Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083811 (3-({1-[3-(1H-Imidazol-2-ylamino)-propyl]-1H-indazo...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.30 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhbitory activity against beta3-transfected 293 cells using alpha-V beta-3 antagonism assay | J Med Chem 43: 41-58 (2000) BindingDB Entry DOI: 10.7270/Q21G0KG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083839 (2-Benzyloxycarbonylamino-3-({1-[3-(4,5-dihydro-1H-...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 3.80 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhbition of Vitronectin receptor (alpha V beta 3) binding | J Med Chem 43: 41-58 (2000) BindingDB Entry DOI: 10.7270/Q21G0KG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083766 (2-(3,5-Dichloro-biphenyl-4-sulfonylamino)-3-({5-[4...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 4.60 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhibition of vitronectin receptor (alpha V beta 3), expressed on human 293 cells, binding to immobilized fibrinogen | J Med Chem 43: 27-40 (2000) BindingDB Entry DOI: 10.7270/Q2571B77 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083823 (3-({1-[3-(1H-Imidazol-2-ylamino)-propyl]-1H-indazo...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 4.70 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhbitory activity against beta3-transfected 293 cells using alpha-V beta-3 antagonism assay | J Med Chem 43: 41-58 (2000) BindingDB Entry DOI: 10.7270/Q21G0KG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083797 (2-(3,5-Dimethyl-biphenyl-4-sulfonylamino)-3-({1-[3...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 4.90 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhbitory activity against beta3-transfected 293 cells using alpha-V beta-3 antagonism assay | J Med Chem 43: 41-58 (2000) BindingDB Entry DOI: 10.7270/Q21G0KG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083788 (2-(2-Chloro-6-methyl-benzenesulfonylamino)-3-({5-[...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 7.10 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhibition of vitronectin receptor (alpha V beta 3), expressed on human 293 cells, binding to immobilized fibrinogen | J Med Chem 43: 27-40 (2000) BindingDB Entry DOI: 10.7270/Q2571B77 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083803 (2-Benzyloxycarbonylamino-3-({1-[3-(4,5-dihydro-1H-...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 7.30 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhbition of Vitronectin receptor (alpha V beta 3) binding | J Med Chem 43: 41-58 (2000) BindingDB Entry DOI: 10.7270/Q21G0KG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083836 (2-(2,6-Dichloro-benzenesulfonylamino)-3-({1-[3-(1H...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 8.5 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhbitory activity against beta3-transfected 293 cells using alpha-V beta-3 antagonism assay | J Med Chem 43: 41-58 (2000) BindingDB Entry DOI: 10.7270/Q21G0KG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083789 (2-(3,5-Dimethyl-biphenyl-4-sulfonylamino)-3-({5-[4...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 8.80 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhibition of vitronectin receptor (alpha V beta 3), expressed on human 293 cells, binding to immobilized fibrinogen | J Med Chem 43: 27-40 (2000) BindingDB Entry DOI: 10.7270/Q2571B77 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083810 (2-(2,6-Dimethyl-benzenesulfonylamino)-3-({1-[3-(1H...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhbitory activity against beta3-transfected 293 cells using alpha-V beta-3 antagonism assay | J Med Chem 43: 41-58 (2000) BindingDB Entry DOI: 10.7270/Q21G0KG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083837 (2-(4-Chloro-benzenesulfonylamino)-3-({1-[3-(1H-imi...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhbitory activity against beta3-transfected 293 cells using alpha-V beta-3 antagonism assay | J Med Chem 43: 41-58 (2000) BindingDB Entry DOI: 10.7270/Q21G0KG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083807 (2-(3,4-Dichloro-benzenesulfonylamino)-3-({1-[3-(1H...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhbitory activity against beta3-transfected 293 cells using alpha-V beta-3 antagonism assay | J Med Chem 43: 41-58 (2000) BindingDB Entry DOI: 10.7270/Q21G0KG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083768 ((S)3-({5-[4-(1H-Imidazol-2-ylamino)-butyl]-4,5-dih...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 10.6 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhibition of vitronectin receptor (alpha V beta 3), expressed on human 293 cells, binding to immobilized fibrinogen | J Med Chem 43: 27-40 (2000) BindingDB Entry DOI: 10.7270/Q2571B77 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083768 ((S)3-({5-[4-(1H-Imidazol-2-ylamino)-butyl]-4,5-dih...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 10.6 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhibition of vitronectin receptor (alpha V beta 3), expressed on human 293 cells, binding to immobilized fibrinogen | J Med Chem 43: 27-40 (2000) BindingDB Entry DOI: 10.7270/Q2571B77 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-IIb/beta-3 (Homo sapiens (Human)) | BDBM50083836 (2-(2,6-Dichloro-benzenesulfonylamino)-3-({1-[3-(1H...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhibition of aggregation of human gel-purified platelets (GPIIbIIIa GPP) | J Med Chem 43: 41-58 (2000) BindingDB Entry DOI: 10.7270/Q21G0KG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083812 (3-({1-[3-(1H-Imidazol-2-ylamino)-propyl]-1H-indazo...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 13 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhbitory activity against beta3-transfected 293 cells using alpha-V beta-3 antagonism assay | J Med Chem 43: 41-58 (2000) BindingDB Entry DOI: 10.7270/Q21G0KG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083769 (3-({5-[4-(1H-Imidazol-2-ylamino)-butyl]-4,5-dihydr...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhibition of vitronectin receptor (alpha V beta 3), expressed on human 293 cells, binding to immobilized fibrinogen | J Med Chem 43: 27-40 (2000) BindingDB Entry DOI: 10.7270/Q2571B77 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083833 (3-({1-[3-(1H-Imidazol-2-ylamino)-propyl]-1H-indazo...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 16 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhbitory activity against beta3-transfected 293 cells using alpha-V beta-3 antagonism assay | J Med Chem 43: 41-58 (2000) BindingDB Entry DOI: 10.7270/Q21G0KG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083783 (2-(2,6-Dichloro-benzenesulfonylamino)-3-({5-[4-(1H...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhibition of vitronectin receptor (alpha V beta 3), expressed on human 293 cells, binding to immobilized fibrinogen | J Med Chem 43: 27-40 (2000) BindingDB Entry DOI: 10.7270/Q2571B77 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-IIb/beta-3 (Homo sapiens (Human)) | BDBM50083811 (3-({1-[3-(1H-Imidazol-2-ylamino)-propyl]-1H-indazo...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 21 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhibition of aggregation of human gel-purified platelets (GPIIbIIIa GPP) | J Med Chem 43: 41-58 (2000) BindingDB Entry DOI: 10.7270/Q21G0KG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083793 (2-Benzyloxycarbonylamino-3-({2-[3-(4,5-dihydro-1H-...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 25 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhbition of Vitronectin receptor (alpha V beta 3) binding | J Med Chem 43: 41-58 (2000) BindingDB Entry DOI: 10.7270/Q21G0KG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083802 (3-({1-[3-(1H-Imidazol-2-ylamino)-propyl]-1H-indazo...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 25 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhbitory activity against beta3-transfected 293 cells using alphaV-beta3 antagonism assay | J Med Chem 43: 41-58 (2000) BindingDB Entry DOI: 10.7270/Q21G0KG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083791 (3-({5-[3-(6-Amino-pyridin-2-yl)-propyl]-4,5-dihydr...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 26 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhibition of vitronectin receptor (alpha V beta 3), expressed on human 293 cells, binding to immobilized fibrinogen | J Med Chem 43: 27-40 (2000) BindingDB Entry DOI: 10.7270/Q2571B77 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083809 (3-({1-[3-(1H-Imidazol-2-ylamino)-propyl]-1H-indazo...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 26 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhbitory activity against beta3-transfected 293 cells using alpha-V beta-3 antagonism assay | J Med Chem 43: 41-58 (2000) BindingDB Entry DOI: 10.7270/Q21G0KG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083814 (3-({1-[3-(1,4,5,6-Tetrahydro-pyrimidin-2-ylamino)-...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 28 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhibition of adhesion of integrin beta3-transfected HEK293 cells to fibrinogen | J Med Chem 43: 41-58 (2000) BindingDB Entry DOI: 10.7270/Q21G0KG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083785 (3-({5-[3-(1H-Imidazol-2-ylcarbamoyl)-propyl]-4,5-d...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 31 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhbitory activity against beta3-transfected 293 cells using alpha-V beta-3 antagonism assay | J Med Chem 43: 41-58 (2000) BindingDB Entry DOI: 10.7270/Q21G0KG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083785 (3-({5-[3-(1H-Imidazol-2-ylcarbamoyl)-propyl]-4,5-d...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 31 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhibition of vitronectin receptor (alpha V beta 3), expressed on human 293 cells, binding to immobilized fibrinogen | J Med Chem 43: 27-40 (2000) BindingDB Entry DOI: 10.7270/Q2571B77 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083775 (3-[(5-{2-[3-(1H-Imidazol-2-yl)-ureido]-ethyl}-4,5-...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 34 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhibition of vitronectin receptor (alpha V beta 3), expressed on human 293 cells, binding to immobilized fibrinogen | J Med Chem 43: 27-40 (2000) BindingDB Entry DOI: 10.7270/Q2571B77 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-IIb/beta-3 (Homo sapiens (Human)) | BDBM50083799 (2-Benzenesulfonylamino-3-({1-[3-(1H-imidazol-2-yla...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 34 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhibition of aggregation of human gel-purified platelets (GPIIbIIIa GPP) | J Med Chem 43: 41-58 (2000) BindingDB Entry DOI: 10.7270/Q21G0KG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083805 (2-(Biphenyl-4-sulfonylamino)-3-({1-[3-(1H-imidazol...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 35 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhbitory activity against beta3-transfected 293 cells using alpha-V beta-3 antagonism assay | J Med Chem 43: 41-58 (2000) BindingDB Entry DOI: 10.7270/Q21G0KG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-IIb/beta-3 (Homo sapiens (Human)) | BDBM50083812 (3-({1-[3-(1H-Imidazol-2-ylamino)-propyl]-1H-indazo...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 39 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhibition of aggregation of human gel-purified platelets (GPIIbIIIa GPP) | J Med Chem 43: 41-58 (2000) BindingDB Entry DOI: 10.7270/Q21G0KG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083799 (2-Benzenesulfonylamino-3-({1-[3-(1H-imidazol-2-yla...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 44 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhbitory activity against beta3-transfected 293 cells using alpha-V beta-3 antagonism assay | J Med Chem 43: 41-58 (2000) BindingDB Entry DOI: 10.7270/Q21G0KG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083780 (2-(3,5-Dimethyl-biphenyl-4-sulfonylamino)-3-({5-[4...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 44 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhibition of vitronectin receptor (alpha V beta 3), expressed on human 293 cells, binding to immobilized fibrinogen | J Med Chem 43: 27-40 (2000) BindingDB Entry DOI: 10.7270/Q2571B77 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083770 (3-({5-[3-(2-Amino-1H-imidazol-4-yl)-propyl]-4,5-di...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 46 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhibition of vitronectin receptor (alpha V beta 3), expressed on human 293 cells, binding to immobilized fibrinogen | J Med Chem 43: 27-40 (2000) BindingDB Entry DOI: 10.7270/Q2571B77 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083813 (3-({1-[3-(Pyridin-2-ylamino)-propyl]-1H-indazole-5...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 48 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhbitory activity against beta3-transfected 293 cells using alpha-V beta-3 antagonism assay | J Med Chem 43: 41-58 (2000) BindingDB Entry DOI: 10.7270/Q21G0KG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083801 (2-Benzyloxycarbonylamino-3-({1-[2-(4,5-dihydro-1H-...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 51 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhbition of Vitronectin receptor (alpha V beta 3) binding | J Med Chem 43: 41-58 (2000) BindingDB Entry DOI: 10.7270/Q21G0KG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083767 (3-({5-[4-(1H-Imidazol-2-ylamino)-butyl]-4,5-dihydr...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 51 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhibition of vitronectin receptor (alpha V beta 3), expressed on human 293 cells, binding to immobilized fibrinogen | J Med Chem 43: 27-40 (2000) BindingDB Entry DOI: 10.7270/Q2571B77 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083816 (3-({1-[3-(1H-Imidazol-2-ylamino)-propyl]-1H-indazo...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 52 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhbitory activity against beta3-transfected 293 cells using alpha-V beta-3 antagonism assay | J Med Chem 43: 41-58 (2000) BindingDB Entry DOI: 10.7270/Q21G0KG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083781 (3-({5-[4-(Pyridin-2-ylamino)-butyl]-4,5-dihydro-is...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 54 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhibition of vitronectin receptor (alpha V beta 3), expressed on human 293 cells, binding to immobilized fibrinogen | J Med Chem 43: 27-40 (2000) BindingDB Entry DOI: 10.7270/Q2571B77 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083828 (2-Benzyloxycarbonylamino-3-({2-[3-(4,5-dihydro-1H-...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 55 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhbition of Vitronectin receptor (alpha V beta 3) binding | J Med Chem 43: 41-58 (2000) BindingDB Entry DOI: 10.7270/Q21G0KG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083794 (3-({1-[2-(1H-Imidazol-2-ylcarbamoyl)-ethyl]-1H-ind...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 56 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhbitory activity against beta3-transfected 293 cells using alpha-V beta-3 antagonism assay | J Med Chem 43: 41-58 (2000) BindingDB Entry DOI: 10.7270/Q21G0KG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-IIb/beta-3 (Homo sapiens (Human)) | BDBM50083821 (3-({1-[3-(4,5-Dihydro-1H-imidazol-2-ylamino)-propy...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 57 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhibition of aggregation of human gel-purified platelets (GPIIbIIIa GPP) | J Med Chem 43: 41-58 (2000) BindingDB Entry DOI: 10.7270/Q21G0KG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083774 (3-({5-[4-(4,5-Dihydro-1H-imidazol-2-ylamino)-butyl...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 62 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhibition of vitronectin receptor (alpha V beta 3), expressed on human 293 cells, binding to immobilized fibrinogen | J Med Chem 43: 27-40 (2000) BindingDB Entry DOI: 10.7270/Q2571B77 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-IIb/beta-3 (Homo sapiens (Human)) | BDBM50083814 (3-({1-[3-(1,4,5,6-Tetrahydro-pyrimidin-2-ylamino)-...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 66 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhibition of aggregation of human gel-purified platelets (GPIIbIIIa GPP) | J Med Chem 43: 41-58 (2000) BindingDB Entry DOI: 10.7270/Q21G0KG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083821 (3-({1-[3-(4,5-Dihydro-1H-imidazol-2-ylamino)-propy...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 70 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhibition of adhesion of integrin beta3-transfected HEK293 cells to fibrinogen | J Med Chem 43: 41-58 (2000) BindingDB Entry DOI: 10.7270/Q21G0KG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083771 (2-(3,5-Dimethyl-isoxazole-4-sulfonylamino)-3-({5-[...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 73 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhibition of vitronectin receptor (alpha V beta 3), expressed on human 293 cells, binding to immobilized fibrinogen | J Med Chem 43: 27-40 (2000) BindingDB Entry DOI: 10.7270/Q2571B77 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50083832 (2-Benzyloxycarbonylamino-3-({1-[3-(1H-imidazol-2-y...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 74 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhbitory activity against beta3-transfected 293 cells using alpha-V beta-3 antagonism assay | J Med Chem 43: 41-58 (2000) BindingDB Entry DOI: 10.7270/Q21G0KG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-IIb/beta-3 (Homo sapiens (Human)) | BDBM50083797 (2-(3,5-Dimethyl-biphenyl-4-sulfonylamino)-3-({1-[3...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 74 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhibition of aggregation of human gel-purified platelets (GPIIbIIIa GPP) | J Med Chem 43: 41-58 (2000) BindingDB Entry DOI: 10.7270/Q21G0KG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-IIb/beta-3 (Homo sapiens (Human)) | BDBM50083810 (2-(2,6-Dimethyl-benzenesulfonylamino)-3-({1-[3-(1H...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 74 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhibition of aggregation of human gel-purified platelets (GPIIbIIIa GPP) | J Med Chem 43: 41-58 (2000) BindingDB Entry DOI: 10.7270/Q21G0KG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-IIb/beta-3 (Homo sapiens (Human)) | BDBM50083823 (3-({1-[3-(1H-Imidazol-2-ylamino)-propyl]-1H-indazo...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 81 | n/a | n/a | n/a | n/a | n/a | n/a |
DuPont Pharmaceuticals Company Curated by ChEMBL | Assay Description Inhibition of aggregation of human gel-purified platelets (GPIIbIIIa GPP) | J Med Chem 43: 41-58 (2000) BindingDB Entry DOI: 10.7270/Q21G0KG2 | |||||||||||
More data for this Ligand-Target Pair |
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