Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Secreted frizzled-related protein 1 (Homo sapiens (Human)) | BDBM50265547![]() (CHEMBL455476 | N-{1-[1-(3,3-Dimethylbutanoyl)-L-pr...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Binding affinity to human purified SARP2 by fluorescent polarization assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Secreted frizzled-related protein 1 (Homo sapiens (Human)) | BDBM50265555![]() ((2S)-N-Phenyl-2-{[4-({[5-(phenylsulfonyl)-2-(trifl...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Binding affinity to human purified SARP2 by fluorescent polarization assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Secreted frizzled-related protein 1 (Homo sapiens (Human)) | BDBM50265554![]() ((2S)-N-(tert-Butyl)-2-{[4-({[5-(phenylsulfonyl)-2-...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Binding affinity to human purified SARP2 by fluorescent polarization assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Secreted frizzled-related protein 1 (Homo sapiens (Human)) | BDBM50265580![]() ((2S)-N,N-Dimethyl-2-{[4-({[5-(phenylsulfonyl)-2-(t...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Binding affinity to human purified SARP2 by fluorescent polarization assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Secreted frizzled-related protein 1 (Homo sapiens (Human)) | BDBM50265583![]() (CHEMBL451431 | N-{1-[1-(3,3-Dimethylbutyl)-L-proly...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Binding affinity to human purified SARP2 by fluorescent polarization assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Secreted frizzled-related protein 1 (Homo sapiens (Human)) | BDBM50265553![]() ((2S)-N-Ethyl-2-{[4-({[5-(phenylsulfonyl)-2-(triflu...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Binding affinity to human purified SARP2 by fluorescent polarization assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Secreted frizzled-related protein 1 (Homo sapiens (Human)) | BDBM50265499![]() (CHEMBL495534 | N-[1-(1H-Imidazol-1-ylacetyl)piperi...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Binding affinity to human purified SARP2 by fluorescent polarization assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Secreted frizzled-related protein 1 (Homo sapiens (Human)) | BDBM50265581![]() (CHEMBL505036 | N-{1-[1-(Morpholin-4-ylcarbonyl)-L-...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Binding affinity to human purified SARP2 by fluorescent polarization assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Secreted frizzled-related protein 1 (Homo sapiens (Human)) | BDBM50265546![]() (CHEMBL447079 | N-{1-[1-(2,2-Dimethylpropanoyl)-L-p...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Binding affinity to human purified SARP2 by fluorescent polarization assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Secreted frizzled-related protein 1 (Homo sapiens (Human)) | BDBM50265584![]() (CHEMBL503281 | N-{1-[1-(Cyclohexylmethyl)-L-prolyl...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Binding affinity to human purified SARP2 by fluorescent polarization assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Secreted frizzled-related protein 1 (Homo sapiens (Human)) | BDBM50265545![]() (CHEMBL500903 | N-[1-(1-Isobutyryl-L-prolyl)piperid...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Binding affinity to human purified SARP2 by fluorescent polarization assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Secreted frizzled-related protein 1 (Homo sapiens (Human)) | BDBM50265549![]() (CHEMBL507695 | N-{1-[1-(Cyclohexylcarbonyl)-L-prol...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 50 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Binding affinity to human purified SARP2 by fluorescent polarization assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Secreted frizzled-related protein 1 (Homo sapiens (Human)) | BDBM50265500![]() ((S)-tert-butyl 2-(4-(5-(phenylsulfonyl)-2-(trifluo...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 60 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Binding affinity to human purified SARP2 by fluorescent polarization assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Secreted frizzled-related protein 1 (Homo sapiens (Human)) | BDBM50265552![]() (CHEMBL454478 | N-[1-(1-Isonicotinoyl-L-prolyl)pipe...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 70 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Binding affinity to human purified SARP2 by fluorescent polarization assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Secreted frizzled-related protein 1 (Homo sapiens (Human)) | BDBM50265550![]() (CHEMBL510748 | N-[1-(1-Benzoyl-L-prolyl)piperidin-...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 70 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Binding affinity to human purified SARP2 by fluorescent polarization assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Secreted frizzled-related protein 1 (Homo sapiens (Human)) | BDBM50265548![]() (CHEMBL501332 | N-[1-(N,N-Dimethylglycyl-L-prolyl)p...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 90 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Binding affinity to human purified SARP2 by fluorescent polarization assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Secreted frizzled-related protein 1 (Homo sapiens (Human)) | BDBM50265505![]() (CHEMBL525899 | N-[1-(5-oxo-L-Prolyl)piperidin-4-yl...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 90 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Binding affinity to human purified SARP2 by fluorescent polarization assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Secreted frizzled-related protein 1 (Homo sapiens (Human)) | BDBM50265480![]() (CHEMBL523726 | N-[1-(Morpholin-4-ylacetyl)piperidi...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Binding affinity to human purified SARP2 by fluorescent polarization assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Secreted frizzled-related protein 1 (Homo sapiens (Human)) | BDBM50265503![]() ((S)-5-(phenylsulfonyl)-N-(1-(pyrrolidine-2-carbony...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 110 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Binding affinity to human purified SARP2 by fluorescent polarization assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Secreted frizzled-related protein 1 (Homo sapiens (Human)) | BDBM50265479![]() (5-(Phenylsulfonyl)-N-[1-(pyrrolidin-1-ylacetyl)pip...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 110 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Binding affinity to human purified SARP2 by fluorescent polarization assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Secreted frizzled-related protein 1 (Homo sapiens (Human)) | BDBM50265551![]() (CHEMBL462363 | N-(1-{1-[4-(Dimethylamino)benzoyl]-...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 110 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Binding affinity to human purified SARP2 by fluorescent polarization assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Secreted frizzled-related protein 1 (Homo sapiens (Human)) | BDBM50265501![]() ((R)-tert-butyl 2-(4-(5-(phenylsulfonyl)-2-(trifluo...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 120 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Binding affinity to human purified SARP2 by fluorescent polarization assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Secreted frizzled-related protein 1 (Homo sapiens (Human)) | BDBM50265582![]() (CHEMBL496581 | N-[1-(1-Methyl-L-prolyl)piperidin-4...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 120 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Binding affinity to human purified SARP2 by fluorescent polarization assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Secreted frizzled-related protein 1 (Homo sapiens (Human)) | BDBM50265502![]() (CHEMBL504979 | tert-Butyl(5S)-2-oxo-5-{[4-({[5-(Ph...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 130 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Binding affinity to human purified SARP2 by fluorescent polarization assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Secreted frizzled-related protein 1 (Homo sapiens (Human)) | BDBM50265481![]() (5-(Phenylsulfonyl)-N-[1-(piperazin-1-ylacetyl)pipe...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 140 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Binding affinity to human purified SARP2 by fluorescent polarization assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Secreted frizzled-related protein 1 (Homo sapiens (Human)) | BDBM50265544![]() (CHEMBL525970 | N-[1-(1-Acetyl-L-prolyl)piperidin-4...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 160 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Binding affinity to human purified SARP2 by fluorescent polarization assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Secreted frizzled-related protein 1 (Homo sapiens (Human)) | BDBM50265504![]() ((R)-5-(phenylsulfonyl)-N-(1-(pyrrolidine-2-carbony...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Binding affinity to human purified SARP2 by fluorescent polarization assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Secreted frizzled-related protein 1 (Homo sapiens (Human)) | BDBM50265468![]() (CHEMBL497177 | N-[1-(N-Methylglycyl)piperidin-4-yl...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Binding affinity to human purified SARP2 by fluorescent polarization assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Secreted frizzled-related protein 1 (Homo sapiens (Human)) | BDBM50265469![]() (CHEMBL497383 | N-[1-(N,N-Dimethylglycyl)piperidin-...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 300 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Binding affinity to human purified SARP2 by fluorescent polarization assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Secreted frizzled-related protein 1 (Homo sapiens (Human)) | BDBM50265467![]() (5-(Phenylsulfonyl)-N-piperidin-4-yl-2-(trifluorome...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 500 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Binding affinity to human purified SARP2 by fluorescent polarization assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Secreted frizzled-related protein 1 (Homo sapiens (Human)) | BDBM50265585![]() (CHEMBL511077 | N-[1-(1-Benzyl-L-prolyl)piperidin-4...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Binding affinity to human purified SARP2 by fluorescent polarization assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50306714![]() (CHEMBL601873 | Isopropyl 1,1-Dimethyl-3-[4-(3-morp...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 5.74E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Inhibition of human ERG | J Med Chem 53: 1774-87 (2010) Article DOI: 10.1021/jm901650u BindingDB Entry DOI: 10.7270/Q24F1QT5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50306735![]() (1-methylethyl 8-fluoro-1,1-dimethyl-3-{[4-(3-morph...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL MMDB PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Inhibition of human ERG | J Med Chem 53: 1774-87 (2010) Article DOI: 10.1021/jm901650u BindingDB Entry DOI: 10.7270/Q24F1QT5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50306744![]() (CHEMBL601221 | Isopropyl 8-Fluoro-1,1-dimethyl-3-[...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Inhibition of human ERG | J Med Chem 53: 1774-87 (2010) Article DOI: 10.1021/jm901650u BindingDB Entry DOI: 10.7270/Q24F1QT5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proto-oncogene Wnt-3 (Homo sapiens (Human)) | BDBM50265480![]() (CHEMBL523726 | N-[1-(Morpholin-4-ylacetyl)piperidi...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 160 | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Antagonist activity at human WNT3 expressed in human U2OS cells assessed as Wnt signaling after 16 to 18 hrs by luciferase reporter gene assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proto-oncogene Wnt-3 (Homo sapiens (Human)) | BDBM50265481![]() (5-(Phenylsulfonyl)-N-[1-(piperazin-1-ylacetyl)pipe...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 250 | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Antagonist activity at human WNT3 expressed in human U2OS cells assessed as Wnt signaling after 16 to 18 hrs by luciferase reporter gene assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proto-oncogene Wnt-3 (Homo sapiens (Human)) | BDBM50265499![]() (CHEMBL495534 | N-[1-(1H-Imidazol-1-ylacetyl)piperi...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 230 | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Antagonist activity at human WNT3 expressed in human U2OS cells assessed as Wnt signaling after 16 to 18 hrs by luciferase reporter gene assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proto-oncogene Wnt-3 (Homo sapiens (Human)) | BDBM50265500![]() ((S)-tert-butyl 2-(4-(5-(phenylsulfonyl)-2-(trifluo...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 60 | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Antagonist activity at human WNT3 expressed in human U2OS cells assessed as Wnt signaling after 16 to 18 hrs by luciferase reporter gene assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proto-oncogene Wnt-3 (Homo sapiens (Human)) | BDBM50265501![]() ((R)-tert-butyl 2-(4-(5-(phenylsulfonyl)-2-(trifluo...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 210 | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Antagonist activity at human WNT3 expressed in human U2OS cells assessed as Wnt signaling after 16 to 18 hrs by luciferase reporter gene assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proto-oncogene Wnt-3 (Homo sapiens (Human)) | BDBM50265502![]() (CHEMBL504979 | tert-Butyl(5S)-2-oxo-5-{[4-({[5-(Ph...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 90 | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Antagonist activity at human WNT3 expressed in human U2OS cells assessed as Wnt signaling after 16 to 18 hrs by luciferase reporter gene assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proto-oncogene Wnt-3 (Homo sapiens (Human)) | BDBM50265503![]() ((S)-5-(phenylsulfonyl)-N-(1-(pyrrolidine-2-carbony...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 350 | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Antagonist activity at human WNT3 expressed in human U2OS cells assessed as Wnt signaling after 16 to 18 hrs by luciferase reporter gene assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proto-oncogene Wnt-3 (Homo sapiens (Human)) | BDBM50265504![]() ((R)-5-(phenylsulfonyl)-N-(1-(pyrrolidine-2-carbony...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 710 | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Antagonist activity at human WNT3 expressed in human U2OS cells assessed as Wnt signaling after 16 to 18 hrs by luciferase reporter gene assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proto-oncogene Wnt-3 (Homo sapiens (Human)) | BDBM50265505![]() (CHEMBL525899 | N-[1-(5-oxo-L-Prolyl)piperidin-4-yl...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 240 | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Antagonist activity at human WNT3 expressed in human U2OS cells assessed as Wnt signaling after 16 to 18 hrs by luciferase reporter gene assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proto-oncogene Wnt-3 (Homo sapiens (Human)) | BDBM50265544![]() (CHEMBL525970 | N-[1-(1-Acetyl-L-prolyl)piperidin-4...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 250 | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Antagonist activity at human WNT3 expressed in human U2OS cells assessed as Wnt signaling after 16 to 18 hrs by luciferase reporter gene assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proto-oncogene Wnt-3 (Homo sapiens (Human)) | BDBM50265545![]() (CHEMBL500903 | N-[1-(1-Isobutyryl-L-prolyl)piperid...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 90 | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Antagonist activity at human WNT3 expressed in human U2OS cells assessed as Wnt signaling after 16 to 18 hrs by luciferase reporter gene assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proto-oncogene Wnt-3 (Homo sapiens (Human)) | BDBM50265546![]() (CHEMBL447079 | N-{1-[1-(2,2-Dimethylpropanoyl)-L-p...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 270 | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Antagonist activity at human WNT3 expressed in human U2OS cells assessed as Wnt signaling after 16 to 18 hrs by luciferase reporter gene assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proto-oncogene Wnt-3 (Homo sapiens (Human)) | BDBM50265547![]() (CHEMBL455476 | N-{1-[1-(3,3-Dimethylbutanoyl)-L-pr...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 120 | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Antagonist activity at human WNT3 expressed in human U2OS cells assessed as Wnt signaling after 16 to 18 hrs by luciferase reporter gene assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proto-oncogene Wnt-3 (Homo sapiens (Human)) | BDBM50265548![]() (CHEMBL501332 | N-[1-(N,N-Dimethylglycyl-L-prolyl)p...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 310 | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Antagonist activity at human WNT3 expressed in human U2OS cells assessed as Wnt signaling after 16 to 18 hrs by luciferase reporter gene assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proto-oncogene Wnt-3 (Homo sapiens (Human)) | BDBM50265549![]() (CHEMBL507695 | N-{1-[1-(Cyclohexylcarbonyl)-L-prol...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 460 | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Antagonist activity at human WNT3 expressed in human U2OS cells assessed as Wnt signaling after 16 to 18 hrs by luciferase reporter gene assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proto-oncogene Wnt-3 (Homo sapiens (Human)) | BDBM50265550![]() (CHEMBL510748 | N-[1-(1-Benzoyl-L-prolyl)piperidin-...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 380 | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Antagonist activity at human WNT3 expressed in human U2OS cells assessed as Wnt signaling after 16 to 18 hrs by luciferase reporter gene assay | J Med Chem 52: 105-16 (2009) Article DOI: 10.1021/jm801144h BindingDB Entry DOI: 10.7270/Q2NZ87HT | |||||||||||
More data for this Ligand-Target Pair |
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