Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Endothelin-1 receptor (RAT) | BDBM50051007 ((2R,3R,4S)-4-Benzo[1,3]dioxol-5-yl-1-dibutylcarbam...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | 0.0340 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Binding affinity towards Endothelin A receptor | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50143784 ((5S,6R,7R)-5-Benzo[1,3]dioxol-5-yl-2-butyl-7-[2-((...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 0.0340 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Binding affinity towards Endothelin A receptor | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50058126 (2-[2-(6-Methyl-benzo[1,3]dioxol-5-yl)-acetyl]-thio...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid UniChem Patents Similars | Article PubMed | 0.430 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Binding affinity towards Endothelin A receptor | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50091105 (4''-Oxazol-2-yl-biphenyl-2-sulfonic acid (3,4-dime...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | 1.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Binding affinity towards Endothelin A receptor | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50108202 ((S)-2-(4,6-Dimethoxy-pyrimidin-2-yloxy)-3-methoxy-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid UniChem Patents Similars | Article PubMed | 6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Binding affinity towards Endothelin A receptor | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50061101 (4-(1,1-Dimethylethyl)-N-(6-(2-hydroxyethoxy)-5-(2-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 6.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Binding affinity towards Endothelin A receptor | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50143792 (3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.0200 | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Inhibitory concentration towards endothelin A receptor in rat. | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50143796 (3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.0200 | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Inhibitory concentration towards endothelin A receptor in rat. | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50143797 (3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.0300 | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Inhibitory concentration towards endothelin A receptor in rat. | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50143802 (3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.0300 | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Inhibitory concentration towards endothelin A receptor in rat. | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50143786 (3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.0300 | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Inhibitory concentration towards endothelin A receptor in rat. | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Homo sapiens (Human)) | BDBM50098777 (3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 0.0400 | n/a | n/a | n/a | n/a | n/a | n/a |
Texas Biotechnology Corporation Curated by ChEMBL | Assay Description Inhibitory concentration was determined against selective Endothelin A receptor | J Med Chem 44: 1211-6 (2001) BindingDB Entry DOI: 10.7270/Q2Z89BN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50143778 (2-{[3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-t...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.0400 | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Inhibitory concentration towards endothelin A receptor in rat. | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50143783 (3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.0400 | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Inhibitory concentration towards endothelin A receptor in rat. | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50098777 (3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.0400 | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Inhibitory concentration towards endothelin A receptor in rat. | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50143773 (3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.0500 | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Inhibitory concentration towards endothelin A receptor in rat. | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50143789 (3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.0500 | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Inhibitory concentration towards endothelin A receptor in rat. | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50143801 (3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.0600 | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Inhibitory concentration towards endothelin A receptor in rat. | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50143785 (3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.0600 | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Inhibitory concentration towards endothelin A receptor in rat. | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50143788 (3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.0700 | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Inhibitory concentration towards endothelin A receptor in rat. | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50143787 (3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.0800 | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Inhibitory concentration towards endothelin A receptor in rat. | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50143780 (3-(3,4-Dimethyl-isoxazol-5-ylsulfamoyl)-thiophene-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.0800 | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Inhibitory concentration towards endothelin A receptor in rat. | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50143793 (3-(3,4-Dimethyl-isoxazol-5-ylsulfamoyl)-thiophene-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.0800 | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Inhibitory concentration towards endothelin A receptor in rat. | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50143794 (3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.0900 | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Inhibitory concentration towards endothelin A receptor in rat. | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50143774 (3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.100 | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Inhibitory concentration towards endothelin A receptor in rat. | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Homo sapiens (Human)) | BDBM50098780 (3-(4-Chloro-5-methyl-isoxazol-3-ylsulfamoyl)-thiop...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | PubMed | n/a | n/a | 0.100 | n/a | n/a | n/a | n/a | n/a | n/a |
Texas Biotechnology Corporation Curated by ChEMBL | Assay Description Inhibitory concentration was determined against selective Endothelin A receptor | J Med Chem 44: 1211-6 (2001) BindingDB Entry DOI: 10.7270/Q2Z89BN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50143772 (2-{[3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-t...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.110 | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Inhibitory concentration towards endothelin A receptor in rat. | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Homo sapiens (Human)) | BDBM50098773 (3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 0.120 | n/a | n/a | n/a | n/a | n/a | n/a |
Texas Biotechnology Corporation Curated by ChEMBL | Assay Description Inhibitory concentration was determined against selective Endothelin A receptor | J Med Chem 44: 1211-6 (2001) BindingDB Entry DOI: 10.7270/Q2Z89BN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Homo sapiens (Human)) | BDBM50098774 (2-[2-(3-Hydroxy-2,4,6-trimethyl-phenyl)-acetyl]-th...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 0.140 | n/a | n/a | n/a | n/a | n/a | n/a |
Texas Biotechnology Corporation Curated by ChEMBL | Assay Description Inhibitory concentration was determined against selective Endothelin A receptor | J Med Chem 44: 1211-6 (2001) BindingDB Entry DOI: 10.7270/Q2Z89BN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Homo sapiens (Human)) | BDBM50098778 (3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 0.140 | n/a | n/a | n/a | n/a | n/a | n/a |
Texas Biotechnology Corporation Curated by ChEMBL | Assay Description Inhibitory concentration was determined against selective Endothelin A receptor | J Med Chem 44: 1211-6 (2001) BindingDB Entry DOI: 10.7270/Q2Z89BN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50143790 (3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.140 | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Inhibitory concentration towards endothelin A receptor in rat. | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50098772 (3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.150 | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Inhibitory concentration towards endothelin A receptor in rat. | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Homo sapiens (Human)) | BDBM50098772 (3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 0.170 | n/a | n/a | n/a | n/a | n/a | n/a |
Texas Biotechnology Corporation Curated by ChEMBL | Assay Description Inhibitory concentration was determined against selective Endothelin A receptor | J Med Chem 44: 1211-6 (2001) BindingDB Entry DOI: 10.7270/Q2Z89BN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Homo sapiens (Human)) | BDBM50098775 (3-(3,4-Dimethyl-isoxazol-5-ylsulfamoyl)-thiophene-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 0.170 | n/a | n/a | n/a | n/a | n/a | n/a |
Texas Biotechnology Corporation Curated by ChEMBL | Assay Description Inhibitory concentration was determined against selective Endothelin A receptor | J Med Chem 44: 1211-6 (2001) BindingDB Entry DOI: 10.7270/Q2Z89BN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Homo sapiens (Human)) | BDBM50098779 (3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 0.190 | n/a | n/a | n/a | n/a | n/a | n/a |
Texas Biotechnology Corporation Curated by ChEMBL | Assay Description Inhibitory concentration was determined against selective Endothelin A receptor | J Med Chem 44: 1211-6 (2001) BindingDB Entry DOI: 10.7270/Q2Z89BN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50143781 (3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-5-met...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.210 | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Inhibitory concentration towards endothelin A receptor in rat. | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50143777 (CHEMBL61425 | TAK-044 | {(2S,5S,8S,11R,14R,17S)-14...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.240 | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Inhibitory concentration towards endothelin A receptor in rat. | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50051007 ((2R,3R,4S)-4-Benzo[1,3]dioxol-5-yl-1-dibutylcarbam...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.310 | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Inhibitory concentration towards endothelin A receptor in rat. | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50143799 (3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.390 | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Inhibitory concentration towards endothelin A receptor in rat. | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Homo sapiens (Human)) | BDBM50098776 (3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 0.430 | n/a | n/a | n/a | n/a | n/a | n/a |
Texas Biotechnology Corporation Curated by ChEMBL | Assay Description Inhibitory concentration was determined against selective Endothelin A receptor | J Med Chem 44: 1211-6 (2001) BindingDB Entry DOI: 10.7270/Q2Z89BN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50143795 (3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.680 | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Inhibitory concentration towards endothelin A receptor in rat. | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50143782 (3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.27 | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Inhibitory concentration towards endothelin A receptor in rat. | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50143791 (3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.37 | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Inhibitory concentration towards endothelin A receptor in rat. | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50058126 (2-[2-(6-Methyl-benzo[1,3]dioxol-5-yl)-acetyl]-thio...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.40 | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Inhibitory concentration towards endothelin A receptor in rat. | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Homo sapiens (Human)) | BDBM50058126 (2-[2-(6-Methyl-benzo[1,3]dioxol-5-yl)-acetyl]-thio...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 1.40 | n/a | n/a | n/a | n/a | n/a | n/a |
Texas Biotechnology Corporation Curated by ChEMBL | Assay Description Inhibitory concentration was determined against selective Endothelin A receptor | J Med Chem 44: 1211-6 (2001) BindingDB Entry DOI: 10.7270/Q2Z89BN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Homo sapiens (Human)) | BDBM50058126 (2-[2-(6-Methyl-benzo[1,3]dioxol-5-yl)-acetyl]-thio...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.40 | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Inhibitory concentration towards Endothelin A receptor in human | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50143798 (3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.47 | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Inhibitory concentration towards endothelin A receptor in rat. | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (RAT) | BDBM50143776 (2-{[3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-t...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.62 | n/a | n/a | n/a | n/a | n/a | n/a |
Encysive Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Inhibitory concentration towards endothelin A receptor in rat. | J Med Chem 47: 1969-86 (2004) Article DOI: 10.1021/jm030528p BindingDB Entry DOI: 10.7270/Q2HD7WD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Homo sapiens (Human)) | BDBM50058132 (2-[2-(6-Methyl-benzo[1,3]dioxol-5-yl)-acetyl]-thio...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 3.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Texas Biotechnology Corporation Curated by ChEMBL | Assay Description Inhibitory concentration was determined against selective Endothelin A receptor | J Med Chem 44: 1211-6 (2001) BindingDB Entry DOI: 10.7270/Q2Z89BN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Homo sapiens (Human)) | BDBM50058106 (3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 3.40 | n/a | n/a | n/a | n/a | n/a | n/a |
Texas Biotechnology Corporation Curated by ChEMBL | Assay Description Inhibitory concentration was determined against selective Endothelin A receptor | J Med Chem 44: 1211-6 (2001) BindingDB Entry DOI: 10.7270/Q2Z89BN4 | |||||||||||
More data for this Ligand-Target Pair |
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