Found 104 hits with Last Name = 'takada' and Initial = 'h' Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Chemerin-like receptor 1
(Homo sapiens (Human)) | BDBM50560538
(CHEMBL4746987)Show SMILES CCCCN([C@H](C)c1ccc(cc1)-c1cc(Cl)ccc1-c1nc(=O)o[nH]1)c1nc2c(cccc2o1)C(O)=O |r| | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet 
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 1.20 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of chemR23 in human CAL1 cells assessed as inhibition of chemerin-induced intracellular calcium ion concentration preincubated for 45 mins... |
Citation and Details
Article DOI: 10.1016/j.bmc.2020.115622
BindingDB Entry DOI: 10.7270/Q2NG4VC4 |
More data for this
Ligand-Target Pair | |
Chemerin-like receptor 1
(Homo sapiens (Human)) | BDBM50560541
(CHEMBL4757632)Show SMILES C[C@@H](N(CC1CC1)c1nc2c(cccc2o1)C(O)=O)c1ccc(cc1)-c1cc(Cl)ccc1-c1nc(=O)o[nH]1 |r| | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 1.30 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of chemR23 in human CAL1 cells assessed as inhibition of chemerin-induced intracellular calcium ion concentration preincubated for 45 mins... |
Citation and Details
Article DOI: 10.1016/j.bmc.2020.115622
BindingDB Entry DOI: 10.7270/Q2NG4VC4 |
More data for this
Ligand-Target Pair | |
Chemerin-like receptor 1
(Homo sapiens (Human)) | BDBM50560540
(CHEMBL4793378)Show SMILES C[C@@H](N(CC1CC1)c1nc2c(cccc2o1)C(O)=O)c1ccc(cc1)-c1cc(F)ccc1-c1nc(=O)o[nH]1 |r| | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 2.30 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of chemR23 in human CAL1 cells assessed as inhibition of chemerin-induced intracellular calcium ion concentration preincubated for 45 mins... |
Citation and Details
Article DOI: 10.1016/j.bmc.2020.115622
BindingDB Entry DOI: 10.7270/Q2NG4VC4 |
More data for this
Ligand-Target Pair | |
Chemerin-like receptor 1
(Homo sapiens (Human)) | BDBM50560537
(CHEMBL4794289)Show SMILES CCCCN([C@H](C)c1ccc(cc1)-c1cc(F)ccc1-c1nc(=O)o[nH]1)c1nc2c(cccc2o1)C(O)=O |r| | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 2.70 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of chemR23 in human CAL1 cells assessed as inhibition of chemerin-induced intracellular calcium ion concentration preincubated for 45 mins... |
Citation and Details
Article DOI: 10.1016/j.bmc.2020.115622
BindingDB Entry DOI: 10.7270/Q2NG4VC4 |
More data for this
Ligand-Target Pair | |
Chemerin-like receptor 1
(Homo sapiens (Human)) | BDBM50560539
(CHEMBL4783675)Show SMILES C[C@@H](N(CC1CC1)c1nc2c(cccc2o1)C(O)=O)c1ccc(cc1)-c1cc(C)ccc1-c1nc(=O)o[nH]1 |r| | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| Purchase
MCE
PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 3.20 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of chemR23 in human CAL1 cells assessed as inhibition of chemerin-induced intracellular calcium ion concentration preincubated for 45 mins... |
Citation and Details
Article DOI: 10.1016/j.bmc.2020.115622
BindingDB Entry DOI: 10.7270/Q2NG4VC4 |
More data for this
Ligand-Target Pair | |
Chemerin-like receptor 1
(Homo sapiens (Human)) | BDBM50603313
(CHEMBL5177967)Show SMILES CCNC(=O)c1ccc(Cl)cc1-c1ccc(cc1)[C@@H](C)N(CC1CC1)c1nc(C(=O)NS(=O)(=O)C2CC2)c(s1)C1CC1 |r| | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 4.80 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
Article DOI: 10.1016/j.bmc.2021.116587
BindingDB Entry DOI: 10.7270/Q28W3JCR |
More data for this
Ligand-Target Pair | |
Chemerin-like receptor 1
(Homo sapiens (Human)) | BDBM50603317
(CHEMBL5204898)Show SMILES CCNC(=O)CCC(=O)N1Cc2ccccc2-c2nnn(CCOCCOCCOCCOCCOCCOCCNC(=O)c3ccc(Cl)cc3-c3ccc(cc3)[C@@H](C)N(CC3CC3)c3nc(C(=O)NS(=O)(=O)C4CC4)c(s3)C3CC3)c2-c2ccccc12 |r| | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 9.10 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
Article DOI: 10.1016/j.bmc.2021.116587
BindingDB Entry DOI: 10.7270/Q28W3JCR |
More data for this
Ligand-Target Pair | |
Chemerin-like receptor 1
(Homo sapiens (Human)) | BDBM50560520
(CHEMBL4796012)Show SMILES CCCCN([C@H](C)c1ccc(cc1)-c1ccccc1-c1nnn[nH]1)c1nc2c(cccc2o1)-c1nccn1C |r| | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of chemR23 in human CAL1 cells assessed as inhibition of chemerin-induced intracellular calcium ion concentration preincubated for 45 mins... |
Citation and Details
Article DOI: 10.1016/j.bmc.2020.115622
BindingDB Entry DOI: 10.7270/Q2NG4VC4 |
More data for this
Ligand-Target Pair | |
Chemerin-like receptor 1
(Homo sapiens (Human)) | BDBM50560542
(CHEMBL4754349)Show SMILES C[C@@H](N(CC1CC1)c1nc2c(cccc2o1)C(O)=O)c1ccc(cc1)-c1ccccc1-c1nc(=O)o[nH]1 |r| | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of chemR23 in human CAL1 cells assessed as inhibition of chemerin-induced intracellular calcium ion concentration preincubated for 45 mins... |
Citation and Details
Article DOI: 10.1016/j.bmc.2020.115622
BindingDB Entry DOI: 10.7270/Q2NG4VC4 |
More data for this
Ligand-Target Pair | |
Chemerin-like receptor 1
(Homo sapiens (Human)) | BDBM50603315
(CHEMBL5202580)Show SMILES C[C@@H](N(CC1CC1)c1nc(C(=O)NS(=O)(=O)C2CC2)c(s1)C1CC1)c1ccc(cc1)-c1cc(Cl)ccc1C(=O)NCCOCCOCCOCCOCCOCCOCCN=[N+]=[N-] |r| | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
Article DOI: 10.1016/j.bmc.2021.116587
BindingDB Entry DOI: 10.7270/Q28W3JCR |
More data for this
Ligand-Target Pair | |
Chemerin-like receptor 1
(Homo sapiens (Human)) | BDBM50560504
(CHEMBL4748968)Show SMILES CCCCN([C@H](C)c1ccc(cc1)-c1ccccc1-c1nnn[nH]1)c1nc2c(cccc2o1)C(=O)N(C)C |r| | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 13 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of chemR23 in human CAL1 cells assessed as inhibition of chemerin-induced intracellular calcium ion concentration preincubated for 45 mins... |
Citation and Details
Article DOI: 10.1016/j.bmc.2020.115622
BindingDB Entry DOI: 10.7270/Q2NG4VC4 |
More data for this
Ligand-Target Pair | |
Chemerin-like receptor 1
(Homo sapiens (Human)) | BDBM50560515
(CHEMBL4745883)Show SMILES CCCCN([C@H](C)c1ccc(cc1)-c1ccccc1-c1nnn[nH]1)c1nc2c(NS(C)(=O)=O)cccc2o1 |r| | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 14 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of chemR23 in human CAL1 cells assessed as inhibition of chemerin-induced intracellular calcium ion concentration preincubated for 45 mins... |
Citation and Details
Article DOI: 10.1016/j.bmc.2020.115622
BindingDB Entry DOI: 10.7270/Q2NG4VC4 |
More data for this
Ligand-Target Pair | |
Chemerin-like receptor 1
(Homo sapiens (Human)) | BDBM50603318
(CHEMBL5183004)Show SMILES [H][C@]12CS[C@@H](CCCCC(=O)NCCOCCOCCOCCOCCC(=O)NCCC(=O)N3Cc4ccccc4-c4nnn(CCOCCOCCOCCOCCOCCOCCNC(=O)c5ccc(Cl)cc5-c5ccc(cc5)[C@@H](C)N(CC5CC5)c5nc(C(=O)NS(=O)(=O)C6CC6)c(s5)C5CC5)c4-c4ccccc34)[C@@]1([H])NC(=O)N2 |r| | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 14 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
Article DOI: 10.1016/j.bmc.2021.116587
BindingDB Entry DOI: 10.7270/Q28W3JCR |
More data for this
Ligand-Target Pair | |
Sodium-dependent phosphate transport protein 2B
(Homo sapiens (Human)) | BDBM50590513
(CHEMBL5170356)Show SMILES CN(CCOCCOCCOCCC(O)=O)Cc1cccc(c1)C(=O)Nc1sc2CC(C)(C)CCc2c1C(=O)Nc1ccc(CCc2ccc(cc2)-c2nnc(C)o2)cc1 | UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 14 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
Article DOI: 10.1016/j.bmc.2022.116944
BindingDB Entry DOI: 10.7270/Q2MW2N4K |
More data for this
Ligand-Target Pair | |
Chemerin-like receptor 1
(Homo sapiens (Human)) | BDBM50560508
(CHEMBL4763169)Show SMILES CCCCN([C@H](C)c1ccc(cc1)-c1ccccc1-c1nnn[nH]1)c1nc2c(cccc2o1)C(=O)NS(C)(=O)=O |r| | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 14 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of chemR23 in human CAL1 cells assessed as inhibition of chemerin-induced intracellular calcium ion concentration preincubated for 45 mins... |
Citation and Details
Article DOI: 10.1016/j.bmc.2020.115622
BindingDB Entry DOI: 10.7270/Q2NG4VC4 |
More data for this
Ligand-Target Pair | |
Sodium-dependent phosphate transport protein 2B
(Homo sapiens (Human)) | BDBM50590497
(CHEMBL5182987)Show SMILES CCC(CC)N(CCN(C)C(=O)CCC(=O)NCCOCCOCCOCCO)Cc1cccc(c1)C(=O)Nc1sc2CC(C)(C)CCc2c1C(=O)c1cnn(c1)-c1ccc(Cl)c(c1)C(F)(F)F | UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
Article DOI: 10.1016/j.bmc.2022.116944
BindingDB Entry DOI: 10.7270/Q2MW2N4K |
More data for this
Ligand-Target Pair | |
Chemerin-like receptor 1
(Homo sapiens (Human)) | BDBM50560507
(CHEMBL4792296)Show SMILES CCCCN([C@H](C)c1ccc(cc1)-c1ccccc1-c1nnn[nH]1)c1nc2c(cccc2o1)C(O)=O |r| | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| Purchase
MCE
PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 17 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of chemR23 in human CAL1 cells assessed as inhibition of chemerin-induced intracellular calcium ion concentration preincubated for 45 mins... |
Citation and Details
Article DOI: 10.1016/j.bmc.2020.115622
BindingDB Entry DOI: 10.7270/Q2NG4VC4 |
More data for this
Ligand-Target Pair | |
Chemerin-like receptor 1
(Homo sapiens (Human)) | BDBM50560513
(CHEMBL4747813)Show SMILES CCCCN([C@H](C)c1ccc(cc1)-c1ccccc1-c1nnn[nH]1)c1nc2c(NC(C)=O)cccc2o1 |r| | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 22 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of chemR23 in human CAL1 cells assessed as inhibition of chemerin-induced intracellular calcium ion concentration preincubated for 45 mins... |
Citation and Details
Article DOI: 10.1016/j.bmc.2020.115622
BindingDB Entry DOI: 10.7270/Q2NG4VC4 |
More data for this
Ligand-Target Pair | |
Chemerin-like receptor 1
(Homo sapiens (Human)) | BDBM50560509
(CHEMBL4752027)Show SMILES CCCCN([C@H](C)c1ccc(cc1)-c1ccccc1-c1nnn[nH]1)c1nc2c(CO)cccc2o1 |r| | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 24 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of chemR23 in human CAL1 cells assessed as inhibition of chemerin-induced intracellular calcium ion concentration preincubated for 45 mins... |
Citation and Details
Article DOI: 10.1016/j.bmc.2020.115622
BindingDB Entry DOI: 10.7270/Q2NG4VC4 |
More data for this
Ligand-Target Pair | |
Sodium-dependent phosphate transport protein 2B
(Homo sapiens (Human)) | BDBM50590511
(CHEMBL5175794)Show SMILES Cc1nnc(o1)-c1ccc(CCc2ccc(NC(=O)c3c(NC(=O)c4cccc(CSCCOCCOCCOCCOCCOCCOCCOCCOCCC(O)=O)c4)sc4CC(C)(C)CCc34)cc2)cc1 | UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 24 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
Article DOI: 10.1016/j.bmc.2022.116944
BindingDB Entry DOI: 10.7270/Q2MW2N4K |
More data for this
Ligand-Target Pair | |
Chemerin-like receptor 1
(Homo sapiens (Human)) | BDBM50560506
(CHEMBL4791896)Show SMILES CCCCN([C@H](C)c1ccc(cc1)-c1ccccc1-c1nnn[nH]1)c1nc2c(cccc2o1)C(=O)N(C)CCO |r| | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 26 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of chemR23 in human CAL1 cells assessed as inhibition of chemerin-induced intracellular calcium ion concentration preincubated for 45 mins... |
Citation and Details
Article DOI: 10.1016/j.bmc.2020.115622
BindingDB Entry DOI: 10.7270/Q2NG4VC4 |
More data for this
Ligand-Target Pair | |
Chemerin-like receptor 1
(Homo sapiens (Human)) | BDBM50560512
(CHEMBL4764426)Show SMILES CCCCN([C@H](C)c1ccc(cc1)-c1ccccc1-c1nnn[nH]1)c1nc2c(N)cccc2o1 |r| | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 27 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of chemR23 in human CAL1 cells assessed as inhibition of chemerin-induced intracellular calcium ion concentration preincubated for 45 mins... |
Citation and Details
Article DOI: 10.1016/j.bmc.2020.115622
BindingDB Entry DOI: 10.7270/Q2NG4VC4 |
More data for this
Ligand-Target Pair | |
Prostacyclin receptor
(Homo sapiens (Human)) | BDBM23954
(5-[(2E,3aS,4R,5R,6aS)-5-hydroxy-4-[(1E,3S)-3-hydro...)Show SMILES [H][C@]12C[C@@H](O)[C@H](\C=C\[C@@H](O)C(C)CC#CC)[C@@]1([H])C\C(C2)=C\CCCC(O)=O Show InChI InChI=1S/C22H32O4/c1-3-4-7-15(2)20(23)11-10-18-19-13-16(8-5-6-9-22(25)26)12-17(19)14-21(18)24/h8,10-11,15,17-21,23-24H,5-7,9,12-14H2,1-2H3,(H,25,26)/b11-10+,16-8+/t15?,17-,18+,19-,20+,21+/m0/s1 | PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
AffyNet
| Purchase
CHEMBL
MCE
PC cid
PC sid
UniChem
Similars
| Article
| n/a | n/a | 27 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Displacement of [3H]-iloprost from Prostaglandin I2 receptor of human platelets |
Bioorg Med Chem Lett 5: 1071-1076 (1995)
Article DOI: 10.1016/0960-894X(95)00168-S
BindingDB Entry DOI: 10.7270/Q29P31MX |
More data for this
Ligand-Target Pair | |
Chemerin-like receptor 1
(Homo sapiens (Human)) | BDBM50560511
(CHEMBL4780439)Show SMILES CCCCN([C@H](C)c1ccc(cc1)-c1ccccc1-c1nnn[nH]1)c1nc2c(COC)cccc2o1 |r| | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 29 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of chemR23 in human CAL1 cells assessed as inhibition of chemerin-induced intracellular calcium ion concentration preincubated for 45 mins... |
Citation and Details
Article DOI: 10.1016/j.bmc.2020.115622
BindingDB Entry DOI: 10.7270/Q2NG4VC4 |
More data for this
Ligand-Target Pair | |
Chemerin-like receptor 1
(Homo sapiens (Human)) | BDBM50560514
(CHEMBL4754029)Show SMILES CCCCN([C@H](C)c1ccc(cc1)-c1ccccc1-c1nnn[nH]1)c1nc2c(NC(=O)N(C)C)cccc2o1 |r| | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 32 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of chemR23 in human CAL1 cells assessed as inhibition of chemerin-induced intracellular calcium ion concentration preincubated for 45 mins... |
Citation and Details
Article DOI: 10.1016/j.bmc.2020.115622
BindingDB Entry DOI: 10.7270/Q2NG4VC4 |
More data for this
Ligand-Target Pair | |
Sodium-dependent phosphate transport protein 2B
(Homo sapiens (Human)) | BDBM50603228
(CHEMBL5194399)Show SMILES CCN(CC)C[C@@H](O)COCCOCCOCCOc1cccc(c1)C(=O)Nc1sc2CC(C)(C)CCc2c1C(=O)N\N=C\c1ccc(Cl)c(c1)C(F)(F)F |r| | UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 33 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01474
BindingDB Entry DOI: 10.7270/Q2ST7TXQ |
More data for this
Ligand-Target Pair | |
Sodium-dependent phosphate transport protein 2B
(Homo sapiens (Human)) | BDBM50603226
(CHEMBL5189512)Show SMILES CCN(CC)CCOCCOCCOc1cccc(c1)C(=O)Nc1sc2CC(C)(C)CCc2c1C(=O)N\N=C\c1ccc(Cl)c(c1)C(F)(F)F | UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01474
BindingDB Entry DOI: 10.7270/Q2ST7TXQ |
More data for this
Ligand-Target Pair | |
Sodium-dependent phosphate transport protein 2B
(Homo sapiens (Human)) | BDBM50590509
(CHEMBL5188991)Show SMILES Cc1cc(NC(=O)c2c(NC(=O)c3cccc(OCCOCCOCCOCCOCCOCCOCC(O)=O)c3)sc3CC(C)(C)CCc23)ccc1CCc1ccc(cc1)-c1ncco1 | UniProtKB/SwissProt
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TBA
| |
Citation and Details
Article DOI: 10.1016/j.bmc.2022.116944
BindingDB Entry DOI: 10.7270/Q2MW2N4K |
More data for this
Ligand-Target Pair | |
Chemerin-like receptor 1
(Homo sapiens (Human)) | BDBM50603314
(CHEMBL5196772)Show SMILES CCCCCCNC(=O)c1ccc(Cl)cc1-c1ccc(cc1)[C@@H](C)N(CC1CC1)c1nc(C(=O)NS(=O)(=O)C2CC2)c(s1)C1CC1 |r| | PDB
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TBA
| |
Citation and Details
Article DOI: 10.1016/j.bmc.2021.116587
BindingDB Entry DOI: 10.7270/Q28W3JCR |
More data for this
Ligand-Target Pair | |
Chemerin-like receptor 1
(Homo sapiens (Human)) | BDBM50560532
(CHEMBL4786002)Show SMILES CCCCN([C@H](C)c1ccc(cc1)-c1cc(C)ccc1-c1nnn[nH]1)c1nc2ccccc2o1 |r| | PDB
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UniChem
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| n/a | n/a | 53 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of chemR23 in human CAL1 cells assessed as inhibition of chemerin-induced intracellular calcium ion concentration preincubated for 45 mins... |
Citation and Details
Article DOI: 10.1016/j.bmc.2020.115622
BindingDB Entry DOI: 10.7270/Q2NG4VC4 |
More data for this
Ligand-Target Pair | |
Chemerin-like receptor 1
(Homo sapiens (Human)) | BDBM50560524
(CHEMBL4752019)Show SMILES CCCCN([C@H](C)c1ccc(cc1)-c1ccc(F)cc1-c1nnn[nH]1)c1nc2ccccc2o1 |r| | PDB
UniProtKB/SwissProt
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UniChem
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| n/a | n/a | 57 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of chemR23 in human CAL1 cells assessed as inhibition of chemerin-induced intracellular calcium ion concentration preincubated for 45 mins... |
Citation and Details
Article DOI: 10.1016/j.bmc.2020.115622
BindingDB Entry DOI: 10.7270/Q2NG4VC4 |
More data for this
Ligand-Target Pair | |
Sodium-dependent phosphate transport protein 2B
(Homo sapiens (Human)) | BDBM50590512
(CHEMBL5173115)Show SMILES Cc1nnc(o1)-c1ccc(CCc2ccc(NC(=O)c3c(NC(=O)c4cccc(COCCOCCOCCOCC(O)=O)c4)sc4CC(C)(C)CCc34)cc2)cc1 | UniProtKB/SwissProt
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TBA
| |
Citation and Details
Article DOI: 10.1016/j.bmc.2022.116944
BindingDB Entry DOI: 10.7270/Q2MW2N4K |
More data for this
Ligand-Target Pair | |
Chemerin-like receptor 1
(Homo sapiens (Human)) | BDBM50560505
(CHEMBL4741497)Show SMILES CCCCN([C@H](C)c1ccc(cc1)-c1ccccc1-c1nnn[nH]1)c1nc2c(cccc2o1)C(=O)N(C)CC |r| | PDB
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UniChem
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| n/a | n/a | 62 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of chemR23 in human CAL1 cells assessed as inhibition of chemerin-induced intracellular calcium ion concentration preincubated for 45 mins... |
Citation and Details
Article DOI: 10.1016/j.bmc.2020.115622
BindingDB Entry DOI: 10.7270/Q2NG4VC4 |
More data for this
Ligand-Target Pair | |
Chemerin-like receptor 1
(Homo sapiens (Human)) | BDBM50560539
(CHEMBL4783675)Show SMILES C[C@@H](N(CC1CC1)c1nc2c(cccc2o1)C(O)=O)c1ccc(cc1)-c1cc(C)ccc1-c1nc(=O)o[nH]1 |r| | PDB
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| n/a | n/a | 63 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of chemR23 expressed in human CAL1 cells assessed as reduction in chemerin-induced chemotaxis incubated for 4 hrs by cell counting based C... |
Citation and Details
Article DOI: 10.1016/j.bmc.2020.115622
BindingDB Entry DOI: 10.7270/Q2NG4VC4 |
More data for this
Ligand-Target Pair | |
Sodium-dependent phosphate transport protein 2B
(Homo sapiens (Human)) | BDBM50590498
(CHEMBL5171732)Show SMILES COCCN(CCOCCOCCOCCOCCOCCOCc1cccc(c1)C(=O)Nc1sc2CC(C)(C)CCc2c1C(=O)N\N=C\c1ccc(Cl)c(c1)C(F)(F)F)CC(O)=O | UniProtKB/SwissProt
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TBA
| |
Citation and Details
Article DOI: 10.1016/j.bmc.2022.116944
BindingDB Entry DOI: 10.7270/Q2MW2N4K |
More data for this
Ligand-Target Pair | |
Sodium-dependent phosphate transport protein 2B
(Homo sapiens (Human)) | BDBM50590498
(CHEMBL5171732)Show SMILES COCCN(CCOCCOCCOCCOCCOCCOCc1cccc(c1)C(=O)Nc1sc2CC(C)(C)CCc2c1C(=O)N\N=C\c1ccc(Cl)c(c1)C(F)(F)F)CC(O)=O | UniProtKB/SwissProt
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TBA
| |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01474
BindingDB Entry DOI: 10.7270/Q2ST7TXQ |
More data for this
Ligand-Target Pair | |
Chemerin-like receptor 1
(Homo sapiens (Human)) | BDBM50560531
(CHEMBL4791613)Show SMILES CCCCN([C@H](C)c1ccc(cc1)-c1cc(Cl)ccc1-c1nnn[nH]1)c1nc2ccccc2o1 |r| | PDB
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UniChem
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| n/a | n/a | 65 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of chemR23 in human CAL1 cells assessed as inhibition of chemerin-induced intracellular calcium ion concentration preincubated for 45 mins... |
Citation and Details
Article DOI: 10.1016/j.bmc.2020.115622
BindingDB Entry DOI: 10.7270/Q2NG4VC4 |
More data for this
Ligand-Target Pair | |
Sodium-dependent phosphate transport protein 2B
(Homo sapiens (Human)) | BDBM50590507
(CHEMBL5206581)Show SMILES COC(=O)c1ccc(CCc2ccc(NC(=O)c3c(NC(=O)c4cccc(OCCOCCOCCOCCOCCOCCOCC(O)=O)c4)sc4CC(C)(C)CCc34)cc2C)cc1 | UniProtKB/SwissProt
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TBA
| |
Citation and Details
Article DOI: 10.1016/j.bmc.2022.116944
BindingDB Entry DOI: 10.7270/Q2MW2N4K |
More data for this
Ligand-Target Pair | |
Chemerin-like receptor 1
(Homo sapiens (Human)) | BDBM50560529
(CHEMBL4746011)Show SMILES CCCCN([C@H](C)c1ccc(cc1)-c1cc(F)ccc1-c1nnn[nH]1)c1nc2ccccc2o1 |r| | PDB
UniProtKB/SwissProt
antibodypedia
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| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 75 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of chemR23 in human CAL1 cells assessed as inhibition of chemerin-induced intracellular calcium ion concentration preincubated for 45 mins... |
Citation and Details
Article DOI: 10.1016/j.bmc.2020.115622
BindingDB Entry DOI: 10.7270/Q2NG4VC4 |
More data for this
Ligand-Target Pair | |
Sodium-dependent phosphate transport protein 2B
(Homo sapiens (Human)) | BDBM50603229
(CHEMBL5172873)Show SMILES CC1(C)CCc2c(C1)sc(NC(=O)c1cccc(OCCOCCOCCOC[C@H](O)CN(CCO)CCO)c1)c2C(=O)N\N=C\c1ccc(Cl)c(c1)C(F)(F)F |r| | UniProtKB/SwissProt
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TBA
| |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01474
BindingDB Entry DOI: 10.7270/Q2ST7TXQ |
More data for this
Ligand-Target Pair | |
Sodium-dependent phosphate transport protein 2B
(Homo sapiens (Human)) | BDBM50603218
(CHEMBL5209124)Show SMILES OC1CCN(Cc2cccc(c2)C(=O)Nc2sc3CCCCc3c2C(=O)N\N=C\c2ccc(Cl)c(c2)C(F)(F)F)CC1 | UniProtKB/SwissProt
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TBA
| |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01474
BindingDB Entry DOI: 10.7270/Q2ST7TXQ |
More data for this
Ligand-Target Pair | |
Chemerin-like receptor 1
(Homo sapiens (Human)) | BDBM50603316
(CHEMBL5190234)Show SMILES C[C@@H](N(CC1CC1)c1nc(C(=O)NS(=O)(=O)C2CC2)c(s1)C1CC1)c1ccc(cc1)-c1cc(Cl)ccc1C(=O)NCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCOCCOCCOCCOCCN=[N+]=[N-] |r| | PDB
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| n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
Article DOI: 10.1016/j.bmc.2021.116587
BindingDB Entry DOI: 10.7270/Q28W3JCR |
More data for this
Ligand-Target Pair | |
Sodium-dependent phosphate transport protein 2B
(Homo sapiens (Human)) | BDBM50590504
(CHEMBL5196753)Show SMILES COC(=O)c1ccc(CCc2ccc(NC(=O)c3c(NC(=O)c4cccc(OCCOCCOCCOCCOCCOCCO)c4)sc4CC(C)(C)CCc34)cc2)cc1 | UniProtKB/SwissProt
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| n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
Article DOI: 10.1016/j.bmc.2022.116944
BindingDB Entry DOI: 10.7270/Q2MW2N4K |
More data for this
Ligand-Target Pair | |
Sodium-dependent phosphate transport protein 2B
(Homo sapiens (Human)) | BDBM50590503
(CHEMBL5202364)Show SMILES CC1(C)CCc2c(C1)sc(NC(=O)c1cccc(COCCOCCOCCOCCOCCOCCO)c1)c2C(=O)Nc1ccc(Cc2ccccc2)cc1 | UniProtKB/SwissProt
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| n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
Article DOI: 10.1016/j.bmc.2022.116944
BindingDB Entry DOI: 10.7270/Q2MW2N4K |
More data for this
Ligand-Target Pair | |
Sodium-dependent phosphate transport protein 2B
(Homo sapiens (Human)) | BDBM50590502
(CHEMBL5206927)Show SMILES CCc1ccc(NC(=O)c2c(NC(=O)c3cccc(COCCOCCOCCOCCOCCOCCO)c3)sc3CC(C)(C)CCc23)cc1 | UniProtKB/SwissProt
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| n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
Article DOI: 10.1016/j.bmc.2022.116944
BindingDB Entry DOI: 10.7270/Q2MW2N4K |
More data for this
Ligand-Target Pair | |
Sodium-dependent phosphate transport protein 2B
(Homo sapiens (Human)) | BDBM50590506
(CHEMBL5187558)Show SMILES CC1(C)CCc2c(C1)sc(NC(=O)c1cccc(OCCOCCOCCOCCOCCOCCO)c1)c2C(=O)Nc1ccc(CCc2ccc(cc2)C(O)=O)cc1 | UniProtKB/SwissProt
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| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
Article DOI: 10.1016/j.bmc.2022.116944
BindingDB Entry DOI: 10.7270/Q2MW2N4K |
More data for this
Ligand-Target Pair | |
Chemerin-like receptor 1
(Homo sapiens (Human)) | BDBM50560522
(CHEMBL4791599)Show SMILES CCCCN([C@H](C)c1ccc(cc1)-c1cccc(F)c1-c1nnn[nH]1)c1nc2ccccc2o1 |r| | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of chemR23 in human CAL1 cells assessed as inhibition of chemerin-induced intracellular calcium ion concentration preincubated for 45 mins... |
Citation and Details
Article DOI: 10.1016/j.bmc.2020.115622
BindingDB Entry DOI: 10.7270/Q2NG4VC4 |
More data for this
Ligand-Target Pair | |
Sodium-dependent phosphate transport protein 2B
(Homo sapiens (Human)) | BDBM50603224
(CHEMBL5192802)Show SMILES CC1(C)CCc2c(C1)sc(NC(=O)c1cccc(OCCOCCOCCO)c1)c2C(=O)N\N=C\c1ccc(Cl)c(c1)C(F)(F)F | UniProtKB/SwissProt
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| PC cid
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| n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01474
BindingDB Entry DOI: 10.7270/Q2ST7TXQ |
More data for this
Ligand-Target Pair | |
Sodium-dependent phosphate transport protein 2B
(Homo sapiens (Human)) | BDBM50603225
(CHEMBL5174328)Show SMILES CC1(C)CCc2c(C1)sc(NC(=O)c1cccc(OCCOCCOCCOCCC(O)=O)c1)c2C(=O)N\N=C\c1ccc(Cl)c(c1)C(F)(F)F | UniProtKB/SwissProt
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| n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01474
BindingDB Entry DOI: 10.7270/Q2ST7TXQ |
More data for this
Ligand-Target Pair | |
Sodium-dependent phosphate transport protein 2B
(Homo sapiens (Human)) | BDBM50590505
(CHEMBL5193730)Show SMILES COC(=O)c1ccc(CCc2ccc(NC(=O)c3c(NC(=O)c4cccc(COCCOCCOCCOCCOCCOCCO)c4)sc4CC(C)(C)CCc34)cc2C)cc1 | UniProtKB/SwissProt
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| n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
Article DOI: 10.1016/j.bmc.2022.116944
BindingDB Entry DOI: 10.7270/Q2MW2N4K |
More data for this
Ligand-Target Pair | |
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