Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Estrogen receptor beta (Homo sapiens (Human)) | BDBM50234790 ((E)-2-chloro-3,4'-dihydroxybiphenyl-4-carbaldehyde...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 12 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universita di Pisa Curated by ChEMBL | Assay Description Displacement of [3H]estradiol from purified full length human ERbeta receptor | J Med Chem 51: 1344-51 (2008) Article DOI: 10.1021/jm701396g BindingDB Entry DOI: 10.7270/Q2HQ40SB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor (Homo sapiens (Human)) | BDBM50234790 ((E)-2-chloro-3,4'-dihydroxybiphenyl-4-carbaldehyde...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 310 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universita di Pisa Curated by ChEMBL | Assay Description Displacement of [3H]estradiol from purified full length human ERalpha receptor | J Med Chem 51: 1344-51 (2008) Article DOI: 10.1021/jm701396g BindingDB Entry DOI: 10.7270/Q2HQ40SB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor beta (Homo sapiens (Human)) | BDBM50234790 ((E)-2-chloro-3,4'-dihydroxybiphenyl-4-carbaldehyde...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 11 | n/a | n/a | n/a | n/a |
Universita di Pisa Curated by ChEMBL | Assay Description Agonist activity at full length human ERbeta receptor expressed in human HEC-1 cells assessed as (ERE)2-pS2-luc reporter gene transcriptional activit... | J Med Chem 51: 1344-51 (2008) Article DOI: 10.1021/jm701396g BindingDB Entry DOI: 10.7270/Q2HQ40SB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor (Homo sapiens (Human)) | BDBM50234790 ((E)-2-chloro-3,4'-dihydroxybiphenyl-4-carbaldehyde...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 26 | n/a | n/a | n/a | n/a |
Universita di Pisa Curated by ChEMBL | Assay Description Agonist activity at full length human ERalpha receptor expressed in human HEC-1 cells assessed as (ERE)2-pS2-luc reporter gene transcriptional activi... | J Med Chem 51: 1344-51 (2008) Article DOI: 10.1021/jm701396g BindingDB Entry DOI: 10.7270/Q2HQ40SB | |||||||||||
More data for this Ligand-Target Pair |