Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50434389 (CHEMBL2387288) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50437067 (CHEMBL2403550) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from recombinant rhesus monkey histamine H3 receptor transfected in CHO cell membranes after 1 hr by scin... | Bioorg Med Chem Lett 23: 4044-7 (2013) Article DOI: 10.1016/j.bmcl.2013.05.068 BindingDB Entry DOI: 10.7270/Q28C9XN0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM50437067 (CHEMBL2403550) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from recombinant rat histamine H3 receptor transfected in CHO cell membranes after 1 hr by scintillation ... | Bioorg Med Chem Lett 23: 4044-7 (2013) Article DOI: 10.1016/j.bmcl.2013.05.068 BindingDB Entry DOI: 10.7270/Q28C9XN0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50434405 (CHEMBL2387306) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50434382 (CHEMBL2387309) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 3.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50434401 (CHEMBL2387314) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50434400 (CHEMBL2387315) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50434392 (CHEMBL2387285) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50434387 (CHEMBL2387290) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50437068 (CHEMBL2403549) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from recombinant rhesus monkey histamine H3 receptor transfected in CHO cell membranes after 1 hr by scin... | Bioorg Med Chem Lett 23: 4044-7 (2013) Article DOI: 10.1016/j.bmcl.2013.05.068 BindingDB Entry DOI: 10.7270/Q28C9XN0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50434388 (CHEMBL2387289) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 8.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM50437068 (CHEMBL2403549) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 11 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from recombinant rat histamine H3 receptor transfected in CHO cell membranes after 1 hr by scintillation ... | Bioorg Med Chem Lett 23: 4044-7 (2013) Article DOI: 10.1016/j.bmcl.2013.05.068 BindingDB Entry DOI: 10.7270/Q28C9XN0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50434393 (CHEMBL2387284) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 11 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50434399 (CHEMBL2387316) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 11 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50434397 (CHEMBL2387318) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 11 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50434396 (CHEMBL2387319) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50434381 (CHEMBL2387310) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 16 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM50435303 (CHEMBL2391167) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 17 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from rat histamine H3 receptor | Bioorg Med Chem Lett 23: 3421-6 (2013) Article DOI: 10.1016/j.bmcl.2013.03.081 BindingDB Entry DOI: 10.7270/Q2HH6MGF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50434383 (CHEMBL2387307) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 18 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50434404 (CHEMBL2387311) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 19 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50434403 (CHEMBL2387312) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 22 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50434394 (CHEMBL2387283) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 23 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50434398 (CHEMBL2387317) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 26 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50434386 (CHEMBL2387291) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 29 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM50434382 (CHEMBL2387309) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 33 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rat histamine H3 receptor transfected in CHO cells after 1 hr by scintillation counting analy... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50434395 (CHEMBL2387282) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 34 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50434391 (CHEMBL2387286) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 36 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM50434381 (CHEMBL2387310) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rat histamine H3 receptor transfected in CHO cells after 1 hr by scintillation counting analy... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50434402 (CHEMBL2387313) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 43 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50434385 (CHEMBL2387292) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 47 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM50435304 (CHEMBL2391166) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 55 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from rat histamine H3 receptor | Bioorg Med Chem Lett 23: 3421-6 (2013) Article DOI: 10.1016/j.bmcl.2013.03.081 BindingDB Entry DOI: 10.7270/Q2HH6MGF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM50437066 (CHEMBL2403551) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 74 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from recombinant rat histamine H3 receptor transfected in CHO cell membranes after 1 hr by scintillation ... | Bioorg Med Chem Lett 23: 4044-7 (2013) Article DOI: 10.1016/j.bmcl.2013.05.068 BindingDB Entry DOI: 10.7270/Q28C9XN0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50434390 (CHEMBL2387287) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM50437069 (CHEMBL2403548) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 93 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from recombinant rat histamine H3 receptor transfected in CHO cell membranes after 1 hr by scintillation ... | Bioorg Med Chem Lett 23: 4044-7 (2013) Article DOI: 10.1016/j.bmcl.2013.05.068 BindingDB Entry DOI: 10.7270/Q28C9XN0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50434384 (CHEMBL2387293) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 115 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50437069 (CHEMBL2403548) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 121 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from recombinant rhesus monkey histamine H3 receptor transfected in CHO cell membranes after 1 hr by scin... | Bioorg Med Chem Lett 23: 4044-7 (2013) Article DOI: 10.1016/j.bmcl.2013.05.068 BindingDB Entry DOI: 10.7270/Q28C9XN0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM50434383 (CHEMBL2387307) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 135 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rat histamine H3 receptor transfected in CHO cells after 1 hr by scintillation counting analy... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50437066 (CHEMBL2403551) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 147 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from recombinant rhesus monkey histamine H3 receptor transfected in CHO cell membranes after 1 hr by scin... | Bioorg Med Chem Lett 23: 4044-7 (2013) Article DOI: 10.1016/j.bmcl.2013.05.068 BindingDB Entry DOI: 10.7270/Q28C9XN0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Homo sapiens (Human)) | BDBM50435303 (CHEMBL2391167) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >9.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Binding affinity to human histamine H1 receptor | Bioorg Med Chem Lett 23: 3421-6 (2013) Article DOI: 10.1016/j.bmcl.2013.03.081 BindingDB Entry DOI: 10.7270/Q2HH6MGF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Homo sapiens (Human)) | BDBM50435304 (CHEMBL2391166) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >9.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Binding affinity to human histamine H1 receptor | Bioorg Med Chem Lett 23: 3421-6 (2013) Article DOI: 10.1016/j.bmcl.2013.03.081 BindingDB Entry DOI: 10.7270/Q2HH6MGF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
11-beta-hydroxysteroid dehydrogenase 1 (Mus musculus (mouse)) | BDBM50433406 (CHEMBL2380643) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi R&D Curated by ChEMBL | Assay Description Inhibition of mouse recombinant 11beta-HSD1 by scintillation proximity assay | Bioorg Med Chem Lett 23: 2414-21 (2013) Article DOI: 10.1016/j.bmcl.2013.02.018 BindingDB Entry DOI: 10.7270/Q2NV9KMN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
11-beta-hydroxysteroid dehydrogenase 1 (Mus musculus (mouse)) | BDBM50433404 (CHEMBL2380641) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi R&D Curated by ChEMBL | Assay Description Inhibition of mouse recombinant 11beta-HSD1 by scintillation proximity assay | Bioorg Med Chem Lett 23: 2414-21 (2013) Article DOI: 10.1016/j.bmcl.2013.02.018 BindingDB Entry DOI: 10.7270/Q2NV9KMN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
11-beta-hydroxysteroid dehydrogenase 1 (Mus musculus (mouse)) | BDBM50433405 (CHEMBL2380642) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi R&D Curated by ChEMBL | Assay Description Inhibition of mouse recombinant 11beta-HSD1 by scintillation proximity assay | Bioorg Med Chem Lett 23: 2414-21 (2013) Article DOI: 10.1016/j.bmcl.2013.02.018 BindingDB Entry DOI: 10.7270/Q2NV9KMN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50499970 (CHEMBL3741505) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi-aventis R&D Curated by ChEMBL | Assay Description Inhibition of DGAT-1 in human Chang cells assessed as lipid level after 6 hrs in presence of substrate [14C]glycerol by HPLC analysis | Bioorg Med Chem Lett 26: 25-32 (2016) Article DOI: 10.1016/j.bmcl.2015.11.046 BindingDB Entry DOI: 10.7270/Q2Z89GDN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
11-beta-hydroxysteroid dehydrogenase 1 (Homo sapiens (Human)) | BDBM50433412 (CHEMBL2380649) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi R&D Curated by ChEMBL | Assay Description Inhibition of human recombinant 11beta-HSD1 by scintillation proximity assay | Bioorg Med Chem Lett 23: 2414-21 (2013) Article DOI: 10.1016/j.bmcl.2013.02.018 BindingDB Entry DOI: 10.7270/Q2NV9KMN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50499970 (CHEMBL3741505) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi-aventis R&D Curated by ChEMBL | Assay Description Inhibition of recombinant human DGAT-1 using 1,2,di(cis-9-octadecenoyl)-sn-glycerol as substrate by Microbeta counter | Bioorg Med Chem Lett 26: 25-32 (2016) Article DOI: 10.1016/j.bmcl.2015.11.046 BindingDB Entry DOI: 10.7270/Q2Z89GDN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
11-beta-hydroxysteroid dehydrogenase 1 (Homo sapiens (Human)) | BDBM50433411 (CHEMBL2380648) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi R&D Curated by ChEMBL | Assay Description Inhibition of human recombinant 11beta-HSD1 by scintillation proximity assay | Bioorg Med Chem Lett 23: 2414-21 (2013) Article DOI: 10.1016/j.bmcl.2013.02.018 BindingDB Entry DOI: 10.7270/Q2NV9KMN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
11-beta-hydroxysteroid dehydrogenase 1 (Homo sapiens (Human)) | BDBM50433400 (CHEMBL2380637) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi R&D Curated by ChEMBL | Assay Description Inhibition of human recombinant 11beta-HSD1 by scintillation proximity assay | Bioorg Med Chem Lett 23: 2414-21 (2013) Article DOI: 10.1016/j.bmcl.2013.02.018 BindingDB Entry DOI: 10.7270/Q2NV9KMN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
11-beta-hydroxysteroid dehydrogenase 1 (Mus musculus (mouse)) | BDBM50433403 (CHEMBL2380640) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi R&D Curated by ChEMBL | Assay Description Inhibition of mouse recombinant 11beta-HSD1 by scintillation proximity assay | Bioorg Med Chem Lett 23: 2414-21 (2013) Article DOI: 10.1016/j.bmcl.2013.02.018 BindingDB Entry DOI: 10.7270/Q2NV9KMN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
11-beta-hydroxysteroid dehydrogenase 1 (Mus musculus (mouse)) | BDBM50433407 (CHEMBL2380644) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi R&D Curated by ChEMBL | Assay Description Inhibition of mouse recombinant 11beta-HSD1 by scintillation proximity assay | Bioorg Med Chem Lett 23: 2414-21 (2013) Article DOI: 10.1016/j.bmcl.2013.02.018 BindingDB Entry DOI: 10.7270/Q2NV9KMN | |||||||||||
More data for this Ligand-Target Pair |
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