Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM26113 (2,4 PDCA | cid_10365 | pyridine carboxylate, 6a | ...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE MMDB PC cid PC sid PDB UniChem Patents | PDB Article PubMed | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using 1 uM hFX-CP as substrate mixture with 3 uM 2OG, 100 u... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM26113 (2,4 PDCA | cid_10365 | pyridine carboxylate, 6a | ...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE MMDB PC cid PC sid PDB UniChem Patents | PDB Article PubMed | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using high 10 uM hFX-CP as substrate mixture with 10 uM 2OG... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM26113 (2,4 PDCA | cid_10365 | pyridine carboxylate, 6a | ...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE MMDB PC cid PC sid PDB UniChem Patents | PDB Article PubMed | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using 1 uM hFX-CP as substrate mixture with 3 uM 2OG, 100 u... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM26113 (2,4 PDCA | cid_10365 | pyridine carboxylate, 6a | ...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE MMDB PC cid PC sid PDB UniChem Patents | PDB Article PubMed | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using 1 uM hFX-CP as substrate mixture with high 200 uM 2OG... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM23223 (7-[8-formyl-1,6,7-trihydroxy-3-methyl-5-(propan-2-...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 250 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using 1 uM hFX-CP as substrate mixture with 3 uM 2OG, 100 u... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM23223 (7-[8-formyl-1,6,7-trihydroxy-3-methyl-5-(propan-2-...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 250 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using 1 uM hFX-CP as substrate mixture with high 200 uM 2OG... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM23223 (7-[8-formyl-1,6,7-trihydroxy-3-methyl-5-(propan-2-...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 260 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using 1 uM hFX-CP as substrate mixture with 3 uM 2OG, 100 u... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM23223 (7-[8-formyl-1,6,7-trihydroxy-3-methyl-5-(propan-2-...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 330 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using high 10 uM hFX-CP as substrate mixture with 10 uM 2OG... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM50270877 ((R)-4-(4-((2-(4-chlorophenyl)-5,5-dimethylcyclohex...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 800 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using 1 uM hFX-CP as substrate mixture with 3 uM 2OG, 100 u... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM50270877 ((R)-4-(4-((2-(4-chlorophenyl)-5,5-dimethylcyclohex...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 1.03E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using 1 uM hFX-CP as substrate mixture with 3 uM 2OG, 100 u... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM50270877 ((R)-4-(4-((2-(4-chlorophenyl)-5,5-dimethylcyclohex...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 1.21E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using high 10 uM hFX-CP as substrate mixture with 10 uM 2OG... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM50162774 (ABT-199 | US11420968, Example ABT-199 | Venetoclax) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.29E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using 1 uM hFX-CP as substrate mixture with 3 uM 2OG, 100 u... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM50270877 ((R)-4-(4-((2-(4-chlorophenyl)-5,5-dimethylcyclohex...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 1.33E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using 1 uM hFX-CP as substrate mixture with high 200 uM 2OG... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM50162774 (ABT-199 | US11420968, Example ABT-199 | Venetoclax) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using 1 uM hFX-CP as substrate mixture with 3 uM 2OG, 100 u... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM50547621 (Blenamax | Bleo-kyowa | Bleocin | Bleomycin | Bleo...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.47E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using 1 uM hFX-CP as substrate mixture with 3 uM 2OG, 100 u... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM50162774 (ABT-199 | US11420968, Example ABT-199 | Venetoclax) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.52E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using 1 uM hFX-CP as substrate mixture with high 200 uM 2OG... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM50162774 (ABT-199 | US11420968, Example ABT-199 | Venetoclax) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.57E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using high 10 uM hFX-CP as substrate mixture with 10 uM 2OG... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM50547621 (Blenamax | Bleo-kyowa | Bleocin | Bleomycin | Bleo...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.65E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using high 10 uM hFX-CP as substrate mixture with 10 uM 2OG... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM50547621 (Blenamax | Bleo-kyowa | Bleocin | Bleomycin | Bleo...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.99E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using 1 uM hFX-CP as substrate mixture with 3 uM 2OG, 100 u... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM21447 (4-(4-{[2-(4-chlorophenyl)phenyl]methyl}piperazin-1...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 2.92E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using 1 uM hFX-CP as substrate mixture with 3 uM 2OG, 100 u... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM21447 (4-(4-{[2-(4-chlorophenyl)phenyl]methyl}piperazin-1...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 2.99E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using high 10 uM hFX-CP as substrate mixture with 10 uM 2OG... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM25150 ((2E)-N-hydroxy-3-[3-(phenylsulfamoyl)phenyl]prop-2...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 3.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using 1 uM hFX-CP as substrate mixture with 3 uM 2OG, 100 u... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM21447 (4-(4-{[2-(4-chlorophenyl)phenyl]methyl}piperazin-1...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 3.38E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using 1 uM hFX-CP as substrate mixture with 3 uM 2OG, 100 u... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM50547623 (CHEBI:31856 | CHEMBL257619) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 3.39E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using high 10 uM hFX-CP as substrate mixture with 10 uM 2OG... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM22449 (CHEMBL356769 | N-(4-{(2R,4R,6S)-4-{[(4,5-diphenyl-...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 3.57E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using high 10 uM hFX-CP as substrate mixture with 10 uM 2OG... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM50547621 (Blenamax | Bleo-kyowa | Bleocin | Bleomycin | Bleo...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.81E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using 1 uM hFX-CP as substrate mixture with high 200 uM 2OG... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM22449 (CHEMBL356769 | N-(4-{(2R,4R,6S)-4-{[(4,5-diphenyl-...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 4.12E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using 1 uM hFX-CP as substrate mixture with 3 uM 2OG, 100 u... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM21447 (4-(4-{[2-(4-chlorophenyl)phenyl]methyl}piperazin-1...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 4.47E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using 1 uM hFX-CP as substrate mixture with high 200 uM 2OG... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM25150 ((2E)-N-hydroxy-3-[3-(phenylsulfamoyl)phenyl]prop-2...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 4.77E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using high 10 uM hFX-CP as substrate mixture with 10 uM 2OG... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM22449 (CHEMBL356769 | N-(4-{(2R,4R,6S)-4-{[(4,5-diphenyl-...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 4.91E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using 1 uM hFX-CP as substrate mixture with 3 uM 2OG, 100 u... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM22449 (CHEMBL356769 | N-(4-{(2R,4R,6S)-4-{[(4,5-diphenyl-...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 5.69E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using 1 uM hFX-CP as substrate mixture with high 200 uM 2OG... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM50326053 (CHEMBL608533 | PKC-412) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 6.02E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using high 10 uM hFX-CP as substrate mixture with 10 uM 2OG... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM50326053 (CHEMBL608533 | PKC-412) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 7.28E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using 1 uM hFX-CP as substrate mixture with 3 uM 2OG, 100 u... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM25150 ((2E)-N-hydroxy-3-[3-(phenylsulfamoyl)phenyl]prop-2...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 7.49E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using 1 uM hFX-CP as substrate mixture with 3 uM 2OG, 100 u... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM50326053 (CHEMBL608533 | PKC-412) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 9.43E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using 1 uM hFX-CP as substrate mixture with 3 uM 2OG, 100 u... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM50547622 (CHEMBL4777255) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 9.44E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using high 10 uM hFX-CP as substrate mixture with 10 uM 2OG... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM50396483 (PLX-4032 | RG 7204 | Ro 5185426 | US10570155, Vemu...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase DrugBank MCE PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 1.05E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using 1 uM hFX-CP as substrate mixture with 3 uM 2OG, 100 u... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM25150 ((2E)-N-hydroxy-3-[3-(phenylsulfamoyl)phenyl]prop-2...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 1.12E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using 1 uM hFX-CP as substrate mixture with high 200 uM 2OG... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM50547622 (CHEMBL4777255) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.19E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using 1 uM hFX-CP as substrate mixture with 3 uM 2OG, 100 u... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM50547623 (CHEBI:31856 | CHEMBL257619) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 1.22E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using 1 uM hFX-CP as substrate mixture with high 200 uM 2OG... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM50326053 (CHEMBL608533 | PKC-412) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 1.24E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using 1 uM hFX-CP as substrate mixture with high 200 uM 2OG... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM50396483 (PLX-4032 | RG 7204 | Ro 5185426 | US10570155, Vemu...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase DrugBank MCE PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 1.29E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using 1 uM hFX-CP as substrate mixture with 3 uM 2OG, 100 u... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM50547622 (CHEMBL4777255) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.32E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using 1 uM hFX-CP as substrate mixture with 3 uM 2OG, 100 u... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM50396483 (PLX-4032 | RG 7204 | Ro 5185426 | US10570155, Vemu...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase DrugBank MCE PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 1.51E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using 1 uM hFX-CP as substrate mixture with high 200 uM 2OG... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM50547622 (CHEMBL4777255) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.64E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using 1 uM hFX-CP as substrate mixture with high 200 uM 2OG... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartyl/asparaginyl beta-hydroxylase (Homo sapiens) | BDBM50396483 (PLX-4032 | RG 7204 | Ro 5185426 | US10570155, Vemu...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase DrugBank MCE PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 1.69E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-His6-tagged human AspH (315-755) expressed in Escherichia coli BL21 (DE3) using high 10 uM hFX-CP as substrate mixture with 10 uM 2OG... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115675 BindingDB Entry DOI: 10.7270/Q2PV6Q0D | |||||||||||
More data for this Ligand-Target Pair |