Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50194360 ((E)-thyl-1-methyl-6,7-dihydro-1H-indol-4(5H)-one O...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 21 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter and Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assay | Bioorg Med Chem Lett 16: 5855-8 (2006) Article DOI: 10.1016/j.bmcl.2006.08.059 BindingDB Entry DOI: 10.7270/Q2057FJJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50194358 ((E)--2-methyl-6,7-dihydro-1H-indol-4(5H)-one O-phe...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 67 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter and Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assay | Bioorg Med Chem Lett 16: 5855-8 (2006) Article DOI: 10.1016/j.bmcl.2006.08.059 BindingDB Entry DOI: 10.7270/Q2057FJJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50198247 (2-(3,4-dimethylphenyl)-3-(4-methoxyphenethyl)-2-me...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 69 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter and Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 mediated ultra-rapid delayed rectifier current Ikur in human atrial cells | Bioorg Med Chem Lett 17: 282-4 (2006) Article DOI: 10.1016/j.bmcl.2006.07.007 BindingDB Entry DOI: 10.7270/Q2S18256 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50198249 (2-(3,4-dimethylphenyl)-3-(4-methoxybenzyloxy)thiaz...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 95 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter and Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 mediated ultra-rapid delayed rectifier current Ikur in human atrial cells | Bioorg Med Chem Lett 17: 282-4 (2006) Article DOI: 10.1016/j.bmcl.2006.07.007 BindingDB Entry DOI: 10.7270/Q2S18256 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50198255 (2-(3,4-dichlorophenyl)-3-(4-methoxybenzyloxy)thiaz...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 113 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter and Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 mediated ultra-rapid delayed rectifier current Ikur in human atrial cells | Bioorg Med Chem Lett 17: 282-4 (2006) Article DOI: 10.1016/j.bmcl.2006.07.007 BindingDB Entry DOI: 10.7270/Q2S18256 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50194319 ((E)-N-(4-chlorophenyl)-2-(3-ethyl-2-methyl-6,7-dih...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 130 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter & Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assay | Bioorg Med Chem Lett 16: 5859-63 (2006) Article DOI: 10.1016/j.bmcl.2006.08.057 BindingDB Entry DOI: 10.7270/Q23X868Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50194321 ((E)-2-(3-ethyl-2-methyl-6,7-dihydro-1H-indol-4(5H)...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 130 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter & Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assay | Bioorg Med Chem Lett 16: 5859-63 (2006) Article DOI: 10.1016/j.bmcl.2006.08.057 BindingDB Entry DOI: 10.7270/Q23X868Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50099574 (2-(3,4-Dimethyl-phenyl)-3-[2-(4-methoxy-phenyl)-et...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 137 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter and Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 mediated ultra-rapid delayed rectifier current Ikur in human atrial cells | Bioorg Med Chem Lett 17: 282-4 (2006) Article DOI: 10.1016/j.bmcl.2006.07.007 BindingDB Entry DOI: 10.7270/Q2S18256 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50189954 (2-(3,4-dimethylphenyl)-3-(2-(4-methoxycyclohexa-2,...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 137 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter & Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Blockade of Kv1.5 channel expressed in LTK cells by patch clamp method | Bioorg Med Chem Lett 16: 4629-32 (2006) Article DOI: 10.1016/j.bmcl.2006.06.001 BindingDB Entry DOI: 10.7270/Q2HQ3ZHZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50198261 (1-(2-(3,4-dimethylphenyl)thiazolidin-3-yl)-3-(4-me...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 150 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter and Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 mediated ultra-rapid delayed rectifier current Ikur in human atrial cells | Bioorg Med Chem Lett 17: 282-4 (2006) Article DOI: 10.1016/j.bmcl.2006.07.007 BindingDB Entry DOI: 10.7270/Q2S18256 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50198260 (1-(2-(3,4-dimethylphenyl)thiazolidin-3-yl)-2-pheno...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 162 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter and Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 mediated ultra-rapid delayed rectifier current Ikur in human atrial cells | Bioorg Med Chem Lett 17: 282-4 (2006) Article DOI: 10.1016/j.bmcl.2006.07.007 BindingDB Entry DOI: 10.7270/Q2S18256 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50198254 (2-(3,4-dimethylphenyl)-3-(2-methoxybenzyloxy)thiaz...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 177 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter and Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 mediated ultra-rapid delayed rectifier current Ikur in human atrial cells | Bioorg Med Chem Lett 17: 282-4 (2006) Article DOI: 10.1016/j.bmcl.2006.07.007 BindingDB Entry DOI: 10.7270/Q2S18256 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50198257 (2-(3,4-dichlorophenyl)-3-(3-methoxybenzyloxy)thiaz...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 179 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter and Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 mediated ultra-rapid delayed rectifier current Ikur in human atrial cells | Bioorg Med Chem Lett 17: 282-4 (2006) Article DOI: 10.1016/j.bmcl.2006.07.007 BindingDB Entry DOI: 10.7270/Q2S18256 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50195804 (1-[1-(3,4-dimethylphenyl)cyclopropyl]-2-[2-(4-meth...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 180 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter & Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assay | Bioorg Med Chem Lett 16: 6213-8 (2006) Article DOI: 10.1016/j.bmcl.2006.09.021 BindingDB Entry DOI: 10.7270/Q21V5DNX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50198256 (2-(4-chlorophenyl)-3-(4-methoxybenzyloxy)thiazolid...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 187 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter and Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 mediated ultra-rapid delayed rectifier current Ikur in human atrial cells | Bioorg Med Chem Lett 17: 282-4 (2006) Article DOI: 10.1016/j.bmcl.2006.07.007 BindingDB Entry DOI: 10.7270/Q2S18256 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50194318 ((E)-2-(3-ethyl-2-methyl-6,7-dihydro-1H-indol-4(5H)...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter & Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assay | Bioorg Med Chem Lett 16: 5859-63 (2006) Article DOI: 10.1016/j.bmcl.2006.08.057 BindingDB Entry DOI: 10.7270/Q23X868Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50198244 (2-(3,4-dichlorophenyl)-3-(2-methoxybenzyloxy)thiaz...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 204 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter and Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 mediated ultra-rapid delayed rectifier current Ikur in human atrial cells | Bioorg Med Chem Lett 17: 282-4 (2006) Article DOI: 10.1016/j.bmcl.2006.07.007 BindingDB Entry DOI: 10.7270/Q2S18256 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50198258 (3-(benzyloxy)-2-(3,4-dimethylphenyl)thiazolidin-4-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 207 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter and Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 mediated ultra-rapid delayed rectifier current Ikur in human atrial cells | Bioorg Med Chem Lett 17: 282-4 (2006) Article DOI: 10.1016/j.bmcl.2006.07.007 BindingDB Entry DOI: 10.7270/Q2S18256 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50198252 (2-(3,4-dimethylphenyl)-3-(3-methoxybenzyloxy)thiaz...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 269 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter and Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 mediated ultra-rapid delayed rectifier current Ikur in human atrial cells | Bioorg Med Chem Lett 17: 282-4 (2006) Article DOI: 10.1016/j.bmcl.2006.07.007 BindingDB Entry DOI: 10.7270/Q2S18256 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50194357 ((E)--2-methyl-6,7-dihydro-1H-indol-4(5H)-one O-4-f...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 275 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter and Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assay | Bioorg Med Chem Lett 16: 5855-8 (2006) Article DOI: 10.1016/j.bmcl.2006.08.059 BindingDB Entry DOI: 10.7270/Q2057FJJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50194325 ((E)-2-(3-ethyl-2-methyl-6,7-dihydro-1H-indol-4(5H)...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 280 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter & Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assay | Bioorg Med Chem Lett 16: 5859-63 (2006) Article DOI: 10.1016/j.bmcl.2006.08.057 BindingDB Entry DOI: 10.7270/Q23X868Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50189955 ((2-(4-methoxyphenethyl)-2H-1,2,3-triazol-4-yl)(3,4...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 294 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter & Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Blockade of Kv1.5 channel expressed in LTK cells by patch clamp method | Bioorg Med Chem Lett 16: 4629-32 (2006) Article DOI: 10.1016/j.bmcl.2006.06.001 BindingDB Entry DOI: 10.7270/Q2HQ3ZHZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50195800 (2-[2-(4-methoxyphenyl)ethyl]-1-[1-(4-methylphenyl)...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 330 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter & Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assay | Bioorg Med Chem Lett 16: 6213-8 (2006) Article DOI: 10.1016/j.bmcl.2006.09.021 BindingDB Entry DOI: 10.7270/Q21V5DNX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50195802 (1-(2,3-dimethylphenyl)-2-[2-(4-methoxyphenyl)ethyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 330 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter & Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assay | Bioorg Med Chem Lett 16: 6213-8 (2006) Article DOI: 10.1016/j.bmcl.2006.09.021 BindingDB Entry DOI: 10.7270/Q21V5DNX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50194361 ((E)--2-methyl-6,7-dihydro-1H-indol-4(5H)-one O-4-(...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 350 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter and Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assay | Bioorg Med Chem Lett 16: 5855-8 (2006) Article DOI: 10.1016/j.bmcl.2006.08.059 BindingDB Entry DOI: 10.7270/Q2057FJJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50194362 ((E)-1-(4-((3-ethyl-1,2-dimethyl-6,7-dihydro-1H-ind...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 368 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter and Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assay | Bioorg Med Chem Lett 16: 5855-8 (2006) Article DOI: 10.1016/j.bmcl.2006.08.059 BindingDB Entry DOI: 10.7270/Q2057FJJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50194324 ((E)-N-(4-acetylphenyl)-2-(2,3-diethyl-1-methyl-6,7...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 370 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter & Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assay | Bioorg Med Chem Lett 16: 5859-63 (2006) Article DOI: 10.1016/j.bmcl.2006.08.057 BindingDB Entry DOI: 10.7270/Q23X868Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50194317 ((E)-N-(4-chlorophenyl)-2-(2,3-dimethyl-6,7-dihydro...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 370 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter & Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assay | Bioorg Med Chem Lett 16: 5859-63 (2006) Article DOI: 10.1016/j.bmcl.2006.08.057 BindingDB Entry DOI: 10.7270/Q23X868Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50198248 (2-(4-chlorophenyl)-3-(3-methoxybenzyloxy)thiazolid...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 380 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter and Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 mediated ultra-rapid delayed rectifier current Ikur in human atrial cells | Bioorg Med Chem Lett 17: 282-4 (2006) Article DOI: 10.1016/j.bmcl.2006.07.007 BindingDB Entry DOI: 10.7270/Q2S18256 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50198246 (3-(4-methoxyphenethyl)-2-methyl-2-p-tolylthiazolid...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 390 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter and Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 mediated ultra-rapid delayed rectifier current Ikur in human atrial cells | Bioorg Med Chem Lett 17: 282-4 (2006) Article DOI: 10.1016/j.bmcl.2006.07.007 BindingDB Entry DOI: 10.7270/Q2S18256 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50195801 (2-[2-(4-methoxyphenyl)ethyl]-1-[1-(4-methylphenyl)...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 400 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter & Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assay | Bioorg Med Chem Lett 16: 6213-8 (2006) Article DOI: 10.1016/j.bmcl.2006.09.021 BindingDB Entry DOI: 10.7270/Q21V5DNX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50194322 ((E)-N-(4-chlorophenyl)-2-(3-ethyl-2-methyl-6,7-dih...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 440 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter & Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assay | Bioorg Med Chem Lett 16: 5859-63 (2006) Article DOI: 10.1016/j.bmcl.2006.08.057 BindingDB Entry DOI: 10.7270/Q23X868Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50198259 (3-(benzyloxy)-2-(3,4-dichlorophenyl)thiazolidin-4-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 463 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter and Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 mediated ultra-rapid delayed rectifier current Ikur in human atrial cells | Bioorg Med Chem Lett 17: 282-4 (2006) Article DOI: 10.1016/j.bmcl.2006.07.007 BindingDB Entry DOI: 10.7270/Q2S18256 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50195805 (1-[1-(4-methylphenyl)cyclopropyl]-2-(3-phenylpropy...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 480 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter & Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assay | Bioorg Med Chem Lett 16: 6213-8 (2006) Article DOI: 10.1016/j.bmcl.2006.09.021 BindingDB Entry DOI: 10.7270/Q21V5DNX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50198251 (3'-(4-methoxyphenethyl)-4-methyl-2,3-dihydrospiro[...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 487 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter and Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 mediated ultra-rapid delayed rectifier current Ikur in human atrial cells | Bioorg Med Chem Lett 17: 282-4 (2006) Article DOI: 10.1016/j.bmcl.2006.07.007 BindingDB Entry DOI: 10.7270/Q2S18256 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50198250 (1-(2-(3,4-dimethylphenyl)thiazolidin-3-yl)-2-(4-me...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 537 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter and Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 mediated ultra-rapid delayed rectifier current Ikur in human atrial cells | Bioorg Med Chem Lett 17: 282-4 (2006) Article DOI: 10.1016/j.bmcl.2006.07.007 BindingDB Entry DOI: 10.7270/Q2S18256 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50194359 ((E)--2-methyl-6,7-dihydro-1H-indol-4(5H)-one O-2-(...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 547 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter and Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assay | Bioorg Med Chem Lett 16: 5855-8 (2006) Article DOI: 10.1016/j.bmcl.2006.08.059 BindingDB Entry DOI: 10.7270/Q2057FJJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50195803 (1-(3,4-dichlorophenyl)-2-[2-(4-methoxyphenyl)ethyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 550 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter & Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assay | Bioorg Med Chem Lett 16: 6213-8 (2006) Article DOI: 10.1016/j.bmcl.2006.09.021 BindingDB Entry DOI: 10.7270/Q21V5DNX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50194323 ((E)-2-(3-ethyl-2-methyl-6,7-dihydro-1H-indol-4(5H)...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 750 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter & Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assay | Bioorg Med Chem Lett 16: 5859-63 (2006) Article DOI: 10.1016/j.bmcl.2006.08.057 BindingDB Entry DOI: 10.7270/Q23X868Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50198245 (5-chloro-3'-(4-methoxyphenethyl)-2,3-dihydrospiro[...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 812 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter and Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 mediated ultra-rapid delayed rectifier current Ikur in human atrial cells | Bioorg Med Chem Lett 17: 282-4 (2006) Article DOI: 10.1016/j.bmcl.2006.07.007 BindingDB Entry DOI: 10.7270/Q2S18256 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50198253 (3-(4-methoxybenzyloxy)-2-phenylthiazolidin-4-one |...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 924 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter and Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 mediated ultra-rapid delayed rectifier current Ikur in human atrial cells | Bioorg Med Chem Lett 17: 282-4 (2006) Article DOI: 10.1016/j.bmcl.2006.07.007 BindingDB Entry DOI: 10.7270/Q2S18256 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50198243 (3-(benzyloxy)-2-(4-chlorophenyl)thiazolidin-4-one ...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 997 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter and Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 mediated ultra-rapid delayed rectifier current Ikur in human atrial cells | Bioorg Med Chem Lett 17: 282-4 (2006) Article DOI: 10.1016/j.bmcl.2006.07.007 BindingDB Entry DOI: 10.7270/Q2S18256 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50194320 ((E)-N-(4-chlorophenyl)-2-(6,7-dihydro-1H-indol-4(5...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter & Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assay | Bioorg Med Chem Lett 16: 5859-63 (2006) Article DOI: 10.1016/j.bmcl.2006.08.057 BindingDB Entry DOI: 10.7270/Q23X868Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50194321 ((E)-2-(3-ethyl-2-methyl-6,7-dihydro-1H-indol-4(5H)...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter & Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of hERG expressed in HEK cells by whole cell patch clamp assay | Bioorg Med Chem Lett 16: 5859-63 (2006) Article DOI: 10.1016/j.bmcl.2006.08.057 BindingDB Entry DOI: 10.7270/Q23X868Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50194360 ((E)-thyl-1-methyl-6,7-dihydro-1H-indol-4(5H)-one O...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter and Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of hERG expressed in HEK cells by whole cell patch clamp assay | Bioorg Med Chem Lett 16: 5855-8 (2006) Article DOI: 10.1016/j.bmcl.2006.08.059 BindingDB Entry DOI: 10.7270/Q2057FJJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50194358 ((E)--2-methyl-6,7-dihydro-1H-indol-4(5H)-one O-phe...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Procter and Gamble Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of hERG expressed in HEK cells by whole cell patch clamp assay | Bioorg Med Chem Lett 16: 5855-8 (2006) Article DOI: 10.1016/j.bmcl.2006.08.059 BindingDB Entry DOI: 10.7270/Q2057FJJ | |||||||||||
More data for this Ligand-Target Pair |