Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Arginase (Leishmania amazonensis) | BDBM50521944 (CHEMBL4204512) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Rio de Janeiro Curated by ChEMBL | Assay Description Competitive inhibition of recombinant Leishmania amazonensis arginase expressed in Escherichia coli assessed as reduction in urea production by measu... | Bioorg Med Chem 27: 3853-3859 (2019) Article DOI: 10.1016/j.bmc.2019.07.022 BindingDB Entry DOI: 10.7270/Q27D2ZJF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Arginase (Leishmania amazonensis) | BDBM50521942 (CHEMBL4216180) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 5.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Rio de Janeiro Curated by ChEMBL | Assay Description Competitive inhibition of recombinant Leishmania amazonensis arginase expressed in Escherichia coli assessed as reduction in urea production by measu... | Bioorg Med Chem 27: 3853-3859 (2019) Article DOI: 10.1016/j.bmc.2019.07.022 BindingDB Entry DOI: 10.7270/Q27D2ZJF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Arginase (Leishmania amazonensis) | BDBM50521943 (CHEMBL4574177) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 2.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Rio de Janeiro Curated by ChEMBL | Assay Description Competitive inhibition of recombinant Leishmania amazonensis arginase expressed in Escherichia coli assessed as reduction in urea production by measu... | Bioorg Med Chem 27: 3853-3859 (2019) Article DOI: 10.1016/j.bmc.2019.07.022 BindingDB Entry DOI: 10.7270/Q27D2ZJF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Arginase (Leishmania amazonensis) | BDBM50521947 (CHEMBL4530523) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 3.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Rio de Janeiro Curated by ChEMBL | Assay Description Competitive inhibition of recombinant Leishmania amazonensis arginase expressed in Escherichia coli assessed as reduction in urea production by measu... | Bioorg Med Chem 27: 3853-3859 (2019) Article DOI: 10.1016/j.bmc.2019.07.022 BindingDB Entry DOI: 10.7270/Q27D2ZJF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Arginase (Leishmania amazonensis) | BDBM50521944 (CHEMBL4204512) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Rio de Janeiro Curated by ChEMBL | Assay Description Inhibition of recombinant Leishmania amazonensis arginase expressed in Escherichia coli assessed as reduction in urea production using L-arginine as ... | Bioorg Med Chem 27: 3853-3859 (2019) Article DOI: 10.1016/j.bmc.2019.07.022 BindingDB Entry DOI: 10.7270/Q27D2ZJF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Arginase (Leishmania amazonensis) | BDBM50521942 (CHEMBL4216180) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Rio de Janeiro Curated by ChEMBL | Assay Description Inhibition of recombinant Leishmania amazonensis arginase expressed in Escherichia coli assessed as reduction in urea production using L-arginine as ... | Bioorg Med Chem 27: 3853-3859 (2019) Article DOI: 10.1016/j.bmc.2019.07.022 BindingDB Entry DOI: 10.7270/Q27D2ZJF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Arginase (Leishmania amazonensis) | BDBM50521947 (CHEMBL4530523) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Rio de Janeiro Curated by ChEMBL | Assay Description Inhibition of recombinant Leishmania amazonensis arginase expressed in Escherichia coli assessed as reduction in urea production using L-arginine as ... | Bioorg Med Chem 27: 3853-3859 (2019) Article DOI: 10.1016/j.bmc.2019.07.022 BindingDB Entry DOI: 10.7270/Q27D2ZJF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Arginase (Leishmania amazonensis) | BDBM50521943 (CHEMBL4574177) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Rio de Janeiro Curated by ChEMBL | Assay Description Inhibition of recombinant Leishmania amazonensis arginase expressed in Escherichia coli assessed as reduction in urea production using L-arginine as ... | Bioorg Med Chem 27: 3853-3859 (2019) Article DOI: 10.1016/j.bmc.2019.07.022 BindingDB Entry DOI: 10.7270/Q27D2ZJF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Arginase (Leishmania amazonensis) | BDBM50521946 (CHEMBL4211729) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Rio de Janeiro Curated by ChEMBL | Assay Description Inhibition of recombinant Leishmania amazonensis arginase expressed in Escherichia coli assessed as reduction in urea production using L-arginine as ... | Bioorg Med Chem 27: 3853-3859 (2019) Article DOI: 10.1016/j.bmc.2019.07.022 BindingDB Entry DOI: 10.7270/Q27D2ZJF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Arginase (Leishmania amazonensis) | BDBM50521945 (CHEMBL4216693) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Rio de Janeiro Curated by ChEMBL | Assay Description Inhibition of recombinant Leishmania amazonensis arginase expressed in Escherichia coli assessed as reduction in urea production using L-arginine as ... | Bioorg Med Chem 27: 3853-3859 (2019) Article DOI: 10.1016/j.bmc.2019.07.022 BindingDB Entry DOI: 10.7270/Q27D2ZJF | |||||||||||
More data for this Ligand-Target Pair |