Found 45 hits with Last Name = 'yasuda-kamatani' and Initial = 'y' Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
Glutamate receptor ionotropic, kainate 1
(RAT) | BDBM50002369
((2S-(2alpha,3beta,4beta))-2-carboxy-4-(1-methyleth...)Show SMILES CC(=C)[C@H]1CN[C@@H]([C@H]1CC(O)=O)C(O)=O |r| Show InChI InChI=1S/C10H15NO4/c1-5(2)7-4-11-9(10(14)15)6(7)3-8(12)13/h6-7,9,11H,1,3-4H2,2H3,(H,12,13)(H,14,15)/t6-,7+,9-/m0/s1 | PDB
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| PDB Article PubMed
| 2.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Suntory Institute for Bioorganic Research
Curated by PDSP Ki Database
| |
Mol Pharmacol 53: 195-201 (1998)
Article DOI: 10.1124/mol.53.2.195 BindingDB Entry DOI: 10.7270/Q2RF5SJH |
More data for this Ligand-Target Pair | 3D Structure (crystal) |
Glutamate receptor ionotropic, NMDA 1
(RAT) | BDBM50004899
((1R,2S)-2-((S)-Amino-carboxy-methyl)-cyclopropanec...)Show InChI InChI=1S/C6H9NO4/c7-4(6(10)11)2-1-3(2)5(8)9/h2-4H,1,7H2,(H,8,9)(H,10,11)/t2-,3+,4-/m0/s1 | PDB
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| 8 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Suntory Institute for Bioorganic Research
Curated by PDSP Ki Database
| |
Mol Pharmacol 53: 195-201 (1998)
Article DOI: 10.1124/mol.53.2.195 BindingDB Entry DOI: 10.7270/Q2RF5SJH |
More data for this Ligand-Target Pair | |
Glutamate receptor ionotropic, kainate 1
(RAT) | BDBM50013055
(2-aminopentanedioateglutamate | L-Glutamate | glut...)Show InChI InChI=1S/C5H9NO4/c6-3(5(9)10)1-2-4(7)8/h3H,1-2,6H2,(H,7,8)(H,9,10)/p-2 | PDB
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| 118 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Suntory Institute for Bioorganic Research
Curated by PDSP Ki Database
| |
Mol Pharmacol 53: 195-201 (1998)
Article DOI: 10.1124/mol.53.2.195 BindingDB Entry DOI: 10.7270/Q2RF5SJH |
More data for this Ligand-Target Pair | |
Glutamate receptor 3
(RAT) | BDBM50013055
(2-aminopentanedioateglutamate | L-Glutamate | glut...)Show InChI InChI=1S/C5H9NO4/c6-3(5(9)10)1-2-4(7)8/h3H,1-2,6H2,(H,7,8)(H,9,10)/p-2 | PDB
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| 118 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Suntory Institute for Bioorganic Research
Curated by PDSP Ki Database
| |
Mol Pharmacol 53: 195-201 (1998)
Article DOI: 10.1124/mol.53.2.195 BindingDB Entry DOI: 10.7270/Q2RF5SJH |
More data for this Ligand-Target Pair | |
Glutamate receptor ionotropic, NMDA 1
(RAT) | BDBM50013055
(2-aminopentanedioateglutamate | L-Glutamate | glut...)Show InChI InChI=1S/C5H9NO4/c6-3(5(9)10)1-2-4(7)8/h3H,1-2,6H2,(H,7,8)(H,9,10)/p-2 | PDB
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| 131 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Suntory Institute for Bioorganic Research
Curated by PDSP Ki Database
| |
Mol Pharmacol 53: 195-201 (1998)
Article DOI: 10.1124/mol.53.2.195 BindingDB Entry DOI: 10.7270/Q2RF5SJH |
More data for this Ligand-Target Pair | |
Glutamate receptor ionotropic, NMDA 1
(RAT) | BDBM50002343
(2-Methylamino-succinic acid | CHEMBL275325 | NMDA)Show InChI InChI=1S/C5H9NO4/c1-6-3(5(9)10)2-4(7)8/h3,6H,2H2,1H3,(H,7,8)(H,9,10) | PDB
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| 5.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Suntory Institute for Bioorganic Research
Curated by PDSP Ki Database
| |
Mol Pharmacol 53: 195-201 (1998)
Article DOI: 10.1124/mol.53.2.195 BindingDB Entry DOI: 10.7270/Q2RF5SJH |
More data for this Ligand-Target Pair | |
Glutamate receptor ionotropic, kainate 1
(RAT) | BDBM50240399
((2R,3R,4S)-3-(carboxymethyl)-4-isopropylpyrrolidin...)Show SMILES CC(C)[C@H]1CN[C@@H]([C@H]1CC(O)=O)C(O)=O |r| Show InChI InChI=1S/C10H17NO4/c1-5(2)7-4-11-9(10(14)15)6(7)3-8(12)13/h5-7,9,11H,3-4H2,1-2H3,(H,12,13)(H,14,15)/t6-,7+,9-/m0/s1 | PDB
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| 6.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Suntory Institute for Bioorganic Research
Curated by PDSP Ki Database
| |
Mol Pharmacol 53: 195-201 (1998)
Article DOI: 10.1124/mol.53.2.195 BindingDB Entry DOI: 10.7270/Q2RF5SJH |
More data for this Ligand-Target Pair | |
Glutamate receptor ionotropic, NMDA 1
(RAT) | BDBM50240399
((2R,3R,4S)-3-(carboxymethyl)-4-isopropylpyrrolidin...)Show SMILES CC(C)[C@H]1CN[C@@H]([C@H]1CC(O)=O)C(O)=O |r| Show InChI InChI=1S/C10H17NO4/c1-5(2)7-4-11-9(10(14)15)6(7)3-8(12)13/h5-7,9,11H,3-4H2,1-2H3,(H,12,13)(H,14,15)/t6-,7+,9-/m0/s1 | PDB
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| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Suntory Institute for Bioorganic Research
Curated by PDSP Ki Database
| |
Mol Pharmacol 53: 195-201 (1998)
Article DOI: 10.1124/mol.53.2.195 BindingDB Entry DOI: 10.7270/Q2RF5SJH |
More data for this Ligand-Target Pair | |
Glutamate receptor ionotropic, NMDA 1
(RAT) | BDBM50093753
((2S,3S)-2-Amino-3-benzyloxy-succinic acid | (2S,3S...)Show InChI InChI=1S/C11H13NO5/c12-8(10(13)14)9(11(15)16)17-6-7-4-2-1-3-5-7/h1-5,8-9H,6,12H2,(H,13,14)(H,15,16)/t8-,9-/m0/s1 | PDB
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| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Suntory Institute for Bioorganic Research
Curated by PDSP Ki Database
| |
Mol Pharmacol 53: 195-201 (1998)
Article DOI: 10.1124/mol.53.2.195 BindingDB Entry DOI: 10.7270/Q2RF5SJH |
More data for this Ligand-Target Pair | |
Glutamate receptor ionotropic, NMDA 1
(RAT) | BDBM85210
(DL-TBzOAsp)Show SMILES N[C@@H]([C@H](OC(=O)c1ccccc1)C(O)=O)C(O)=O |r| Show InChI InChI=1S/C11H11NO6/c12-7(9(13)14)8(10(15)16)18-11(17)6-4-2-1-3-5-6/h1-5,7-8H,12H2,(H,13,14)(H,15,16)/t7-,8-/m0/s1 | PDB
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| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Suntory Institute for Bioorganic Research
Curated by PDSP Ki Database
| |
Mol Pharmacol 53: 195-201 (1998)
Article DOI: 10.1124/mol.53.2.195 BindingDB Entry DOI: 10.7270/Q2RF5SJH |
More data for this Ligand-Target Pair | |
Glutamate receptor ionotropic, NMDA 1
(RAT) | BDBM85209
(DL-THA)Show InChI InChI=1S/C4H7NO5/c5-1(3(7)8)2(6)4(9)10/h1-2,6H,5H2,(H,7,8)(H,9,10)/t1-,2-/m0/s1 | PDB
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| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Suntory Institute for Bioorganic Research
Curated by PDSP Ki Database
| |
Mol Pharmacol 53: 195-201 (1998)
Article DOI: 10.1124/mol.53.2.195 BindingDB Entry DOI: 10.7270/Q2RF5SJH |
More data for this Ligand-Target Pair | |
Glutamate receptor ionotropic, NMDA 1
(RAT) | BDBM85211
(t-2,4-PDC | t-PDC)Show InChI InChI=1S/C6H9NO4/c8-5(9)3-1-4(6(10)11)7-2-3/h3-4,7H,1-2H2,(H,8,9)(H,10,11)/t3-,4+/m1/s1 | PDB
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| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Suntory Institute for Bioorganic Research
Curated by PDSP Ki Database
| |
Mol Pharmacol 53: 195-201 (1998)
Article DOI: 10.1124/mol.53.2.195 BindingDB Entry DOI: 10.7270/Q2RF5SJH |
More data for this Ligand-Target Pair | |
Glutamate receptor ionotropic, kainate 1
(RAT) | BDBM85211
(t-2,4-PDC | t-PDC)Show InChI InChI=1S/C6H9NO4/c8-5(9)3-1-4(6(10)11)7-2-3/h3-4,7H,1-2H2,(H,8,9)(H,10,11)/t3-,4+/m1/s1 | PDB
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| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Suntory Institute for Bioorganic Research
Curated by PDSP Ki Database
| |
Mol Pharmacol 53: 195-201 (1998)
Article DOI: 10.1124/mol.53.2.195 BindingDB Entry DOI: 10.7270/Q2RF5SJH |
More data for this Ligand-Target Pair | |
Glutamate receptor ionotropic, kainate 1
(RAT) | BDBM85209
(DL-THA)Show InChI InChI=1S/C4H7NO5/c5-1(3(7)8)2(6)4(9)10/h1-2,6H,5H2,(H,7,8)(H,9,10)/t1-,2-/m0/s1 | PDB
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| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Suntory Institute for Bioorganic Research
Curated by PDSP Ki Database
| |
Mol Pharmacol 53: 195-201 (1998)
Article DOI: 10.1124/mol.53.2.195 BindingDB Entry DOI: 10.7270/Q2RF5SJH |
More data for this Ligand-Target Pair | |
Glutamate receptor ionotropic, kainate 1
(RAT) | BDBM85210
(DL-TBzOAsp)Show SMILES N[C@@H]([C@H](OC(=O)c1ccccc1)C(O)=O)C(O)=O |r| Show InChI InChI=1S/C11H11NO6/c12-7(9(13)14)8(10(15)16)18-11(17)6-4-2-1-3-5-6/h1-5,7-8H,12H2,(H,13,14)(H,15,16)/t7-,8-/m0/s1 | PDB
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| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Suntory Institute for Bioorganic Research
Curated by PDSP Ki Database
| |
Mol Pharmacol 53: 195-201 (1998)
Article DOI: 10.1124/mol.53.2.195 BindingDB Entry DOI: 10.7270/Q2RF5SJH |
More data for this Ligand-Target Pair | |
Glutamate receptor ionotropic, kainate 1
(RAT) | BDBM50093753
((2S,3S)-2-Amino-3-benzyloxy-succinic acid | (2S,3S...)Show InChI InChI=1S/C11H13NO5/c12-8(10(13)14)9(11(15)16)17-6-7-4-2-1-3-5-7/h1-5,8-9H,6,12H2,(H,13,14)(H,15,16)/t8-,9-/m0/s1 | PDB
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| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Suntory Institute for Bioorganic Research
Curated by PDSP Ki Database
| |
Mol Pharmacol 53: 195-201 (1998)
Article DOI: 10.1124/mol.53.2.195 BindingDB Entry DOI: 10.7270/Q2RF5SJH |
More data for this Ligand-Target Pair | |
Glutamate receptor 3
(RAT) | BDBM85209
(DL-THA)Show InChI InChI=1S/C4H7NO5/c5-1(3(7)8)2(6)4(9)10/h1-2,6H,5H2,(H,7,8)(H,9,10)/t1-,2-/m0/s1 | PDB
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| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Suntory Institute for Bioorganic Research
Curated by PDSP Ki Database
| |
Mol Pharmacol 53: 195-201 (1998)
Article DOI: 10.1124/mol.53.2.195 BindingDB Entry DOI: 10.7270/Q2RF5SJH |
More data for this Ligand-Target Pair | |
Glutamate receptor 3
(RAT) | BDBM85210
(DL-TBzOAsp)Show SMILES N[C@@H]([C@H](OC(=O)c1ccccc1)C(O)=O)C(O)=O |r| Show InChI InChI=1S/C11H11NO6/c12-7(9(13)14)8(10(15)16)18-11(17)6-4-2-1-3-5-6/h1-5,7-8H,12H2,(H,13,14)(H,15,16)/t7-,8-/m0/s1 | PDB
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| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Suntory Institute for Bioorganic Research
Curated by PDSP Ki Database
| |
Mol Pharmacol 53: 195-201 (1998)
Article DOI: 10.1124/mol.53.2.195 BindingDB Entry DOI: 10.7270/Q2RF5SJH |
More data for this Ligand-Target Pair | |
Glutamate receptor 3
(RAT) | BDBM50240399
((2R,3R,4S)-3-(carboxymethyl)-4-isopropylpyrrolidin...)Show SMILES CC(C)[C@H]1CN[C@@H]([C@H]1CC(O)=O)C(O)=O |r| Show InChI InChI=1S/C10H17NO4/c1-5(2)7-4-11-9(10(14)15)6(7)3-8(12)13/h5-7,9,11H,3-4H2,1-2H3,(H,12,13)(H,14,15)/t6-,7+,9-/m0/s1 | PDB
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| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Suntory Institute for Bioorganic Research
Curated by PDSP Ki Database
| |
Mol Pharmacol 53: 195-201 (1998)
Article DOI: 10.1124/mol.53.2.195 BindingDB Entry DOI: 10.7270/Q2RF5SJH |
More data for this Ligand-Target Pair | |
Glutamate receptor 3
(RAT) | BDBM50093753
((2S,3S)-2-Amino-3-benzyloxy-succinic acid | (2S,3S...)Show InChI InChI=1S/C11H13NO5/c12-8(10(13)14)9(11(15)16)17-6-7-4-2-1-3-5-7/h1-5,8-9H,6,12H2,(H,13,14)(H,15,16)/t8-,9-/m0/s1 | PDB
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| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Suntory Institute for Bioorganic Research
Curated by PDSP Ki Database
| |
Mol Pharmacol 53: 195-201 (1998)
Article DOI: 10.1124/mol.53.2.195 BindingDB Entry DOI: 10.7270/Q2RF5SJH |
More data for this Ligand-Target Pair | |
Glutamate receptor 3
(RAT) | BDBM85211
(t-2,4-PDC | t-PDC)Show InChI InChI=1S/C6H9NO4/c8-5(9)3-1-4(6(10)11)7-2-3/h3-4,7H,1-2H2,(H,8,9)(H,10,11)/t3-,4+/m1/s1 | PDB
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| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Suntory Institute for Bioorganic Research
Curated by PDSP Ki Database
| |
Mol Pharmacol 53: 195-201 (1998)
Article DOI: 10.1124/mol.53.2.195 BindingDB Entry DOI: 10.7270/Q2RF5SJH |
More data for this Ligand-Target Pair | |
Excitatory amino acid transporter 2
(Homo sapiens (Human)) | BDBM50093754
((2S, 3S)-3-Amino-2-(naphthalen-1-ylmethoxy)-pentan...)Show SMILES N[C@@H]([C@H](OCc1cccc2ccccc12)C(O)=O)C(O)=O Show InChI InChI=1S/C15H15NO5/c16-12(14(17)18)13(15(19)20)21-8-10-6-3-5-9-4-1-2-7-11(9)10/h1-7,12-13H,8,16H2,(H,17,18)(H,19,20)/t12-,13-/m0/s1 | PDB
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| n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute for Bioorganic Research
Curated by ChEMBL
| Assay Description Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 2 |
Bioorg Med Chem Lett 10: 2407-10 (2001)
Checked by Author BindingDB Entry DOI: 10.7270/Q2CR5TVN |
More data for this Ligand-Target Pair | |
Excitatory amino acid transporter 2
(Homo sapiens (Human)) | BDBM50093752
((2S, 3S)-3-Amino-2-methoxy-pentanedioic acid | CHE...)Show InChI InChI=1S/C5H9NO5/c1-11-3(5(9)10)2(6)4(7)8/h2-3H,6H2,1H3,(H,7,8)(H,9,10)/t2-,3-/m0/s1 | PDB
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| n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute for Bioorganic Research
Curated by ChEMBL
| Assay Description Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 2 |
Bioorg Med Chem Lett 10: 2407-10 (2001)
Checked by Author BindingDB Entry DOI: 10.7270/Q2CR5TVN |
More data for this Ligand-Target Pair | |
Excitatory amino acid transporter 2
(Homo sapiens (Human)) | BDBM50093755
((2S, 3S)-3-Amino-2-(naphthalen-2-ylmethoxy)-pentan...)Show SMILES N[C@@H]([C@H](OCc1ccc2ccccc2c1)C(O)=O)C(O)=O Show InChI InChI=1S/C15H15NO5/c16-12(14(17)18)13(15(19)20)21-8-9-5-6-10-3-1-2-4-11(10)7-9/h1-7,12-13H,8,16H2,(H,17,18)(H,19,20)/t12-,13-/m0/s1 | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
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| PubMed
| n/a | n/a | 2.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute for Bioorganic Research
Curated by ChEMBL
| Assay Description Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 2 |
Bioorg Med Chem Lett 10: 2407-10 (2001)
Checked by Author BindingDB Entry DOI: 10.7270/Q2CR5TVN |
More data for this Ligand-Target Pair | |
Excitatory amino acid transporter 2
(Homo sapiens (Human)) | BDBM50093753
((2S,3S)-2-Amino-3-benzyloxy-succinic acid | (2S,3S...)Show InChI InChI=1S/C11H13NO5/c12-8(10(13)14)9(11(15)16)17-6-7-4-2-1-3-5-7/h1-5,8-9H,6,12H2,(H,13,14)(H,15,16)/t8-,9-/m0/s1 | PDB
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| n/a | n/a | 3.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute for Bioorganic Research
Curated by ChEMBL
| Assay Description Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 2 |
Bioorg Med Chem Lett 10: 2407-10 (2001)
Checked by Author BindingDB Entry DOI: 10.7270/Q2CR5TVN |
More data for this Ligand-Target Pair | |
Excitatory amino acid transporter 3
(Homo sapiens (Human)) | BDBM50093754
((2S, 3S)-3-Amino-2-(naphthalen-1-ylmethoxy)-pentan...)Show SMILES N[C@@H]([C@H](OCc1cccc2ccccc12)C(O)=O)C(O)=O Show InChI InChI=1S/C15H15NO5/c16-12(14(17)18)13(15(19)20)21-8-10-6-3-5-9-4-1-2-7-11(9)10/h1-7,12-13H,8,16H2,(H,17,18)(H,19,20)/t12-,13-/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| CHEMBL KEGG PC cid PC sid UniChem
Similars
| PubMed
| n/a | n/a | 4.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute for Bioorganic Research
Curated by ChEMBL
| Assay Description Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 3 |
Bioorg Med Chem Lett 10: 2407-10 (2001)
Checked by Author BindingDB Entry DOI: 10.7270/Q2CR5TVN |
More data for this Ligand-Target Pair | |
Excitatory amino acid transporter 3
(Homo sapiens (Human)) | BDBM50093755
((2S, 3S)-3-Amino-2-(naphthalen-2-ylmethoxy)-pentan...)Show SMILES N[C@@H]([C@H](OCc1ccc2ccccc2c1)C(O)=O)C(O)=O Show InChI InChI=1S/C15H15NO5/c16-12(14(17)18)13(15(19)20)21-8-9-5-6-10-3-1-2-4-11(10)7-9/h1-7,12-13H,8,16H2,(H,17,18)(H,19,20)/t12-,13-/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| CHEMBL KEGG PC cid PC sid UniChem
Similars
| PubMed
| n/a | n/a | 6.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute for Bioorganic Research
Curated by ChEMBL
| Assay Description Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 3 |
Bioorg Med Chem Lett 10: 2407-10 (2001)
Checked by Author BindingDB Entry DOI: 10.7270/Q2CR5TVN |
More data for this Ligand-Target Pair | |
Excitatory amino acid transporter 3
(Homo sapiens (Human)) | BDBM50093753
((2S,3S)-2-Amino-3-benzyloxy-succinic acid | (2S,3S...)Show InChI InChI=1S/C11H13NO5/c12-8(10(13)14)9(11(15)16)17-6-7-4-2-1-3-5-7/h1-5,8-9H,6,12H2,(H,13,14)(H,15,16)/t8-,9-/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE KEGG MMDB PC cid PC sid PDB UniChem
Patents
Similars
| PubMed
| n/a | n/a | 7.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute for Bioorganic Research
Curated by ChEMBL
| Assay Description Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 3 |
Bioorg Med Chem Lett 10: 2407-10 (2001)
Checked by Author BindingDB Entry DOI: 10.7270/Q2CR5TVN |
More data for this Ligand-Target Pair | |
Excitatory amino acid transporter 2
(Homo sapiens (Human)) | BDBM50247191
((2S,3S)-2-Amino-3-benzyloxy-succinic acid | CHEMBL...)Show InChI InChI=1S/C11H13NO5/c12-8(10(13)14)9(11(15)16)17-6-7-4-2-1-3-5-7/h1-5,8-9H,6,12H2,(H,13,14)(H,15,16) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid PDB UniChem
Similars
| PubMed
| n/a | n/a | 7.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute for Bioorganic Research
Curated by ChEMBL
| Assay Description Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 2 |
Bioorg Med Chem Lett 10: 2407-10 (2001)
Checked by Author BindingDB Entry DOI: 10.7270/Q2CR5TVN |
More data for this Ligand-Target Pair | |
Excitatory amino acid transporter 3
(Homo sapiens (Human)) | BDBM50247191
((2S,3S)-2-Amino-3-benzyloxy-succinic acid | CHEMBL...)Show InChI InChI=1S/C11H13NO5/c12-8(10(13)14)9(11(15)16)17-6-7-4-2-1-3-5-7/h1-5,8-9H,6,12H2,(H,13,14)(H,15,16) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid PDB UniChem
Similars
| PubMed
| n/a | n/a | 8.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute for Bioorganic Research
Curated by ChEMBL
| Assay Description Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 3 |
Bioorg Med Chem Lett 10: 2407-10 (2001)
Checked by Author BindingDB Entry DOI: 10.7270/Q2CR5TVN |
More data for this Ligand-Target Pair | |
Excitatory amino acid transporter 3
(Homo sapiens (Human)) | BDBM50093752
((2S, 3S)-3-Amino-2-methoxy-pentanedioic acid | CHE...)Show InChI InChI=1S/C5H9NO5/c1-11-3(5(9)10)2(6)4(7)8/h2-3H,6H2,1H3,(H,7,8)(H,9,10)/t2-,3-/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| CHEMBL KEGG PC cid PC sid UniChem
Similars
| PubMed
| n/a | n/a | 8.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute for Bioorganic Research
Curated by ChEMBL
| Assay Description Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 3 |
Bioorg Med Chem Lett 10: 2407-10 (2001)
Checked by Author BindingDB Entry DOI: 10.7270/Q2CR5TVN |
More data for this Ligand-Target Pair | |
Excitatory amino acid transporter 1
(Homo sapiens (Human)) | BDBM50093754
((2S, 3S)-3-Amino-2-(naphthalen-1-ylmethoxy)-pentan...)Show SMILES N[C@@H]([C@H](OCc1cccc2ccccc12)C(O)=O)C(O)=O Show InChI InChI=1S/C15H15NO5/c16-12(14(17)18)13(15(19)20)21-8-10-6-3-5-9-4-1-2-7-11(9)10/h1-7,12-13H,8,16H2,(H,17,18)(H,19,20)/t12-,13-/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| CHEMBL KEGG PC cid PC sid UniChem
Similars
| PubMed
| n/a | n/a | 1.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute for Bioorganic Research
Curated by ChEMBL
| Assay Description Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 1 |
Bioorg Med Chem Lett 10: 2407-10 (2001)
Checked by Author BindingDB Entry DOI: 10.7270/Q2CR5TVN |
More data for this Ligand-Target Pair | |
Excitatory amino acid transporter 1
(Homo sapiens (Human)) | BDBM50093755
((2S, 3S)-3-Amino-2-(naphthalen-2-ylmethoxy)-pentan...)Show SMILES N[C@@H]([C@H](OCc1ccc2ccccc2c1)C(O)=O)C(O)=O Show InChI InChI=1S/C15H15NO5/c16-12(14(17)18)13(15(19)20)21-8-9-5-6-10-3-1-2-4-11(10)7-9/h1-7,12-13H,8,16H2,(H,17,18)(H,19,20)/t12-,13-/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| CHEMBL KEGG PC cid PC sid UniChem
Similars
| PubMed
| n/a | n/a | 1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute for Bioorganic Research
Curated by ChEMBL
| Assay Description Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 1 |
Bioorg Med Chem Lett 10: 2407-10 (2001)
Checked by Author BindingDB Entry DOI: 10.7270/Q2CR5TVN |
More data for this Ligand-Target Pair | |
Excitatory amino acid transporter 3
(Homo sapiens (Human)) | BDBM50093753
((2S,3S)-2-Amino-3-benzyloxy-succinic acid | (2S,3S...)Show InChI InChI=1S/C11H13NO5/c12-8(10(13)14)9(11(15)16)17-6-7-4-2-1-3-5-7/h1-5,8-9H,6,12H2,(H,13,14)(H,15,16)/t8-,9-/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE KEGG MMDB PC cid PC sid PDB UniChem
Patents
Similars
| PubMed
| n/a | n/a | 2.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute for Bioorganic Research
Curated by ChEMBL
| Assay Description Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 3 |
Bioorg Med Chem Lett 10: 2407-10 (2001)
Checked by Author BindingDB Entry DOI: 10.7270/Q2CR5TVN |
More data for this Ligand-Target Pair | |
Excitatory amino acid transporter 1
(Homo sapiens (Human)) | BDBM50093753
((2S,3S)-2-Amino-3-benzyloxy-succinic acid | (2S,3S...)Show InChI InChI=1S/C11H13NO5/c12-8(10(13)14)9(11(15)16)17-6-7-4-2-1-3-5-7/h1-5,8-9H,6,12H2,(H,13,14)(H,15,16)/t8-,9-/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE KEGG MMDB PC cid PC sid PDB UniChem
Patents
Similars
| PubMed
| n/a | n/a | 2.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute for Bioorganic Research
Curated by ChEMBL
| Assay Description Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 1 |
Bioorg Med Chem Lett 10: 2407-10 (2001)
Checked by Author BindingDB Entry DOI: 10.7270/Q2CR5TVN |
More data for this Ligand-Target Pair | |
Excitatory amino acid transporter 1
(Homo sapiens (Human)) | BDBM50247191
((2S,3S)-2-Amino-3-benzyloxy-succinic acid | CHEMBL...)Show InChI InChI=1S/C11H13NO5/c12-8(10(13)14)9(11(15)16)17-6-7-4-2-1-3-5-7/h1-5,8-9H,6,12H2,(H,13,14)(H,15,16) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid PDB UniChem
Similars
| PubMed
| n/a | n/a | 4.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute for Bioorganic Research
Curated by ChEMBL
| Assay Description Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 1 |
Bioorg Med Chem Lett 10: 2407-10 (2001)
Checked by Author BindingDB Entry DOI: 10.7270/Q2CR5TVN |
More data for this Ligand-Target Pair | |
Excitatory amino acid transporter 2
(Homo sapiens (Human)) | BDBM50093753
((2S,3S)-2-Amino-3-benzyloxy-succinic acid | (2S,3S...)Show InChI InChI=1S/C11H13NO5/c12-8(10(13)14)9(11(15)16)17-6-7-4-2-1-3-5-7/h1-5,8-9H,6,12H2,(H,13,14)(H,15,16)/t8-,9-/m0/s1 | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE KEGG MMDB PC cid PC sid PDB UniChem
Patents
Similars
| PubMed
| n/a | n/a | 6.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute for Bioorganic Research
Curated by ChEMBL
| Assay Description Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 2 |
Bioorg Med Chem Lett 10: 2407-10 (2001)
Checked by Author BindingDB Entry DOI: 10.7270/Q2CR5TVN |
More data for this Ligand-Target Pair | |
Excitatory amino acid transporter 1
(Homo sapiens (Human)) | BDBM50093752
((2S, 3S)-3-Amino-2-methoxy-pentanedioic acid | CHE...)Show InChI InChI=1S/C5H9NO5/c1-11-3(5(9)10)2(6)4(7)8/h2-3H,6H2,1H3,(H,7,8)(H,9,10)/t2-,3-/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| CHEMBL KEGG PC cid PC sid UniChem
Similars
| PubMed
| n/a | n/a | 6.90E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute for Bioorganic Research
Curated by ChEMBL
| Assay Description Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 1 |
Bioorg Med Chem Lett 10: 2407-10 (2001)
Checked by Author BindingDB Entry DOI: 10.7270/Q2CR5TVN |
More data for this Ligand-Target Pair | |
Excitatory amino acid transporter 3
(Homo sapiens (Human)) | BDBM50093753
((2S,3S)-2-Amino-3-benzyloxy-succinic acid | (2S,3S...)Show InChI InChI=1S/C11H13NO5/c12-8(10(13)14)9(11(15)16)17-6-7-4-2-1-3-5-7/h1-5,8-9H,6,12H2,(H,13,14)(H,15,16)/t8-,9-/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE KEGG MMDB PC cid PC sid PDB UniChem
Patents
Similars
| PubMed
| n/a | n/a | 1.61E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute for Bioorganic Research
Curated by ChEMBL
| Assay Description Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 3 |
Bioorg Med Chem Lett 10: 2407-10 (2001)
Checked by Author BindingDB Entry DOI: 10.7270/Q2CR5TVN |
More data for this Ligand-Target Pair | |
Excitatory amino acid transporter 3
(Homo sapiens (Human)) | BDBM50093753
((2S,3S)-2-Amino-3-benzyloxy-succinic acid | (2S,3S...)Show InChI InChI=1S/C11H13NO5/c12-8(10(13)14)9(11(15)16)17-6-7-4-2-1-3-5-7/h1-5,8-9H,6,12H2,(H,13,14)(H,15,16)/t8-,9-/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE KEGG MMDB PC cid PC sid PDB UniChem
Patents
Similars
| PubMed
| n/a | n/a | 1.61E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute for Bioorganic Research
Curated by ChEMBL
| Assay Description Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 3 |
Bioorg Med Chem Lett 10: 2407-10 (2001)
Checked by Author BindingDB Entry DOI: 10.7270/Q2CR5TVN |
More data for this Ligand-Target Pair | |
Excitatory amino acid transporter 2
(Homo sapiens (Human)) | BDBM50093753
((2S,3S)-2-Amino-3-benzyloxy-succinic acid | (2S,3S...)Show InChI InChI=1S/C11H13NO5/c12-8(10(13)14)9(11(15)16)17-6-7-4-2-1-3-5-7/h1-5,8-9H,6,12H2,(H,13,14)(H,15,16)/t8-,9-/m0/s1 | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE KEGG MMDB PC cid PC sid PDB UniChem
Patents
Similars
| PubMed
| n/a | n/a | 2.21E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute for Bioorganic Research
Curated by ChEMBL
| Assay Description Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 2 |
Bioorg Med Chem Lett 10: 2407-10 (2001)
Checked by Author BindingDB Entry DOI: 10.7270/Q2CR5TVN |
More data for this Ligand-Target Pair | |
Excitatory amino acid transporter 2
(Homo sapiens (Human)) | BDBM50093753
((2S,3S)-2-Amino-3-benzyloxy-succinic acid | (2S,3S...)Show InChI InChI=1S/C11H13NO5/c12-8(10(13)14)9(11(15)16)17-6-7-4-2-1-3-5-7/h1-5,8-9H,6,12H2,(H,13,14)(H,15,16)/t8-,9-/m0/s1 | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE KEGG MMDB PC cid PC sid PDB UniChem
Patents
Similars
| PubMed
| n/a | n/a | 2.21E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute for Bioorganic Research
Curated by ChEMBL
| Assay Description Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 2 |
Bioorg Med Chem Lett 10: 2407-10 (2001)
Checked by Author BindingDB Entry DOI: 10.7270/Q2CR5TVN |
More data for this Ligand-Target Pair | |
Excitatory amino acid transporter 1
(Homo sapiens (Human)) | BDBM50093753
((2S,3S)-2-Amino-3-benzyloxy-succinic acid | (2S,3S...)Show InChI InChI=1S/C11H13NO5/c12-8(10(13)14)9(11(15)16)17-6-7-4-2-1-3-5-7/h1-5,8-9H,6,12H2,(H,13,14)(H,15,16)/t8-,9-/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE KEGG MMDB PC cid PC sid PDB UniChem
Patents
Similars
| PubMed
| n/a | n/a | 6.37E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute for Bioorganic Research
Curated by ChEMBL
| Assay Description Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 1 |
Bioorg Med Chem Lett 10: 2407-10 (2001)
Checked by Author BindingDB Entry DOI: 10.7270/Q2CR5TVN |
More data for this Ligand-Target Pair | |
Excitatory amino acid transporter 1
(Homo sapiens (Human)) | BDBM50093753
((2S,3S)-2-Amino-3-benzyloxy-succinic acid | (2S,3S...)Show InChI InChI=1S/C11H13NO5/c12-8(10(13)14)9(11(15)16)17-6-7-4-2-1-3-5-7/h1-5,8-9H,6,12H2,(H,13,14)(H,15,16)/t8-,9-/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE KEGG MMDB PC cid PC sid PDB UniChem
Patents
Similars
| PubMed
| n/a | n/a | 6.37E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute for Bioorganic Research
Curated by ChEMBL
| Assay Description Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 1 |
Bioorg Med Chem Lett 10: 2407-10 (2001)
Checked by Author BindingDB Entry DOI: 10.7270/Q2CR5TVN |
More data for this Ligand-Target Pair | |
Excitatory amino acid transporter 1
(Homo sapiens (Human)) | BDBM50093753
((2S,3S)-2-Amino-3-benzyloxy-succinic acid | (2S,3S...)Show InChI InChI=1S/C11H13NO5/c12-8(10(13)14)9(11(15)16)17-6-7-4-2-1-3-5-7/h1-5,8-9H,6,12H2,(H,13,14)(H,15,16)/t8-,9-/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE KEGG MMDB PC cid PC sid PDB UniChem
Patents
Similars
| PubMed
| n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute for Bioorganic Research
Curated by ChEMBL
| Assay Description Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 1 |
Bioorg Med Chem Lett 10: 2407-10 (2001)
Checked by Author BindingDB Entry DOI: 10.7270/Q2CR5TVN |
More data for this Ligand-Target Pair | |