Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Renin (Homo sapiens (Human)) | BDBM50392953 (CHEMBL2152353) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.900 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of human recombinant renin compound treated for 10 mins before substrate addition measured after 90 mins by fluorescence method | ACS Med Chem Lett 3: 754-758 (2012) Article DOI: 10.1021/ml300168e BindingDB Entry DOI: 10.7270/Q29S1S41 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Renin (Homo sapiens (Human)) | BDBM17950 ((2S,4S,5S,7S)-5-amino-N-(2-carbamoyl-2,2-dimethyle...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE MMDB PC cid PC sid PDB UniChem Patents Similars | DrugBank MMDB PDB Article PubMed | n/a | n/a | 1.5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of human recombinant renin compound treated for 10 mins before substrate addition measured after 90 mins by fluorescence method | ACS Med Chem Lett 3: 754-758 (2012) Article DOI: 10.1021/ml300168e BindingDB Entry DOI: 10.7270/Q29S1S41 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Renin (Homo sapiens (Human)) | BDBM50392953 (CHEMBL2152353) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.90 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of human plasma renin activity after 60 mins by competitive RIA | ACS Med Chem Lett 3: 754-758 (2012) Article DOI: 10.1021/ml300168e BindingDB Entry DOI: 10.7270/Q29S1S41 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Renin (Homo sapiens (Human)) | BDBM17950 ((2S,4S,5S,7S)-5-amino-N-(2-carbamoyl-2,2-dimethyle...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE MMDB PC cid PC sid PDB UniChem Patents Similars | DrugBank MMDB PDB Article PubMed | n/a | n/a | 2.90 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of human plasma renin activity after 60 mins by competitive RIA | ACS Med Chem Lett 3: 754-758 (2012) Article DOI: 10.1021/ml300168e BindingDB Entry DOI: 10.7270/Q29S1S41 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Type-1 angiotensin II receptor (Bos taurus) | BDBM50049128 (5-(1-Hydroxy-ethyl)-2-propyl-3-[2'-(2H-tetrazol-5-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 4.90 | n/a | n/a | n/a | n/a | n/a | n/a |
Sankyo Company, Ltd. Curated by ChEMBL | Assay Description In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortex | J Med Chem 39: 323-38 (1996) Article DOI: 10.1021/jm950450f BindingDB Entry DOI: 10.7270/Q28S4P18 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Tryptase beta-2 (Homo sapiens (Human)) | BDBM50184499 (CHEMBL208638 | N-(2-(3-(4-(aminomethyl)phenyl)prop...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Mochida Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of human beta tryptase | Bioorg Med Chem Lett 16: 2986-90 (2006) Article DOI: 10.1016/j.bmcl.2006.02.064 BindingDB Entry DOI: 10.7270/Q2QC0322 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (Bos taurus) | BDBM50049118 (2-Ethyl-5-(1-hydroxy-1-methyl-ethyl)-3-[2'-(2H-tet...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Sankyo Company, Ltd. Curated by ChEMBL | Assay Description In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortex | J Med Chem 39: 323-38 (1996) Article DOI: 10.1021/jm950450f BindingDB Entry DOI: 10.7270/Q28S4P18 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Renin (Macaca fascicularis) | BDBM50392953 (CHEMBL2152353) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.30 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of cynomolgus monkey plasma renin activity after 60 mins by competitive RIA | ACS Med Chem Lett 3: 754-758 (2012) Article DOI: 10.1021/ml300168e BindingDB Entry DOI: 10.7270/Q29S1S41 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (Bos taurus) | BDBM50049123 (5-Hydroxymethyl-2-propyl-3-[2'-(2H-tetrazol-5-yl)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 6.90 | n/a | n/a | n/a | n/a | n/a | n/a |
Sankyo Company, Ltd. Curated by ChEMBL | Assay Description In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortex | J Med Chem 39: 323-38 (1996) Article DOI: 10.1021/jm950450f BindingDB Entry DOI: 10.7270/Q28S4P18 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Renin (Macaca fascicularis) | BDBM17950 ((2S,4S,5S,7S)-5-amino-N-(2-carbamoyl-2,2-dimethyle...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE MMDB PC cid PC sid PDB UniChem Patents Similars | MMDB PDB Article PubMed | n/a | n/a | 8 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of cynomolgus monkey plasma renin activity after 60 mins by competitive RIA | ACS Med Chem Lett 3: 754-758 (2012) Article DOI: 10.1021/ml300168e BindingDB Entry DOI: 10.7270/Q29S1S41 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Type-1 angiotensin II receptor (Bos taurus) | BDBM50241364 (4-(1-hydroxy-1-methylethyl)-2-propyl-1-{[2'-(1H-te...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | n/a | n/a | 8.10 | n/a | n/a | n/a | n/a | n/a | n/a |
Sankyo Company, Ltd. Curated by ChEMBL | Assay Description In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortex | J Med Chem 39: 323-38 (1996) Article DOI: 10.1021/jm950450f BindingDB Entry DOI: 10.7270/Q28S4P18 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Type-1 angiotensin II receptor (Bos taurus) | BDBM50049107 (2-Propyl-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmet...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.10 | n/a | n/a | n/a | n/a | n/a | n/a |
Sankyo Company, Ltd. Curated by ChEMBL | Assay Description In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortex | J Med Chem 39: 323-38 (1996) Article DOI: 10.1021/jm950450f BindingDB Entry DOI: 10.7270/Q28S4P18 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (Bos taurus) | BDBM50049109 (2-Butyl-5-(1-hydroxy-1-methyl-ethyl)-3-[2'-(2H-tet...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 9.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Sankyo Company, Ltd. Curated by ChEMBL | Assay Description In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortex | J Med Chem 39: 323-38 (1996) Article DOI: 10.1021/jm950450f BindingDB Entry DOI: 10.7270/Q28S4P18 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (Bos taurus) | BDBM50049124 (5-Methyl-2-propyl-3-[2'-(1H-tetrazol-5-yl)-bipheny...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
Sankyo Company, Ltd. Curated by ChEMBL | Assay Description In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortex | J Med Chem 39: 323-38 (1996) Article DOI: 10.1021/jm950450f BindingDB Entry DOI: 10.7270/Q28S4P18 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (Bos taurus) | BDBM50049116 (5-Ethyl-2-propyl-3-(2'-tetrazol-1-yl-biphenyl-4-yl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
Sankyo Company, Ltd. Curated by ChEMBL | Assay Description In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortex | J Med Chem 39: 323-38 (1996) Article DOI: 10.1021/jm950450f BindingDB Entry DOI: 10.7270/Q28S4P18 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (Bos taurus) | BDBM50006909 (2-Butyl-5-chloro-3-[2'-(1H-tetrazol-5-yl)-biphenyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Patents Similars | Article | n/a | n/a | 22 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of [125l]-All binding to bovine adrenal cortex | Bioorg Med Chem Lett 4: 177-182 (1994) Article DOI: 10.1016/S0960-894X(01)81143-4 BindingDB Entry DOI: 10.7270/Q2BG2NZQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (Bos taurus) | BDBM50006909 (2-Butyl-5-chloro-3-[2'-(1H-tetrazol-5-yl)-biphenyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 22 | n/a | n/a | n/a | n/a | n/a | n/a |
Sankyo Company, Ltd. Curated by ChEMBL | Assay Description In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortex | J Med Chem 39: 323-38 (1996) Article DOI: 10.1021/jm950450f BindingDB Entry DOI: 10.7270/Q28S4P18 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (Bos taurus) | BDBM50049112 (3-(2'-Carboxy-biphenyl-4-ylmethyl)-5-(1-hydroxy-et...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 28 | n/a | n/a | n/a | n/a | n/a | n/a |
Sankyo Company, Ltd. Curated by ChEMBL | Assay Description In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortex | J Med Chem 39: 323-38 (1996) Article DOI: 10.1021/jm950450f BindingDB Entry DOI: 10.7270/Q28S4P18 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (Bos taurus) | BDBM50049132 (3-(2'-Carboxy-biphenyl-4-ylmethyl)-5-(1-hydroxy-1-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 28 | n/a | n/a | n/a | n/a | n/a | n/a |
Sankyo Company, Ltd. Curated by ChEMBL | Assay Description In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortex | J Med Chem 39: 323-38 (1996) Article DOI: 10.1021/jm950450f BindingDB Entry DOI: 10.7270/Q28S4P18 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (Bos taurus) | BDBM50049122 (2-Butyl-3-(2'-carboxy-biphenyl-4-ylmethyl)-5-(1-hy...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
Sankyo Company, Ltd. Curated by ChEMBL | Assay Description In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortex | J Med Chem 39: 323-38 (1996) Article DOI: 10.1021/jm950450f BindingDB Entry DOI: 10.7270/Q28S4P18 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (Bos taurus) | BDBM50049117 (3-(2'-Carboxy-biphenyl-4-ylmethyl)-2-ethyl-5-(1-hy...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 37 | n/a | n/a | n/a | n/a | n/a | n/a |
Sankyo Company, Ltd. Curated by ChEMBL | Assay Description In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortex | J Med Chem 39: 323-38 (1996) Article DOI: 10.1021/jm950450f BindingDB Entry DOI: 10.7270/Q28S4P18 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (Bos taurus) | BDBM50049130 (5-Isopropyl-2-propyl-3-[2'-(1H-tetrazol-5-yl)-biph...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 46 | n/a | n/a | n/a | n/a | n/a | n/a |
Sankyo Company, Ltd. Curated by ChEMBL | Assay Description In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortex | J Med Chem 39: 323-38 (1996) Article DOI: 10.1021/jm950450f BindingDB Entry DOI: 10.7270/Q28S4P18 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (Bos taurus) | BDBM50049113 (5-Isopropenyl-2-propyl-3-[2'-(2H-tetrazol-5-yl)-bi...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 50 | n/a | n/a | n/a | n/a | n/a | n/a |
Sankyo Company, Ltd. Curated by ChEMBL | Assay Description In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortex | J Med Chem 39: 323-38 (1996) Article DOI: 10.1021/jm950450f BindingDB Entry DOI: 10.7270/Q28S4P18 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (Bos taurus) | BDBM50049106 (3-(2'-Carboxy-biphenyl-4-ylmethyl)-5-(1-hydroxy-1-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 51 | n/a | n/a | n/a | n/a | n/a | n/a |
Sankyo Company, Ltd. Curated by ChEMBL | Assay Description In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortex | J Med Chem 39: 323-38 (1996) Article DOI: 10.1021/jm950450f BindingDB Entry DOI: 10.7270/Q28S4P18 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Tryptase beta-2 (Homo sapiens (Human)) | BDBM16127 (2,2 -methanediylbis(1H-benzimidazole-6-carboximida...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 51 | n/a | n/a | n/a | n/a | n/a | n/a |
Mochida Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of human beta tryptase | Bioorg Med Chem Lett 16: 2986-90 (2006) Article DOI: 10.1016/j.bmcl.2006.02.064 BindingDB Entry DOI: 10.7270/Q2QC0322 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (Bos taurus) | BDBM50049108 (3-(2'-Carboxy-biphenyl-4-ylmethyl)-5-hydroxymethyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 58 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of [125l]-All binding to bovine adrenal cortex | Bioorg Med Chem Lett 4: 177-182 (1994) Article DOI: 10.1016/S0960-894X(01)81143-4 BindingDB Entry DOI: 10.7270/Q2BG2NZQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (Bos taurus) | BDBM50049108 (3-(2'-Carboxy-biphenyl-4-ylmethyl)-5-hydroxymethyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 58 | n/a | n/a | n/a | n/a | n/a | n/a |
Sankyo Company, Ltd. Curated by ChEMBL | Assay Description In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortex | J Med Chem 39: 323-38 (1996) Article DOI: 10.1021/jm950450f BindingDB Entry DOI: 10.7270/Q28S4P18 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (Bos taurus) | BDBM50049126 (3-(2'-Carboxy-biphenyl-4-ylmethyl)-2-propyl-3H-imi...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 60 | n/a | n/a | n/a | n/a | n/a | n/a |
Sankyo Company, Ltd. Curated by ChEMBL | Assay Description In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortex | J Med Chem 39: 323-38 (1996) Article DOI: 10.1021/jm950450f BindingDB Entry DOI: 10.7270/Q28S4P18 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (Bos taurus) | BDBM50282291 (2-Butyl-3-(2'-carboxy-biphenyl-4-ylmethyl)-5-hydro...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article | n/a | n/a | 65 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of [125l]-All binding to bovine adrenal cortex | Bioorg Med Chem Lett 4: 177-182 (1994) Article DOI: 10.1016/S0960-894X(01)81143-4 BindingDB Entry DOI: 10.7270/Q2BG2NZQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Tryptase beta-2 (Homo sapiens (Human)) | BDBM50184504 (CHEMBL380668 | N-(2-(3-(4-(aminomethyl)phenyl)prop...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 73 | n/a | n/a | n/a | n/a | n/a | n/a |
Mochida Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of human beta tryptase | Bioorg Med Chem Lett 16: 2986-90 (2006) Article DOI: 10.1016/j.bmcl.2006.02.064 BindingDB Entry DOI: 10.7270/Q2QC0322 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (Bos taurus) | BDBM50049103 (3-(2'-Carboxy-biphenyl-4-ylmethyl)-5-ethyl-2-propy...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
Sankyo Company, Ltd. Curated by ChEMBL | Assay Description In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortex | J Med Chem 39: 323-38 (1996) Article DOI: 10.1021/jm950450f BindingDB Entry DOI: 10.7270/Q28S4P18 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (Bos taurus) | BDBM50049110 (2-Propyl-1-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmet...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
Sankyo Company, Ltd. Curated by ChEMBL | Assay Description In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortex | J Med Chem 39: 323-38 (1996) Article DOI: 10.1021/jm950450f BindingDB Entry DOI: 10.7270/Q28S4P18 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (Bos taurus) | BDBM50049129 (3-(2'-Carboxy-biphenyl-4-ylmethyl)-5-(1-ethyl-1-hy...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 110 | n/a | n/a | n/a | n/a | n/a | n/a |
Sankyo Company, Ltd. Curated by ChEMBL | Assay Description In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortex | J Med Chem 39: 323-38 (1996) Article DOI: 10.1021/jm950450f BindingDB Entry DOI: 10.7270/Q28S4P18 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (Bos taurus) | BDBM50049104 (3-(2'-Carboxy-biphenyl-4-ylmethyl)-5-methyl-2-prop...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 110 | n/a | n/a | n/a | n/a | n/a | n/a |
Sankyo Company, Ltd. Curated by ChEMBL | Assay Description In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortex | J Med Chem 39: 323-38 (1996) Article DOI: 10.1021/jm950450f BindingDB Entry DOI: 10.7270/Q28S4P18 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (Bos taurus) | BDBM50009714 (CHEMBL191 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazol-5...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 120 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of [125l]-All binding to bovine adrenal cortex | Bioorg Med Chem Lett 4: 177-182 (1994) Article DOI: 10.1016/S0960-894X(01)81143-4 BindingDB Entry DOI: 10.7270/Q2BG2NZQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Tryptase beta-2 (Homo sapiens (Human)) | BDBM50184505 (CHEMBL415045 | N-(2-((3-(4-(aminomethyl)phenyl)pro...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 120 | n/a | n/a | n/a | n/a | n/a | n/a |
Mochida Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of human beta tryptase | Bioorg Med Chem Lett 16: 2986-90 (2006) Article DOI: 10.1016/j.bmcl.2006.02.064 BindingDB Entry DOI: 10.7270/Q2QC0322 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (Bos taurus) | BDBM50009714 (CHEMBL191 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazol-5...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 120 | n/a | n/a | n/a | n/a | n/a | n/a |
Sankyo Company, Ltd. Curated by ChEMBL | Assay Description In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortex | J Med Chem 39: 323-38 (1996) Article DOI: 10.1021/jm950450f BindingDB Entry DOI: 10.7270/Q28S4P18 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (Bos taurus) | BDBM50009505 (2-Butyl-3-(2'-carboxy-biphenyl-4-ylmethyl)-5-chlor...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 130 | n/a | n/a | n/a | n/a | n/a | n/a |
Sankyo Company, Ltd. Curated by ChEMBL | Assay Description In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortex | J Med Chem 39: 323-38 (1996) Article DOI: 10.1021/jm950450f BindingDB Entry DOI: 10.7270/Q28S4P18 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (Bos taurus) | BDBM50009505 (2-Butyl-3-(2'-carboxy-biphenyl-4-ylmethyl)-5-chlor...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article | n/a | n/a | 130 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of [125l]-All binding to bovine adrenal cortex | Bioorg Med Chem Lett 4: 177-182 (1994) Article DOI: 10.1016/S0960-894X(01)81143-4 BindingDB Entry DOI: 10.7270/Q2BG2NZQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Tryptase beta-2 (Homo sapiens (Human)) | BDBM50184508 (CHEMBL207193 | N-(2-(3-(4-(aminomethyl)phenyl)prop...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 130 | n/a | n/a | n/a | n/a | n/a | n/a |
Mochida Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of human beta tryptase | Bioorg Med Chem Lett 16: 2986-90 (2006) Article DOI: 10.1016/j.bmcl.2006.02.064 BindingDB Entry DOI: 10.7270/Q2QC0322 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (Bos taurus) | BDBM50282290 (3-(2'-Carboxy-biphenyl-4-ylmethyl)-2-ethyl-5-hydro...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 150 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of [125l]-All binding to bovine adrenal cortex | Bioorg Med Chem Lett 4: 177-182 (1994) Article DOI: 10.1016/S0960-894X(01)81143-4 BindingDB Entry DOI: 10.7270/Q2BG2NZQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Tryptase beta-2 (Homo sapiens (Human)) | BDBM50184512 (CHEMBL438621 | N-(2-(3-(4-(aminomethyl)phenyl)prop...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 190 | n/a | n/a | n/a | n/a | n/a | n/a |
Mochida Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of human beta tryptase | Bioorg Med Chem Lett 16: 2986-90 (2006) Article DOI: 10.1016/j.bmcl.2006.02.064 BindingDB Entry DOI: 10.7270/Q2QC0322 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Tryptase beta-2 (Homo sapiens (Human)) | BDBM50184513 (CHEMBL208526 | N-(2-(3-(4-(aminomethyl)phenyl)prop...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
Mochida Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of human beta tryptase | Bioorg Med Chem Lett 16: 2986-90 (2006) Article DOI: 10.1016/j.bmcl.2006.02.064 BindingDB Entry DOI: 10.7270/Q2QC0322 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (Bos taurus) | BDBM50049115 (5-(1-Hydroxy-1-methyl-ethyl)-2-propyl-3-[2'-(2H-te...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
Sankyo Company, Ltd. Curated by ChEMBL | Assay Description In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortex | J Med Chem 39: 323-38 (1996) Article DOI: 10.1021/jm950450f BindingDB Entry DOI: 10.7270/Q28S4P18 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Tryptase beta-2 (Homo sapiens (Human)) | BDBM50184514 (CHEMBL379328 | N-(2-(3-(4-(aminomethyl)phenyl)prop...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 210 | n/a | n/a | n/a | n/a | n/a | n/a |
Mochida Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of human beta tryptase | Bioorg Med Chem Lett 16: 2986-90 (2006) Article DOI: 10.1016/j.bmcl.2006.02.064 BindingDB Entry DOI: 10.7270/Q2QC0322 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (Bos taurus) | BDBM50049125 (3-(2'-Carboxy-biphenyl-4-ylmethyl)-5-isopropenyl-2...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 270 | n/a | n/a | n/a | n/a | n/a | n/a |
Sankyo Company, Ltd. Curated by ChEMBL | Assay Description In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortex | J Med Chem 39: 323-38 (1996) Article DOI: 10.1021/jm950450f BindingDB Entry DOI: 10.7270/Q28S4P18 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Tryptase beta-2 (Homo sapiens (Human)) | BDBM50184500 (CHEMBL377266 | N-(2-(3-(4-(aminomethyl)phenyl)prop...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 270 | n/a | n/a | n/a | n/a | n/a | n/a |
Mochida Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of human beta tryptase | Bioorg Med Chem Lett 16: 2986-90 (2006) Article DOI: 10.1016/j.bmcl.2006.02.064 BindingDB Entry DOI: 10.7270/Q2QC0322 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (Bos taurus) | BDBM50049119 (1-(2'-Carboxy-biphenyl-4-ylmethyl)-2-propyl-1H-imi...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 320 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of [125l]-All binding to bovine adrenal cortex | Bioorg Med Chem Lett 4: 177-182 (1994) Article DOI: 10.1016/S0960-894X(01)81143-4 BindingDB Entry DOI: 10.7270/Q2BG2NZQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (Bos taurus) | BDBM50049119 (1-(2'-Carboxy-biphenyl-4-ylmethyl)-2-propyl-1H-imi...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 320 | n/a | n/a | n/a | n/a | n/a | n/a |
Sankyo Company, Ltd. Curated by ChEMBL | Assay Description In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortex | J Med Chem 39: 323-38 (1996) Article DOI: 10.1021/jm950450f BindingDB Entry DOI: 10.7270/Q28S4P18 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (Bos taurus) | BDBM50049111 (3-(2'-Carboxy-biphenyl-4-ylmethyl)-5-isopropyl-2-p...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 360 | n/a | n/a | n/a | n/a | n/a | n/a |
Sankyo Company, Ltd. Curated by ChEMBL | Assay Description In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortex | J Med Chem 39: 323-38 (1996) Article DOI: 10.1021/jm950450f BindingDB Entry DOI: 10.7270/Q28S4P18 | |||||||||||
More data for this Ligand-Target Pair |
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