Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sodium-dependent dopamine transporter (Rattus norvegicus (rat)) | BDBM22418 (Cocaine | Cocaine (-) | methyl (1R,2R,3S,5S)-3-(be...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase DrugBank KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article | 280 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity to inhibit [3H]mazindol binding in rat corpus striatum P2 synaptosomes | Bioorg Med Chem Lett 4: 303-308 (1994) Article DOI: 10.1016/S0960-894X(01)80133-5 BindingDB Entry DOI: 10.7270/Q2F47PNG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent dopamine transporter (Rattus norvegicus (rat)) | BDBM50283380 (3-Benzoyloxy-8-carboxymethyl-8-aza-bicyclo[3.2.1]o...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | 380 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity to inhibit [3H]mazindol binding in rat corpus striatum P2 synaptosomes | Bioorg Med Chem Lett 4: 303-308 (1994) Article DOI: 10.1016/S0960-894X(01)80133-5 BindingDB Entry DOI: 10.7270/Q2F47PNG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent dopamine transporter (Rattus norvegicus (rat)) | BDBM50283377 (3-Benzoyloxy-8-methoxycarbonylmethyl-8-aza-bicyclo...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | 480 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity to inhibit [3H]mazindol binding in rat corpus striatum P2 synaptosomes | Bioorg Med Chem Lett 4: 303-308 (1994) Article DOI: 10.1016/S0960-894X(01)80133-5 BindingDB Entry DOI: 10.7270/Q2F47PNG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent dopamine transporter (Rattus norvegicus (rat)) | BDBM50283376 (3-Benzoyloxy-8-(2-hydroxy-ethyl)-8-aza-bicyclo[3.2...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | 700 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity to inhibit [3H]mazindol binding in rat corpus striatum P2 synaptosomes | Bioorg Med Chem Lett 4: 303-308 (1994) Article DOI: 10.1016/S0960-894X(01)80133-5 BindingDB Entry DOI: 10.7270/Q2F47PNG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent dopamine transporter (Rattus norvegicus (rat)) | BDBM50283381 (3-Benzoyloxy-8-nitro-8-aza-bicyclo[3.2.1]octane-2-...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | 7.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity to inhibit [3H]mazindol binding in rat corpus striatum P2 synaptosomes | Bioorg Med Chem Lett 4: 303-308 (1994) Article DOI: 10.1016/S0960-894X(01)80133-5 BindingDB Entry DOI: 10.7270/Q2F47PNG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent dopamine transporter (Rattus norvegicus (rat)) | BDBM50283378 (Benzoic acid 5-oxo-6,7-diaza-tricyclo[5.3.0.0*4,8*...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | 4.49E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity to inhibit [3H]mazindol binding in rat corpus striatum P2 synaptosomes | Bioorg Med Chem Lett 4: 303-308 (1994) Article DOI: 10.1016/S0960-894X(01)80133-5 BindingDB Entry DOI: 10.7270/Q2F47PNG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent dopamine transporter (Rattus norvegicus (rat)) | BDBM50283375 (3-Benzoyloxy-8-nitroso-8-aza-bicyclo[3.2.1]octane-...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | 9.95E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity to inhibit [3H]mazindol binding in rat corpus striatum P2 synaptosomes | Bioorg Med Chem Lett 4: 303-308 (1994) Article DOI: 10.1016/S0960-894X(01)80133-5 BindingDB Entry DOI: 10.7270/Q2F47PNG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent dopamine transporter (Rattus norvegicus (rat)) | BDBM50283379 (8-Acetylamino-3-benzoyloxy-8-aza-bicyclo[3.2.1]oct...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | >1.00E+6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity to inhibit [3H]mazindol binding in rat corpus striatum P2 synaptosomes | Bioorg Med Chem Lett 4: 303-308 (1994) Article DOI: 10.1016/S0960-894X(01)80133-5 BindingDB Entry DOI: 10.7270/Q2F47PNG | |||||||||||
More data for this Ligand-Target Pair |