Found 86 hits with Last Name = 'araki' and Initial = 'l' Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
Histamine H3 receptor
(Homo sapiens (Human)) | BDBM50121205
(CHEBI:18295 | Histamine)Show InChI InChI=1S/C5H9N3/c6-2-1-5-3-7-4-8-5/h3-4H,1-2,6H2,(H,7,8) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| Purchase
MCE KEGG PC cid PC sid PDB UniChem
Patents
| Article PubMed
| 34 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University
Curated by ChEMBL
| Assay Description Histamine H3 receptor competition binding using [3H]Na-methylhistamine |
J Med Chem 46: 3162-5 (2003)
Article DOI: 10.1021/jm0300025 BindingDB Entry DOI: 10.7270/Q24B343F |
More data for this Ligand-Target Pair | |
Histamine H4 receptor
(Homo sapiens (Human)) | BDBM50170163
(CHEMBL321860)Show InChI InChI=1S/C11H16N6O/c1-13-11(16-6-12)15-4-8-2-3-10(18-8)9-5-14-7-17-9/h5,7-8,10H,2-4H2,1H3,(H,14,17)(H2,13,15,16)/t8-,10-/m1/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| 126 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University
Curated by ChEMBL
| Assay Description Histamine H4 receptor competition binding using [3H]Na-methylhistamine |
J Med Chem 46: 3162-5 (2003)
Article DOI: 10.1021/jm0300025 BindingDB Entry DOI: 10.7270/Q24B343F |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Homo sapiens (Human)) | BDBM50474242
(CHEMBL106931)Show InChI InChI=1S/C8H13N3O/c9-3-6-1-2-8(12-6)7-4-10-5-11-7/h4-6,8H,1-3,9H2,(H,10,11)/t6-,8-/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 219 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University
Curated by ChEMBL
| Assay Description Histamine H3 receptor competition binding using [3H]Na-methylhistamine |
J Med Chem 46: 3162-5 (2003)
Article DOI: 10.1021/jm0300025 BindingDB Entry DOI: 10.7270/Q24B343F |
More data for this Ligand-Target Pair | |
Histamine H4 receptor
(Homo sapiens (Human)) | BDBM50474249
(CHEMBL106158)Show SMILES C\N=C(\NC[C@@H]1CC[C@@H](O1)c1c[nH]cn1)NC#N Show InChI InChI=1S/C11H16N6O/c1-13-11(16-6-12)15-4-8-2-3-10(18-8)9-5-14-7-17-9/h5,7-8,10H,2-4H2,1H3,(H,14,17)(H2,13,15,16)/t8-,10+/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 224 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University
Curated by ChEMBL
| Assay Description Histamine H4 receptor competition binding using [3H]Na-methylhistamine |
J Med Chem 46: 3162-5 (2003)
Article DOI: 10.1021/jm0300025 BindingDB Entry DOI: 10.7270/Q24B343F |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Homo sapiens (Human)) | BDBM50474240
(Imifuramine)Show InChI InChI=1S/C8H13N3O/c9-3-6-1-2-8(12-6)7-4-10-5-11-7/h4-6,8H,1-3,9H2,(H,10,11)/t6-,8-/m1/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 229 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University
Curated by ChEMBL
| Assay Description Histamine H3 receptor competition binding using [3H]Na-methylhistamine |
J Med Chem 46: 3162-5 (2003)
Article DOI: 10.1021/jm0300025 BindingDB Entry DOI: 10.7270/Q24B343F |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Homo sapiens (Human)) | BDBM50474250
(CHEMBL105803)Show InChI InChI=1S/C15H18N2O2/c1-2-4-12(5-3-1)9-18-10-13-6-7-15(19-13)14-8-16-11-17-14/h1-5,8,11,13,15H,6-7,9-10H2,(H,16,17)/t13-,15-/m1/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 245 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University
Curated by ChEMBL
| Assay Description Histamine H3 receptor competition binding using [3H]Na-methylhistamine |
J Med Chem 46: 3162-5 (2003)
Article DOI: 10.1021/jm0300025 BindingDB Entry DOI: 10.7270/Q24B343F |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Homo sapiens (Human)) | BDBM50474252
(CHEMBL320331)Show InChI InChI=1S/C15H18N2O2/c1-2-4-12(5-3-1)9-18-10-13-6-7-15(19-13)14-8-16-11-17-14/h1-5,8,11,13,15H,6-7,9-10H2,(H,16,17)/t13-,15+/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 331 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University
Curated by ChEMBL
| Assay Description Histamine H3 receptor competition binding using [3H]Na-methylhistamine |
J Med Chem 46: 3162-5 (2003)
Article DOI: 10.1021/jm0300025 BindingDB Entry DOI: 10.7270/Q24B343F |
More data for this Ligand-Target Pair | |
Histamine H4 receptor
(Homo sapiens (Human)) | BDBM50474252
(CHEMBL320331)Show InChI InChI=1S/C15H18N2O2/c1-2-4-12(5-3-1)9-18-10-13-6-7-15(19-13)14-8-16-11-17-14/h1-5,8,11,13,15H,6-7,9-10H2,(H,16,17)/t13-,15+/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 437 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University
Curated by ChEMBL
| Assay Description Histamine H4 receptor competition binding using [3H]Na-methylhistamine |
J Med Chem 46: 3162-5 (2003)
Article DOI: 10.1021/jm0300025 BindingDB Entry DOI: 10.7270/Q24B343F |
More data for this Ligand-Target Pair | |
Histamine H4 receptor
(Homo sapiens (Human)) | BDBM50474240
(Imifuramine)Show InChI InChI=1S/C8H13N3O/c9-3-6-1-2-8(12-6)7-4-10-5-11-7/h4-6,8H,1-3,9H2,(H,10,11)/t6-,8-/m1/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 891 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University
Curated by ChEMBL
| Assay Description Histamine H4 receptor competition binding using [3H]Na-methylhistamine |
J Med Chem 46: 3162-5 (2003)
Article DOI: 10.1021/jm0300025 BindingDB Entry DOI: 10.7270/Q24B343F |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Homo sapiens (Human)) | BDBM50474247
(CHEMBL109130)Show InChI InChI=1S/C8H11N3O/c9-3-6-1-2-8(12-6)7-4-10-5-11-7/h1-2,4-6,8H,3,9H2,(H,10,11)/t6-,8-/m1/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 1.02E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University
Curated by ChEMBL
| Assay Description Histamine H3 receptor competition binding using [3H]Na-methylhistamine |
J Med Chem 46: 3162-5 (2003)
Article DOI: 10.1021/jm0300025 BindingDB Entry DOI: 10.7270/Q24B343F |
More data for this Ligand-Target Pair | |
Histamine H4 receptor
(Homo sapiens (Human)) | BDBM50474250
(CHEMBL105803)Show InChI InChI=1S/C15H18N2O2/c1-2-4-12(5-3-1)9-18-10-13-6-7-15(19-13)14-8-16-11-17-14/h1-5,8,11,13,15H,6-7,9-10H2,(H,16,17)/t13-,15-/m1/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 1.05E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University
Curated by ChEMBL
| Assay Description Histamine H4 receptor competition binding using [3H]Na-methylhistamine |
J Med Chem 46: 3162-5 (2003)
Article DOI: 10.1021/jm0300025 BindingDB Entry DOI: 10.7270/Q24B343F |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Homo sapiens (Human)) | BDBM50474244
(CHEMBL106913)Show InChI InChI=1S/C8H13N3O/c9-3-6-1-2-8(12-6)7-4-10-5-11-7/h4-6,8H,1-3,9H2,(H,10,11)/t6-,8+/m1/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 1.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University
Curated by ChEMBL
| Assay Description Histamine H3 receptor competition binding using [3H]Na-methylhistamine |
J Med Chem 46: 3162-5 (2003)
Article DOI: 10.1021/jm0300025 BindingDB Entry DOI: 10.7270/Q24B343F |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Homo sapiens (Human)) | BDBM50474248
(CHEMBL321920)Show InChI InChI=1S/C8H13N3O/c9-3-6-1-2-8(12-6)7-4-10-5-11-7/h4-6,8H,1-3,9H2,(H,10,11)/t6-,8+/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 2.04E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University
Curated by ChEMBL
| Assay Description Histamine H3 receptor competition binding using [3H]Na-methylhistamine |
J Med Chem 46: 3162-5 (2003)
Article DOI: 10.1021/jm0300025 BindingDB Entry DOI: 10.7270/Q24B343F |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Homo sapiens (Human)) | BDBM50170163
(CHEMBL321860)Show InChI InChI=1S/C11H16N6O/c1-13-11(16-6-12)15-4-8-2-3-10(18-8)9-5-14-7-17-9/h5,7-8,10H,2-4H2,1H3,(H,14,17)(H2,13,15,16)/t8-,10-/m1/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| 2.19E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University
Curated by ChEMBL
| Assay Description Histamine H3 receptor competition binding using [3H]Na-methylhistamine |
J Med Chem 46: 3162-5 (2003)
Article DOI: 10.1021/jm0300025 BindingDB Entry DOI: 10.7270/Q24B343F |
More data for this Ligand-Target Pair | |
Histamine H4 receptor
(Homo sapiens (Human)) | BDBM50474248
(CHEMBL321920)Show InChI InChI=1S/C8H13N3O/c9-3-6-1-2-8(12-6)7-4-10-5-11-7/h4-6,8H,1-3,9H2,(H,10,11)/t6-,8+/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 2.51E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University
Curated by ChEMBL
| Assay Description Histamine H4 receptor competition binding using [3H]Na-methylhistamine |
J Med Chem 46: 3162-5 (2003)
Article DOI: 10.1021/jm0300025 BindingDB Entry DOI: 10.7270/Q24B343F |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Homo sapiens (Human)) | BDBM50474246
(CHEMBL319658)Show InChI InChI=1S/C8H11N3O/c9-3-6-1-2-8(12-6)7-4-10-5-11-7/h1-2,4-6,8H,3,9H2,(H,10,11)/t6-,8-/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 2.51E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University
Curated by ChEMBL
| Assay Description Histamine H3 receptor competition binding using [3H]Na-methylhistamine |
J Med Chem 46: 3162-5 (2003)
Article DOI: 10.1021/jm0300025 BindingDB Entry DOI: 10.7270/Q24B343F |
More data for this Ligand-Target Pair | |
Histamine H4 receptor
(Homo sapiens (Human)) | BDBM50474244
(CHEMBL106913)Show InChI InChI=1S/C8H13N3O/c9-3-6-1-2-8(12-6)7-4-10-5-11-7/h4-6,8H,1-3,9H2,(H,10,11)/t6-,8+/m1/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 6.46E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University
Curated by ChEMBL
| Assay Description Histamine H4 receptor competition binding using [3H]Na-methylhistamine |
J Med Chem 46: 3162-5 (2003)
Article DOI: 10.1021/jm0300025 BindingDB Entry DOI: 10.7270/Q24B343F |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Homo sapiens (Human)) | BDBM50474253
(CHEMBL1632410)Show SMILES C(OCc1ccccc1)[C@H]1CC[C@H](O1)c1c[nH]cn1 |r| Show InChI InChI=1S/C15H18N2O2/c1-2-4-12(5-3-1)9-18-10-13-6-7-15(19-13)14-8-16-11-17-14/h1-5,8,11,13,15H,6-7,9-10H2,(H,16,17)/t13-,15+/m1/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 6.92E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University
Curated by ChEMBL
| Assay Description Histamine H3 receptor competition binding using [3H]Na-methylhistamine |
J Med Chem 46: 3162-5 (2003)
Article DOI: 10.1021/jm0300025 BindingDB Entry DOI: 10.7270/Q24B343F |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Homo sapiens (Human)) | BDBM50474249
(CHEMBL106158)Show SMILES C\N=C(\NC[C@@H]1CC[C@@H](O1)c1c[nH]cn1)NC#N Show InChI InChI=1S/C11H16N6O/c1-13-11(16-6-12)15-4-8-2-3-10(18-8)9-5-14-7-17-9/h5,7-8,10H,2-4H2,1H3,(H,14,17)(H2,13,15,16)/t8-,10+/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 7.08E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University
Curated by ChEMBL
| Assay Description Histamine H3 receptor competition binding using [3H]Na-methylhistamine |
J Med Chem 46: 3162-5 (2003)
Article DOI: 10.1021/jm0300025 BindingDB Entry DOI: 10.7270/Q24B343F |
More data for this Ligand-Target Pair | |
Histamine H4 receptor
(Homo sapiens (Human)) | BDBM50474251
(CHEMBL108649)Show InChI InChI=1S/C11H16N6O/c1-13-11(16-6-12)15-4-8-2-3-10(18-8)9-5-14-7-17-9/h5,7-8,10H,2-4H2,1H3,(H,14,17)(H2,13,15,16)/t8-,10+/m1/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 8.13E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University
Curated by ChEMBL
| Assay Description Histamine H4 receptor competition binding using [3H]Na-methylhistamine |
J Med Chem 46: 3162-5 (2003)
Article DOI: 10.1021/jm0300025 BindingDB Entry DOI: 10.7270/Q24B343F |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Homo sapiens (Human)) | BDBM50474251
(CHEMBL108649)Show InChI InChI=1S/C11H16N6O/c1-13-11(16-6-12)15-4-8-2-3-10(18-8)9-5-14-7-17-9/h5,7-8,10H,2-4H2,1H3,(H,14,17)(H2,13,15,16)/t8-,10+/m1/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 8.13E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University
Curated by ChEMBL
| Assay Description Histamine H3 receptor competition binding using [3H]Na-methylhistamine |
J Med Chem 46: 3162-5 (2003)
Article DOI: 10.1021/jm0300025 BindingDB Entry DOI: 10.7270/Q24B343F |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Homo sapiens (Human)) | BDBM50474241
(CHEMBL322256)Show InChI InChI=1S/C15H18N2O2/c1-2-4-12(5-3-1)9-18-10-13-6-7-15(19-13)14-8-16-11-17-14/h1-5,8,11,13,15H,6-7,9-10H2,(H,16,17)/t13-,15-/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 1.05E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University
Curated by ChEMBL
| Assay Description Compound was tested for H3 receptor competition binding using [3H]- Na-methylhistamine |
J Med Chem 46: 3162-5 (2003)
Article DOI: 10.1021/jm0300025 BindingDB Entry DOI: 10.7270/Q24B343F |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Homo sapiens (Human)) | BDBM50474245
(CHEMBL320279)Show InChI InChI=1S/C8H11N3O/c9-3-6-1-2-8(12-6)7-4-10-5-11-7/h1-2,4-6,8H,3,9H2,(H,10,11)/t6-,8+/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 1.15E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University
Curated by ChEMBL
| Assay Description Histamine H3 receptor competition binding using [3H]Na-methylhistamine |
J Med Chem 46: 3162-5 (2003)
Article DOI: 10.1021/jm0300025 BindingDB Entry DOI: 10.7270/Q24B343F |
More data for this Ligand-Target Pair | |
Histamine H4 receptor
(Homo sapiens (Human)) | BDBM50474247
(CHEMBL109130)Show InChI InChI=1S/C8H11N3O/c9-3-6-1-2-8(12-6)7-4-10-5-11-7/h1-2,4-6,8H,3,9H2,(H,10,11)/t6-,8-/m1/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 1.17E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University
Curated by ChEMBL
| Assay Description Histamine H4 receptor competition binding using [3H]Na-methylhistamine |
J Med Chem 46: 3162-5 (2003)
Article DOI: 10.1021/jm0300025 BindingDB Entry DOI: 10.7270/Q24B343F |
More data for this Ligand-Target Pair | |
Histamine H4 receptor
(Homo sapiens (Human)) | BDBM50474239
(CHEMBL107877)Show InChI InChI=1S/C8H11N3O/c9-3-6-1-2-8(12-6)7-4-10-5-11-7/h1-2,4-6,8H,3,9H2,(H,10,11)/t6-,8+/m1/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 1.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University
Curated by ChEMBL
| Assay Description Histamine H4 receptor competition binding using [3H]Na-methylhistamine |
J Med Chem 46: 3162-5 (2003)
Article DOI: 10.1021/jm0300025 BindingDB Entry DOI: 10.7270/Q24B343F |
More data for this Ligand-Target Pair | |
Histamine H4 receptor
(Homo sapiens (Human)) | BDBM50474242
(CHEMBL106931)Show InChI InChI=1S/C8H13N3O/c9-3-6-1-2-8(12-6)7-4-10-5-11-7/h4-6,8H,1-3,9H2,(H,10,11)/t6-,8-/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 1.29E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University
Curated by ChEMBL
| Assay Description Histamine H4 receptor competition binding using [3H]Na-methylhistamine |
J Med Chem 46: 3162-5 (2003)
Article DOI: 10.1021/jm0300025 BindingDB Entry DOI: 10.7270/Q24B343F |
More data for this Ligand-Target Pair | |
Histamine H4 receptor
(Homo sapiens (Human)) | BDBM50474253
(CHEMBL1632410)Show SMILES C(OCc1ccccc1)[C@H]1CC[C@H](O1)c1c[nH]cn1 |r| Show InChI InChI=1S/C15H18N2O2/c1-2-4-12(5-3-1)9-18-10-13-6-7-15(19-13)14-8-16-11-17-14/h1-5,8,11,13,15H,6-7,9-10H2,(H,16,17)/t13-,15+/m1/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 1.35E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University
Curated by ChEMBL
| Assay Description Histamine H4 receptor competition binding using [3H]Na-methylhistamine |
J Med Chem 46: 3162-5 (2003)
Article DOI: 10.1021/jm0300025 BindingDB Entry DOI: 10.7270/Q24B343F |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Homo sapiens (Human)) | BDBM50474243
(CHEMBL106570)Show InChI InChI=1S/C11H16N6O/c1-13-11(16-6-12)15-4-8-2-3-10(18-8)9-5-14-7-17-9/h5,7-8,10H,2-4H2,1H3,(H,14,17)(H2,13,15,16)/t8-,10-/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 1.86E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University
Curated by ChEMBL
| Assay Description Histamine H3 receptor competition binding using [3H]Na-methylhistamine |
J Med Chem 46: 3162-5 (2003)
Article DOI: 10.1021/jm0300025 BindingDB Entry DOI: 10.7270/Q24B343F |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Homo sapiens (Human)) | BDBM50474239
(CHEMBL107877)Show InChI InChI=1S/C8H11N3O/c9-3-6-1-2-8(12-6)7-4-10-5-11-7/h1-2,4-6,8H,3,9H2,(H,10,11)/t6-,8+/m1/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University
Curated by ChEMBL
| Assay Description Compound was tested for H3 receptor competition binding using [3H]- Na-methylhistamine |
J Med Chem 46: 3162-5 (2003)
Article DOI: 10.1021/jm0300025 BindingDB Entry DOI: 10.7270/Q24B343F |
More data for this Ligand-Target Pair | |
Histamine H4 receptor
(Homo sapiens (Human)) | BDBM50474243
(CHEMBL106570)Show InChI InChI=1S/C11H16N6O/c1-13-11(16-6-12)15-4-8-2-3-10(18-8)9-5-14-7-17-9/h5,7-8,10H,2-4H2,1H3,(H,14,17)(H2,13,15,16)/t8-,10-/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 2.04E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University
Curated by ChEMBL
| Assay Description Histamine H4 receptor competition binding using [3H]Na-methylhistamine |
J Med Chem 46: 3162-5 (2003)
Article DOI: 10.1021/jm0300025 BindingDB Entry DOI: 10.7270/Q24B343F |
More data for this Ligand-Target Pair | |
Histamine H4 receptor
(Homo sapiens (Human)) | BDBM50474241
(CHEMBL322256)Show InChI InChI=1S/C15H18N2O2/c1-2-4-12(5-3-1)9-18-10-13-6-7-15(19-13)14-8-16-11-17-14/h1-5,8,11,13,15H,6-7,9-10H2,(H,16,17)/t13-,15-/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 2.14E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University
Curated by ChEMBL
| Assay Description Histamine H4 receptor competition binding using [3H]Na-methylhistamine |
J Med Chem 46: 3162-5 (2003)
Article DOI: 10.1021/jm0300025 BindingDB Entry DOI: 10.7270/Q24B343F |
More data for this Ligand-Target Pair | |
Histamine H4 receptor
(Homo sapiens (Human)) | BDBM50474245
(CHEMBL320279)Show InChI InChI=1S/C8H11N3O/c9-3-6-1-2-8(12-6)7-4-10-5-11-7/h1-2,4-6,8H,3,9H2,(H,10,11)/t6-,8+/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 2.19E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University
Curated by ChEMBL
| Assay Description Histamine H4 receptor competition binding using [3H]Na-methylhistamine |
J Med Chem 46: 3162-5 (2003)
Article DOI: 10.1021/jm0300025 BindingDB Entry DOI: 10.7270/Q24B343F |
More data for this Ligand-Target Pair | |
Histamine H4 receptor
(Homo sapiens (Human)) | BDBM50474246
(CHEMBL319658)Show InChI InChI=1S/C8H11N3O/c9-3-6-1-2-8(12-6)7-4-10-5-11-7/h1-2,4-6,8H,3,9H2,(H,10,11)/t6-,8-/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| <1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University
Curated by ChEMBL
| Assay Description Histamine H4 receptor competition binding using [3H]Na-methylhistamine |
J Med Chem 46: 3162-5 (2003)
Article DOI: 10.1021/jm0300025 BindingDB Entry DOI: 10.7270/Q24B343F |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Homo sapiens (Human)) | BDBM50214615
(CHEBI:64177 | Clobenpropit)Show InChI InChI=1S/C14H17ClN4S/c15-12-5-3-11(4-6-12)8-18-14(16)20-7-1-2-13-9-17-10-19-13/h3-6,9-10H,1-2,7-8H2,(H2,16,18)(H,17,19) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| Purchase
KEGG PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 0.794 | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University of Pharmaceutical Sciences
Curated by ChEMBL
| Assay Description Antagonist activity at human histamine H3 receptor expressed in CHO cells assessed as inhibition of forskolin/R-alpha-methylhistamine-induced cAMP ac... |
Bioorg Med Chem Lett 23: 6415-20 (2013)
Article DOI: 10.1016/j.bmcl.2013.09.052 BindingDB Entry DOI: 10.7270/Q2R78J5R |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Homo sapiens (Human)) | BDBM50494136
(CHEMBL2441945)Show InChI InChI=1S/C20H30N4S/c21-17-19-10-8-18(9-11-19)7-2-3-12-23-20(22)25-16-6-15-24-13-4-1-5-14-24/h8-11H,1-7,12-16H2,(H2,22,23) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University of Pharmaceutical Sciences
Curated by ChEMBL
| Assay Description Antagonist activity at human histamine H3 receptor expressed in CHO cells assessed as inhibition of forskolin/R-alpha-methylhistamine-induced cAMP ac... |
Bioorg Med Chem Lett 23: 6415-20 (2013)
Article DOI: 10.1016/j.bmcl.2013.09.052 BindingDB Entry DOI: 10.7270/Q2R78J5R |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Homo sapiens (Human)) | BDBM50494138
(CHEMBL2441946)Show InChI InChI=1S/C18H36N4S/c19-18(23-17-9-16-22-13-6-2-7-14-22)20-10-3-8-15-21-11-4-1-5-12-21/h1-17H2,(H2,19,20) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 6.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University of Pharmaceutical Sciences
Curated by ChEMBL
| Assay Description Antagonist activity at human histamine H3 receptor expressed in CHO cells assessed as inhibition of forskolin/R-alpha-methylhistamine-induced cAMP ac... |
Bioorg Med Chem Lett 23: 6415-20 (2013)
Article DOI: 10.1016/j.bmcl.2013.09.052 BindingDB Entry DOI: 10.7270/Q2R78J5R |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Homo sapiens (Human)) | BDBM50494132
(CHEMBL2441941)Show InChI InChI=1S/C18H28ClN3S/c19-17-9-7-16(8-10-17)6-4-11-21-18(20)23-15-5-14-22-12-2-1-3-13-22/h7-10H,1-6,11-15H2,(H2,20,21) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 6.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University of Pharmaceutical Sciences
Curated by ChEMBL
| Assay Description Antagonist activity at human histamine H3 receptor expressed in CHO cells assessed as inhibition of forskolin/R-alpha-methylhistamine-induced cAMP ac... |
Bioorg Med Chem Lett 23: 6415-20 (2013)
Article DOI: 10.1016/j.bmcl.2013.09.052 BindingDB Entry DOI: 10.7270/Q2R78J5R |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Homo sapiens (Human)) | BDBM50494137
(CHEMBL2441942)Show InChI InChI=1S/C19H30ClN3S/c20-18-10-8-17(9-11-18)7-2-3-12-22-19(21)24-16-6-15-23-13-4-1-5-14-23/h8-11H,1-7,12-16H2,(H2,21,22) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 6.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University of Pharmaceutical Sciences
Curated by ChEMBL
| Assay Description Antagonist activity at human histamine H3 receptor expressed in CHO cells assessed as inhibition of forskolin/R-alpha-methylhistamine-induced cAMP ac... |
Bioorg Med Chem Lett 23: 6415-20 (2013)
Article DOI: 10.1016/j.bmcl.2013.09.052 BindingDB Entry DOI: 10.7270/Q2R78J5R |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Homo sapiens (Human)) | BDBM50494141
(CHEMBL2441940)Show InChI InChI=1S/C17H26ClN3S/c18-16-7-5-15(6-8-16)9-10-20-17(19)22-14-4-13-21-11-2-1-3-12-21/h5-8H,1-4,9-14H2,(H2,19,20) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 7.90 | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University of Pharmaceutical Sciences
Curated by ChEMBL
| Assay Description Antagonist activity at human histamine H3 receptor expressed in CHO cells assessed as inhibition of forskolin/R-alpha-methylhistamine-induced cAMP ac... |
Bioorg Med Chem Lett 23: 6415-20 (2013)
Article DOI: 10.1016/j.bmcl.2013.09.052 BindingDB Entry DOI: 10.7270/Q2R78J5R |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Homo sapiens (Human)) | BDBM50494127
(CHEMBL2441944)Show SMILES Cl.FC(F)(F)c1ccc(CCCCNC(=N)SCCCN2CCCCC2)cc1 Show InChI InChI=1S/C20H30F3N3S/c21-20(22,23)18-10-8-17(9-11-18)7-2-3-12-25-19(24)27-16-6-15-26-13-4-1-5-14-26/h8-11H,1-7,12-16H2,(H2,24,25) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 16 | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University of Pharmaceutical Sciences
Curated by ChEMBL
| Assay Description Antagonist activity at human histamine H3 receptor expressed in CHO cells assessed as inhibition of forskolin/R-alpha-methylhistamine-induced cAMP ac... |
Bioorg Med Chem Lett 23: 6415-20 (2013)
Article DOI: 10.1016/j.bmcl.2013.09.052 BindingDB Entry DOI: 10.7270/Q2R78J5R |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Homo sapiens (Human)) | BDBM50494135
(CHEMBL2441933)Show InChI InChI=1S/C15H22ClN3S/c16-14-6-4-13(5-7-14)12-18-15(17)20-11-3-10-19-8-1-2-9-19/h4-7H,1-3,8-12H2,(H2,17,18) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University of Pharmaceutical Sciences
Curated by ChEMBL
| Assay Description Antagonist activity at human histamine H3 receptor expressed in CHO cells assessed as inhibition of forskolin/R-alpha-methylhistamine-induced cAMP ac... |
Bioorg Med Chem Lett 23: 6415-20 (2013)
Article DOI: 10.1016/j.bmcl.2013.09.052 BindingDB Entry DOI: 10.7270/Q2R78J5R |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Homo sapiens (Human)) | BDBM50494131
(CHEMBL2441943)Show InChI InChI=1S/C20H33N3S/c21-20(24-18-10-17-23-15-8-3-9-16-23)22-14-7-2-6-13-19-11-4-1-5-12-19/h1,4-5,11-12H,2-3,6-10,13-18H2,(H2,21,22) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 32 | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University of Pharmaceutical Sciences
Curated by ChEMBL
| Assay Description Antagonist activity at human histamine H3 receptor expressed in CHO cells assessed as inhibition of forskolin/R-alpha-methylhistamine-induced cAMP ac... |
Bioorg Med Chem Lett 23: 6415-20 (2013)
Article DOI: 10.1016/j.bmcl.2013.09.052 BindingDB Entry DOI: 10.7270/Q2R78J5R |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Homo sapiens (Human)) | BDBM50494139
(CHEMBL2441938)Show InChI InChI=1S/C16H24ClN3S/c17-15-6-4-14(5-7-15)8-9-19-16(18)21-13-3-12-20-10-1-2-11-20/h4-7H,1-3,8-13H2,(H2,18,19) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 32 | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University of Pharmaceutical Sciences
Curated by ChEMBL
| Assay Description Antagonist activity at human histamine H3 receptor expressed in CHO cells assessed as inhibition of forskolin/R-alpha-methylhistamine-induced cAMP ac... |
Bioorg Med Chem Lett 23: 6415-20 (2013)
Article DOI: 10.1016/j.bmcl.2013.09.052 BindingDB Entry DOI: 10.7270/Q2R78J5R |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Homo sapiens (Human)) | BDBM50494142
(CHEMBL2441935)Show InChI InChI=1S/C16H24ClN3S/c17-15-7-5-14(6-8-15)13-19-16(18)21-12-4-11-20-9-2-1-3-10-20/h5-8H,1-4,9-13H2,(H2,18,19) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 79 | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University of Pharmaceutical Sciences
Curated by ChEMBL
| Assay Description Antagonist activity at human histamine H3 receptor expressed in CHO cells assessed as inhibition of forskolin/R-alpha-methylhistamine-induced cAMP ac... |
Bioorg Med Chem Lett 23: 6415-20 (2013)
Article DOI: 10.1016/j.bmcl.2013.09.052 BindingDB Entry DOI: 10.7270/Q2R78J5R |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Homo sapiens (Human)) | BDBM50494130
(CHEMBL2441947)Show InChI InChI=1S/C19H29ClN2O/c20-18-11-9-17(10-12-18)7-2-3-13-21-19(23)8-6-16-22-14-4-1-5-15-22/h9-12H,1-8,13-16H2,(H,21,23) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 126 | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University of Pharmaceutical Sciences
Curated by ChEMBL
| Assay Description Antagonist activity at human histamine H3 receptor expressed in CHO cells assessed as inhibition of forskolin/R-alpha-methylhistamine-induced cAMP ac... |
Bioorg Med Chem Lett 23: 6415-20 (2013)
Article DOI: 10.1016/j.bmcl.2013.09.052 BindingDB Entry DOI: 10.7270/Q2R78J5R |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Homo sapiens (Human)) | BDBM50494129
(CHEMBL2441948)Show InChI InChI=1S/C20H29F3N2O/c21-20(22,23)18-11-9-17(10-12-18)7-2-3-13-24-19(26)8-6-16-25-14-4-1-5-15-25/h9-12H,1-8,13-16H2,(H,24,26) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 126 | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University of Pharmaceutical Sciences
Curated by ChEMBL
| Assay Description Antagonist activity at human histamine H3 receptor expressed in CHO cells assessed as inhibition of forskolin/R-alpha-methylhistamine-induced cAMP ac... |
Bioorg Med Chem Lett 23: 6415-20 (2013)
Article DOI: 10.1016/j.bmcl.2013.09.052 BindingDB Entry DOI: 10.7270/Q2R78J5R |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Homo sapiens (Human)) | BDBM50494128
(CHEMBL2441939)Show InChI InChI=1S/C16H24ClN3OS/c17-15-4-2-14(3-5-15)6-7-19-16(18)22-13-1-8-20-9-11-21-12-10-20/h2-5H,1,6-13H2,(H2,18,19) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 316 | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University of Pharmaceutical Sciences
Curated by ChEMBL
| Assay Description Antagonist activity at human histamine H3 receptor expressed in CHO cells assessed as inhibition of forskolin/R-alpha-methylhistamine-induced cAMP ac... |
Bioorg Med Chem Lett 23: 6415-20 (2013)
Article DOI: 10.1016/j.bmcl.2013.09.052 BindingDB Entry DOI: 10.7270/Q2R78J5R |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Homo sapiens (Human)) | BDBM50494126
(CHEMBL2441949)Show InChI InChI=1S/C19H29ClN2O/c20-18-11-9-17(10-12-18)7-2-3-8-19(23)21-13-6-16-22-14-4-1-5-15-22/h9-12H,1-8,13-16H2,(H,21,23) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 316 | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University of Pharmaceutical Sciences
Curated by ChEMBL
| Assay Description Antagonist activity at human histamine H3 receptor expressed in CHO cells assessed as inhibition of forskolin/R-alpha-methylhistamine-induced cAMP ac... |
Bioorg Med Chem Lett 23: 6415-20 (2013)
Article DOI: 10.1016/j.bmcl.2013.09.052 BindingDB Entry DOI: 10.7270/Q2R78J5R |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Homo sapiens (Human)) | BDBM50494134
(CHEMBL2441936)Show InChI InChI=1S/C16H25ClN4S/c1-20-8-10-21(11-9-20)7-2-12-22-16(18)19-13-14-3-5-15(17)6-4-14/h3-6H,2,7-13H2,1H3,(H2,18,19) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 1.26E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University of Pharmaceutical Sciences
Curated by ChEMBL
| Assay Description Antagonist activity at human histamine H3 receptor expressed in CHO cells assessed as inhibition of forskolin/R-alpha-methylhistamine-induced cAMP ac... |
Bioorg Med Chem Lett 23: 6415-20 (2013)
Article DOI: 10.1016/j.bmcl.2013.09.052 BindingDB Entry DOI: 10.7270/Q2R78J5R |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Homo sapiens (Human)) | BDBM50494140
(CHEMBL2441934)Show InChI InChI=1S/C15H22ClN3OS/c16-14-4-2-13(3-5-14)12-18-15(17)21-11-1-6-19-7-9-20-10-8-19/h2-5H,1,6-12H2,(H2,17,18) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 1.59E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Osaka University of Pharmaceutical Sciences
Curated by ChEMBL
| Assay Description Antagonist activity at human histamine H3 receptor expressed in CHO cells assessed as inhibition of forskolin/R-alpha-methylhistamine-induced cAMP ac... |
Bioorg Med Chem Lett 23: 6415-20 (2013)
Article DOI: 10.1016/j.bmcl.2013.09.052 BindingDB Entry DOI: 10.7270/Q2R78J5R |
More data for this Ligand-Target Pair | |