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