Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50583031 (CHEMBL5081078) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 36 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at rat GluN1/GluN2C NMDA receptor expressed in Xenopus oocytes measured after 4 days in presence of L-glutamte by two-electrode volt... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c01810 BindingDB Entry DOI: 10.7270/Q21R6VFZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50583020 (CHEMBL5087374) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 40 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at rat GluN1/GluN2C NMDA receptor expressed in Xenopus oocytes measured after 4 days in presence of L-glutamte by two-electrode volt... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c01810 BindingDB Entry DOI: 10.7270/Q21R6VFZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50583019 (CHEMBL5081008) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 63 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at rat GluN1/GluN2C NMDA receptor expressed in Xenopus oocytes measured after 4 days in presence of L-glutamte by two-electrode volt... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c01810 BindingDB Entry DOI: 10.7270/Q21R6VFZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50583032 (CHEMBL5090386) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 74 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at rat GluN1/GluN2C NMDA receptor expressed in Xenopus oocytes measured after 4 days in presence of L-glutamte by two-electrode volt... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c01810 BindingDB Entry DOI: 10.7270/Q21R6VFZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50220152 ((1S,2R)-2-((S)-Amino-carboxy-methyl)-cyclopropanec...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 110 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at rat recombinant wild type GluN1/GluN2C receptor expressed in Xenopus laevis oocytes by two electrode voltage clamp technique | J Med Chem 56: 4071-81 (2013) Article DOI: 10.1021/jm400346a BindingDB Entry DOI: 10.7270/Q20G3MHR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50583021 (CHEMBL5091289) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 110 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at rat GluN1/GluN2C NMDA receptor expressed in Xenopus oocytes measured after 4 days in presence of L-glutamte by two-electrode volt... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c01810 BindingDB Entry DOI: 10.7270/Q21R6VFZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50583023 (CHEMBL5081203) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 120 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at rat GluN1/GluN2C NMDA receptor expressed in Xenopus oocytes measured after 4 days in presence of L-glutamte by two-electrode volt... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c01810 BindingDB Entry DOI: 10.7270/Q21R6VFZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50432711 (CHEMBL2348224) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 124 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at rat recombinant wild type GluN1/GluN2C receptor expressed in Xenopus laevis oocytes by two electrode voltage clamp technique | J Med Chem 56: 4071-81 (2013) Article DOI: 10.1021/jm400346a BindingDB Entry DOI: 10.7270/Q20G3MHR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50583022 (CHEMBL5085583) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 140 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at rat GluN1/GluN2C NMDA receptor expressed in Xenopus oocytes measured after 4 days in presence of L-glutamte by two-electrode volt... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c01810 BindingDB Entry DOI: 10.7270/Q21R6VFZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM23167 ((2R)-2-amino-3-hydroxypropanoic acid | CHEMBL28512...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | n/a | n/a | n/a | n/a | 190 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at rat GluN1/GluN2C NMDA receptor expressed in Xenopus oocytes measured after 4 days in presence of L-glutamte by two-electrode volt... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c01810 BindingDB Entry DOI: 10.7270/Q21R6VFZ | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM18133 (2-aminoacetic acid | CHEMBL773 | Glycine | [14C]Gl...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | n/a | 210 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at rat GluN1/GluN2C NMDA receptor expressed in Xenopus oocytes measured after 4 days in presence of L-glutamte by two-electrode volt... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c01810 BindingDB Entry DOI: 10.7270/Q21R6VFZ | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50436093 (CHEMBL2397268) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 300 | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Activity at rat recombinant GluN1/GluN2C receptor assessed as potentiation of glycine/glutamate-induced activation by two-electrode voltage clamp tec... | J Med Chem 56: 5351-81 (2014) Article DOI: 10.1021/jm400177t BindingDB Entry DOI: 10.7270/Q26W9CH4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50238357 (CHEMBL4100452) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 340 | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Positive allosteric modulation of recombinant rat GluN1/GluN2C receptor expressed in xenopus laevis oocyte assessed as potentiation of glutamate and ... | J Med Chem 60: 5556-5585 (2017) Article DOI: 10.1021/acs.jmedchem.7b00239 BindingDB Entry DOI: 10.7270/Q298898H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50238354 (CHEMBL4070902) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 350 | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Positive allosteric modulation of recombinant rat GluN1/GluN2C receptor expressed in xenopus laevis oocyte assessed as potentiation of glutamate and ... | J Med Chem 60: 5556-5585 (2017) Article DOI: 10.1021/acs.jmedchem.7b00239 BindingDB Entry DOI: 10.7270/Q298898H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50238363 (CHEMBL4099510) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 350 | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Positive allosteric modulation of recombinant rat GluN1/GluN2C receptor expressed in xenopus laevis oocyte assessed as potentiation of glutamate and ... | J Med Chem 60: 5556-5585 (2017) Article DOI: 10.1021/acs.jmedchem.7b00239 BindingDB Entry DOI: 10.7270/Q298898H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50238335 (CHEMBL4083076) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 380 | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Positive allosteric modulation of recombinant rat GluN1/GluN2C receptor expressed in xenopus laevis oocyte assessed as potentiation of glutamate and ... | J Med Chem 60: 5556-5585 (2017) Article DOI: 10.1021/acs.jmedchem.7b00239 BindingDB Entry DOI: 10.7270/Q298898H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50545698 (CHEMBL4637429) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 398 | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Positive allosteric modulation of recombinant rat GluN1a/GluN2C receptor expressed in Xenopus laevis oocytes assessed as increase in glycine/L-glutam... | J Med Chem 63: 7569-7600 (2020) Article DOI: 10.1021/acs.jmedchem.9b01733 BindingDB Entry DOI: 10.7270/Q26D5XJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50545700 (CHEMBL4633060) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 398 | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Positive allosteric modulation of recombinant rat GluN1a/GluN2C receptor expressed in Xenopus laevis oocytes assessed as increase in glycine/L-glutam... | J Med Chem 63: 7569-7600 (2020) Article DOI: 10.1021/acs.jmedchem.9b01733 BindingDB Entry DOI: 10.7270/Q26D5XJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50545699 (CHEMBL4636021) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 398 | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Positive allosteric modulation of recombinant rat GluN1a/GluN2C receptor expressed in Xenopus laevis oocytes assessed as increase in glycine/L-glutam... | J Med Chem 63: 7569-7600 (2020) Article DOI: 10.1021/acs.jmedchem.9b01733 BindingDB Entry DOI: 10.7270/Q26D5XJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50436094 (CHEMBL2397267) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 400 | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Activity at rat recombinant GluN1/GluN2C receptor assessed as potentiation of glycine/glutamate-induced activation by two-electrode voltage clamp tec... | J Med Chem 56: 5351-81 (2014) Article DOI: 10.1021/jm400177t BindingDB Entry DOI: 10.7270/Q26W9CH4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50238350 (CHEMBL4063861) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 420 | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Positive allosteric modulation of recombinant rat GluN1/GluN2C receptor expressed in xenopus laevis oocyte assessed as potentiation of glutamate and ... | J Med Chem 60: 5556-5585 (2017) Article DOI: 10.1021/acs.jmedchem.7b00239 BindingDB Entry DOI: 10.7270/Q298898H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50238355 (CHEMBL4091770) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 480 | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Positive allosteric modulation of recombinant rat GluN1/GluN2C receptor expressed in xenopus laevis oocyte assessed as potentiation of glutamate and ... | J Med Chem 60: 5556-5585 (2017) Article DOI: 10.1021/acs.jmedchem.7b00239 BindingDB Entry DOI: 10.7270/Q298898H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50238364 (CHEMBL4064008) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 480 | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Positive allosteric modulation of recombinant rat GluN1/GluN2C receptor expressed in xenopus laevis oocyte assessed as potentiation of glutamate and ... | J Med Chem 60: 5556-5585 (2017) Article DOI: 10.1021/acs.jmedchem.7b00239 BindingDB Entry DOI: 10.7270/Q298898H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50432710 (CHEMBL2348221) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 540 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at rat recombinant wild type GluN1/GluN2C receptor expressed in Xenopus laevis oocytes by two electrode voltage clamp technique | J Med Chem 56: 4071-81 (2013) Article DOI: 10.1021/jm400346a BindingDB Entry DOI: 10.7270/Q20G3MHR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50238341 (CHEMBL4064435) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 690 | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Effect on synaptosomal uptake inhibition of 5-hydroxytryptamine (5-HT) | J Med Chem 60: 5556-5585 (2017) Article DOI: 10.1021/acs.jmedchem.7b00239 BindingDB Entry DOI: 10.7270/Q298898H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50238356 (CHEMBL4062279) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 700 | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Positive allosteric modulation of recombinant rat GluN1/GluN2C receptor expressed in xenopus laevis oocyte assessed as potentiation of glutamate and ... | J Med Chem 60: 5556-5585 (2017) Article DOI: 10.1021/acs.jmedchem.7b00239 BindingDB Entry DOI: 10.7270/Q298898H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50436095 (CHEMBL2397266) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 700 | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Activity at rat recombinant GluN1/GluN2C receptor assessed as potentiation of glycine/glutamate-induced activation by two-electrode voltage clamp tec... | J Med Chem 56: 5351-81 (2014) Article DOI: 10.1021/jm400177t BindingDB Entry DOI: 10.7270/Q26W9CH4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50238359 (CHEMBL4091772) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 710 | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Positive allosteric modulation of recombinant rat GluN1/GluN2C receptor expressed in xenopus laevis oocyte assessed as potentiation of glutamate and ... | J Med Chem 60: 5556-5585 (2017) Article DOI: 10.1021/acs.jmedchem.7b00239 BindingDB Entry DOI: 10.7270/Q298898H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50583033 (CHEMBL5092220) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 750 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at rat GluN1/GluN2C NMDA receptor expressed in Xenopus oocytes measured after 4 days in presence of L-glutamte by two-electrode volt... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c01810 BindingDB Entry DOI: 10.7270/Q21R6VFZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50545716 (CHEMBL4636029) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 794 | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Positive allosteric modulation of recombinant rat GluN1a/GluN2C receptor expressed in Xenopus laevis oocytes assessed as increase in glycine/L-glutam... | J Med Chem 63: 7569-7600 (2020) Article DOI: 10.1021/acs.jmedchem.9b01733 BindingDB Entry DOI: 10.7270/Q26D5XJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50436082 (CHEMBL2397103 | US10273214, Example 1391) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 900 | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Activity at rat recombinant GluN1/GluN2C receptor assessed as potentiation of glycine/glutamate-induced activation by two-electrode voltage clamp tec... | J Med Chem 56: 5351-81 (2014) Article DOI: 10.1021/jm400177t BindingDB Entry DOI: 10.7270/Q26W9CH4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50238338 (CHEMBL4068612) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 900 | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Positive allosteric modulation of recombinant rat GluN1/GluN2C receptor expressed in xenopus laevis oocyte assessed as potentiation of glutamate and ... | J Med Chem 60: 5556-5585 (2017) Article DOI: 10.1021/acs.jmedchem.7b00239 BindingDB Entry DOI: 10.7270/Q298898H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50436098 (CHEMBL2397262) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 900 | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Activity at rat recombinant GluN1/GluN2C receptor assessed as potentiation of glycine/glutamate-induced activation by two-electrode voltage clamp tec... | J Med Chem 56: 5351-81 (2014) Article DOI: 10.1021/jm400177t BindingDB Entry DOI: 10.7270/Q26W9CH4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50238372 (CHEMBL4083995) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 920 | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Positive allosteric modulation of recombinant rat GluN1/GluN2C receptor expressed in xenopus laevis oocyte assessed as potentiation of glutamate and ... | J Med Chem 60: 5556-5585 (2017) Article DOI: 10.1021/acs.jmedchem.7b00239 BindingDB Entry DOI: 10.7270/Q298898H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50238352 (CHEMBL4061206) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 940 | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Positive allosteric modulation of recombinant rat GluN1/GluN2C receptor expressed in xenopus laevis oocyte assessed as potentiation of glutamate and ... | J Med Chem 60: 5556-5585 (2017) Article DOI: 10.1021/acs.jmedchem.7b00239 BindingDB Entry DOI: 10.7270/Q298898H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50238351 (CHEMBL4091645) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 970 | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Positive allosteric modulation of recombinant rat GluN1/GluN2C receptor expressed in xenopus laevis oocyte assessed as potentiation of glutamate and ... | J Med Chem 60: 5556-5585 (2017) Article DOI: 10.1021/acs.jmedchem.7b00239 BindingDB Entry DOI: 10.7270/Q298898H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50237806 (CHEMBL4099073) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Positive allosteric modulation of recombinant rat GluN1/GluN2C receptor expressed in xenopus laevis oocyte assessed as potentiation of glutamate and ... | J Med Chem 60: 5556-5585 (2017) Article DOI: 10.1021/acs.jmedchem.7b00239 BindingDB Entry DOI: 10.7270/Q298898H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50436088 (CHEMBL2397121) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Activity at rat recombinant GluN1/GluN2C receptor assessed as potentiation of glycine/glutamate-induced activation by two-electrode voltage clamp tec... | J Med Chem 56: 5351-81 (2014) Article DOI: 10.1021/jm400177t BindingDB Entry DOI: 10.7270/Q26W9CH4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50238338 (CHEMBL4068612) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Positive allosteric modulation of recombinant rat GluN1a/GluN2C receptor expressed in Xenopus laevis oocytes assessed as increase in glycine/L-glutam... | J Med Chem 63: 7569-7600 (2020) Article DOI: 10.1021/acs.jmedchem.9b01733 BindingDB Entry DOI: 10.7270/Q26D5XJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50545701 (CHEMBL4648608) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Positive allosteric modulation of recombinant rat GluN1a/GluN2C receptor expressed in Xenopus laevis oocytes assessed as increase in glycine/L-glutam... | J Med Chem 63: 7569-7600 (2020) Article DOI: 10.1021/acs.jmedchem.9b01733 BindingDB Entry DOI: 10.7270/Q26D5XJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50436090 (CHEMBL2397119 | US10273214, Example 1180-31) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Activity at rat recombinant GluN1/GluN2C receptor assessed as potentiation of glycine/glutamate-induced activation by two-electrode voltage clamp tec... | J Med Chem 56: 5351-81 (2014) Article DOI: 10.1021/jm400177t BindingDB Entry DOI: 10.7270/Q26W9CH4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50238339 (CHEMBL4096621) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Positive allosteric modulation of recombinant rat GluN1/GluN2C receptor expressed in xenopus laevis oocyte assessed as potentiation of glutamate and ... | J Med Chem 60: 5556-5585 (2017) Article DOI: 10.1021/acs.jmedchem.7b00239 BindingDB Entry DOI: 10.7270/Q298898H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50545714 (CHEMBL4641889) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.26E+3 | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Positive allosteric modulation of recombinant rat GluN1a/GluN2C receptor expressed in Xenopus laevis oocytes assessed as increase in glycine/L-glutam... | J Med Chem 63: 7569-7600 (2020) Article DOI: 10.1021/acs.jmedchem.9b01733 BindingDB Entry DOI: 10.7270/Q26D5XJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50436102 (CHEMBL2397256 | US10273214, Example 1180-26) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.26E+3 | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Positive allosteric modulation of recombinant rat GluN1a/GluN2C receptor expressed in Xenopus laevis oocytes assessed as increase in glycine/L-glutam... | J Med Chem 63: 7569-7600 (2020) Article DOI: 10.1021/acs.jmedchem.9b01733 BindingDB Entry DOI: 10.7270/Q26D5XJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50545718 (CHEMBL4638424) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.26E+3 | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Positive allosteric modulation of recombinant rat GluN1a/GluN2C receptor expressed in Xenopus laevis oocytes assessed as increase in glycine/L-glutam... | J Med Chem 63: 7569-7600 (2020) Article DOI: 10.1021/acs.jmedchem.9b01733 BindingDB Entry DOI: 10.7270/Q26D5XJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50436102 (CHEMBL2397256 | US10273214, Example 1180-26) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Positive allosteric modulation of recombinant rat GluN1/GluN2C receptor expressed in xenopus laevis oocyte assessed as potentiation of glutamate and ... | J Med Chem 60: 5556-5585 (2017) Article DOI: 10.1021/acs.jmedchem.7b00239 BindingDB Entry DOI: 10.7270/Q298898H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50238370 (CHEMBL4101706) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Positive allosteric modulation of recombinant rat GluN1/GluN2C receptor expressed in xenopus laevis oocyte assessed as potentiation of glutamate and ... | J Med Chem 60: 5556-5585 (2017) Article DOI: 10.1021/acs.jmedchem.7b00239 BindingDB Entry DOI: 10.7270/Q298898H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50436102 (CHEMBL2397256 | US10273214, Example 1180-26) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Activity at rat recombinant GluN1/GluN2C receptor assessed as potentiation of glycine/glutamate-induced activation by two-electrode voltage clamp tec... | J Med Chem 56: 5351-81 (2014) Article DOI: 10.1021/jm400177t BindingDB Entry DOI: 10.7270/Q26W9CH4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50583027 (CHEMBL5076681) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at rat GluN1/GluN2C NMDA receptor expressed in Xenopus oocytes measured after 4 days in presence of L-glutamte by two-electrode volt... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c01810 BindingDB Entry DOI: 10.7270/Q21R6VFZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat)) | BDBM50583034 (CHEMBL5075942) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at rat GluN1/GluN2C NMDA receptor expressed in Xenopus oocytes measured after 4 days in presence of L-glutamte by two-electrode volt... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c01810 BindingDB Entry DOI: 10.7270/Q21R6VFZ | |||||||||||
More data for this Ligand-Target Pair |
Displayed 1 to 50 (of 201 total ) | Next | Last >> |