Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
DNA-(apurinic or apyrimidinic site) endonuclease (Homo sapiens (Human)) | BDBM203861 ((5-(acetylamino)-2-[2-(4-isothiocyanato-3-sulfophe...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 250 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Universidade de Lisboa | Assay Description In this assay, the complementary single-stranded oligonucleotides at 100 μm were mixed at a 1:1 ratio and annealed in assay buffer (50 mm Tris pH ... | Chem Biol Drug Des 88: 915-925 (2016) Article DOI: 10.1111/cbdd.12826 BindingDB Entry DOI: 10.7270/Q2Q52NGR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA-(apurinic or apyrimidinic site) endonuclease (Homo sapiens (Human)) | BDBM203862 (6-amino-4-hydroxy-5-[(4-nitro-2-sulfophenyl)azo]-2...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.76E+3 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Universidade de Lisboa | Assay Description In this assay, the complementary single-stranded oligonucleotides at 100 μm were mixed at a 1:1 ratio and annealed in assay buffer (50 mm Tris pH ... | Chem Biol Drug Des 88: 915-925 (2016) Article DOI: 10.1111/cbdd.12826 BindingDB Entry DOI: 10.7270/Q2Q52NGR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA-(apurinic or apyrimidinic site) endonuclease (Homo sapiens (Human)) | BDBM203863 (6-amino-5-[(4-amino-2-sulfophenyl)azo]-4-hydroxy-2...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 8.85E+3 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Universidade de Lisboa | Assay Description In this assay, the complementary single-stranded oligonucleotides at 100 μm were mixed at a 1:1 ratio and annealed in assay buffer (50 mm Tris pH ... | Chem Biol Drug Des 88: 915-925 (2016) Article DOI: 10.1111/cbdd.12826 BindingDB Entry DOI: 10.7270/Q2Q52NGR | |||||||||||
More data for this Ligand-Target Pair |