Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM19331 (CHEMBL266063 | N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.300 | n/a | 3 | n/a | n/a | n/a | n/a |
CNRS | Assay Description Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co... | J Med Chem 50: 5790-5806 (2007) Article DOI: 10.1021/jm0704550 BindingDB Entry DOI: 10.7270/Q2HD7SZ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM19331 (CHEMBL266063 | N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.300 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Antagonist activity at human GHSR1a receptor expressed in CHO cells assessed as reduction of ghrelin-induced intracellular calcium mobilization | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM19331 (CHEMBL266063 | N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.300 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM19333 (N-[(1R)-1-{4-[(2,4-dimethoxyphenyl)methyl]-5-[2-(1...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.5 | n/a | 0.600 | n/a | n/a | n/a | n/a |
CNRS | Assay Description Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co... | J Med Chem 50: 5790-5806 (2007) Article DOI: 10.1021/jm0704550 BindingDB Entry DOI: 10.7270/Q2HD7SZ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM19331 (CHEMBL266063 | N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.600 | n/a | n/a | n/a | n/a | n/a | n/a |
Universités Montpellier 1 Curated by ChEMBL | Assay Description Displacement of 125I-His9-ghrelin from human GHSR1a expressed in LLCPK1 cells | J Med Chem 51: 689-93 (2008) Article DOI: 10.1021/jm701292s BindingDB Entry DOI: 10.7270/Q2N0168Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM19332 (N-[(1R)-2-(1H-indol-3-yl)-1-{4-[(4-methoxyphenyl)m...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.600 | n/a | 1.60 | n/a | n/a | n/a | n/a |
CNRS | Assay Description Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co... | J Med Chem 50: 5790-5806 (2007) Article DOI: 10.1021/jm0704550 BindingDB Entry DOI: 10.7270/Q2HD7SZ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50232281 ((R)-N-((4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4-t...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.700 | n/a | n/a | n/a | n/a | n/a | n/a |
Universités Montpellier 1 Curated by ChEMBL | Assay Description Displacement of 125I-His9-ghrelin from human GHSR1a expressed in LLCPK1 cells | J Med Chem 51: 689-93 (2008) Article DOI: 10.1021/jm701292s BindingDB Entry DOI: 10.7270/Q2N0168Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM19334 (N-[(1R)-1-{4-[(2,4-dimethoxyphenyl)methyl]-5-(2-ph...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.900 | n/a | 6.10 | n/a | n/a | n/a | n/a |
CNRS | Assay Description Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co... | J Med Chem 50: 5790-5806 (2007) Article DOI: 10.1021/jm0704550 BindingDB Entry DOI: 10.7270/Q2HD7SZ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50232297 ((R)-N-((4-(2,4-dimethoxybenzyl)-5-phenethyl-4H-1,2...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.10 | n/a | n/a | n/a | n/a | n/a | n/a |
Universités Montpellier 1 Curated by ChEMBL | Assay Description Displacement of 125I-His9-ghrelin from human GHSR1a expressed in LLCPK1 cells | J Med Chem 51: 689-93 (2008) Article DOI: 10.1021/jm701292s BindingDB Entry DOI: 10.7270/Q2N0168Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50232283 ((R)-N-((5-(2-(1H-indol-3-yl)ethyl)-4-(2,4-dimethox...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.80 | n/a | n/a | n/a | n/a | n/a | n/a |
Universités Montpellier 1 Curated by ChEMBL | Assay Description Displacement of 125I-His9-ghrelin from human GHSR1a expressed in LLCPK1 cells | J Med Chem 51: 689-93 (2008) Article DOI: 10.1021/jm701292s BindingDB Entry DOI: 10.7270/Q2N0168Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50227177 ((R)-pyridin-2-yl 1-(5-(2-(1H-indol-3-yl)ethyl)-4-(...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.90 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50232270 ((R)-N-((5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxyben...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.90 | n/a | n/a | n/a | n/a | n/a | n/a |
Universités Montpellier 1 Curated by ChEMBL | Assay Description Displacement of 125I-His9-ghrelin from human GHSR1a expressed in LLCPK1 cells | J Med Chem 51: 689-93 (2008) Article DOI: 10.1021/jm701292s BindingDB Entry DOI: 10.7270/Q2N0168Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50232266 ((R)-N-((4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4-t...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universités Montpellier 1 Curated by ChEMBL | Assay Description Displacement of 125I-His9-ghrelin from human GHSR1a expressed in LLCPK1 cells | J Med Chem 51: 689-93 (2008) Article DOI: 10.1021/jm701292s BindingDB Entry DOI: 10.7270/Q2N0168Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50232295 ((R)-N-((4-(2,4-dimethoxybenzyl)-5-phenethyl-4H-1,2...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Universités Montpellier 1 Curated by ChEMBL | Assay Description Displacement of 125I-His9-ghrelin from human GHSR1a expressed in LLCPK1 cells | J Med Chem 51: 689-93 (2008) Article DOI: 10.1021/jm701292s BindingDB Entry DOI: 10.7270/Q2N0168Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM19312 ((2S)-N-[(1R)-1-{4-[(2,4-dimethoxyphenyl)methyl]-5-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.60 | 11 | n/a | n/a | n/a | 7.3 | 25 |
CNRS | Assay Description Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co... | J Med Chem 50: 5790-5806 (2007) Article DOI: 10.1021/jm0704550 BindingDB Entry DOI: 10.7270/Q2HD7SZ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM19312 ((2S)-N-[(1R)-1-{4-[(2,4-dimethoxyphenyl)methyl]-5-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.60 | n/a | n/a | n/a | n/a | n/a | n/a |
Universités Montpellier 1 Curated by ChEMBL | Assay Description Displacement of 125I-His9-ghrelin from human GHSR1a expressed in LLCPK1 cells | J Med Chem 51: 689-93 (2008) Article DOI: 10.1021/jm701292s BindingDB Entry DOI: 10.7270/Q2N0168Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM19294 (2-amino-N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(1H-indo...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 6 | 4 | n/a | n/a | n/a | 7.3 | 25 |
CNRS | Assay Description Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co... | J Med Chem 50: 5790-5806 (2007) Article DOI: 10.1021/jm0704550 BindingDB Entry DOI: 10.7270/Q2HD7SZ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM19294 (2-amino-N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(1H-indo...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM19349 (N-[(1R)-2-(1H-indol-3-yl)-1-{4-[(4-methoxyphenyl)m...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 6 | 51 | n/a | n/a | n/a | n/a | n/a |
CNRS | Assay Description Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co... | J Med Chem 50: 5790-5806 (2007) Article DOI: 10.1021/jm0704550 BindingDB Entry DOI: 10.7270/Q2HD7SZ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM19294 (2-amino-N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(1H-indo...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Universités Montpellier I et II Curated by ChEMBL | Assay Description Displacement of [125I-His9]ghrelin from human GHS1a receptor expressed in LLC PK1 cells | J Med Chem 50: 1939-57 (2007) Article DOI: 10.1021/jm070024h BindingDB Entry DOI: 10.7270/Q2251HW6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM19294 (2-amino-N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(1H-indo...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
Universités Montpellier 1 Curated by ChEMBL | Assay Description Displacement of 125I-His9-ghrelin from human GHSR1a expressed in LLCPK1 cells | J Med Chem 51: 689-93 (2008) Article DOI: 10.1021/jm701292s BindingDB Entry DOI: 10.7270/Q2N0168Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM19318 (N-[(1R)-1-{4-[(2,4-dimethoxyphenyl)methyl]-5-[2-(1...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 6.5 | n/a | 5.30 | n/a | n/a | 7.3 | 25 |
CNRS | Assay Description Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co... | J Med Chem 50: 5790-5806 (2007) Article DOI: 10.1021/jm0704550 BindingDB Entry DOI: 10.7270/Q2HD7SZ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM19323 ((3R)-N-[(1R)-2-(1H-indol-3-yl)-1-{4-[(4-methoxyphe...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 7 | n/a | 36 | n/a | n/a | n/a | n/a |
CNRS | Assay Description Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co... | J Med Chem 50: 5790-5806 (2007) Article DOI: 10.1021/jm0704550 BindingDB Entry DOI: 10.7270/Q2HD7SZ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50227171 ((S)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxyb...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50232274 ((R)-N-((5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxyben...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.90 | n/a | n/a | n/a | n/a | n/a | n/a |
Universités Montpellier 1 Curated by ChEMBL | Assay Description Displacement of 125I-His9-ghrelin from human GHSR1a expressed in LLCPK1 cells | J Med Chem 51: 689-93 (2008) Article DOI: 10.1021/jm701292s BindingDB Entry DOI: 10.7270/Q2N0168Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50227180 ((R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxyb...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 8 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50227167 ((S)-N-((R)-1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-meth...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM19308 ((2S)-N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(1H-indol-3...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 9 | 6 | n/a | n/a | n/a | 7.3 | 25 |
CNRS | Assay Description Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co... | J Med Chem 50: 5790-5806 (2007) Article DOI: 10.1021/jm0704550 BindingDB Entry DOI: 10.7270/Q2HD7SZ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM19310 ((2S)-N-[(1R)-2-(1H-indol-3-yl)-1-{4-[(4-methoxyphe...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 9.5 | 13 | n/a | n/a | n/a | 7.3 | 25 |
CNRS | Assay Description Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co... | J Med Chem 50: 5790-5806 (2007) Article DOI: 10.1021/jm0704550 BindingDB Entry DOI: 10.7270/Q2HD7SZ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM19321 ((3S)-N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(1H-indol-3...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 10 | n/a | 2.5 | n/a | n/a | 7.3 | 25 |
CNRS | Assay Description Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co... | J Med Chem 50: 5790-5806 (2007) Article DOI: 10.1021/jm0704550 BindingDB Entry DOI: 10.7270/Q2HD7SZ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50232264 (CHEMBL249638 | N-((R)-(4-(4-methoxybenzyl)-5-phene...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
Universités Montpellier 1 Curated by ChEMBL | Assay Description Displacement of 125I-His9-ghrelin from human GHSR1a expressed in LLCPK1 cells | J Med Chem 51: 689-93 (2008) Article DOI: 10.1021/jm701292s BindingDB Entry DOI: 10.7270/Q2N0168Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50208662 ((R)-N-(1-(4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50208646 ((R)-N-(1-(5-(3-(1H-indol-3-yl)propyl)-4-phenethyl-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Universités Montpellier I et II Curated by ChEMBL | Assay Description Displacement of [125I-His9]ghrelin from human GHS1a receptor expressed in LLC PK1 cells | J Med Chem 50: 1939-57 (2007) Article DOI: 10.1021/jm070024h BindingDB Entry DOI: 10.7270/Q2251HW6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50208662 ((R)-N-(1-(4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Universités Montpellier I et II Curated by ChEMBL | Assay Description Displacement of [125I-His9]ghrelin from human GHS1a receptor expressed in LLC PK1 cells | J Med Chem 50: 1939-57 (2007) Article DOI: 10.1021/jm070024h BindingDB Entry DOI: 10.7270/Q2251HW6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM19326 ((2S)-N-[(1R)-2-(1H-indol-3-yl)-1-{4-[(4-methoxyphe...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 11 | 27 | n/a | n/a | n/a | n/a | n/a |
CNRS | Assay Description Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co... | J Med Chem 50: 5790-5806 (2007) Article DOI: 10.1021/jm0704550 BindingDB Entry DOI: 10.7270/Q2HD7SZ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50232263 ((R)-N-((4-(2,4-dimethoxybenzyl)-5-phenethyl-4H-1,2...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 11.8 | n/a | n/a | n/a | n/a | n/a | n/a |
Universités Montpellier 1 Curated by ChEMBL | Assay Description Displacement of 125I-His9-ghrelin from human GHSR1a expressed in LLCPK1 cells | J Med Chem 51: 689-93 (2008) Article DOI: 10.1021/jm701292s BindingDB Entry DOI: 10.7270/Q2N0168Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50208678 ((R)-N-(1-(4-(4-methoxybenzyl)-5-(3-phenylpropyl)-4...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Universités Montpellier I et II Curated by ChEMBL | Assay Description Displacement of [125I-His9]ghrelin from human GHS1a receptor expressed in LLC PK1 cells | J Med Chem 50: 1939-57 (2007) Article DOI: 10.1021/jm070024h BindingDB Entry DOI: 10.7270/Q2251HW6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50208678 ((R)-N-(1-(4-(4-methoxybenzyl)-5-(3-phenylpropyl)-4...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM19319 (N-[(1R)-1-{4-benzyl-5-[2-(1H-indol-3-yl)ethyl]-4H-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 13 | n/a | 9.90 | n/a | n/a | 7.3 | 25 |
CNRS | Assay Description Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co... | J Med Chem 50: 5790-5806 (2007) Article DOI: 10.1021/jm0704550 BindingDB Entry DOI: 10.7270/Q2HD7SZ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50232268 ((R)-N-((4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4-t...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 14 | n/a | n/a | n/a | n/a | n/a | n/a |
Universités Montpellier 1 Curated by ChEMBL | Assay Description Displacement of 125I-His9-ghrelin from human GHSR1a expressed in LLCPK1 cells | J Med Chem 51: 689-93 (2008) Article DOI: 10.1021/jm701292s BindingDB Entry DOI: 10.7270/Q2N0168Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50208670 ((R)-N-(1-(4-(2-(1H-indol-3-yl)ethyl)-5-(3-(1H-indo...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 14 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Universités Montpellier I et II Curated by ChEMBL | Assay Description Displacement of [125I-His9]ghrelin from human GHS1a receptor expressed in LLC PK1 cells | J Med Chem 50: 1939-57 (2007) Article DOI: 10.1021/jm070024h BindingDB Entry DOI: 10.7270/Q2251HW6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM19293 ((R)-N-(1-(5-(2-(1H-Indol-3-yl)ethyl)-4-benzyl-4H-1...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Universités Montpellier I et II Curated by ChEMBL | Assay Description Displacement of [125I-His9]ghrelin from human GHS1a receptor expressed in LLC PK1 cells | J Med Chem 50: 1939-57 (2007) Article DOI: 10.1021/jm070024h BindingDB Entry DOI: 10.7270/Q2251HW6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM19293 ((R)-N-(1-(5-(2-(1H-Indol-3-yl)ethyl)-4-benzyl-4H-1...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 15 | n/a | 64 | n/a | n/a | 7.3 | 25 |
CNRS | Assay Description Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co... | J Med Chem 50: 5790-5806 (2007) Article DOI: 10.1021/jm0704550 BindingDB Entry DOI: 10.7270/Q2HD7SZ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM19322 ((3S)-N-[(1R)-2-(1H-indol-3-yl)-1-{4-[(4-methoxyphe...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 16 | 10 | n/a | n/a | n/a | 7.3 | 25 |
CNRS | Assay Description Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co... | J Med Chem 50: 5790-5806 (2007) Article DOI: 10.1021/jm0704550 BindingDB Entry DOI: 10.7270/Q2HD7SZ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 5 activator 1 (Homo sapiens (Human)) | BDBM50424266 (CHEMBL2314466) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 17 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ Paris Descartes Curated by ChEMBL | Assay Description Inhibition of recombinant human CDK5/p25 after 30 mins by scintillation counting | Bioorg Med Chem Lett 23: 125-31 (2012) Article DOI: 10.1016/j.bmcl.2012.10.141 BindingDB Entry DOI: 10.7270/Q2J38TVS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50208689 ((R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(3-methoxyb...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Universités Montpellier I et II Curated by ChEMBL | Assay Description Displacement of [125I-His9]ghrelin from human GHS1a receptor expressed in LLC PK1 cells | J Med Chem 50: 1939-57 (2007) Article DOI: 10.1021/jm070024h BindingDB Entry DOI: 10.7270/Q2251HW6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50208689 ((R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(3-methoxyb...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a | n/a |
Universités Montpellier 1 Curated by ChEMBL | Assay Description Displacement of 125I-His9-ghrelin from human GHSR1a expressed in LLCPK1 cells | J Med Chem 51: 689-93 (2008) Article DOI: 10.1021/jm701292s BindingDB Entry DOI: 10.7270/Q2N0168Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM19344 (N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(1H-indol-3-yl)e...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 18 | n/a | 8.70 | n/a | n/a | n/a | n/a |
CNRS | Assay Description Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co... | J Med Chem 50: 5790-5806 (2007) Article DOI: 10.1021/jm0704550 BindingDB Entry DOI: 10.7270/Q2HD7SZ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM19350 (N-[(1R)-2-(1H-indol-3-yl)-1-{4-[(4-methoxyphenyl)m...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 18 | n/a | 390 | n/a | n/a | n/a | n/a |
CNRS | Assay Description Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co... | J Med Chem 50: 5790-5806 (2007) Article DOI: 10.1021/jm0704550 BindingDB Entry DOI: 10.7270/Q2HD7SZ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50232293 ((R)-N-((5-(2-(1H-indol-3-yl)ethyl)-4-(2,4-dimethox...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 18.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Universités Montpellier 1 Curated by ChEMBL | Assay Description Displacement of 125I-His9-ghrelin from human GHSR1a expressed in LLCPK1 cells | J Med Chem 51: 689-93 (2008) Article DOI: 10.1021/jm701292s BindingDB Entry DOI: 10.7270/Q2N0168Z | |||||||||||
More data for this Ligand-Target Pair |
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