Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
C-X-C chemokine receptor type 1 (Homo sapiens (Human)) | BDBM50150572![]() (1-(2-Bromo-phenyl)-3-(2,4-dihydroxy-phenyl)-urea |...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 22 | n/a | n/a | n/a | n/a | n/a | n/a |
Johnson and Johnson Pharmaceutical Research and Development Curated by ChEMBL | Assay Description Inhibitory concentration against interleukin-8 receptor of human neutrophils by using [125I]-IL-8 (0.125 nM) as radioligand | Bioorg Med Chem Lett 14: 4307-11 (2004) Article DOI: 10.1016/j.bmcl.2004.05.080 BindingDB Entry DOI: 10.7270/Q23F4P4M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 1 (Homo sapiens (Human)) | BDBM50150573![]() (1-{4-[5-(4-Chloro-phenyl)-isoxazol-3-yl]-phenoxyme...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Johnson and Johnson Pharmaceutical Research and Development Curated by ChEMBL | Assay Description Inhibitory concentration against interleukin-8 receptor of human neutrophils by using [125I]-IL-8 (0.125 nM) as radioligand | Bioorg Med Chem Lett 14: 4307-11 (2004) Article DOI: 10.1016/j.bmcl.2004.05.080 BindingDB Entry DOI: 10.7270/Q23F4P4M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 1 (Homo sapiens (Human)) | BDBM50150561![]() (1-(3-{4-[3-(4-Fluoro-phenyl)-isoxazol-5-yl]-phenox...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Johnson and Johnson Pharmaceutical Research and Development Curated by ChEMBL | Assay Description Inhibitory concentration against interleukin-8 receptor of human neutrophils by using [125I]-IL-8 (0.125 nM) as radioligand | Bioorg Med Chem Lett 14: 4307-11 (2004) Article DOI: 10.1016/j.bmcl.2004.05.080 BindingDB Entry DOI: 10.7270/Q23F4P4M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 1 (Homo sapiens (Human)) | BDBM50150558![]() (1-(3-{4-[3-(4-Chloro-phenyl)-isoxazol-5-yl]-phenox...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Johnson and Johnson Pharmaceutical Research and Development Curated by ChEMBL | Assay Description Inhibitory concentration against interleukin-8 receptor of human neutrophils by using [125I]-IL-8 (0.125 nM) as radioligand | Bioorg Med Chem Lett 14: 4307-11 (2004) Article DOI: 10.1016/j.bmcl.2004.05.080 BindingDB Entry DOI: 10.7270/Q23F4P4M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 1 (Homo sapiens (Human)) | BDBM50150555![]() (1-(3-{4-[3-(4-Chloro-phenyl)-[1,2,4]oxadiazol-5-yl...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Johnson and Johnson Pharmaceutical Research and Development Curated by ChEMBL | Assay Description Inhibitory concentration against interleukin-8 receptor of human neutrophils by using [125I]-IL-8 (0.125 nM) as radioligand | Bioorg Med Chem Lett 14: 4307-11 (2004) Article DOI: 10.1016/j.bmcl.2004.05.080 BindingDB Entry DOI: 10.7270/Q23F4P4M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 1 (Homo sapiens (Human)) | BDBM50150563![]() (CHEMBL183061 | {4-[5-(4-Chloro-phenyl)-isoxazol-3-...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Johnson and Johnson Pharmaceutical Research and Development Curated by ChEMBL | Assay Description Inhibitory concentration against interleukin-8 receptor of human neutrophils by using [125I]-IL-8 (0.125 nM) as radioligand | Bioorg Med Chem Lett 14: 4307-11 (2004) Article DOI: 10.1016/j.bmcl.2004.05.080 BindingDB Entry DOI: 10.7270/Q23F4P4M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sporulation kinase A (Bacillus subtilis (strain 168)) | BDBM50471725![]() (CHEMBL327734) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The R. W. Johnson Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of autophosphorylation of the two-component signal transduction system kinase was measured using the KinA/Spo0F regulatory system of Bacil... | J Med Chem 41: 2939-45 (1998) Article DOI: 10.1021/jm9803572 BindingDB Entry DOI: 10.7270/Q2VM4G0W | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 1 (Homo sapiens (Human)) | BDBM50150553![]() (1-Methyl-4-{3-[4-(3-phenyl-isoxazol-5-yl)-phenoxy]...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Johnson and Johnson Pharmaceutical Research and Development Curated by ChEMBL | Assay Description Inhibitory concentration against interleukin-8 receptor of human neutrophils by using [125I]-IL-8 (0.125 nM) as radioligand | Bioorg Med Chem Lett 14: 4307-11 (2004) Article DOI: 10.1016/j.bmcl.2004.05.080 BindingDB Entry DOI: 10.7270/Q23F4P4M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 1 (Homo sapiens (Human)) | BDBM50150559![]() (CHEMBL182361 | {4-[5-(4-Fluoro-phenyl)-isoxazol-3-...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Johnson and Johnson Pharmaceutical Research and Development Curated by ChEMBL | Assay Description Inhibitory concentration against interleukin-8 receptor of human neutrophils by using [125I]-IL-8 (0.125 nM) as radioligand | Bioorg Med Chem Lett 14: 4307-11 (2004) Article DOI: 10.1016/j.bmcl.2004.05.080 BindingDB Entry DOI: 10.7270/Q23F4P4M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 1 (Homo sapiens (Human)) | BDBM50150558![]() (1-(3-{4-[3-(4-Chloro-phenyl)-isoxazol-5-yl]-phenox...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Johnson and Johnson Pharmaceutical Research and Development Curated by ChEMBL | Assay Description Inhibition of interleukin-8 induced elastase release from human neutrophils | Bioorg Med Chem Lett 14: 4307-11 (2004) Article DOI: 10.1016/j.bmcl.2004.05.080 BindingDB Entry DOI: 10.7270/Q23F4P4M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sporulation kinase A (Bacillus subtilis (strain 168)) | BDBM50215968![]() (CHEMBL57324) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 3.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
R.W. Johnson Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of histidine protein kinase (KinA) phosphorylation in the presence of response regulator (Spo0F) | Bioorg Med Chem Lett 8: 1923-8 (1998) BindingDB Entry DOI: 10.7270/Q27S7QZM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sporulation kinase A (Bacillus subtilis (strain 168)) | BDBM50063753![]() (CHEMBL12131 | Closantel | N-(5-chloro-4-((4-chloro...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 3.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The R. W. Johnson Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of autophosphorylation of the two-component signal transduction system kinase was measured using the KinA/Spo0F regulatory system of Bacil... | J Med Chem 41: 2939-45 (1998) Article DOI: 10.1021/jm9803572 BindingDB Entry DOI: 10.7270/Q2VM4G0W | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 1 (Homo sapiens (Human)) | BDBM50150561![]() (1-(3-{4-[3-(4-Fluoro-phenyl)-isoxazol-5-yl]-phenox...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Johnson and Johnson Pharmaceutical Research and Development Curated by ChEMBL | Assay Description Inhibition of interleukin-8 induced elastase release from human neutrophils | Bioorg Med Chem Lett 14: 4307-11 (2004) Article DOI: 10.1016/j.bmcl.2004.05.080 BindingDB Entry DOI: 10.7270/Q23F4P4M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 1 (Homo sapiens (Human)) | BDBM50150569![]() ((3-{4-[3-(4-Chloro-phenyl)-isoxazol-5-yl]-phenoxy}...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Johnson and Johnson Pharmaceutical Research and Development Curated by ChEMBL | Assay Description Inhibitory concentration against interleukin-8 receptor of human neutrophils by using [125I]-IL-8 (0.125 nM) as radioligand | Bioorg Med Chem Lett 14: 4307-11 (2004) Article DOI: 10.1016/j.bmcl.2004.05.080 BindingDB Entry DOI: 10.7270/Q23F4P4M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 1 (Homo sapiens (Human)) | BDBM50150559![]() (CHEMBL182361 | {4-[5-(4-Fluoro-phenyl)-isoxazol-3-...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Johnson and Johnson Pharmaceutical Research and Development Curated by ChEMBL | Assay Description Inhibition of interleukin-8 induced elastase release from human neutrophils | Bioorg Med Chem Lett 14: 4307-11 (2004) Article DOI: 10.1016/j.bmcl.2004.05.080 BindingDB Entry DOI: 10.7270/Q23F4P4M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 1 (Homo sapiens (Human)) | BDBM50150574![]() (CHEMBL413959 | {2-[5-(4-Chloro-phenyl)-isoxazol-3-...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Johnson and Johnson Pharmaceutical Research and Development Curated by ChEMBL | Assay Description Inhibitory concentration against interleukin-8 receptor of human neutrophils by using [125I]-IL-8 (0.125 nM) as radioligand | Bioorg Med Chem Lett 14: 4307-11 (2004) Article DOI: 10.1016/j.bmcl.2004.05.080 BindingDB Entry DOI: 10.7270/Q23F4P4M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 1 (Homo sapiens (Human)) | BDBM50150555![]() (1-(3-{4-[3-(4-Chloro-phenyl)-[1,2,4]oxadiazol-5-yl...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Johnson and Johnson Pharmaceutical Research and Development Curated by ChEMBL | Assay Description Inhibition of interleukin-8 induced elastase release from human neutrophils | Bioorg Med Chem Lett 14: 4307-11 (2004) Article DOI: 10.1016/j.bmcl.2004.05.080 BindingDB Entry DOI: 10.7270/Q23F4P4M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sporulation kinase A (Bacillus subtilis (strain 168)) | BDBM50215967![]() (CHEMBL56579) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 4.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
R.W. Johnson Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of histidine protein kinase (KinA) phosphorylation in the presence of response regulator (Spo0F) | Bioorg Med Chem Lett 8: 1923-8 (1998) BindingDB Entry DOI: 10.7270/Q27S7QZM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sporulation kinase A (Bacillus subtilis (strain 168)) | BDBM50471718![]() (CHEMBL98026) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The R. W. Johnson Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of autophosphorylation of the two-component signal transduction system kinase was measured using the KinA/Spo0F regulatory system of Bacil... | J Med Chem 41: 2939-45 (1998) Article DOI: 10.1021/jm9803572 BindingDB Entry DOI: 10.7270/Q2VM4G0W | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 1 (Homo sapiens (Human)) | BDBM50150567![]() (1-[4-(5-Phenyl-isoxazol-3-yl)-phenoxymethyl]-piper...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Johnson and Johnson Pharmaceutical Research and Development Curated by ChEMBL | Assay Description Inhibitory concentration against interleukin-8 receptor of human neutrophils by using [125I]-IL-8 (0.125 nM) as radioligand | Bioorg Med Chem Lett 14: 4307-11 (2004) Article DOI: 10.1016/j.bmcl.2004.05.080 BindingDB Entry DOI: 10.7270/Q23F4P4M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 1 (Homo sapiens (Human)) | BDBM50150556![]() (1-Methyl-4-(3-{4-[3-(3-trifluoromethyl-phenyl)-iso...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Johnson and Johnson Pharmaceutical Research and Development Curated by ChEMBL | Assay Description Inhibitory concentration against interleukin-8 receptor of human neutrophils by using [125I]-IL-8 (0.125 nM) as radioligand | Bioorg Med Chem Lett 14: 4307-11 (2004) Article DOI: 10.1016/j.bmcl.2004.05.080 BindingDB Entry DOI: 10.7270/Q23F4P4M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sporulation kinase A (Bacillus subtilis (strain 168)) | BDBM50218645![]() (CHEMBL288462) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 6.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The R. W. Johnson Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of KinA/Sp0F system two component (TCS) from Bacillus subtilis. | Bioorg Med Chem Lett 11: 1545-8 (2001) BindingDB Entry DOI: 10.7270/Q2V69MSM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 1 (Homo sapiens (Human)) | BDBM50150566![]() (1-Methyl-4-[4-(5-phenyl-isoxazol-3-yl)-phenoxymeth...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Johnson and Johnson Pharmaceutical Research and Development Curated by ChEMBL | Assay Description Inhibitory concentration against interleukin-8 receptor of human neutrophils by using [125I]-IL-8 (0.125 nM) as radioligand | Bioorg Med Chem Lett 14: 4307-11 (2004) Article DOI: 10.1016/j.bmcl.2004.05.080 BindingDB Entry DOI: 10.7270/Q23F4P4M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 1 (Homo sapiens (Human)) | BDBM50150568![]() (CHEMBL183819 | Dimethyl-{3-[4-(3-phenyl-isoxazol-5...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Johnson and Johnson Pharmaceutical Research and Development Curated by ChEMBL | Assay Description Inhibitory concentration against interleukin-8 receptor of human neutrophils by using [125I]-IL-8 (0.125 nM) as radioligand | Bioorg Med Chem Lett 14: 4307-11 (2004) Article DOI: 10.1016/j.bmcl.2004.05.080 BindingDB Entry DOI: 10.7270/Q23F4P4M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 1 (Homo sapiens (Human)) | BDBM50150570![]() (1-Methyl-4-[4-(5-phenyl-isoxazol-3-yl)-phenoxymeth...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Johnson and Johnson Pharmaceutical Research and Development Curated by ChEMBL | Assay Description Inhibitory concentration against interleukin-8 receptor of human neutrophils by using [125I]-IL-8 (0.125 nM) as radioligand | Bioorg Med Chem Lett 14: 4307-11 (2004) Article DOI: 10.1016/j.bmcl.2004.05.080 BindingDB Entry DOI: 10.7270/Q23F4P4M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sporulation kinase A (Bacillus subtilis (strain 168)) | BDBM50218644![]() (CHEMBL416972) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 7.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The R. W. Johnson Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of KinA/Sp0F system two component (TCS) from Bacillus subtilis. | Bioorg Med Chem Lett 11: 1545-8 (2001) BindingDB Entry DOI: 10.7270/Q2V69MSM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 1 (Homo sapiens (Human)) | BDBM50150560![]() (CHEMBL184583 | {3-[5-(4-Chloro-phenyl)-isoxazol-3-...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Johnson and Johnson Pharmaceutical Research and Development Curated by ChEMBL | Assay Description Inhibitory concentration against interleukin-8 receptor of human neutrophils by using [125I]-IL-8 (0.125 nM) as radioligand | Bioorg Med Chem Lett 14: 4307-11 (2004) Article DOI: 10.1016/j.bmcl.2004.05.080 BindingDB Entry DOI: 10.7270/Q23F4P4M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 1 (Homo sapiens (Human)) | BDBM50150565![]() (1-(2-{4-[5-(4-Chloro-phenyl)-isoxazol-3-yl]-phenox...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Johnson and Johnson Pharmaceutical Research and Development Curated by ChEMBL | Assay Description Inhibitory concentration against interleukin-8 receptor of human neutrophils by using [125I]-IL-8 (0.125 nM) as radioligand | Bioorg Med Chem Lett 14: 4307-11 (2004) Article DOI: 10.1016/j.bmcl.2004.05.080 BindingDB Entry DOI: 10.7270/Q23F4P4M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sporulation initiation phosphotransferase F/kinase A (Bacillus subtilis (strain 168)) | BDBM50215963![]() (CHEMBL57687) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 9.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
R.W. Johnson Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of histidine protein kinase (KinA) phosphorylation in the presence of response regulator (Spo0F) | Bioorg Med Chem Lett 8: 1923-8 (1998) BindingDB Entry DOI: 10.7270/Q27S7QZM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sporulation kinase A (Bacillus subtilis (strain 168)) | BDBM50471730![]() (CHEMBL101786) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 9.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The R. W. Johnson Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of autophosphorylation of the two-component signal transduction system kinase was measured using the KinA/Spo0F regulatory system of Bacil... | J Med Chem 41: 2939-45 (1998) Article DOI: 10.1021/jm9803572 BindingDB Entry DOI: 10.7270/Q2VM4G0W | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sporulation kinase A (Bacillus subtilis (strain 168)) | BDBM50471728![]() (CHEMBL100719) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 9.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The R. W. Johnson Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of autophosphorylation of the two-component signal transduction system kinase was measured using the KinA/Spo0F regulatory system of Bacil... | J Med Chem 41: 2939-45 (1998) Article DOI: 10.1021/jm9803572 BindingDB Entry DOI: 10.7270/Q2VM4G0W | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 1 (Homo sapiens (Human)) | BDBM50150571![]() (1-(3-{4-[3-(3-Chloro-phenyl)-isoxazol-5-yl]-phenox...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Johnson and Johnson Pharmaceutical Research and Development Curated by ChEMBL | Assay Description Inhibitory concentration against interleukin-8 receptor of human neutrophils by using [125I]-IL-8 (0.125 nM) as radioligand | Bioorg Med Chem Lett 14: 4307-11 (2004) Article DOI: 10.1016/j.bmcl.2004.05.080 BindingDB Entry DOI: 10.7270/Q23F4P4M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sporulation kinase A (Bacillus subtilis (strain 168)) | BDBM50218648![]() (CHEMBL290098) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The R. W. Johnson Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of KinA/Sp0F system two component (TCS) from Bacillus subtilis. | Bioorg Med Chem Lett 11: 1545-8 (2001) BindingDB Entry DOI: 10.7270/Q2V69MSM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sporulation kinase A (Bacillus subtilis (strain 168)) | BDBM50218640![]() (CHEMBL38683) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The R. W. Johnson Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of KinA/Sp0F system two component (TCS) from Bacillus subtilis. | Bioorg Med Chem Lett 11: 1545-8 (2001) BindingDB Entry DOI: 10.7270/Q2V69MSM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 1 (Homo sapiens (Human)) | BDBM50150557![]() (1-(3-{4-[3-(4-Fluoro-phenyl)-[1,2,4]oxadiazol-5-yl...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.05E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Johnson and Johnson Pharmaceutical Research and Development Curated by ChEMBL | Assay Description Inhibitory concentration against interleukin-8 receptor of human neutrophils by using [125I]-IL-8 (0.125 nM) as radioligand | Bioorg Med Chem Lett 14: 4307-11 (2004) Article DOI: 10.1016/j.bmcl.2004.05.080 BindingDB Entry DOI: 10.7270/Q23F4P4M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 1 (Homo sapiens (Human)) | BDBM50150564![]() (CHEMBL425882 | Dimethyl-[4-(5-phenyl-isoxazol-3-yl...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.06E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Johnson and Johnson Pharmaceutical Research and Development Curated by ChEMBL | Assay Description Inhibitory concentration against interleukin-8 receptor of human neutrophils by using [125I]-IL-8 (0.125 nM) as radioligand | Bioorg Med Chem Lett 14: 4307-11 (2004) Article DOI: 10.1016/j.bmcl.2004.05.080 BindingDB Entry DOI: 10.7270/Q23F4P4M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 1 (Homo sapiens (Human)) | BDBM50150575![]() (1-Methyl-4-[4-(5-pyridin-2-yl-isoxazol-3-yl)-pheno...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.15E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Johnson and Johnson Pharmaceutical Research and Development Curated by ChEMBL | Assay Description Inhibitory concentration against interleukin-8 receptor of human neutrophils by using [125I]-IL-8 (0.125 nM) as radioligand | Bioorg Med Chem Lett 14: 4307-11 (2004) Article DOI: 10.1016/j.bmcl.2004.05.080 BindingDB Entry DOI: 10.7270/Q23F4P4M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sporulation kinase A (Bacillus subtilis (strain 168)) | BDBM50218643![]() (CHEMBL39634) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The R. W. Johnson Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of KinA/Sp0F system two component (TCS) from Bacillus subtilis. | Bioorg Med Chem Lett 11: 1545-8 (2001) BindingDB Entry DOI: 10.7270/Q2V69MSM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 1 (Homo sapiens (Human)) | BDBM50150562![]() (CHEMBL184401 | Dimethyl-{4-[5-(4-nitro-phenyl)-iso...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.21E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Johnson and Johnson Pharmaceutical Research and Development Curated by ChEMBL | Assay Description Inhibitory concentration against interleukin-8 receptor of human neutrophils by using [125I]-IL-8 (0.125 nM) as radioligand | Bioorg Med Chem Lett 14: 4307-11 (2004) Article DOI: 10.1016/j.bmcl.2004.05.080 BindingDB Entry DOI: 10.7270/Q23F4P4M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sporulation kinase A (Bacillus subtilis (strain 168)) | BDBM50218655![]() (CHEMBL38914) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The R. W. Johnson Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of KinA/Sp0F system two component (TCS) from Bacillus subtilis. | Bioorg Med Chem Lett 11: 1545-8 (2001) BindingDB Entry DOI: 10.7270/Q2V69MSM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sporulation kinase A (Bacillus subtilis (strain 168)) | BDBM50218647![]() (CHEMBL38867) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.54E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The R. W. Johnson Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of KinA/Sp0F system two component (TCS) from Bacillus subtilis. | Bioorg Med Chem Lett 11: 1545-8 (2001) BindingDB Entry DOI: 10.7270/Q2V69MSM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sporulation kinase A (Bacillus subtilis (strain 168)) | BDBM50218659![]() (CHEMBL43691) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 1.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The R. W. Johnson Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of KinA/Sp0F system two component (TCS) from Bacillus subtilis. | Bioorg Med Chem Lett 11: 1545-8 (2001) BindingDB Entry DOI: 10.7270/Q2V69MSM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sporulation kinase A (Bacillus subtilis (strain 168)) | BDBM50471723![]() (CHEMBL98273) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.90E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The R. W. Johnson Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of autophosphorylation of the two-component signal transduction system kinase was measured using the KinA/Spo0F regulatory system of Bacil... | J Med Chem 41: 2939-45 (1998) Article DOI: 10.1021/jm9803572 BindingDB Entry DOI: 10.7270/Q2VM4G0W | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sporulation kinase A (Bacillus subtilis (strain 168)) | BDBM50065970![]() (CHEMBL57656 | N-(3,4-Dichloro-phenyl)-2-hydroxy-3,...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The R. W. Johnson Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of autophosphorylation of the two-component signal transduction system kinase was measured using the KinA/Spo0F regulatory system of Bacil... | J Med Chem 41: 2939-45 (1998) Article DOI: 10.1021/jm9803572 BindingDB Entry DOI: 10.7270/Q2VM4G0W | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sporulation kinase A (Bacillus subtilis (strain 168)) | BDBM50065970![]() (CHEMBL57656 | N-(3,4-Dichloro-phenyl)-2-hydroxy-3,...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
R.W. Johnson Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of histidine protein kinase (KinA) phosphorylation in the presence of response regulator (Spo0F) | Bioorg Med Chem Lett 8: 1923-8 (1998) BindingDB Entry DOI: 10.7270/Q27S7QZM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 1 (Homo sapiens (Human)) | BDBM50150576![]() (1-Methyl-4-(3-{4-[3-(4-phenoxy-phenyl)-isoxazol-5-...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.27E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Johnson and Johnson Pharmaceutical Research and Development Curated by ChEMBL | Assay Description Inhibitory concentration against interleukin-8 receptor of human neutrophils by using [125I]-IL-8 (0.125 nM) as radioligand | Bioorg Med Chem Lett 14: 4307-11 (2004) Article DOI: 10.1016/j.bmcl.2004.05.080 BindingDB Entry DOI: 10.7270/Q23F4P4M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sporulation kinase A (Bacillus subtilis (strain 168)) | BDBM50218653![]() (CHEMBL39178) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 2.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The R. W. Johnson Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of KinA/Sp0F system two component (TCS) from Bacillus subtilis. | Bioorg Med Chem Lett 11: 1545-8 (2001) BindingDB Entry DOI: 10.7270/Q2V69MSM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 1 (Homo sapiens (Human)) | BDBM50150554![]() (4-(3-{4-[3-(4-Chloro-phenyl)-[1,2,4]oxadiazol-5-yl...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >2.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Johnson and Johnson Pharmaceutical Research and Development Curated by ChEMBL | Assay Description Inhibitory concentration against interleukin-8 receptor of human neutrophils by using [125I]-IL-8 (0.125 nM) as radioligand | Bioorg Med Chem Lett 14: 4307-11 (2004) Article DOI: 10.1016/j.bmcl.2004.05.080 BindingDB Entry DOI: 10.7270/Q23F4P4M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sporulation kinase A (Bacillus subtilis (strain 168)) | BDBM50471716![]() (CHEMBL431272) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The R. W. Johnson Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of autophosphorylation of the two-component signal transduction system kinase was measured using the KinA/Spo0F regulatory system of Bacil... | J Med Chem 41: 2939-45 (1998) Article DOI: 10.1021/jm9803572 BindingDB Entry DOI: 10.7270/Q2VM4G0W | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sporulation kinase A (Bacillus subtilis (strain 168)) | BDBM50100895![]() (2-(4-(4-carbamimidoylphenoxy)phenyl)-1H-indole-6-c...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid PDB UniChem Patents Similars | PubMed | n/a | n/a | 3.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The R. W. Johnson Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of KinA/Sp0F system two component system (TCS) from Bacillus subtilis | Bioorg Med Chem Lett 11: 1545-8 (2001) BindingDB Entry DOI: 10.7270/Q2V69MSM | |||||||||||
More data for this Ligand-Target Pair |
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