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| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM498079 ((5'S)-N-{[5- (Ethylsulfonyl)pyridin- 2-yl]methyl}-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet  | PC cid PC sid UniChem | US Patent | 3.27 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Eli Lilly and Company US Patent | Assay Description Receptor competition binding assays are run in a buffer made up of DPBS (1 L) (Hyclone #SH30028.03), 2.2 g BSA Fraction v (Roche #9048-46-8), 100 mL ... | US Patent US11008336 (2021) BindingDB Entry DOI: 10.7270/Q2W380G1 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM498077 (N-[4- (Ethylsulfonyl)benzyl]- 5'-methyl-1-{1-[6- (...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 4.42 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Eli Lilly and Company US Patent | Assay Description Receptor competition binding assays are run in a buffer made up of DPBS (1 L) (Hyclone #SH30028.03), 2.2 g BSA Fraction v (Roche #9048-46-8), 100 mL ... | US Patent US11008336 (2021) BindingDB Entry DOI: 10.7270/Q2W380G1 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM498074 ((5′S)—N-[4-(Ethylsulfonyl)benzyl]-5′-m...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 5.88 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Eli Lilly and Company US Patent | Assay Description Receptor competition binding assays are run in a buffer made up of DPBS (1 L) (Hyclone #SH30028.03), 2.2 g BSA Fraction v (Roche #9048-46-8), 100 mL ... | US Patent US11008336 (2021) BindingDB Entry DOI: 10.7270/Q2W380G1 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM438836 (1'-[1-(4- Cyanophenyl)ethyl]- 5,5- spirocyclopropa...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Eli Lilly and Company US Patent | Assay Description His-tagged human RAR-related orphan receptor alpha (hRORa), human RAR-related orphan receptor beta (hRORb), and human RAR-related orphan receptor gam... | US Patent US10603320 (2020) BindingDB Entry DOI: 10.7270/Q2154M2H | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM498076 ((5'S)-N-{[5- (Ethylsulfonyl)pyridin- 2-yl]methyl}-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 6.04 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Eli Lilly and Company US Patent | Assay Description Receptor competition binding assays are run in a buffer made up of DPBS (1 L) (Hyclone #SH30028.03), 2.2 g BSA Fraction v (Roche #9048-46-8), 100 mL ... | US Patent US11008336 (2021) BindingDB Entry DOI: 10.7270/Q2W380G1 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM438835 (N-{[5-(Ethylsulfonyl)pyridin-2-yl]methyl}-1″...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 6.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Eli Lilly and Company US Patent | Assay Description His-tagged human RAR-related orphan receptor alpha (hRORa), human RAR-related orphan receptor beta (hRORb), and human RAR-related orphan receptor gam... | US Patent US10603320 (2020) BindingDB Entry DOI: 10.7270/Q2154M2H | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM438834 (N-{[5-(Ethylsulfonyl)pyridin-2-yl]methyl}-5′...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 6.96 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Eli Lilly and Company US Patent | Assay Description His-tagged human RAR-related orphan receptor alpha (hRORa), human RAR-related orphan receptor beta (hRORb), and human RAR-related orphan receptor gam... | US Patent US10603320 (2020) BindingDB Entry DOI: 10.7270/Q2154M2H | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM498078 (N-{[5- (Ethylsulfonyl)pyridin- 2-yl]methyl}-5'- me...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 10.8 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Eli Lilly and Company US Patent | Assay Description Receptor competition binding assays are run in a buffer made up of DPBS (1 L) (Hyclone #SH30028.03), 2.2 g BSA Fraction v (Roche #9048-46-8), 100 mL ... | US Patent US11008336 (2021) BindingDB Entry DOI: 10.7270/Q2W380G1 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM498080 (1-[(1S)-1-(4- Cyanophenyl)ethyl]- N-[4- (ethylsulf...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 15.8 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Eli Lilly and Company US Patent | Assay Description Receptor competition binding assays are run in a buffer made up of DPBS (1 L) (Hyclone #SH30028.03), 2.2 g BSA Fraction v (Roche #9048-46-8), 100 mL ... | US Patent US11008336 (2021) BindingDB Entry DOI: 10.7270/Q2W380G1 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM498081 ((5'S)-N-[4- (Ethylsulfonyl)benzyl]- 5'-methyl-1-{1...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 151 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Eli Lilly and Company US Patent | Assay Description Receptor competition binding assays are run in a buffer made up of DPBS (1 L) (Hyclone #SH30028.03), 2.2 g BSA Fraction v (Roche #9048-46-8), 100 mL ... | US Patent US11008336 (2021) BindingDB Entry DOI: 10.7270/Q2W380G1 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Nuclear receptor ROR-alpha (Homo sapiens (Human)) | BDBM498081 ((5'S)-N-[4- (Ethylsulfonyl)benzyl]- 5'-methyl-1-{1...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 698 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Eli Lilly and Company US Patent | Assay Description Receptor competition binding assays are run in a buffer made up of DPBS (1 L) (Hyclone #SH30028.03), 2.2 g BSA Fraction v (Roche #9048-46-8), 100 mL ... | US Patent US11008336 (2021) BindingDB Entry DOI: 10.7270/Q2W380G1 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Nuclear receptor ROR-alpha (Homo sapiens (Human)) | BDBM498076 ((5'S)-N-{[5- (Ethylsulfonyl)pyridin- 2-yl]methyl}-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 1.05E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Eli Lilly and Company US Patent | Assay Description Receptor competition binding assays are run in a buffer made up of DPBS (1 L) (Hyclone #SH30028.03), 2.2 g BSA Fraction v (Roche #9048-46-8), 100 mL ... | US Patent US11008336 (2021) BindingDB Entry DOI: 10.7270/Q2W380G1 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM498076 ((5'S)-N-{[5- (Ethylsulfonyl)pyridin- 2-yl]methyl}-...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 1.14E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Eli Lilly and Company US Patent | Assay Description Receptor competition binding assays are run in a buffer made up of DPBS (1 L) (Hyclone #SH30028.03), 2.2 g BSA Fraction v (Roche #9048-46-8), 100 mL ... | US Patent US11008336 (2021) BindingDB Entry DOI: 10.7270/Q2W380G1 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Nuclear receptor ROR-alpha (Homo sapiens (Human)) | BDBM498074 ((5′S)—N-[4-(Ethylsulfonyl)benzyl]-5′-m...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 3.11E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Eli Lilly and Company US Patent | Assay Description Receptor competition binding assays are run in a buffer made up of DPBS (1 L) (Hyclone #SH30028.03), 2.2 g BSA Fraction v (Roche #9048-46-8), 100 mL ... | US Patent US11008336 (2021) BindingDB Entry DOI: 10.7270/Q2W380G1 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Nuclear receptor ROR-alpha (Homo sapiens (Human)) | BDBM498080 (1-[(1S)-1-(4- Cyanophenyl)ethyl]- N-[4- (ethylsulf...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 3.27E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Eli Lilly and Company US Patent | Assay Description Receptor competition binding assays are run in a buffer made up of DPBS (1 L) (Hyclone #SH30028.03), 2.2 g BSA Fraction v (Roche #9048-46-8), 100 mL ... | US Patent US11008336 (2021) BindingDB Entry DOI: 10.7270/Q2W380G1 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Nuclear receptor ROR-alpha (Homo sapiens (Human)) | BDBM438835 (N-{[5-(Ethylsulfonyl)pyridin-2-yl]methyl}-1″...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 3.46E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Eli Lilly and Company US Patent | Assay Description His-tagged human RAR-related orphan receptor alpha (hRORa), human RAR-related orphan receptor beta (hRORb), and human RAR-related orphan receptor gam... | US Patent US10603320 (2020) BindingDB Entry DOI: 10.7270/Q2154M2H | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM498082 ((5'S)-N-{[5- (Ethylsulfonyl)pyridin- 2-yl]methyl}-...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 4.47E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Eli Lilly and Company US Patent | Assay Description Receptor competition binding assays are run in a buffer made up of DPBS (1 L) (Hyclone #SH30028.03), 2.2 g BSA Fraction v (Roche #9048-46-8), 100 mL ... | US Patent US11008336 (2021) BindingDB Entry DOI: 10.7270/Q2W380G1 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM498078 (N-{[5- (Ethylsulfonyl)pyridin- 2-yl]methyl}-5'- me...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 4.84E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Eli Lilly and Company US Patent | Assay Description Receptor competition binding assays are run in a buffer made up of DPBS (1 L) (Hyclone #SH30028.03), 2.2 g BSA Fraction v (Roche #9048-46-8), 100 mL ... | US Patent US11008336 (2021) BindingDB Entry DOI: 10.7270/Q2W380G1 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Nuclear receptor ROR-alpha (Homo sapiens (Human)) | BDBM438834 (N-{[5-(Ethylsulfonyl)pyridin-2-yl]methyl}-5′...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 5.68E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Eli Lilly and Company US Patent | Assay Description His-tagged human RAR-related orphan receptor alpha (hRORa), human RAR-related orphan receptor beta (hRORb), and human RAR-related orphan receptor gam... | US Patent US10603320 (2020) BindingDB Entry DOI: 10.7270/Q2154M2H | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Nuclear receptor ROR-alpha (Homo sapiens (Human)) | BDBM498082 ((5'S)-N-{[5- (Ethylsulfonyl)pyridin- 2-yl]methyl}-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 9.53E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Eli Lilly and Company US Patent | Assay Description Receptor competition binding assays are run in a buffer made up of DPBS (1 L) (Hyclone #SH30028.03), 2.2 g BSA Fraction v (Roche #9048-46-8), 100 mL ... | US Patent US11008336 (2021) BindingDB Entry DOI: 10.7270/Q2W380G1 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM498074 ((5′S)—N-[4-(Ethylsulfonyl)benzyl]-5′-m...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | >1.25E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Eli Lilly and Company US Patent | Assay Description Receptor competition binding assays are run in a buffer made up of DPBS (1 L) (Hyclone #SH30028.03), 2.2 g BSA Fraction v (Roche #9048-46-8), 100 mL ... | US Patent US11008336 (2021) BindingDB Entry DOI: 10.7270/Q2W380G1 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM498079 ((5'S)-N-{[5- (Ethylsulfonyl)pyridin- 2-yl]methyl}-...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | >1.25E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Eli Lilly and Company US Patent | Assay Description Receptor competition binding assays are run in a buffer made up of DPBS (1 L) (Hyclone #SH30028.03), 2.2 g BSA Fraction v (Roche #9048-46-8), 100 mL ... | US Patent US11008336 (2021) BindingDB Entry DOI: 10.7270/Q2W380G1 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| RAR related orphan receptor B isoform 1 (Human) | BDBM438836 (1'-[1-(4- Cyanophenyl)ethyl]- 5,5- spirocyclopropa...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | >1.25E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Eli Lilly and Company US Patent | Assay Description His-tagged human RAR-related orphan receptor alpha (hRORa), human RAR-related orphan receptor beta (hRORb), and human RAR-related orphan receptor gam... | US Patent US10603320 (2020) BindingDB Entry DOI: 10.7270/Q2154M2H | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| RAR related orphan receptor B isoform 1 (Human) | BDBM438835 (N-{[5-(Ethylsulfonyl)pyridin-2-yl]methyl}-1″...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | >1.25E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Eli Lilly and Company US Patent | Assay Description His-tagged human RAR-related orphan receptor alpha (hRORa), human RAR-related orphan receptor beta (hRORb), and human RAR-related orphan receptor gam... | US Patent US10603320 (2020) BindingDB Entry DOI: 10.7270/Q2154M2H | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM498077 (N-[4- (Ethylsulfonyl)benzyl]- 5'-methyl-1-{1-[6- (...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | >1.25E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Eli Lilly and Company US Patent | Assay Description Receptor competition binding assays are run in a buffer made up of DPBS (1 L) (Hyclone #SH30028.03), 2.2 g BSA Fraction v (Roche #9048-46-8), 100 mL ... | US Patent US11008336 (2021) BindingDB Entry DOI: 10.7270/Q2W380G1 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| RAR related orphan receptor B isoform 1 (Human) | BDBM438834 (N-{[5-(Ethylsulfonyl)pyridin-2-yl]methyl}-5′...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | >1.25E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Eli Lilly and Company US Patent | Assay Description His-tagged human RAR-related orphan receptor alpha (hRORa), human RAR-related orphan receptor beta (hRORb), and human RAR-related orphan receptor gam... | US Patent US10603320 (2020) BindingDB Entry DOI: 10.7270/Q2154M2H | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Nuclear receptor ROR-alpha (Homo sapiens (Human)) | BDBM498079 ((5'S)-N-{[5- (Ethylsulfonyl)pyridin- 2-yl]methyl}-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 1.93E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Eli Lilly and Company US Patent | Assay Description Receptor competition binding assays are run in a buffer made up of DPBS (1 L) (Hyclone #SH30028.03), 2.2 g BSA Fraction v (Roche #9048-46-8), 100 mL ... | US Patent US11008336 (2021) BindingDB Entry DOI: 10.7270/Q2W380G1 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Nuclear receptor ROR-alpha (Homo sapiens (Human)) | BDBM438836 (1'-[1-(4- Cyanophenyl)ethyl]- 5,5- spirocyclopropa...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | >2.04E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Eli Lilly and Company US Patent | Assay Description His-tagged human RAR-related orphan receptor alpha (hRORa), human RAR-related orphan receptor beta (hRORb), and human RAR-related orphan receptor gam... | US Patent US10603320 (2020) BindingDB Entry DOI: 10.7270/Q2154M2H | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Nuclear receptor ROR-alpha (Homo sapiens (Human)) | BDBM498078 (N-{[5- (Ethylsulfonyl)pyridin- 2-yl]methyl}-5'- me...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | >2.04E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Eli Lilly and Company US Patent | Assay Description Receptor competition binding assays are run in a buffer made up of DPBS (1 L) (Hyclone #SH30028.03), 2.2 g BSA Fraction v (Roche #9048-46-8), 100 mL ... | US Patent US11008336 (2021) BindingDB Entry DOI: 10.7270/Q2W380G1 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Nuclear receptor ROR-alpha (Homo sapiens (Human)) | BDBM498077 (N-[4- (Ethylsulfonyl)benzyl]- 5'-methyl-1-{1-[6- (...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | >2.04E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Eli Lilly and Company US Patent | Assay Description Receptor competition binding assays are run in a buffer made up of DPBS (1 L) (Hyclone #SH30028.03), 2.2 g BSA Fraction v (Roche #9048-46-8), 100 mL ... | US Patent US11008336 (2021) BindingDB Entry DOI: 10.7270/Q2W380G1 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM498080 (1-[(1S)-1-(4- Cyanophenyl)ethyl]- N-[4- (ethylsulf...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | >2.27E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Eli Lilly and Company US Patent | Assay Description Receptor competition binding assays are run in a buffer made up of DPBS (1 L) (Hyclone #SH30028.03), 2.2 g BSA Fraction v (Roche #9048-46-8), 100 mL ... | US Patent US11008336 (2021) BindingDB Entry DOI: 10.7270/Q2W380G1 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Cyclic GMP-AMP synthase (Homo sapiens) | BDBM639724 (3-[[6,7-Dichloro-3-(1H-pyrazol-4-yl)-1H-indol-4-yl...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | n/a | n/a | 3.22 | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Cyclic GMP-AMP synthase (Homo sapiens) | BDBM639875 ((S)—N-(5,6-Dichloro-8-(cyanomethoxy)-9-(1H-py...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | n/a | n/a | 3.38 | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Cyclic GMP-AMP synthase (Homo sapiens) | BDBM639703 (N-[6, 7-Dichloro-3-(1H-pyrazol-4-yl)-1H-indol-4-yl...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | n/a | n/a | 3.56 | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Cyclic GMP-AMP synthase (Homo sapiens) | BDBM639763 ((S)—N-(5,6-Dichloro-8-(cyanomethoxy)-9-(1H-py...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | n/a | n/a | 3.76 | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Cyclic GMP-AMP synthase (Homo sapiens) | BDBM639676 (3-[[6,7-Dichloro-3-(1H-pyrazol-4-yl)-1H-indol-4-yl...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | n/a | n/a | 4.33 | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Cyclic GMP-AMP synthase (Homo sapiens) | BDBM639869 (3-((6,7-Dichloro-2-(hydroxymethyl)-3-(1H-pyrazol-4...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | n/a | n/a | 4.74 | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Cyclic GMP-AMP synthase (Homo sapiens) | BDBM639655 (6,7-Dichloro-N-(2-fluoroethyl)-3-(1H-pyrazol-4-yl)...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | n/a | n/a | 4.91 | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Cyclic GMP-AMP synthase (Homo sapiens) | BDBM639685 (N-((6,7-Dichloro-4-(cyanomethoxy)-3-(1H-pyrazol-4-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | n/a | n/a | 5.11 | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Cyclic GMP-AMP synthase (Homo sapiens) | BDBM639781 (3-[[6,7-Dichloro-3-(1H-pyrazol-4-yl)-1H-indazol-4-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | n/a | n/a | 5.20 | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Cyclic GMP-AMP synthase (Homo sapiens) | BDBM639702 (N-(6,7-Dichloro-3-(1H-pyrazol-4-yl)-1H-indol-4-yl)...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | n/a | n/a | 5.67 | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Cyclic GMP-AMP synthase (Homo sapiens) | BDBM639874 ((S)—N-(5,6-Dichloro-8-ethoxy-9-(1H-pyrazol-4-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | n/a | n/a | 6.14 | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Cyclic GMP-AMP synthase (Homo sapiens) | BDBM639734 (2-((6,7-Dichloro-2-(5-methyl-1,3,4-thiadiazol-2-yl...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | n/a | n/a | 6.77 | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Cyclic GMP-AMP synthase (Homo sapiens) | BDBM639879 (3,4-Dichloro-1-(3-hydroxypropoxy)-10-(1H-pyrazol-4...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | n/a | n/a | 6.95 | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Cyclic GMP-AMP synthase (Homo sapiens) | BDBM639810 (2-((6,7-Dichloro-2-(2-methoxyacetyl)-10-(1H-pyrazo...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | n/a | n/a | 7.20 | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Cyclic GMP-AMP synthase (Homo sapiens) | BDBM639768 (N-(5,6-Dichloro-9-(1H-pyrazol-4-yl)-2,3-dihydro-1H...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | n/a | n/a | 7.69 | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Cyclic GMP-AMP synthase (Homo sapiens) | BDBM639870 (6,7-Dichloro-9-(3-hydroxypropoxy)-2-methyl-10-(1H-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | n/a | n/a | 7.89 | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Cyclic GMP-AMP synthase (Homo sapiens) | BDBM639811 (US20230391786, Example 280) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | n/a | n/a | 8.70 | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Cyclic GMP-AMP synthase (Homo sapiens) | BDBM639812 (US20230391786, Example 281) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | n/a | n/a | 8.90 | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Cyclic GMP-AMP synthase (Homo sapiens) | BDBM639728 (22-[6, 7-Dichloro-1-[1-(2-hydroxy ethyl)triazol-4-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | n/a | n/a | 8.93 | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
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