Found 49 hits Enz. Inhib. hit(s) with Target = 'Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]' Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626350
(2-[[[4-cyano-7-(4-isopropyl-2- thienyl)-2,3-dihyd...)Show SMILES CC(C)c1csc(c1)-c1cc(NCC(=C)C(O)=O)c(C#N)c2CCOc12 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet 
| PC cid
PC sid
UniChem
| | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626318
(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)Show SMILES CC(C)c1ccc(cc1)-c1cc(NCC(=C)C(O)=O)c(C#N)c2CCOc12 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626358
(2-[[[7-cyano-4-[4- (trifluoromethoxy)phenyl]-1,3-...)Show SMILES ONC(=O)C(=C)CNc1cc(-c2ccc(OC(F)(F)F)cc2)c2ncsc2c1C#N | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 80 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626324
(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)Show SMILES CC(C)c1ccc(cc1)-c1cc(NCC(=C)C(=O)NO)c(C#N)c2CCOc12 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626361
(2-[[[4-cyano-7-[4-(pentafluoro- lambda6-sulfanyl)...)Show SMILES OC(=O)C(=C)CNc1cc(c2OCCc2c1C#N)-c1ccc(cc1)S(F)(F)(F)(F)F | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 120 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626354
(2-[[[4-cyano-2,2-dideuterio-7-[4- (trifluorometho...)Show SMILES ONC(=O)C(=C)CNc1cc(c2OCCc2c1C#N)-c1ccc(OC(F)(F)F)cc1 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 140 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626355
(2-[[[4-cyano-7-[4-(pentafluoro- lambda6-sulfanyl)...)Show SMILES ONC(=O)C(=C)CNc1cc(c2OCCc2c1C#N)-c1ccc(cc1)S(F)(F)(F)(F)F | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 160 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626354
(2-[[[4-cyano-2,2-dideuterio-7-[4- (trifluorometho...)Show SMILES ONC(=O)C(=C)CNc1cc(c2OCCc2c1C#N)-c1ccc(OC(F)(F)F)cc1 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 180 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626319
(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)Show SMILES CC(C)c1ccc(cc1)-c1cc(NCC(=C)C(N)=O)c(C#N)c2CCOc12 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626364
(2-[[[4-cyano-7-(5-isopropylthiazol- 2-yl)-2,3-dih...)Show SMILES CC(C)c1cnc(s1)-c1cc(NCC(=C)C(O)=O)c(C#N)c2CCOc12 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626362
(2-[[[4-(hydroxymethyl)-7-[4- (trifluoromethoxy)ph...)Show SMILES OCc1c2CCOc2c(cc1NCC(=C)C(=O)NO)-c1ccc(OC(F)(F)F)cc1 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 240 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626360
(2-[[[4-cyano-7-[4- (trifluoromethoxy)phenyl]-2,3-...)Show SMILES NC(=O)C(=C)CNc1cc(c2OCCc2c1C#N)-c1ccc(OC(F)(F)F)cc1 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 320 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626359
(2-[[[4-cyano-7-[4- (trifluoromethoxy)phenyl]-2,3-...)Show SMILES CN(O)C(=O)C(=C)CNc1cc(c2OCCc2c1C#N)-c1ccc(OC(F)(F)F)cc1 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 490 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626363
(2-[[[4-cyano-7-[4-(pentafluoro- lambda6-sulfanyl)...)Show SMILES NC(=O)C(=C)CNc1cc(c2OCCc2c1C#N)-c1ccc(cc1)S(F)(F)(F)(F)F | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 580 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626352
(2-[[[4-(hydroxymethyl)-7-[4- (trifluoromethoxy)ph...)Show SMILES NC(=O)C(=C)CNc1cc(c2OCCc2c1CO)-c1ccc(OC(F)(F)F)cc1 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 590 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626353
(2-[[[4-cyano-7-(3-isopropylpyrazol- 1-yl)-2,3-dih...)Show SMILES CC(C)c1ccn(n1)-c1cc(NCC(=C)C(=O)NO)c(C#N)c2CCOc12 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626349
(2-[[[4-cyano-7-(4-isopropylthiazol- 2-yl)-2,3-dih...)Show SMILES CC(C)c1csc(n1)-c1cc(NCC(=C)C(=O)NO)c(C#N)c2CCOc12 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626365
(2-[[[7-cyano-4-[4-(pentafluoro- lambda6-sulfanyl)...)Show SMILES ONC(=O)C(=C)CNc1cc(-c2ccc(cc2)S(F)(F)(F)(F)F)c2ncsc2c1C#N | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626347
(2-[[[4-cyano-7-(5-isopropylthiazol- 2-yl)-2,3-dih...)Show SMILES CC(C)c1cnc(s1)-c1cc(NCC(=C)C(=O)NO)c(C#N)c2CCOc12 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626336
(2-[[[4-fluoro-7-(4-isopropylphenyl)- 2,3-dihydrob...)Show SMILES CC(C)c1ccc(cc1)-c1cc(NCC(=C)C(O)=O)c(F)c2CCOc12 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | n/a | n/a | 30 | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626337
(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrofu...)Show SMILES CC(C)c1ccc(cc1)-c1nc(NCC(=C)C(O)=O)c(C#N)c2CCOc12 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | n/a | n/a | 100 | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626338
(2-[[[7-cyano-4-[4-(1,1- difluoroethyl)phenyl]-1,3...)Show SMILES CC(F)(F)c1ccc(cc1)-c1cc(NCC(=C)C(O)=O)c(C#N)c2scnc12 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626339
(2-[[[6-methoxy-5-[(E)-2-[trans-4- (trifluoromethy...)Show SMILES COc1ncc(NCC(=C)C(O)=O)cc1\C=C\[C@H]1CC[C@@H](CC1)C(F)(F)F |r,wU:17.17,wD:20.24,(3.33,3.85,;2,4.62,;.67,3.85,;-.67,4.62,;-2,3.85,;-2,2.31,;-3.33,1.54,;-4.67,2.31,;-6,1.54,;-6,,;-7.34,2.31,;-8.67,1.54,;-7.34,3.85,;-.67,1.54,;.67,2.31,;2,1.54,;2,,;3.33,-.77,;4.67,,;6,-.77,;6,-2.31,;4.67,-3.08,;3.33,-2.31,;7.34,-3.08,;8.67,-2.31,;7.34,-4.62,;8.67,-3.85,)| | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626341
(2-[[[4-cyano-7-(2,6-difluoro-4- isopropyl-phenyl)...)Show SMILES CC(C)c1cc(F)c(c(F)c1)-c1cc(NCC(=C)C(O)=O)c(C#N)c2CCOc12 |(8,-1.99,;6.67,-2.76,;6.67,-4.3,;5.33,-1.99,;5.33,-.45,;4,.32,;4,1.86,;2.67,-.45,;2.67,-1.99,;1.33,-2.76,;4,-2.76,;1.33,.32,;,-.45,;-1.33,.32,;-2.67,-.45,;-4,.32,;-5.33,-.45,;-5.33,-1.99,;-6.67,.32,;-8,-.45,;-6.67,1.86,;-1.33,1.86,;-2.67,2.63,;-4,3.4,;,2.63,;.32,4.14,;1.85,4.3,;2.48,2.89,;1.33,1.86,)| | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626342
(2-[[[4-cyano-7-(2-fluoro-4- isopropyl-phenyl)-2,3...)Show SMILES CC(C)c1ccc(c(F)c1)-c1cc(NCC(=C)C(O)=O)c(C#N)c2CCOc12 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | n/a | n/a | 40 | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626343
(2-[[[4-carbamoyl-7-(4- isopropylphenyl)-2,3- dih...)Show SMILES CC(C)c1ccc(cc1)-c1cc(NCC(=C)C(O)=O)c(C(N)=O)c2CCOc12 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | n/a | n/a | 700 | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626344
(2-[[[7-cyano-4-[4- (trifluoromethoxy)phenyl]-1,3-...)Show SMILES NC(=O)C(=C)CNc1cc(-c2ccc(OC(F)(F)F)cc2)c2ncsc2c1C#N | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626345
(2-[[[4-cyano-7-(5-isopropyl-2- pyridyl)-2,3-dihyd...)Show SMILES CC(C)c1ccc(nc1)-c1cc(NCC(=C)C(O)=O)c(C#N)c2CCOc12 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | n/a | n/a | 3.40E+3 | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626346
(2-[[[7-(4-isopropylphenyl)-4- methylsulfonyl-2,3-...)Show SMILES CC(C)c1ccc(cc1)-c1cc(NCC(=C)C(O)=O)c(c2CCOc12)S(C)(=O)=O | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626335
(2-[[[4-(4-isopropylphenyl)-6,7- dihydrofuro[3,2-d...)Show SMILES CC(C)c1ccc(cc1)-c1nc(NCC(=C)C(O)=O)nc2CCOc12 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | n/a | n/a | 40 | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626334
(2-[[[4-cyano-7-[4-(1,1- difluoroethyl)phenyl]-2,3...)Show SMILES CC(F)(F)c1ccc(cc1)-c1cc(NCC(=C)C(O)=O)c(C#N)c2CCOc12 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | n/a | n/a | 230 | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626333
(2-[[[4-cyano-7-[4- (trifluoromethoxy)phenyl]-2,3-...)Show SMILES OC(=O)C(=C)CNc1cc(c2OCCc2c1C#N)-c1ccc(OC(F)(F)F)cc1 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | n/a | n/a | 60 | n/a | n/a | n/a | n/a |
TBA
| |
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More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626332
(US11787775, Compound 16-D)Show SMILES C[C@H](c1ccc(cc1)-c1cc(NCC(=C)C(O)=O)c(C#N)c2CCOc12)C(F)(F)F |r| | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | n/a | n/a | 100 | n/a | n/a | n/a | n/a |
TBA
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Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626331
(US11787775, Compound 16-C)Show SMILES C[C@@H](c1ccc(cc1)-c1cc(NCC(=C)C(O)=O)c(C#N)c2CCOc12)C(F)(F)F |r| | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | n/a | n/a | 10 | n/a | n/a | n/a | n/a |
TBA
| |
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Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626330
(2-[[[4-cyano-7-[4- (trifluoromethyl)phenyl]-2,3- ...)Show SMILES OC(=O)C(=C)CNc1cc(c2OCCc2c1C#N)-c1ccc(cc1)C(F)(F)F | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | n/a | n/a | 250 | n/a | n/a | n/a | n/a |
TBA
| |
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Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626329
(2-[[[4-(hydroxymethyl)-7-(4- isopropylphenyl)-2,3...)Show SMILES CC(C)c1ccc(cc1)-c1cc(NCC(=C)C(=O)NO)c(CO)c2CCOc12 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | n/a | n/a | 890 | n/a | n/a | n/a | n/a |
TBA
| |
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Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626328
(2-[[[4-(hydroxymethyl)-7-(4- isopropylphenyl)-2,3...)Show SMILES CC(C)c1ccc(cc1)-c1cc(NCC(=C)C(N)=O)c(CO)c2CCOc12 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | n/a | n/a | 180 | n/a | n/a | n/a | n/a |
TBA
| |
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Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626327
(2-[[[4-(hydroxymethyl)-7-(4- isopropylphenyl)-2,3...)Show SMILES CC(C)c1ccc(cc1)-c1cc(NCC(=C)C(O)=O)c(CO)c2CCOc12 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | n/a | n/a | 750 | n/a | n/a | n/a | n/a |
TBA
| |
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Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626326
(7-(4-isopropylphenyl)-5-[(2- methylene-3-oxo-buty...)Show SMILES CC(C)c1ccc(cc1)-c1cc(NCC(=C)C(C)=O)c(C#N)c2CCOc12 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | n/a | n/a | 80 | n/a | n/a | n/a | n/a |
TBA
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Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626325
(1-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)Show SMILES CC(C)c1ccc(cc1)-c1cc(NCC(=C)B(O)O)c(C#N)c2CCOc12 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | n/a | n/a | 2.10E+3 | n/a | n/a | n/a | n/a |
TBA
| |
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Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626324
(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)Show SMILES CC(C)c1ccc(cc1)-c1cc(NCC(=C)C(=O)NO)c(C#N)c2CCOc12 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | n/a | n/a | 280 | n/a | n/a | n/a | n/a |
TBA
| |
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Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626323
(US11787775, Compound 8 | methyl 2-[[[4-cyano-7-(4-...)Show SMILES COC(=O)C(=C)CNc1cc(c2OCCc2c1C#N)-c1ccc(cc1)C(C)C | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a |
TBA
| |
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Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626322
(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)Show SMILES CC(C)c1ccc(cc1)-c1cc(N(C)CC(=C)C(O)=O)c(C#N)c2CCOc12 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | n/a | n/a | 430 | n/a | n/a | n/a | n/a |
TBA
| |
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Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626321
(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)Show SMILES CC(C)c1ccc(cc1)-c1cc(NCC(=C)C(=O)N(C)C)c(C#N)c2CCOc12 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a |
TBA
| |
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Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626320
(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)Show SMILES CNC(=O)C(=C)CNc1cc(c2OCCc2c1C#N)-c1ccc(cc1)C(C)C | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a |
TBA
| |
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Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626319
(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)Show SMILES CC(C)c1ccc(cc1)-c1cc(NCC(=C)C(N)=O)c(C#N)c2CCOc12 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | n/a | n/a | 160 | n/a | n/a | n/a | n/a |
TBA
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Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626318
(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)Show SMILES CC(C)c1ccc(cc1)-c1cc(NCC(=C)C(O)=O)c(C#N)c2CCOc12 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | n/a | n/a | 30 | n/a | n/a | n/a | n/a |
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Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626316
(2-[[[7-(4-isopropylphenyl)-2,3- dihydrobenzofuran...)Show SMILES CC(C)c1ccc(cc1)-c1cc(NCC(=C)C(O)=O)cc2CCOc12 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | n/a | n/a | 50 | n/a | n/a | n/a | n/a |
TBA
| |
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Ligand-Target Pair | |
Transcriptional enhancer factor TEF-3/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626317
(2-[[[7-(4-isopropylphenyl)-2,3- dihydrobenzofuran...)Show SMILES CC(C)c1ccc(cc1)-c1cc(NCC(=C)C(N)=O)cc2CCOc12 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | n/a | n/a | 90 | n/a | n/a | n/a | n/a |
TBA
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